Basic Information

Name	[ICD-11: 2A00-2F9Z]
Protein Number	183
Molecule Number	3267

Active subnetwork

Terpenoid-protein target Activity Association

ID	Uniport	Pref_name	Gene name	value	unit	type
TKC118419	O00329	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform	None	4	nM	IC50
TKC118419	O00329	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform	None	9	nM	IC50
TKC118419	O00329	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform	None	9	nM	IC50
TKC118419	O00329	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform	None	5.5	nM	Kd
TKC001229	O14684	Prostaglandin E synthase	None	5000	nM	IC50
TKC011412	O14684	Prostaglandin E synthase	None	5000	nM	IC50
TKC051154	O14684	Prostaglandin E synthase	None	3000	nM	IC50
TKC051154	O14684	Prostaglandin E synthase	None	3000	nM	IC50
TKC061939	O14684	Prostaglandin E synthase	None	10000	nM	IC50
TKC061968	O14684	Prostaglandin E synthase	None	10000	nM	IC50
TKC061969	O14684	Prostaglandin E synthase	None	10000	nM	IC50
TKC065375	O14684	Prostaglandin E synthase	None	3000	nM	IC50
TKC095567	O14684	Prostaglandin E synthase	None	400	nM	IC50
TKC139366	O14684	Prostaglandin E synthase	None	3000	nM	IC50
TKC139366	O14684	Prostaglandin E synthase	None	10000	nM	IC50
TKC141601	O14684	Prostaglandin E synthase	None	1100	nM	IC50
TKC141602	O14684	Prostaglandin E synthase	None	1200	nM	IC50
TKC141622	O14684	Prostaglandin E synthase	None	900	nM	IC50
TKC141805	O14684	Prostaglandin E synthase	None	5000	nM	IC50
TKC141805	O14684	Prostaglandin E synthase	None	5000	nM	IC50
TKC141805	O14684	Prostaglandin E synthase	None	5000	nM	IC50
TKC142203	O14684	Prostaglandin E synthase	None	8500	nM	IC50
TKC142208	O14684	Prostaglandin E synthase	None	10000	nM	IC50
TKC150635	O14684	Prostaglandin E synthase	None	3000	nM	IC50
TKC152813	O14684	Prostaglandin E synthase	None	400	nM	IC50
TKC156572	O14684	Prostaglandin E synthase	None	900	nM	IC50
TKC174442	O14684	Prostaglandin E synthase	None	1000	nM	IC50
TKC005454	O14746	Telomerase reverse transcriptase	None	75	%	Inhibition
TKC014568	O14746	Telomerase reverse transcriptase	None	65	%	Inhibition
TKC035208	O14746	Telomerase reverse transcriptase	None	65000	nM	IC50
TKC066096	O14746	Telomerase reverse transcriptase	None	780	nM	IC50
TKC134702	O14746	Telomerase reverse transcriptase	None	4000	nM	IC50
TKC118419	O14757	Serine/threonine-protein kinase Chk1	None	87	%	Activity
TKC117625	O14763	Tumor necrosis factor receptor superfamily member 10B	None	2800	nM	EC50
TKC148385	O14786	Neuropilin-1	None	>95000	nM	IC50
TKC020117	O15151	Protein Mdm4	None	3580	nM	IC50
TKC011761	O15530	3-phosphoinositide-dependent protein kinase 1	None	46	%	Inhibition
TKC118419	O15530	3-phosphoinositide-dependent protein kinase 1	None	91	%	Activity
TKC076129	O43570	Carbonic anhydrase 12	None	2150	nM	Ki
TKC118419	O75116	Rho-associated protein kinase 2	None	99	%	Activity
TKC001786	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	4110	nM	Potency
TKC002916	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC005454	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	20596	nM	Potency
TKC005835	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	18356	nM	Potency
TKC005842	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	20596	nM	Potency
TKC008286	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	651	nM	Potency
TKC012100	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC012116	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	7308	nM	Potency
TKC013799	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	106	%	Activity
TKC014800	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	2593	nM	Potency
TKC014807	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	3264	nM	Potency
TKC016277	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	2909	nM	Potency
TKC016338	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	6513	nM	Potency
TKC016340	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	16360	nM	Potency
TKC016371	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	14581	nM	Potency
TKC016414	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC016544	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	14581	nM	Potency
TKC019863	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC020031	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC022945	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	1458	nM	Potency
TKC022996	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	88	%	Activity
TKC023041	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	107	%	Activity
TKC030034	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	116	nM	Potency
TKC031180	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	18356	nM	Potency
TKC032619	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	16360	nM	Potency
TKC035580	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	18356	nM	Potency
TKC037521	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	20596	nM	Potency
TKC038268	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	1836	nM	Potency
TKC038273	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	6513	nM	Potency
TKC039202	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	16360	nM	Potency
TKC040128	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC041149	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	46	nM	Potency
TKC041159	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	366	nM	Potency
TKC041160	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	184	nM	Potency
TKC041436	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	259	nM	Potency
TKC044085	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	164	nM	Potency
TKC048330	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	102	%	Activity
TKC048922	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC048923	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	25929	nM	Potency
TKC053726	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	109	%	Activity
TKC053815	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	10323	nM	Potency
TKC053879	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	731	nM	Potency
TKC056482	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	102	%	Activity
TKC058736	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	99	%	Activity
TKC058739	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	99	%	Activity
TKC058743	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	102	%	Activity
TKC059913	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	99	%	Activity
TKC060929	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	1300	nM	Potency
TKC062669	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	651	nM	Potency
TKC062670	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	116	nM	Potency
TKC065891	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	146	nM	Potency
TKC066096	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	4611	nM	Potency
TKC066954	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	98	%	Activity
TKC067542	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC070444	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	5805	nM	Potency
TKC072319	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	95	%	Activity
TKC075769	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	231	nM	Potency
TKC076529	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	14581	nM	Potency
TKC077689	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	101	%	Activity
TKC078094	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	206	nM	Potency
TKC082378	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	8200	nM	Potency
TKC087533	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	20596	nM	Potency
TKC090566	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	130	nM	Potency
TKC090726	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	5805	nM	Potency
TKC092297	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	14581	nM	Potency
TKC092591	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	581	nM	Potency
TKC093161	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	23109	nM	Potency
TKC093162	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	18356	nM	Potency
TKC095493	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	8200	nM	Potency
TKC096901	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	1458	nM	Potency
TKC096920	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	259	nM	Potency
TKC098410	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	6513	nM	Potency
TKC101519	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	46	nM	Potency
TKC101598	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	103	nM	Potency
TKC101922	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	291	nM	Potency
TKC101978	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	106	%	Activity
TKC102593	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	3981	nM	Potency
TKC102941	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	20596	nM	Potency
TKC103159	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	82	nM	Potency
TKC103207	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	731	nM	Potency
TKC103369	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	10323	nM	Potency
TKC103381	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	9200	nM	Potency
TKC103725	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC104088	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	18356	nM	Potency
TKC104414	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC104558	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC105753	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC106013	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	37	nM	Potency
TKC106026	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC107557	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	18356	nM	Potency
TKC107625	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	12995	nM	Potency
TKC108316	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	3663	nM	Potency
TKC108793	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC109519	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	18	nM	Potency
TKC109594	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	82	nM	Potency
TKC109881	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	206	nM	Potency
TKC110956	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	820	nM	Potency
TKC112576	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	130	nM	Potency
TKC113063	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	20596	nM	Potency
TKC114015	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC117617	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	1300	nM	Potency
TKC117638	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	1032	nM	Potency
TKC117993	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	1158	nM	Potency
TKC118131	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	920	nM	Potency
TKC118419	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	19953	nM	Potency
TKC122884	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	96	%	Activity
TKC122980	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	99	%	Activity
TKC122982	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	101	%	Activity
TKC123088	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	102	%	Activity
TKC129004	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	5	nM	Potency
TKC129193	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC132374	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC132609	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	18356	nM	Potency
TKC134702	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	1458	nM	Potency
TKC134744	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	12995	nM	Potency
TKC135702	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	2311	nM	Potency
TKC136632	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC138054	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	105	%	Activity
TKC143227	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	20596	nM	Potency
TKC143885	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	18356	nM	Potency
TKC145932	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	105	%	Activity
TKC148160	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	103	%	Activity
TKC149344	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	106	%	Activity
TKC151303	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	731	nM	Potency
TKC151443	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC151609	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	20596	nM	Potency
TKC151966	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	106	%	Activity
TKC151971	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	93	%	Activity
TKC152765	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	104	%	Activity
TKC156644	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	6513	nM	Potency
TKC159332	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	3663	nM	Potency
TKC162991	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	5	nM	Potency
TKC168160	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	18356	nM	Potency
TKC174441	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	16360	nM	Potency
TKC197335	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	206	nM	Potency
TKC197337	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	7	nM	Potency
TKC197340	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	7	nM	Potency
TKC202992	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	41	nM	Potency
TKC205407	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	184	nM	Potency
TKC205699	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	2311	nM	Potency
TKC205700	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	2311	nM	Potency
TKC205928	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	366	nM	Potency
TKC206362	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	2311	nM	Potency
TKC206395	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	37	nM	Potency
TKC206589	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	50119	nM	Potency
TKC206652	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	206	nM	Potency
TKC206660	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	1458	nM	Potency
TKC206686	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	25929	nM	Potency
TKC206688	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	29093	nM	Potency
TKC206754	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	5174	nM	Potency
TKC206777	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	23109	nM	Potency
TKC206780	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	18356	nM	Potency
TKC206781	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	9200	nM	Potency
TKC206783	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	39811	nM	Potency
TKC206816	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	23109	nM	Potency
TKC206872	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	2060	nM	Potency
TKC206876	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	4611	nM	Potency
TKC206884	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	16360	nM	Potency
TKC206889	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	1636	nM	Potency
TKC207267	O75874	Isocitrate dehydrogenase [NADP] cytoplasmic	None	517	nM	Potency
TKC002908	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	89125	nM	Potency
TKC005454	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	79433	nM	Potency
TKC008359	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	79433	nM	Potency
TKC008529	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC011709	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC013304	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	19953	nM	Potency
TKC013323	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	35481	nM	Potency
TKC014568	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	28184	nM	Potency
TKC016544	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	31623	nM	Potency
TKC018288	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	44668	nM	Potency
TKC019887	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC019913	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC020944	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	20	nM	Potency
TKC023148	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	1778	nM	Potency
TKC026870	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	10000	nM	Potency
TKC027192	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	28184	nM	Potency
TKC030469	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	56234	nM	Potency
TKC034632	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC034640	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	63096	nM	Potency
TKC034641	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	63096	nM	Potency
TKC035272	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	10000	nM	Potency
TKC035984	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	19953	nM	Potency
TKC038756	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	89125	nM	Potency
TKC039332	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	22387	nM	Potency
TKC041411	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	3981	nM	Potency
TKC044884	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC047194	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	79433	nM	Potency
TKC048330	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	8913	nM	Potency
TKC048341	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	355	nM	Potency
TKC053095	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC053825	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	63096	nM	Potency
TKC055972	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	79433	nM	Potency
TKC057133	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	35481	nM	Potency
TKC062321	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	89125	nM	Potency
TKC062333	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	56234	nM	Potency
TKC066332	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	44668	nM	Potency
TKC068076	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	56234	nM	Potency
TKC070979	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	1122019	nM	Potency
TKC079223	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC083025	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	56234	nM	Potency
TKC083534	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC084630	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	63096	nM	Potency
TKC087533	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	355	nM	Potency
TKC087664	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	79433	nM	Potency
TKC088815	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	447	nM	Potency
TKC091895	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	22387	nM	Potency
TKC092297	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	28184	nM	Potency
TKC092943	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	7943	nM	Potency
TKC093162	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	79433	nM	Potency
TKC095638	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	35481	nM	Potency
TKC096012	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	56234	nM	Potency
TKC097727	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	251	nM	Potency
TKC097937	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC098345	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	79433	nM	Potency
TKC099703	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	56234	nM	Potency
TKC100636	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	22387	nM	Potency
TKC100649	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	12589	nM	Potency
TKC100701	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	22387	nM	Potency
TKC101111	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	22387	nM	Potency
TKC102080	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	251	nM	Potency
TKC102145	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	35481	nM	Potency
TKC102173	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	316	nM	Potency
TKC102204	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC102540	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	44668	nM	Potency
TKC102743	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC103257	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	44668	nM	Potency
TKC103542	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	70795	nM	Potency
TKC103736	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	89125	nM	Potency
TKC103799	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	56234	nM	Potency
TKC103984	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	79433	nM	Potency
TKC104293	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	89125	nM	Potency
TKC104404	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	79433	nM	Potency
TKC104435	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	63096	nM	Potency
TKC104602	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC104656	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC105153	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	44668	nM	Potency
TKC105168	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC105343	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	112202	nM	Potency
TKC105360	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC105378	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC105424	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC105530	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	44668	nM	Potency
TKC105784	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	44668	nM	Potency
TKC105891	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	22387	nM	Potency
TKC106426	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	7943	nM	Potency
TKC106621	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	25119	nM	Potency
TKC106952	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	3548	nM	Potency
TKC107104	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	25119	nM	Potency
TKC107201	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	31623	nM	Potency
TKC107332	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC107499	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	5012	nM	Potency
TKC107525	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	22387	nM	Potency
TKC107625	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC107818	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC107830	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC107871	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	56234	nM	Potency
TKC107944	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	100000	nM	Potency
TKC108295	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	63096	nM	Potency
TKC108732	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	25119	nM	Potency
TKC110162	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	44668	nM	Potency
TKC111464	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	79433	nM	Potency
TKC112754	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	89125	nM	Potency
TKC112759	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	50119	nM	Potency
TKC112784	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	79433	nM	Potency
TKC112792	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	63096	nM	Potency
TKC112826	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	10000	nM	Potency
TKC112920	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	7080	nM	Potency
TKC112929	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC113146	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	44668	nM	Potency
TKC113149	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC114819	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	35481	nM	Potency
TKC115263	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	17783	nM	Potency
TKC115268	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	44668	nM	Potency
TKC115284	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	56234	nM	Potency
TKC117710	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	31623	nM	Potency
TKC118419	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC118895	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	89125	nM	Potency
TKC122892	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	56234	nM	Potency
TKC123129	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	79433	nM	Potency
TKC134702	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	8913	nM	Potency
TKC134744	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	35481	nM	Potency
TKC135961	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	89125	nM	Potency
TKC138780	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	56234	nM	Potency
TKC139094	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	5012	nM	Potency
TKC140412	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	3981	nM	Potency
TKC141824	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	794	nM	Potency
TKC145824	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	316	nM	Potency
TKC146423	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	100000	nM	Potency
TKC147252	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	35481	nM	Potency
TKC147290	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC148482	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC148601	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	44668	nM	Potency
TKC151321	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	251	nM	Potency
TKC151327	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	5012	nM	Potency
TKC151519	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	15849	nM	Potency
TKC151675	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	31623	nM	Potency
TKC205806	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	31623	nM	Potency
TKC205926	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	25119	nM	Potency
TKC206042	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	28184	nM	Potency
TKC206365	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	100000	nM	Potency
TKC206387	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC206622	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	35481	nM	Potency
TKC206754	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	35481	nM	Potency
TKC206758	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	35481	nM	Potency
TKC206760	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	56234	nM	Potency
TKC206765	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	7080	nM	Potency
TKC206766	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	39811	nM	Potency
TKC206767	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	7943	nM	Potency
TKC206771	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	89125	nM	Potency
TKC206777	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	3162	nM	Potency
TKC206781	O94782	Ubiquitin carboxyl-terminal hydrolase 1	None	44668	nM	Potency
TKC118419	O96013	Serine/threonine-protein kinase PAK 4	None	90	%	Activity
TKC118419	O96017	Serine/threonine-protein kinase Chk2	None	90	%	Activity
TKC010047	P00441	Superoxide dismutase [Cu-Zn]	None	56600	nM	IC50
TKC151761	P00519	Tyrosine-protein kinase ABL1	None	>10000	nM	IC50
TKC200866	P00519	Tyrosine-protein kinase ABL1	None	>10000	nM	IC50
TKC007127	P00533	Epidermal growth factor receptor	None	19	%	Inhibition
TKC025462	P00533	Epidermal growth factor receptor	None	>200	ug.mL-1	IC50
TKC025466	P00533	Epidermal growth factor receptor	None	>200	ug.mL-1	IC50
TKC025475	P00533	Epidermal growth factor receptor	None	197	ug.mL-1	IC50
TKC071640	P00533	Epidermal growth factor receptor	None	>20000	nM	IC50
TKC076041	P00533	Epidermal growth factor receptor	None	75	%	Inhibition
TKC077689	P00533	Epidermal growth factor receptor	None	>20000	nM	IC50
TKC106319	P00533	Epidermal growth factor receptor	None	56	nM	IC50
TKC108557	P00533	Epidermal growth factor receptor	None	0.82	nM	Kd
TKC151761	P00533	Epidermal growth factor receptor	None	>10000	nM	IC50
TKC200866	P00533	Epidermal growth factor receptor	None	>10000	nM	IC50
TKC055903	P00734	Prothrombin	None	4	nM	IC50
TKC055903	P00734	Prothrombin	None	50	nM	IC50
TKC064786	P00734	Prothrombin	None	130	nM	IC50
TKC064787	P00734	Prothrombin	None	70	nM	IC50
TKC101989	P00734	Prothrombin	None	4000	nM	IC50
TKC106074	P00734	Prothrombin	None	>50000	nM	IC50
TKC106074	P00734	Prothrombin	None	>50000	nM	IC50
TKC122980	P00734	Prothrombin	None	9200	nM	IC50
TKC139119	P00734	Prothrombin	None	90	nM	IC50
TKC141433	P00734	Prothrombin	None	18	nM	IC50
TKC005744	P00742	Coagulation factor X	None	27900	nM	IC50
TKC012492	P00742	Coagulation factor X	None	13385	nM	Ki
TKC013400	P00742	Coagulation factor X	None	2500	nM	IC50
TKC013430	P00742	Coagulation factor X	None	11418	nM	IC50
TKC055903	P00742	Coagulation factor X	None	>20000	nM	IC50
TKC107140	P00742	Coagulation factor X	None	7991	nM	Ki
TKC124270	P00742	Coagulation factor X	None	27558	nM	Ki
TKC128698	P00742	Coagulation factor X	None	7200	nM	IC50
TKC128699	P00742	Coagulation factor X	None	7165	nM	IC50
TKC205733	P00742	Coagulation factor X	None	1023	nM	IC50
TKC073833	P00749	Urokinase-type plasminogen activator	None	58479	nM	Potency
TKC076529	P00749	Urokinase-type plasminogen activator	None	23281	nM	Potency
TKC082279	P00749	Urokinase-type plasminogen activator	None	52119	nM	Potency
TKC076129	P00915	Carbonic anhydrase 1	None	8010	nM	Ki
TKC104783	P00915	Carbonic anhydrase 1	None	2210	nM	Ki
TKC105780	P00915	Carbonic anhydrase 1	None	1470	nM	Ki
TKC076129	P00918	Carbonic anhydrase 2	None	6130	nM	Ki
TKC104783	P00918	Carbonic anhydrase 2	None	1280	nM	Ki
TKC105780	P00918	Carbonic anhydrase 2	None	970	nM	Ki
TKC112756	P00918	Carbonic anhydrase 2	None	>10000	nM	IC50
TKC143885	P01106	Myc proto-oncogene protein	None	4000000	nM	IC50
TKC117397	P01112	GTPase HRas	None	2	ug.mL-1	IC50
TKC051021	P01375	Tumor necrosis factor	None	9	nM	Kd
TKC051029	P01375	Tumor necrosis factor	None	9	nM	Kd
TKC055869	P01375	Tumor necrosis factor	None	10880	nM	IC50
TKC063751	P01375	Tumor necrosis factor	None	19	nM	Kd
TKC064986	P01375	Tumor necrosis factor	None	3	nM	Kd
TKC075769	P01375	Tumor necrosis factor	None	376	nM	Potency
TKC101833	P01375	Tumor necrosis factor	None	8	nM	Kd
TKC145547	P01375	Tumor necrosis factor	None	2	nM	Kd
TKC148618	P01375	Tumor necrosis factor	None	17	nM	Kd
TKC151763	P01375	Tumor necrosis factor	None	8	nM	Kd
TKC151876	P01375	Tumor necrosis factor	None	6	%	Inhibition
TKC013753	P03372	Estrogen receptor	None	8913	nM	Potency
TKC019072	P03372	Estrogen receptor	None	78	%	Activity
TKC022931	P03372	Estrogen receptor	None	1995	nM	Potency
TKC022961	P03372	Estrogen receptor	None	54	%	Activity
TKC028029	P03372	Estrogen receptor	None	0	%	Activity
TKC028034	P03372	Estrogen receptor	None	<0	%	Activity
TKC028037	P03372	Estrogen receptor	None	1	%	Activity
TKC028038	P03372	Estrogen receptor	None	<0	%	Activity
TKC028041	P03372	Estrogen receptor	None	<0	%	Activity
TKC034016	P03372	Estrogen receptor	None	51	%	Activity
TKC034337	P03372	Estrogen receptor	None	2800000	nM	IC50
TKC034640	P03372	Estrogen receptor	None	>1000000	nM	Ki
TKC035208	P03372	Estrogen receptor	None	39	%	Activity
TKC035272	P03372	Estrogen receptor	None	2551	nM	IC50
TKC035462	P03372	Estrogen receptor	None	42	%	Activity
TKC066169	P03372	Estrogen receptor	None	39811	nM	Potency
TKC075769	P03372	Estrogen receptor	None	251	nM	Potency
TKC079320	P03372	Estrogen receptor	None	<0	%	Activity
TKC079321	P03372	Estrogen receptor	None	<0	%	Activity
TKC087664	P03372	Estrogen receptor	None	3162	nM	Potency
TKC087988	P03372	Estrogen receptor	None	631	nM	Potency
TKC087991	P03372	Estrogen receptor	None	4467	nM	Potency
TKC092297	P03372	Estrogen receptor	None	15849	nM	Potency
TKC092348	P03372	Estrogen receptor	None	8913	nM	Potency
TKC096012	P03372	Estrogen receptor	None	126	nM	Potency
TKC100644	P03372	Estrogen receptor	None	31623	nM	Potency
TKC101365	P03372	Estrogen receptor	None	12570	nM	EC50
TKC102448	P03372	Estrogen receptor	None	2550	nM	EC50
TKC107086	P03372	Estrogen receptor	None	8913	nM	Potency
TKC107735	P03372	Estrogen receptor	None	50119	nM	Potency
TKC111727	P03372	Estrogen receptor	None	0	nM	Ki
TKC111738	P03372	Estrogen receptor	None	1	nM	EC50
TKC111738	P03372	Estrogen receptor	None	166	nM	IC50
TKC111738	P03372	Estrogen receptor	None	210	nM	IC50
TKC111738	P03372	Estrogen receptor	None	96	nM	IC50
TKC112923	P03372	Estrogen receptor	None	26	nM	EC50
TKC115268	P03372	Estrogen receptor	None	15849	nM	Potency
TKC129821	P03372	Estrogen receptor	None	70	%	Activity
TKC151345	P03372	Estrogen receptor	None	35	%	Activity
TKC151713	P03372	Estrogen receptor	None	40	%	Activity
TKC151765	P03372	Estrogen receptor	None	81	%	Activity
TKC206549	P03372	Estrogen receptor	None	3548	nM	Potency
TKC206608	P03372	Estrogen receptor	None	8170	nM	EC50
TKC206652	P03372	Estrogen receptor	None	112	nM	Potency
TKC206725	P03372	Estrogen receptor	None	8	nM	Ki
TKC206726	P03372	Estrogen receptor	None	72	nM	EC50
TKC206759	P03372	Estrogen receptor	None	>10000	nM	IC50
TKC206759	P03372	Estrogen receptor	None	>10000	nM	IC50
TKC206760	P03372	Estrogen receptor	None	25119	nM	Potency
TKC206764	P03372	Estrogen receptor	None	0	%	RBA
TKC206770	P03372	Estrogen receptor	None	5012	nM	Potency
TKC206779	P03372	Estrogen receptor	None	6310	nM	Potency
TKC206812	P03372	Estrogen receptor	None	62000	nM	IC50
TKC206812	P03372	Estrogen receptor	None	39811	nM	Potency
TKC206816	P03372	Estrogen receptor	None	>1000	nM	IC50
TKC206816	P03372	Estrogen receptor	None	>1000	nM	IC50
TKC020117	P03956	Interstitial collagenase	None	95	%	Inhibition
TKC013753	P04150	Glucocorticoid receptor	None	5012	nM	Potency
TKC019368	P04150	Glucocorticoid receptor	None	10000	nM	Potency
TKC021365	P04150	Glucocorticoid receptor	None	5623	nM	Potency
TKC021425	P04150	Glucocorticoid receptor	None	5623	nM	Potency
TKC023246	P04150	Glucocorticoid receptor	None	>3210	nM	Ki
TKC023246	P04150	Glucocorticoid receptor	None	2465	nM	Ki
TKC030239	P04150	Glucocorticoid receptor	None	30	nM	Ki
TKC030239	P04150	Glucocorticoid receptor	None	69	%	Inhibition
TKC035272	P04150	Glucocorticoid receptor	None	44668	nM	Potency
TKC048937	P04150	Glucocorticoid receptor	None	56	%	Inhibition
TKC063171	P04150	Glucocorticoid receptor	None	56	%	Inhibition
TKC074866	P04150	Glucocorticoid receptor	None	25119	nM	Potency
TKC075769	P04150	Glucocorticoid receptor	None	562	nM	Potency
TKC081853	P04150	Glucocorticoid receptor	None	84	%	Activity
TKC087664	P04150	Glucocorticoid receptor	None	4	nM	Potency
TKC087988	P04150	Glucocorticoid receptor	None	1995	nM	Potency
TKC092297	P04150	Glucocorticoid receptor	None	794	nM	Potency
TKC096011	P04150	Glucocorticoid receptor	None	1	nM	Ki
TKC106250	P04150	Glucocorticoid receptor	None	298700	nM	EC50
TKC106877	P04150	Glucocorticoid receptor	None	2465	nM	Ki
TKC106878	P04150	Glucocorticoid receptor	None	>2465	nM	Ki
TKC106878	P04150	Glucocorticoid receptor	None	3210	nM	Ki
TKC106879	P04150	Glucocorticoid receptor	None	3210	nM	Ki
TKC107086	P04150	Glucocorticoid receptor	None	8913	nM	Potency
TKC109619	P04150	Glucocorticoid receptor	None	298700	nM	EC50
TKC111727	P04150	Glucocorticoid receptor	None	17884	nM	Ki
TKC114511	P04150	Glucocorticoid receptor	None	252	nM	Ki
TKC115268	P04150	Glucocorticoid receptor	None	50119	nM	Potency
TKC122884	P04150	Glucocorticoid receptor	None	11220	nM	Potency
TKC134780	P04150	Glucocorticoid receptor	None	4	nM	Potency
TKC136411	P04150	Glucocorticoid receptor	None	1	nM	Potency
TKC183618	P04150	Glucocorticoid receptor	None	70	%	Activity
TKC206652	P04150	Glucocorticoid receptor	None	355	nM	Potency
TKC206672	P04150	Glucocorticoid receptor	None	50119	nM	Potency
TKC206688	P04150	Glucocorticoid receptor	None	501	nM	Potency
TKC206690	P04150	Glucocorticoid receptor	None	28184	nM	Potency
TKC206759	P04150	Glucocorticoid receptor	None	1457	nM	Ki
TKC206760	P04150	Glucocorticoid receptor	None	39811	nM	Potency
TKC206770	P04150	Glucocorticoid receptor	None	2818	nM	Potency
TKC206779	P04150	Glucocorticoid receptor	None	23	nM	Ki
TKC206812	P04150	Glucocorticoid receptor	None	224	nM	Ki
TKC206816	P04150	Glucocorticoid receptor	None	31	nM	Ki
TKC206816	P04150	Glucocorticoid receptor	None	31	nM	Ki
TKC206816	P04150	Glucocorticoid receptor	None	31	nM	Ki
TKC206816	P04150	Glucocorticoid receptor	None	31	nM	Ki
TKC206816	P04150	Glucocorticoid receptor	None	31	nM	Ki
TKC206816	P04150	Glucocorticoid receptor	None	>1000	nM	IC50
TKC206816	P04150	Glucocorticoid receptor	None	>1000	nM	IC50
TKC206816	P04150	Glucocorticoid receptor	None	31	nM	Ki
TKC025462	P04626	Receptor tyrosine-protein kinase erbB-2	None	>200	ug.mL-1	IC50
TKC025466	P04626	Receptor tyrosine-protein kinase erbB-2	None	>200	ug.mL-1	IC50
TKC025475	P04626	Receptor tyrosine-protein kinase erbB-2	None	125	ug.mL-1	IC50
TKC026211	P04626	Receptor tyrosine-protein kinase erbB-2	None	6	ug.mL-1	IC50
TKC026214	P04626	Receptor tyrosine-protein kinase erbB-2	None	8	ug.mL-1	IC50
TKC026217	P04626	Receptor tyrosine-protein kinase erbB-2	None	4	ug.mL-1	IC50
TKC026229	P04626	Receptor tyrosine-protein kinase erbB-2	None	8	ug.mL-1	IC50
TKC012971	P04637	Cellular tumor antigen p53	None	15849	nM	Potency
TKC013753	P04637	Cellular tumor antigen p53	None	13	nM	Potency
TKC014568	P04637	Cellular tumor antigen p53	None	2512	nM	Potency
TKC016418	P04637	Cellular tumor antigen p53	None	15849	nM	Potency
TKC018710	P04637	Cellular tumor antigen p53	None	5	nM	Potency
TKC020116	P04637	Cellular tumor antigen p53	None	1585	nM	Potency
TKC020117	P04637	Cellular tumor antigen p53	None	12589	nM	Potency
TKC020732	P04637	Cellular tumor antigen p53	None	3162	nM	Potency
TKC022945	P04637	Cellular tumor antigen p53	None	10000	nM	Potency
TKC032619	P04637	Cellular tumor antigen p53	None	15849	nM	Potency
TKC034083	P04637	Cellular tumor antigen p53	None	31623	nM	Potency
TKC035272	P04637	Cellular tumor antigen p53	None	12589	nM	Potency
TKC039869	P04637	Cellular tumor antigen p53	None	25119	nM	Potency
TKC052854	P04637	Cellular tumor antigen p53	None	25119	nM	Potency
TKC062321	P04637	Cellular tumor antigen p53	None	10000	nM	Potency
TKC075769	P04637	Cellular tumor antigen p53	None	159	nM	Potency
TKC084075	P04637	Cellular tumor antigen p53	None	8	nM	Potency
TKC091895	P04637	Cellular tumor antigen p53	None	50119	nM	Potency
TKC092297	P04637	Cellular tumor antigen p53	None	15849	nM	Potency
TKC095493	P04637	Cellular tumor antigen p53	None	3162	nM	Potency
TKC100636	P04637	Cellular tumor antigen p53	None	1585	nM	Potency
TKC100701	P04637	Cellular tumor antigen p53	None	10000	nM	Potency
TKC101020	P04637	Cellular tumor antigen p53	None	12589	nM	Potency
TKC101618	P04637	Cellular tumor antigen p53	None	12589	nM	Potency
TKC102204	P04637	Cellular tumor antigen p53	None	31623	nM	Potency
TKC102540	P04637	Cellular tumor antigen p53	None	31623	nM	Potency
TKC103149	P04637	Cellular tumor antigen p53	None	12589	nM	Potency
TKC103210	P04637	Cellular tumor antigen p53	None	40	nM	Potency
TKC103257	P04637	Cellular tumor antigen p53	None	10000	nM	Potency
TKC103736	P04637	Cellular tumor antigen p53	None	2512	nM	Potency
TKC104070	P04637	Cellular tumor antigen p53	None	63	nM	Potency
TKC104071	P04637	Cellular tumor antigen p53	None	50	nM	Potency
TKC104072	P04637	Cellular tumor antigen p53	None	126	nM	Potency
TKC104073	P04637	Cellular tumor antigen p53	None	63	nM	Potency
TKC104114	P04637	Cellular tumor antigen p53	None	79	nM	Potency
TKC105153	P04637	Cellular tumor antigen p53	None	5012	nM	Potency
TKC105168	P04637	Cellular tumor antigen p53	None	12589	nM	Potency
TKC105360	P04637	Cellular tumor antigen p53	None	15849	nM	Potency
TKC105424	P04637	Cellular tumor antigen p53	None	25119	nM	Potency
TKC105784	P04637	Cellular tumor antigen p53	None	25119	nM	Potency
TKC105891	P04637	Cellular tumor antigen p53	None	10000	nM	Potency
TKC106232	P04637	Cellular tumor antigen p53	None	15849	nM	Potency
TKC107086	P04637	Cellular tumor antigen p53	None	12589	nM	Potency
TKC107104	P04637	Cellular tumor antigen p53	None	12589	nM	Potency
TKC107201	P04637	Cellular tumor antigen p53	None	19953	nM	Potency
TKC107332	P04637	Cellular tumor antigen p53	None	10000	nM	Potency
TKC107525	P04637	Cellular tumor antigen p53	None	31623	nM	Potency
TKC107627	P04637	Cellular tumor antigen p53	None	25119	nM	Potency
TKC107818	P04637	Cellular tumor antigen p53	None	12589	nM	Potency
TKC108536	P04637	Cellular tumor antigen p53	None	5	nM	Potency
TKC108732	P04637	Cellular tumor antigen p53	None	19953	nM	Potency
TKC109484	P04637	Cellular tumor antigen p53	None	20	nM	Potency
TKC109519	P04637	Cellular tumor antigen p53	None	10000	nM	Potency
TKC109561	P04637	Cellular tumor antigen p53	None	159	nM	Potency
TKC109569	P04637	Cellular tumor antigen p53	None	32	nM	Potency
TKC110010	P04637	Cellular tumor antigen p53	None	56234	nM	Potency
TKC112576	P04637	Cellular tumor antigen p53	None	50	nM	Potency
TKC112784	P04637	Cellular tumor antigen p53	None	31623	nM	Potency
TKC112792	P04637	Cellular tumor antigen p53	None	25119	nM	Potency
TKC115268	P04637	Cellular tumor antigen p53	None	70795	nM	Potency
TKC117625	P04637	Cellular tumor antigen p53	None	3162	nM	Potency
TKC117993	P04637	Cellular tumor antigen p53	None	501	nM	Potency
TKC117994	P04637	Cellular tumor antigen p53	None	40	nM	Potency
TKC118006	P04637	Cellular tumor antigen p53	None	100	nM	Potency
TKC118895	P04637	Cellular tumor antigen p53	None	31623	nM	Potency
TKC132609	P04637	Cellular tumor antigen p53	None	11220	nM	Potency
TKC134635	P04637	Cellular tumor antigen p53	None	56234	nM	Potency
TKC138777	P04637	Cellular tumor antigen p53	None	15849	nM	Potency
TKC140757	P04637	Cellular tumor antigen p53	None	31623	nM	Potency
TKC147290	P04637	Cellular tumor antigen p53	None	12589	nM	Potency
TKC148482	P04637	Cellular tumor antigen p53	None	19953	nM	Potency
TKC149827	P04637	Cellular tumor antigen p53	None	1000	nM	Potency
TKC150706	P04637	Cellular tumor antigen p53	None	31623	nM	Potency
TKC151237	P04637	Cellular tumor antigen p53	None	35481	nM	Potency
TKC151303	P04637	Cellular tumor antigen p53	None	31623	nM	Potency
TKC151571	P04637	Cellular tumor antigen p53	None	6310	nM	Potency
TKC151758	P04637	Cellular tumor antigen p53	None	19953	nM	Potency
TKC173955	P04637	Cellular tumor antigen p53	None	31623	nM	Potency
TKC206652	P04637	Cellular tumor antigen p53	None	32	nM	Potency
TKC206657	P04637	Cellular tumor antigen p53	None	8	nM	Potency
TKC206760	P04637	Cellular tumor antigen p53	None	31623	nM	Potency
TKC206760	P04637	Cellular tumor antigen p53	None	15000	nM	Kd
TKC206812	P04637	Cellular tumor antigen p53	None	31623	nM	Potency
TKC206872	P04637	Cellular tumor antigen p53	None	631	nM	Potency
TKC206889	P04637	Cellular tumor antigen p53	None	501	nM	Potency
TKC206901	P04637	Cellular tumor antigen p53	None	2512	nM	Potency
TKC017481	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	5000	nM	IC50
TKC023239	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	124	ug.mL-1	IC50
TKC023241	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>128	ug.mL-1	IC50
TKC025769	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	4	ug.mL-1	IC50
TKC027669	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	44000	nM	IC50
TKC027670	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	44000	nM	IC50
TKC027671	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	3000	nM	IC50
TKC027672	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	4000	nM	IC50
TKC045766	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	19000	nM	IC50
TKC045769	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	17000	nM	IC50
TKC045770	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	5000	nM	IC50
TKC045946	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	5000	nM	IC50
TKC045992	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	18000	nM	IC50
TKC046480	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	9000	nM	IC50
TKC049704	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100	ug.mL-1	IC50
TKC052207	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100	ug.mL-1	IC50
TKC055009	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100	ug.mL-1	IC50
TKC055012	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100	ug.mL-1	IC50
TKC055482	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	54	ug.mL-1	IC50
TKC063713	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100	ug.mL-1	IC50
TKC063714	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100	ug.mL-1	IC50
TKC063989	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100	ug.mL-1	IC50
TKC063990	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100	ug.mL-1	IC50
TKC063991	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100	ug.mL-1	IC50
TKC075769	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	400	nM	IC50
TKC075769	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	290	nM	IC50
TKC075769	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	189	nM	Ki
TKC075769	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	268	nM	Ki
TKC091539	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	18000	nM	IC50
TKC091545	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	14000	nM	IC50
TKC091549	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	6000	nM	IC50
TKC101866	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	117000	nM	IC50
TKC102035	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100000	nM	IC50
TKC102240	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100000	nM	IC50
TKC105362	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	6000	nM	IC50
TKC107166	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	5000	nM	IC50
TKC107681	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	5	nM	IC50
TKC107785	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	22	ug.mL-1	IC50
TKC108159	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100000	nM	IC50
TKC109568	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	18	nM	IC50
TKC112576	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	6000	nM	IC50
TKC112576	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	97	nM	Ki
TKC113001	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	54	ug.mL-1	IC50
TKC117375	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>128000	nM	IC50
TKC117612	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	196	nM	Ki
TKC141213	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	60	ug.mL-1	IC50
TKC149884	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	1090	nM	IC50
TKC164053	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100000	nM	IC50
TKC164226	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	59	ug.mL-1	IC50
TKC164227	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	59	ug.mL-1	IC50
TKC164286	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100000	nM	IC50
TKC171641	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100000	nM	IC50
TKC173723	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	60	ug.mL-1	IC50
TKC173962	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100000	nM	IC50
TKC175484	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100	ug.mL-1	IC50
TKC176831	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	54	ug.mL-1	IC50
TKC194807	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	>100	ug.mL-1	IC50
TKC206652	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	8	nM	IC50
TKC206652	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	89	nM	Ki
TKC206660	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	8	nM	IC50
TKC206661	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	7	nM	IC50
TKC206662	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	87	nM	IC50
TKC206872	P05023	Sodium/potassium-transporting ATPase subunit alpha-1	None	139	nM	Ki
TKC022945	P05067	Amyloid-beta precursor protein	None	23109	nM	Potency
TKC027272	P05067	Amyloid-beta precursor protein	None	>300000	nM	EC50
TKC027273	P05067	Amyloid-beta precursor protein	None	65400	nM	EC50
TKC050321	P05067	Amyloid-beta precursor protein	None	100	%	Activity
TKC050560	P05067	Amyloid-beta precursor protein	None	0	%	Inhibition
TKC051308	P05067	Amyloid-beta precursor protein	None	0	%	Inhibition
TKC059731	P05067	Amyloid-beta precursor protein	None	39	%	Activity
TKC060461	P05067	Amyloid-beta precursor protein	None	65	%	Activity
TKC077689	P05067	Amyloid-beta precursor protein	None	100	%	Activity
TKC102625	P05067	Amyloid-beta precursor protein	None	0	%	Inhibition
TKC111348	P05067	Amyloid-beta precursor protein	None	17	%	Activity
TKC113610	P05067	Amyloid-beta precursor protein	None	20	%	Activity
TKC113764	P05067	Amyloid-beta precursor protein	None	71900	nM	IC50
TKC113765	P05067	Amyloid-beta precursor protein	None	28000	nM	IC50
TKC113766	P05067	Amyloid-beta precursor protein	None	34300	nM	IC50
TKC113767	P05067	Amyloid-beta precursor protein	None	55	%	Inhibition
TKC113768	P05067	Amyloid-beta precursor protein	None	43500	nM	IC50
TKC113769	P05067	Amyloid-beta precursor protein	None	1200	nM	IC50
TKC118380	P05067	Amyloid-beta precursor protein	None	13400	nM	IC50
TKC118381	P05067	Amyloid-beta precursor protein	None	10100	nM	IC50
TKC118419	P05067	Amyloid-beta precursor protein	None	231	nM	Potency
TKC123071	P05067	Amyloid-beta precursor protein	None	20	%	Activity
TKC150909	P05067	Amyloid-beta precursor protein	None	0	%	Activity
TKC152398	P05067	Amyloid-beta precursor protein	None	100000	nM	IC50
TKC179988	P05067	Amyloid-beta precursor protein	None	8	hr	TIME
TKC206799	P05067	Amyloid-beta precursor protein	None	95900	nM	IC50
TKC012929	P05771	Protein kinase C beta type	None	2	nM	Ki
TKC055602	P05771	Protein kinase C beta type	None	>150000	nM	IC50
TKC075924	P05771	Protein kinase C beta type	None	90	%	Inhibition
TKC090435	P05771	Protein kinase C beta type	None	0.2	nM	Kd
TKC103074	P05771	Protein kinase C beta type	None	>150000	nM	IC50
TKC104128	P05771	Protein kinase C beta type	None	>150000	nM	IC50
TKC104703	P05771	Protein kinase C beta type	None	>150000	nM	IC50
TKC105956	P05771	Protein kinase C beta type	None	2	nM	Ki
TKC123088	P05771	Protein kinase C beta type	None	>150000	nM	IC50
TKC151276	P05771	Protein kinase C beta type	None	>150000	nM	IC50
TKC151326	P05771	Protein kinase C beta type	None	1	nM	Kd
TKC151326	P05771	Protein kinase C beta type	None	1.3	nM	Kd
TKC151326	P05771	Protein kinase C beta type	None	1.3	nM	Kd
TKC151326	P05771	Protein kinase C beta type	None	1.8	nM	Ki
TKC151326	P05771	Protein kinase C beta type	None	1.3	nM	Kd
TKC151326	P05771	Protein kinase C beta type	None	1.3	nM	Kd
TKC152742	P05771	Protein kinase C beta type	None	>150000	nM	IC50
TKC026717	P06239	Tyrosine-protein kinase Lck	None	80	ug.mL-1	IC50
TKC046110	P06239	Tyrosine-protein kinase Lck	None	45	%	Activity
TKC105249	P06239	Tyrosine-protein kinase Lck	None	92	ug.mL-1	IC50
TKC111609	P06239	Tyrosine-protein kinase Lck	None	47	%	Activity
TKC111658	P06239	Tyrosine-protein kinase Lck	None	42	%	Activity
TKC118419	P06239	Tyrosine-protein kinase Lck	None	95	%	Inhibition
TKC023246	P06401	Progesterone receptor	None	<354	nM	IC50
TKC048937	P06401	Progesterone receptor	None	64	%	Inhibition
TKC063171	P06401	Progesterone receptor	None	66	%	Inhibition
TKC106878	P06401	Progesterone receptor	None	35	nM	EC50
TKC114511	P06401	Progesterone receptor	None	224	nM	Ki
TKC206759	P06401	Progesterone receptor	None	0	%	Binding
TKC206812	P06401	Progesterone receptor	None	201	nM	Ki
TKC206816	P06401	Progesterone receptor	None	0	nM	EC50
TKC206816	P06401	Progesterone receptor	None	1.6	nM	IC50
TKC206816	P06401	Progesterone receptor	None	>10000	nM	EC50
TKC206816	P06401	Progesterone receptor	None	1.8	nM	EC50
TKC206816	P06401	Progesterone receptor	None	0.92	nM	EC50
TKC206816	P06401	Progesterone receptor	None	3.5	nM	Ki
TKC206816	P06401	Progesterone receptor	None	0.92	nM	EC50
TKC206816	P06401	Progesterone receptor	None	1.5	nM	EC50
TKC206816	P06401	Progesterone receptor	None	3.5	nM	Ki
TKC206816	P06401	Progesterone receptor	None	2.9	nM	EC50
TKC206816	P06401	Progesterone receptor	None	2.9	nM	EC50
TKC206816	P06401	Progesterone receptor	None	5	nM	IC50
TKC206816	P06401	Progesterone receptor	None	1.8	nM	EC50
TKC206816	P06401	Progesterone receptor	None	2	nM	EC50
TKC206816	P06401	Progesterone receptor	None	0.5	nM	EC50
TKC206816	P06401	Progesterone receptor	None	0.2	nM	IC50
TKC206816	P06401	Progesterone receptor	None	17	nM	IC50
TKC206816	P06401	Progesterone receptor	None	3.5	nM	Ki
TKC206816	P06401	Progesterone receptor	None	3.5	nM	Ki
TKC206816	P06401	Progesterone receptor	None	0.9	nM	EC50
TKC206816	P06401	Progesterone receptor	None	>10000	nM	IC50
TKC206816	P06401	Progesterone receptor	None	3.5	nM	Ki
TKC046324	P06493	Cyclin-dependent kinase 1	None	>100000	nM	IC50
TKC117541	P06493	Cyclin-dependent kinase 1	None	34	%	Activity
TKC005454	P06746	DNA polymerase beta	None	22387	nM	Potency
TKC009499	P06746	DNA polymerase beta	None	39811	nM	Potency
TKC011384	P06746	DNA polymerase beta	None	17783	nM	Potency
TKC011921	P06746	DNA polymerase beta	None	>100000	nM	IC50
TKC012100	P06746	DNA polymerase beta	None	79433	nM	Potency
TKC014568	P06746	DNA polymerase beta	None	19953	nM	Potency
TKC018339	P06746	DNA polymerase beta	None	44668	nM	Potency
TKC020574	P06746	DNA polymerase beta	None	25119	nM	Potency
TKC021477	P06746	DNA polymerase beta	None	19953	nM	Potency
TKC023619	P06746	DNA polymerase beta	None	28184	nM	Potency
TKC025405	P06746	DNA polymerase beta	None	25119	nM	Potency
TKC026600	P06746	DNA polymerase beta	None	45200	nM	IC50
TKC028718	P06746	DNA polymerase beta	None	39811	nM	Potency
TKC031572	P06746	DNA polymerase beta	None	141	nM	Potency
TKC035272	P06746	DNA polymerase beta	None	316	nM	Potency
TKC036999	P06746	DNA polymerase beta	None	50119	nM	Potency
TKC039202	P06746	DNA polymerase beta	None	19953	nM	Potency
TKC042797	P06746	DNA polymerase beta	None	>200000	nM	IC50
TKC051128	P06746	DNA polymerase beta	None	21500	nM	IC50
TKC054329	P06746	DNA polymerase beta	None	25119	nM	Potency
TKC056469	P06746	DNA polymerase beta	None	39811	nM	Potency
TKC056482	P06746	DNA polymerase beta	None	18600	nM	IC50
TKC063474	P06746	DNA polymerase beta	None	89125	nM	Potency
TKC064644	P06746	DNA polymerase beta	None	13000	nM	IC50
TKC072319	P06746	DNA polymerase beta	None	26500	nM	IC50
TKC077689	P06746	DNA polymerase beta	None	3000	nM	IC50
TKC077689	P06746	DNA polymerase beta	None	50119	nM	Potency
TKC077689	P06746	DNA polymerase beta	None	26250	nM	IC50
TKC077689	P06746	DNA polymerase beta	None	8800	nM	IC50
TKC077689	P06746	DNA polymerase beta	None	8800	nM	IC50
TKC103150	P06746	DNA polymerase beta	None	22387	nM	Potency
TKC104194	P06746	DNA polymerase beta	None	25119	nM	Potency
TKC105717	P06746	DNA polymerase beta	None	44668	nM	Potency
TKC108694	P06746	DNA polymerase beta	None	>50000	nM	IC50
TKC113063	P06746	DNA polymerase beta	None	50119	nM	Potency
TKC122980	P06746	DNA polymerase beta	None	26300	nM	IC50
TKC122982	P06746	DNA polymerase beta	None	43400	nM	IC50
TKC123088	P06746	DNA polymerase beta	None	3162	nM	Potency
TKC123088	P06746	DNA polymerase beta	None	33700	nM	IC50
TKC123088	P06746	DNA polymerase beta	None	43600	nM	IC50
TKC134702	P06746	DNA polymerase beta	None	100000	nM	Potency
TKC139229	P06746	DNA polymerase beta	None	2200	nM	IC50
TKC139322	P06746	DNA polymerase beta	None	12600	nM	IC50
TKC150598	P06746	DNA polymerase beta	None	89125	nM	Potency
TKC151609	P06746	DNA polymerase beta	None	89125	nM	Potency
TKC206764	P06746	DNA polymerase beta	None	100000	nM	Potency
TKC206771	P06746	DNA polymerase beta	None	4467	nM	Potency
TKC021518	P07477	Trypsin-1	None	>200000	nM	IC50
TKC021519	P07477	Trypsin-1	None	>200000	nM	IC50
TKC055903	P07477	Trypsin-1	None	70	nM	IC50
TKC105803	P07477	Trypsin-1	None	>200000	nM	IC50
TKC130567	P07477	Trypsin-1	None	>200000	nM	IC50
TKC006863	P07900	Heat shock protein HSP 90-alpha	None	1000	nM	Kd
TKC006886	P07900	Heat shock protein HSP 90-alpha	None	28	nM	Kd
TKC006887	P07900	Heat shock protein HSP 90-alpha	None	1739	nM	Kd
TKC022121	P07900	Heat shock protein HSP 90-alpha	None	2388	nM	Kd
TKC022128	P07900	Heat shock protein HSP 90-alpha	None	5925	nM	Kd
TKC023022	P07900	Heat shock protein HSP 90-alpha	None	12	nM	Kd
TKC023024	P07900	Heat shock protein HSP 90-alpha	None	26	nM	Kd
TKC044085	P07900	Heat shock protein HSP 90-alpha	None	<195	nM	AC50
TKC052570	P07900	Heat shock protein HSP 90-alpha	None	49	nM	Kd
TKC061684	P07900	Heat shock protein HSP 90-alpha	None	33	nM	Kd
TKC066096	P07900	Heat shock protein HSP 90-alpha	None	1408	nM	AC50
TKC066096	P07900	Heat shock protein HSP 90-alpha	None	12	%	Inhibition
TKC096901	P07900	Heat shock protein HSP 90-alpha	None	2295	nM	AC50
TKC104518	P07900	Heat shock protein HSP 90-alpha	None	348	nM	Kd
TKC118419	P07900	Heat shock protein HSP 90-alpha	None	363	nM	AC50
TKC129193	P07900	Heat shock protein HSP 90-alpha	None	3791	nM	AC50
TKC143885	P07900	Heat shock protein HSP 90-alpha	None	649	nM	AC50
TKC161438	P07900	Heat shock protein HSP 90-alpha	None	73	nM	Kd
TKC035272	P07947	Tyrosine-protein kinase Yes	None	30748	nM	Potency
TKC149924	P08047	Transcription factor Sp1	None	8	ug.mL-1	IC50
TKC024886	P08069	Insulin-like growth factor 1 receptor	None	11800	nM	IC50
TKC025690	P08069	Insulin-like growth factor 1 receptor	None	3310	nM	IC50
TKC115259	P08069	Insulin-like growth factor 1 receptor	None	3160	nM	IC50
TKC115261	P08069	Insulin-like growth factor 1 receptor	None	2420	nM	IC50
TKC115272	P08069	Insulin-like growth factor 1 receptor	None	>100000	nM	IC50
TKC115273	P08069	Insulin-like growth factor 1 receptor	None	2300	nM	IC50
TKC152148	P08069	Insulin-like growth factor 1 receptor	None	2770	nM	IC50
TKC152157	P08069	Insulin-like growth factor 1 receptor	None	2460	nM	IC50
TKC174547	P08069	Insulin-like growth factor 1 receptor	None	>100000	nM	IC50
TKC002306	P08183	ATP-dependent translocase ABCB1	None	193	uM	ED50
TKC005454	P08183	ATP-dependent translocase ABCB1	None	50	%	Inhibition
TKC013426	P08183	ATP-dependent translocase ABCB1	None	195	uM	ED50
TKC013736	P08183	ATP-dependent translocase ABCB1	None	35	%	Inhibition
TKC014568	P08183	ATP-dependent translocase ABCB1	None	50	%	Inhibition
TKC014669	P08183	ATP-dependent translocase ABCB1	None	323	%	Inhibition
TKC014732	P08183	ATP-dependent translocase ABCB1	None	81	%	Activity
TKC014741	P08183	ATP-dependent translocase ABCB1	None	133	%	Activity
TKC014744	P08183	ATP-dependent translocase ABCB1	None	98	%	Activity
TKC014745	P08183	ATP-dependent translocase ABCB1	None	127	%	Activity
TKC014746	P08183	ATP-dependent translocase ABCB1	None	53	%	Activity
TKC016483	P08183	ATP-dependent translocase ABCB1	None	95	%	Activity
TKC016484	P08183	ATP-dependent translocase ABCB1	None	80	%	Activity
TKC030239	P08183	ATP-dependent translocase ABCB1	None	50000	nM	IC50
TKC035661	P08183	ATP-dependent translocase ABCB1	None	3010	nM	Ki
TKC035738	P08183	ATP-dependent translocase ABCB1	None	74	%	Activity
TKC035739	P08183	ATP-dependent translocase ABCB1	None	780	nM	Ki
TKC035741	P08183	ATP-dependent translocase ABCB1	None	73	%	Activity
TKC035744	P08183	ATP-dependent translocase ABCB1	None	302	nM	Ki
TKC035812	P08183	ATP-dependent translocase ABCB1	None	3715	nM	Ki
TKC035818	P08183	ATP-dependent translocase ABCB1	None	1349	nM	Ki
TKC035819	P08183	ATP-dependent translocase ABCB1	None	1445	nM	Ki
TKC035822	P08183	ATP-dependent translocase ABCB1	None	73	%	Activity
TKC035829	P08183	ATP-dependent translocase ABCB1	None	420	nM	Ki
TKC035830	P08183	ATP-dependent translocase ABCB1	None	73	%	Activity
TKC035835	P08183	ATP-dependent translocase ABCB1	None	11220	nM	Ki
TKC035836	P08183	ATP-dependent translocase ABCB1	None	910	nM	Ki
TKC035847	P08183	ATP-dependent translocase ABCB1	None	3467	nM	Ki
TKC035853	P08183	ATP-dependent translocase ABCB1	None	510	nM	Ki
TKC035858	P08183	ATP-dependent translocase ABCB1	None	1500	nM	Ki
TKC035900	P08183	ATP-dependent translocase ABCB1	None	1622	nM	Ki
TKC035901	P08183	ATP-dependent translocase ABCB1	None	9772	nM	Ki
TKC040325	P08183	ATP-dependent translocase ABCB1	None	37	%	Activity
TKC040351	P08183	ATP-dependent translocase ABCB1	None	7720	nM	Ki
TKC040363	P08183	ATP-dependent translocase ABCB1	None	630	nM	Ki
TKC040410	P08183	ATP-dependent translocase ABCB1	None	280	nM	Ki
TKC040411	P08183	ATP-dependent translocase ABCB1	None	290	nM	Ki
TKC040416	P08183	ATP-dependent translocase ABCB1	None	72	%	Activity
TKC041926	P08183	ATP-dependent translocase ABCB1	None	6918	nM	Ki
TKC041927	P08183	ATP-dependent translocase ABCB1	None	8460	nM	Ki
TKC041928	P08183	ATP-dependent translocase ABCB1	None	4250	nM	Ki
TKC051988	P08183	ATP-dependent translocase ABCB1	None	95	%	Survival
TKC053751	P08183	ATP-dependent translocase ABCB1	None	88	%	Survival
TKC059890	P08183	ATP-dependent translocase ABCB1	None	106	%	Activity
TKC062844	P08183	ATP-dependent translocase ABCB1	None	119	%	Activity
TKC062846	P08183	ATP-dependent translocase ABCB1	None	119	%	Activity
TKC062848	P08183	ATP-dependent translocase ABCB1	None	118	%	Activity
TKC062849	P08183	ATP-dependent translocase ABCB1	None	100	%	Activity
TKC064191	P08183	ATP-dependent translocase ABCB1	None	98	%	Activity
TKC064201	P08183	ATP-dependent translocase ABCB1	None	123	%	Activity
TKC064204	P08183	ATP-dependent translocase ABCB1	None	132	%	Activity
TKC071640	P08183	ATP-dependent translocase ABCB1	None	100	%	Survival
TKC071920	P08183	ATP-dependent translocase ABCB1	None	3450	nM	Ki
TKC071921	P08183	ATP-dependent translocase ABCB1	None	100000	nM	Ki
TKC071922	P08183	ATP-dependent translocase ABCB1	None	7413	nM	Ki
TKC075769	P08183	ATP-dependent translocase ABCB1	None	50000	nM	IC50
TKC091804	P08183	ATP-dependent translocase ABCB1	None	104	%	Survival
TKC094919	P08183	ATP-dependent translocase ABCB1	None	51	%	Activity
TKC102063	P08183	ATP-dependent translocase ABCB1	None	708	nM	Ki
TKC102759	P08183	ATP-dependent translocase ABCB1	None	1738	nM	Ki
TKC103014	P08183	ATP-dependent translocase ABCB1	None	500	nM	Ki
TKC103015	P08183	ATP-dependent translocase ABCB1	None	250	nM	Ki
TKC103787	P08183	ATP-dependent translocase ABCB1	None	169	%	Activity
TKC103802	P08183	ATP-dependent translocase ABCB1	None	25040	nM	Ki
TKC103872	P08183	ATP-dependent translocase ABCB1	None	700	nM	Ki
TKC104215	P08183	ATP-dependent translocase ABCB1	None	4160	nM	Ki
TKC104474	P08183	ATP-dependent translocase ABCB1	None	6918	nM	Ki
TKC104565	P08183	ATP-dependent translocase ABCB1	None	1259	nM	Ki
TKC104744	P08183	ATP-dependent translocase ABCB1	None	1220	nM	Ki
TKC105215	P08183	ATP-dependent translocase ABCB1	None	610	nM	Ki
TKC105268	P08183	ATP-dependent translocase ABCB1	None	2344	nM	Ki
TKC105449	P08183	ATP-dependent translocase ABCB1	None	390	nM	Ki
TKC105680	P08183	ATP-dependent translocase ABCB1	None	2070	nM	Ki
TKC105741	P08183	ATP-dependent translocase ABCB1	None	3970	nM	Ki
TKC106435	P08183	ATP-dependent translocase ABCB1	None	70	%	Activity
TKC106816	P08183	ATP-dependent translocase ABCB1	None	7586	nM	Ki
TKC106971	P08183	ATP-dependent translocase ABCB1	None	1023	nM	Ki
TKC107081	P08183	ATP-dependent translocase ABCB1	None	101	%	Activity
TKC107643	P08183	ATP-dependent translocase ABCB1	None	68	%	Activity
TKC108026	P08183	ATP-dependent translocase ABCB1	None	724	nM	Ki
TKC108212	P08183	ATP-dependent translocase ABCB1	None	7040	nM	Ki
TKC108240	P08183	ATP-dependent translocase ABCB1	None	2188	nM	Ki
TKC108294	P08183	ATP-dependent translocase ABCB1	None	7586	nM	Ki
TKC108609	P08183	ATP-dependent translocase ABCB1	None	2884	nM	Ki
TKC108638	P08183	ATP-dependent translocase ABCB1	None	7586	nM	Ki
TKC108654	P08183	ATP-dependent translocase ABCB1	None	1698	nM	Ki
TKC108810	P08183	ATP-dependent translocase ABCB1	None	74	%	Activity
TKC111264	P08183	ATP-dependent translocase ABCB1	None	73	%	Inhibition
TKC112787	P08183	ATP-dependent translocase ABCB1	None	40	%	Activity
TKC117216	P08183	ATP-dependent translocase ABCB1	None	57	%	Inhibition
TKC122884	P08183	ATP-dependent translocase ABCB1	None	8200	nM	IC50
TKC132270	P08183	ATP-dependent translocase ABCB1	None	114	%	Activity
TKC145296	P08183	ATP-dependent translocase ABCB1	None	104	%	Activity
TKC145307	P08183	ATP-dependent translocase ABCB1	None	117	%	Activity
TKC146761	P08183	ATP-dependent translocase ABCB1	None	25	10'-6 cm/s	Papp
TKC151523	P08183	ATP-dependent translocase ABCB1	None	19140	nM	IC50
TKC151761	P08183	ATP-dependent translocase ABCB1	None	700	nM	Km
TKC151761	P08183	ATP-dependent translocase ABCB1	None	53900	nM	IC50
TKC151761	P08183	ATP-dependent translocase ABCB1	None	2596	nM	IC50
TKC151761	P08183	ATP-dependent translocase ABCB1	None	2600	nM	IC50
TKC151825	P08183	ATP-dependent translocase ABCB1	None	86	%	Activity
TKC153609	P08183	ATP-dependent translocase ABCB1	None	89	%	Activity
TKC156278	P08183	ATP-dependent translocase ABCB1	None	470	nM	Ki
TKC156279	P08183	ATP-dependent translocase ABCB1	None	570	nM	Ki
TKC156536	P08183	ATP-dependent translocase ABCB1	None	290	nM	Ki
TKC156584	P08183	ATP-dependent translocase ABCB1	None	68	%	Activity
TKC156701	P08183	ATP-dependent translocase ABCB1	None	640	nM	Ki
TKC160583	P08183	ATP-dependent translocase ABCB1	None	74	%	Activity
TKC200866	P08183	ATP-dependent translocase ABCB1	None	700	nM	Km
TKC200866	P08183	ATP-dependent translocase ABCB1	None	53900	nM	IC50
TKC200866	P08183	ATP-dependent translocase ABCB1	None	2596	nM	IC50
TKC200866	P08183	ATP-dependent translocase ABCB1	None	2600	nM	IC50
TKC205544	P08183	ATP-dependent translocase ABCB1	None	429	nm/s	Papp
TKC205880	P08183	ATP-dependent translocase ABCB1	None	2512	nM	Ki
TKC206549	P08183	ATP-dependent translocase ABCB1	None	80200	nM	IC50
TKC206671	P08183	ATP-dependent translocase ABCB1	None	66	%	Activity
TKC206759	P08183	ATP-dependent translocase ABCB1	None	668	nm/s	Papp
TKC206816	P08183	ATP-dependent translocase ABCB1	None	21200	nM	EC50
TKC206816	P08183	ATP-dependent translocase ABCB1	None	192200	nM	IC50
TKC206816	P08183	ATP-dependent translocase ABCB1	None	47863	nM	IC50
TKC206849	P08183	ATP-dependent translocase ABCB1	None	88	%	Activity
TKC207219	P08183	ATP-dependent translocase ABCB1	None	5740	nM	Ki
TKC207258	P08183	ATP-dependent translocase ABCB1	None	18197	nM	Ki
TKC030239	P08235	Mineralocorticoid receptor	None	2.9	nM	EC50
TKC030239	P08235	Mineralocorticoid receptor	None	0.5	nM	Kd
TKC114511	P08235	Mineralocorticoid receptor	None	1880	nM	IC50
TKC206688	P08235	Mineralocorticoid receptor	None	1	nM	Kd
TKC206812	P08235	Mineralocorticoid receptor	None	39	nM	Ki
TKC206816	P08235	Mineralocorticoid receptor	None	0	nM	Kd
TKC206816	P08235	Mineralocorticoid receptor	None	14	nM	IC50
TKC206816	P08235	Mineralocorticoid receptor	None	14	nM	IC50
TKC206816	P08235	Mineralocorticoid receptor	None	14	nM	IC50
TKC206816	P08235	Mineralocorticoid receptor	None	14	nM	IC50
TKC206816	P08235	Mineralocorticoid receptor	None	>14	nM	IC50
TKC009193	P08253	72 kDa type IV collagenase	None	33260	nM	IC50
TKC020117	P08253	72 kDa type IV collagenase	None	90	%	Inhibition
TKC023429	P08253	72 kDa type IV collagenase	None	0	ug.mL-1	IC50
TKC020712	P08581	Hepatocyte growth factor receptor	None	>20000	nM	IC50
TKC024886	P08581	Hepatocyte growth factor receptor	None	3120	nM	IC50
TKC025690	P08581	Hepatocyte growth factor receptor	None	>100000	nM	IC50
TKC033871	P08581	Hepatocyte growth factor receptor	None	50000	nM	IC50
TKC082039	P08581	Hepatocyte growth factor receptor	None	5500	nM	IC50
TKC115259	P08581	Hepatocyte growth factor receptor	None	34000	nM	IC50
TKC115261	P08581	Hepatocyte growth factor receptor	None	47600	nM	IC50
TKC115272	P08581	Hepatocyte growth factor receptor	None	>100000	nM	IC50
TKC115273	P08581	Hepatocyte growth factor receptor	None	27500	nM	IC50
TKC152148	P08581	Hepatocyte growth factor receptor	None	78000	nM	IC50
TKC152157	P08581	Hepatocyte growth factor receptor	None	71500	nM	IC50
TKC174547	P08581	Hepatocyte growth factor receptor	None	>100000	nM	IC50
TKC000602	P08684	Cytochrome P450 3A4	None	>100000	nM	IC50
TKC003636	P08684	Cytochrome P450 3A4	None	>100000	nM	IC50
TKC003637	P08684	Cytochrome P450 3A4	None	>100000	nM	IC50
TKC004452	P08684	Cytochrome P450 3A4	None	>100000	nM	IC50
TKC004454	P08684	Cytochrome P450 3A4	None	>100000	nM	IC50
TKC004758	P08684	Cytochrome P450 3A4	None	>100000	nM	IC50
TKC005454	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC008359	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC011075	P08684	Cytochrome P450 3A4	None	2512	nM	Potency
TKC011412	P08684	Cytochrome P450 3A4	None	4300	nM	Ki
TKC011526	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC012971	P08684	Cytochrome P450 3A4	None	25119	nM	AC50
TKC013304	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC013736	P08684	Cytochrome P450 3A4	None	8700	nM	Km
TKC013753	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC016418	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC020117	P08684	Cytochrome P450 3A4	None	631	nM	Potency
TKC023263	P08684	Cytochrome P450 3A4	None	5070	nM	IC50
TKC025230	P08684	Cytochrome P450 3A4	None	>10000	nM	IC50
TKC025231	P08684	Cytochrome P450 3A4	None	>10000	nM	IC50
TKC030239	P08684	Cytochrome P450 3A4	None	>19953	nM	Potency
TKC030239	P08684	Cytochrome P450 3A4	None	>50000	nM	IC50
TKC031954	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC032619	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC032983	P08684	Cytochrome P450 3A4	None	98200	nM	IC50
TKC034078	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC034083	P08684	Cytochrome P450 3A4	None	7943	nM	Potency
TKC034640	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC034641	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC034979	P08684	Cytochrome P450 3A4	None	20000	nM	Ki
TKC035272	P08684	Cytochrome P450 3A4	None	31623	nM	AC50
TKC037686	P08684	Cytochrome P450 3A4	None	42600	nM	IC50
TKC038725	P08684	Cytochrome P450 3A4	None	1995	nM	Potency
TKC039868	P08684	Cytochrome P450 3A4	None	10	%	Drug metabolism
TKC039869	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC040026	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC040094	P08684	Cytochrome P450 3A4	None	8800	nM	IC50
TKC040829	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC045513	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC053825	P08684	Cytochrome P450 3A4	None	3981	nM	Potency
TKC055066	P08684	Cytochrome P450 3A4	None	2512	nM	Potency
TKC055209	P08684	Cytochrome P450 3A4	None	2512	nM	Potency
TKC057133	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC062321	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC062327	P08684	Cytochrome P450 3A4	None	1585	nM	Potency
TKC062332	P08684	Cytochrome P450 3A4	None	1585	nM	Potency
TKC062333	P08684	Cytochrome P450 3A4	None	6310	nM	Potency
TKC066013	P08684	Cytochrome P450 3A4	None	7943	nM	Potency
TKC066332	P08684	Cytochrome P450 3A4	None	1259	nM	Potency
TKC068076	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC074866	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC075769	P08684	Cytochrome P450 3A4	None	>50000	nM	IC50
TKC077034	P08684	Cytochrome P450 3A4	None	62500	nM	IC50
TKC077038	P08684	Cytochrome P450 3A4	None	21800	nM	IC50
TKC078496	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC079001	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC087664	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC087991	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC088678	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC090094	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC092297	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC092348	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC095493	P08684	Cytochrome P450 3A4	None	1585	nM	AC50
TKC096012	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC097717	P08684	Cytochrome P450 3A4	None	48400	nM	IC50
TKC098345	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC100636	P08684	Cytochrome P450 3A4	None	398	nM	Potency
TKC100649	P08684	Cytochrome P450 3A4	None	3981	nM	Potency
TKC100701	P08684	Cytochrome P450 3A4	None	1995	nM	Potency
TKC101020	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC101092	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC101111	P08684	Cytochrome P450 3A4	None	2512	nM	Potency
TKC101617	P08684	Cytochrome P450 3A4	None	7943	nM	AC50
TKC101618	P08684	Cytochrome P450 3A4	None	6	nM	Potency
TKC101907	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC101920	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC102032	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC102120	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC102204	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC102407	P08684	Cytochrome P450 3A4	None	5012	nM	Potency
TKC102439	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC102540	P08684	Cytochrome P450 3A4	None	3981	nM	Potency
TKC102743	P08684	Cytochrome P450 3A4	None	1000	nM	Potency
TKC103023	P08684	Cytochrome P450 3A4	None	19953	nM	Potency
TKC103041	P08684	Cytochrome P450 3A4	None	19953	nM	Potency
TKC103149	P08684	Cytochrome P450 3A4	None	3981	nM	AC50
TKC103257	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC103736	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC103799	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC104091	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC104293	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC104404	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC104435	P08684	Cytochrome P450 3A4	None	2512	nM	Potency
TKC104602	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC104656	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC104664	P08684	Cytochrome P450 3A4	None	398	nM	Potency
TKC104767	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC104977	P08684	Cytochrome P450 3A4	None	7943	nM	Potency
TKC104979	P08684	Cytochrome P450 3A4	None	1259	nM	Potency
TKC105033	P08684	Cytochrome P450 3A4	None	12589	nM	AC50
TKC105034	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC105037	P08684	Cytochrome P450 3A4	None	12589	nM	AC50
TKC105153	P08684	Cytochrome P450 3A4	None	501	nM	Potency
TKC105168	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC105295	P08684	Cytochrome P450 3A4	None	2512	nM	Potency
TKC105346	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC105378	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC105424	P08684	Cytochrome P450 3A4	None	2512	nM	Potency
TKC105530	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC105784	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC106184	P08684	Cytochrome P450 3A4	None	5012	nM	Potency
TKC106198	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC106212	P08684	Cytochrome P450 3A4	None	2512	nM	AC50
TKC106232	P08684	Cytochrome P450 3A4	None	1995	nM	AC50
TKC106240	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC106301	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC106358	P08684	Cytochrome P450 3A4	None	3981	nM	Potency
TKC106426	P08684	Cytochrome P450 3A4	None	12589	nM	AC50
TKC106840	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC107021	P08684	Cytochrome P450 3A4	None	3162	nM	Potency
TKC107067	P08684	Cytochrome P450 3A4	None	5012	nM	Potency
TKC107104	P08684	Cytochrome P450 3A4	None	2512	nM	Potency
TKC107201	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC107332	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC107525	P08684	Cytochrome P450 3A4	None	2512	nM	Potency
TKC107593	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC107818	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC107830	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC107944	P08684	Cytochrome P450 3A4	None	2512	nM	Potency
TKC108109	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC108295	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC108732	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC109561	P08684	Cytochrome P450 3A4	None	3162	nM	AC50
TKC110481	P08684	Cytochrome P450 3A4	None	1	uL/mg/min	Vmax/Km
TKC110956	P08684	Cytochrome P450 3A4	None	26	pmol/min	Drug metabolism
TKC111349	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC111738	P08684	Cytochrome P450 3A4	None	1995	nM	Potency
TKC112653	P08684	Cytochrome P450 3A4	None	>100000	nM	IC50
TKC112655	P08684	Cytochrome P450 3A4	None	>100000	nM	IC50
TKC112745	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC112754	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC112906	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC112909	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC112914	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC113125	P08684	Cytochrome P450 3A4	None	2512	nM	Potency
TKC113146	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC113149	P08684	Cytochrome P450 3A4	None	1585	nM	Potency
TKC113150	P08684	Cytochrome P450 3A4	None	3162	nM	Potency
TKC114511	P08684	Cytochrome P450 3A4	None	3162	nM	Potency
TKC114819	P08684	Cytochrome P450 3A4	None	3981	nM	Potency
TKC115268	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC117710	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC118004	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC122904	P08684	Cytochrome P450 3A4	None	9	pmol/min	Vmax
TKC122980	P08684	Cytochrome P450 3A4	None	>100000	nM	IC50
TKC132834	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC134571	P08684	Cytochrome P450 3A4	None	35500	nM	IC50
TKC135244	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC135961	P08684	Cytochrome P450 3A4	None	39811	nM	Potency
TKC138777	P08684	Cytochrome P450 3A4	None	2512	nM	Potency
TKC138780	P08684	Cytochrome P450 3A4	None	25119	nM	Potency
TKC141032	P08684	Cytochrome P450 3A4	None	5012	nM	Potency
TKC146761	P08684	Cytochrome P450 3A4	None	125000	nM	IC50
TKC147290	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC148482	P08684	Cytochrome P450 3A4	None	1585	nM	Potency
TKC148601	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC150706	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC151522	P08684	Cytochrome P450 3A4	None	3981	nM	Potency
TKC151523	P08684	Cytochrome P450 3A4	None	23200	nM	Ki
TKC151571	P08684	Cytochrome P450 3A4	None	12589	nM	AC50
TKC151675	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC151758	P08684	Cytochrome P450 3A4	None	316	nM	Potency
TKC151875	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC205806	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC205809	P08684	Cytochrome P450 3A4	None	66	%	Activity
TKC206114	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC206365	P08684	Cytochrome P450 3A4	None	1000	nM	Potency
TKC206386	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC206452	P08684	Cytochrome P450 3A4	None	12589	nM	AC50
TKC206453	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC206687	P08684	Cytochrome P450 3A4	None	1000	nM	Potency
TKC206688	P08684	Cytochrome P450 3A4	None	7943	nM	Potency
TKC206689	P08684	Cytochrome P450 3A4	None	25	nM	Potency
TKC206690	P08684	Cytochrome P450 3A4	None	10000	nM	Potency
TKC206754	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC206759	P08684	Cytochrome P450 3A4	None	10000	nM	IC50
TKC206760	P08684	Cytochrome P450 3A4	None	31623	nM	Potency
TKC206777	P08684	Cytochrome P450 3A4	None	15849	nM	Potency
TKC206783	P08684	Cytochrome P450 3A4	None	12589	nM	AC50
TKC206812	P08684	Cytochrome P450 3A4	None	1000	nM	Potency
TKC206816	P08684	Cytochrome P450 3A4	None	3981	nM	Potency
TKC206884	P08684	Cytochrome P450 3A4	None	12589	nM	Potency
TKC206901	P08684	Cytochrome P450 3A4	None	7943	nM	AC50
TKC207071	P08684	Cytochrome P450 3A4	None	7500	nM	Km
TKC207099	P08684	Cytochrome P450 3A4	None	5012	nM	Potency
TKC207209	P08684	Cytochrome P450 3A4	None	19953	nM	Potency
TKC207282	P08684	Cytochrome P450 3A4	None	3162	nM	AC50
TKC112785	P08912	Muscarinic acetylcholine receptor M5	None	>10000	nM	Ki
TKC206544	P08912	Muscarinic acetylcholine receptor M5	None	>10000	nM	Ki
TKC041411	P09211	Glutathione S-transferase P	None	500	nM	IC50
TKC107855	P09211	Glutathione S-transferase P	None	8500	nM	IC50
TKC020117	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	-67	%	Inhibition
TKC024485	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>50000	nM	IC50
TKC024587	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	600	nM	IC50
TKC024956	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	18000	nM	IC50
TKC024992	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	450	nM	IC50
TKC024993	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	14000	nM	IC50
TKC025965	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>150000	nM	IC50
TKC026303	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	4600	nM	IC50
TKC026309	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	680	nM	IC50
TKC027255	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>67	%	Activity
TKC034201	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>200000	nM	IC50
TKC040026	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	72	%	Inhibition
TKC051154	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	2700	nM	IC50
TKC056482	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>64	%	Activity
TKC058811	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	42000	nM	IC50
TKC058812	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>93	%	Activity
TKC064374	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	42000	nM	IC50
TKC064407	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>72	%	Activity
TKC065375	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>70	%	Activity
TKC071640	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>60	%	Activity
TKC076350	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	100	%	Activity
TKC077689	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	100	%	Activity
TKC077703	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>86	%	Activity
TKC078194	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	31800	nM	IC50
TKC082039	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	48	%	Inhibition
TKC088678	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	24800	nM	IC50
TKC089448	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	35	%	Inhibition
TKC094647	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	97	%	Activity
TKC107943	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	2000	nM	IC50
TKC123028	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	30400	nM	IC50
TKC124303	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	750	nM	IC50
TKC133309	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>200000	nM	IC50
TKC133656	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	25100	nM	IC50
TKC134278	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>200000	nM	IC50
TKC139322	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>67	%	Activity
TKC139366	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	3000	nM	IC50
TKC141401	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	42000	nM	IC50
TKC141499	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	25700	nM	IC50
TKC141805	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>53	%	Activity
TKC142849	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>70	%	Activity
TKC142897	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	30600	nM	IC50
TKC142922	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>61	%	Activity
TKC143539	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	100	%	Activity
TKC145848	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	42000	nM	IC50
TKC145932	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>56	%	Activity
TKC145968	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	100	%	Activity
TKC146774	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>63	%	Activity
TKC149759	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>73	%	Activity
TKC150706	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>62	%	Activity
TKC066096	P09936	Ubiquitin carboxyl-terminal hydrolase isozyme L1	None	6800	nM	IC50
TKC087988	P0DMS8	Adenosine receptor A3	None	2357	nM	Ki
TKC096012	P0DMS8	Adenosine receptor A3	None	2982	nM	Ki
TKC205544	P0DMS8	Adenosine receptor A3	None	95	nM	IC50
TKC206779	P0DMS8	Adenosine receptor A3	None	2674	nM	Ki
TKC013304	P10145	Interleukin-8	None	74978	nM	Potency
TKC013753	P10145	Interleukin-8	None	422	nM	Potency
TKC018710	P10145	Interleukin-8	None	33492	nM	Potency
TKC066169	P10145	Interleukin-8	None	42163	nM	Potency
TKC075769	P10145	Interleukin-8	None	299	nM	Potency
TKC087664	P10145	Interleukin-8	None	37578	nM	Potency
TKC087991	P10145	Interleukin-8	None	422	nM	Potency
TKC092297	P10145	Interleukin-8	None	66824	nM	Potency
TKC104088	P10145	Interleukin-8	None	817	nM	IC50
TKC107086	P10145	Interleukin-8	None	66824	nM	Potency
TKC107735	P10145	Interleukin-8	None	66824	nM	Potency
TKC115268	P10145	Interleukin-8	None	66824	nM	Potency
TKC132609	P10145	Interleukin-8	None	7490	nM	IC50
TKC136411	P10145	Interleukin-8	None	74978	nM	Potency
TKC206759	P10145	Interleukin-8	None	74978	nM	Potency
TKC206760	P10145	Interleukin-8	None	74978	nM	Potency
TKC206770	P10145	Interleukin-8	None	74978	nM	Potency
TKC206812	P10145	Interleukin-8	None	66824	nM	Potency
TKC206816	P10145	Interleukin-8	None	74978	nM	Potency
TKC206884	P10145	Interleukin-8	None	74978	nM	Potency
TKC001669	P10275	Androgen receptor	None	260	nM	IC50
TKC006934	P10275	Androgen receptor	None	50119	nM	Potency
TKC013304	P10275	Androgen receptor	None	70795	nM	Potency
TKC019571	P10275	Androgen receptor	None	19953	nM	Potency
TKC021325	P10275	Androgen receptor	None	31623	nM	Potency
TKC021332	P10275	Androgen receptor	None	31623	nM	Potency
TKC023246	P10275	Androgen receptor	None	449	nM	IC50
TKC030239	P10275	Androgen receptor	None	14	nM	Potency
TKC035272	P10275	Androgen receptor	None	15849	nM	Potency
TKC056140	P10275	Androgen receptor	None	50	%	Activity
TKC066169	P10275	Androgen receptor	None	3981	nM	Potency
TKC074867	P10275	Androgen receptor	None	28184	nM	Potency
TKC075769	P10275	Androgen receptor	None	355	nM	Potency
TKC079001	P10275	Androgen receptor	None	1	nM	Potency
TKC096012	P10275	Androgen receptor	None	178	nM	Potency
TKC100644	P10275	Androgen receptor	None	35481	nM	Potency
TKC102407	P10275	Androgen receptor	None	44668	nM	Potency
TKC106878	P10275	Androgen receptor	None	238	nM	IC50
TKC107086	P10275	Androgen receptor	None	17783	nM	Potency
TKC107735	P10275	Androgen receptor	None	3981	nM	Potency
TKC111738	P10275	Androgen receptor	None	17783	nM	Potency
TKC112923	P10275	Androgen receptor	None	212	nM	IC50
TKC114095	P10275	Androgen receptor	None	1790	nM	IC50
TKC114511	P10275	Androgen receptor	None	315	nM	Ki
TKC115268	P10275	Androgen receptor	None	35481	nM	Potency
TKC115284	P10275	Androgen receptor	None	1	nM	Ki
TKC117154	P10275	Androgen receptor	None	580	nM	IC50
TKC120161	P10275	Androgen receptor	None	44668	nM	Potency
TKC122884	P10275	Androgen receptor	None	39811	nM	Potency
TKC122892	P10275	Androgen receptor	None	10000	nM	IC50
TKC134780	P10275	Androgen receptor	None	2	nM	Potency
TKC147240	P10275	Androgen receptor	None	50	%	Activity
TKC206652	P10275	Androgen receptor	None	50	nM	Potency
TKC206688	P10275	Androgen receptor	None	224	nM	Potency
TKC206690	P10275	Androgen receptor	None	36	nM	Potency
TKC206759	P10275	Androgen receptor	None	2	nM	Potency
TKC206759	P10275	Androgen receptor	None	3.9	nM	IC50
TKC206759	P10275	Androgen receptor	None	4.7	nM	IC50
TKC206759	P10275	Androgen receptor	None	4.2	nM	IC50
TKC206759	P10275	Androgen receptor	None	29	nM	Ki
TKC206759	P10275	Androgen receptor	None	1.1	nM	EC50
TKC206759	P10275	Androgen receptor	None	2.7	nM	IC50
TKC206759	P10275	Androgen receptor	None	2.7	nM	IC50
TKC206759	P10275	Androgen receptor	None	2.7	nM	IC50
TKC206759	P10275	Androgen receptor	None	30	nM	IC50
TKC206759	P10275	Androgen receptor	None	4.57	nM	IC50
TKC206770	P10275	Androgen receptor	None	224	nM	Potency
TKC206779	P10275	Androgen receptor	None	2	nM	Potency
TKC206812	P10275	Androgen receptor	None	220	nM	IC50
TKC206816	P10275	Androgen receptor	None	9	nM	Ki
TKC206816	P10275	Androgen receptor	None	8.5	nM	Ki
TKC206816	P10275	Androgen receptor	None	8.5	nM	Ki
TKC206816	P10275	Androgen receptor	None	8.5	nM	Ki
TKC206816	P10275	Androgen receptor	None	8.5	nM	Ki
TKC206816	P10275	Androgen receptor	None	37	nM	IC50
TKC206816	P10275	Androgen receptor	None	8.5	nM	Ki
TKC206816	P10275	Androgen receptor	None	35	nM	Ki
TKC206816	P10275	Androgen receptor	None	14	nM	IC50
TKC013755	P10276	Retinoic acid receptor alpha	None	7	nM	IC50
TKC013755	P10276	Retinoic acid receptor alpha	None	191	nM	EC50
TKC013755	P10276	Retinoic acid receptor alpha	None	220	nM	EC50
TKC013755	P10276	Retinoic acid receptor alpha	None	22	nM	Ki
TKC013755	P10276	Retinoic acid receptor alpha	None	102	nM	EC50
TKC013755	P10276	Retinoic acid receptor alpha	None	23	nM	EC50
TKC013755	P10276	Retinoic acid receptor alpha	None	45	nM	EC50
TKC013755	P10276	Retinoic acid receptor alpha	None	191	nM	EC50
TKC013755	P10276	Retinoic acid receptor alpha	None	93	nM	Kd
TKC013755	P10276	Retinoic acid receptor alpha	None	102	nM	EC50
TKC013755	P10276	Retinoic acid receptor alpha	None	21	nM	EC50
TKC013755	P10276	Retinoic acid receptor alpha	None	102	nM	EC50
TKC013755	P10276	Retinoic acid receptor alpha	None	191	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	0	nM	Ki
TKC096012	P10276	Retinoic acid receptor alpha	None	7	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	350	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	240	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	240	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	436	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	350	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	563	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	7	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	15	nM	Kd
TKC096012	P10276	Retinoic acid receptor alpha	None	5	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	27	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	2.3	nM	Kd
TKC096012	P10276	Retinoic acid receptor alpha	None	15	nM	Kd
TKC096012	P10276	Retinoic acid receptor alpha	None	350	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	3.3	nM	Ki
TKC096012	P10276	Retinoic acid receptor alpha	None	15	nM	Kd
TKC096012	P10276	Retinoic acid receptor alpha	None	15	nM	Kd
TKC096012	P10276	Retinoic acid receptor alpha	None	16	nM	Kd
TKC096012	P10276	Retinoic acid receptor alpha	None	0.78	nM	IC50
TKC096012	P10276	Retinoic acid receptor alpha	None	0.89	nM	IC50
TKC096012	P10276	Retinoic acid receptor alpha	None	9000	nM	IC50
TKC096012	P10276	Retinoic acid receptor alpha	None	17	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	5	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	350	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	5	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	50	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	1	nM	EC50
TKC096012	P10276	Retinoic acid receptor alpha	None	15	nM	Kd
TKC206482	P10276	Retinoic acid receptor alpha	None	102	nM	EC50
TKC035272	P10415	Apoptosis regulator Bcl-2	None	170	nM	Ki
TKC035272	P10415	Apoptosis regulator Bcl-2	None	260	nM	IC50
TKC035272	P10415	Apoptosis regulator Bcl-2	None	320	nM	Ki
TKC035272	P10415	Apoptosis regulator Bcl-2	None	440	nM	Ki
TKC035272	P10415	Apoptosis regulator Bcl-2	None	440	nM	Ki
TKC035272	P10415	Apoptosis regulator Bcl-2	None	1191	nM	IC50
TKC035272	P10415	Apoptosis regulator Bcl-2	None	450	nM	Ki
TKC035272	P10415	Apoptosis regulator Bcl-2	None	320	nM	Ki
TKC035272	P10415	Apoptosis regulator Bcl-2	None	600	nM	IC50
TKC035272	P10415	Apoptosis regulator Bcl-2	None	420	nM	Ki
TKC035272	P10415	Apoptosis regulator Bcl-2	None	10100	nM	Ki
TKC035272	P10415	Apoptosis regulator Bcl-2	None	4800	nM	Kd
TKC035272	P10415	Apoptosis regulator Bcl-2	None	2110	nM	IC50
TKC035272	P10415	Apoptosis regulator Bcl-2	None	558	nM	Ki
TKC035272	P10415	Apoptosis regulator Bcl-2	None	320	nM	Ki
TKC134945	P10415	Apoptosis regulator Bcl-2	None	1460	nM	Ki
TKC151761	P10415	Apoptosis regulator Bcl-2	None	>10000	nM	GI50
TKC200866	P10415	Apoptosis regulator Bcl-2	None	>10000	nM	GI50
TKC057132	P10613	Lanosterol 14-alpha demethylase	None	7400	nM	Km
TKC008286	P11021	Endoplasmic reticulum chaperone BiP	None	31623	nM	Potency
TKC012929	P11021	Endoplasmic reticulum chaperone BiP	None	10000	nM	Potency
TKC013738	P11021	Endoplasmic reticulum chaperone BiP	None	25119	nM	Potency
TKC030466	P11021	Endoplasmic reticulum chaperone BiP	None	63096	nM	Potency
TKC032619	P11021	Endoplasmic reticulum chaperone BiP	None	14689	nM	Potency
TKC035272	P11021	Endoplasmic reticulum chaperone BiP	None	46452	nM	Potency
TKC035984	P11021	Endoplasmic reticulum chaperone BiP	None	17	nM	Potency
TKC039869	P11021	Endoplasmic reticulum chaperone BiP	None	50119	nM	Potency
TKC084075	P11021	Endoplasmic reticulum chaperone BiP	None	11220	nM	Potency
TKC092297	P11021	Endoplasmic reticulum chaperone BiP	None	44668	nM	Potency
TKC105022	P11021	Endoplasmic reticulum chaperone BiP	None	7080	nM	Potency
TKC105153	P11021	Endoplasmic reticulum chaperone BiP	None	28184	nM	Potency
TKC107627	P11021	Endoplasmic reticulum chaperone BiP	None	11220	nM	Potency
TKC149827	P11021	Endoplasmic reticulum chaperone BiP	None	12589	nM	Potency
TKC151404	P11021	Endoplasmic reticulum chaperone BiP	None	10000	nM	Potency
TKC206622	P11021	Endoplasmic reticulum chaperone BiP	None	36898	nM	Potency
TKC206544	P11229	Muscarinic acetylcholine receptor M1	None	>10000	nM	Ki
TKC011761	P11309	Serine/threonine-protein kinase pim-1	None	11	%	Inhibition
TKC024886	P11309	Serine/threonine-protein kinase pim-1	None	20300	nM	IC50
TKC025690	P11309	Serine/threonine-protein kinase pim-1	None	>100000	nM	IC50
TKC115259	P11309	Serine/threonine-protein kinase pim-1	None	>100000	nM	IC50
TKC115261	P11309	Serine/threonine-protein kinase pim-1	None	>100000	nM	IC50
TKC115272	P11309	Serine/threonine-protein kinase pim-1	None	>100000	nM	IC50
TKC115273	P11309	Serine/threonine-protein kinase pim-1	None	>100000	nM	IC50
TKC118419	P11309	Serine/threonine-protein kinase pim-1	None	87	%	Activity
TKC152148	P11309	Serine/threonine-protein kinase pim-1	None	>100000	nM	IC50
TKC152157	P11309	Serine/threonine-protein kinase pim-1	None	>100000	nM	IC50
TKC174547	P11309	Serine/threonine-protein kinase pim-1	None	>100000	nM	IC50
TKC151761	P11362	Fibroblast growth factor receptor 1	None	>10000	nM	IC50
TKC200866	P11362	Fibroblast growth factor receptor 1	None	>10000	nM	IC50
TKC014892	P11387	DNA topoisomerase 1	None	3	ug.mL-1	MIC
TKC014893	P11387	DNA topoisomerase 1	None	13	ug.mL-1	MIC
TKC017201	P11387	DNA topoisomerase 1	None	13	ug.mL-1	MIC
TKC048122	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC048308	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC048324	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC048330	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC048341	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC049414	P11387	DNA topoisomerase 1	None	25000	nM	IC50
TKC049417	P11387	DNA topoisomerase 1	None	55000	nM	IC50
TKC056419	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC056423	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC056425	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC056427	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC056430	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC058891	P11387	DNA topoisomerase 1	None	23800	nM	IC50
TKC058895	P11387	DNA topoisomerase 1	None	48600	nM	IC50
TKC058897	P11387	DNA topoisomerase 1	None	45100	nM	IC50
TKC058919	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC058921	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC058935	P11387	DNA topoisomerase 1	None	109300	nM	IC50
TKC058949	P11387	DNA topoisomerase 1	None	250000	nM	IC50
TKC058950	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC058953	P11387	DNA topoisomerase 1	None	23800	nM	IC50
TKC058979	P11387	DNA topoisomerase 1	None	23800	nM	IC50
TKC059000	P11387	DNA topoisomerase 1	None	53700	nM	IC50
TKC059030	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC059045	P11387	DNA topoisomerase 1	None	131700	nM	IC50
TKC059148	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC059149	P11387	DNA topoisomerase 1	None	23800	nM	IC50
TKC059160	P11387	DNA topoisomerase 1	None	23800	nM	IC50
TKC059165	P11387	DNA topoisomerase 1	None	23800	nM	IC50
TKC059317	P11387	DNA topoisomerase 1	None	250000	nM	IC50
TKC059337	P11387	DNA topoisomerase 1	None	23800	nM	IC50
TKC059344	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC059345	P11387	DNA topoisomerase 1	None	23800	nM	IC50
TKC059425	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC072969	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC072970	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC096715	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC100727	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC103324	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC105545	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC137826	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC137841	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC138033	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC138054	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC143022	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC143033	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC143055	P11387	DNA topoisomerase 1	None	23800	nM	IC50
TKC143114	P11387	DNA topoisomerase 1	None	250000	nM	IC50
TKC143115	P11387	DNA topoisomerase 1	None	23800	nM	IC50
TKC145932	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC146257	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC147779	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC147805	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC148618	P11387	DNA topoisomerase 1	None	106000	nM	IC50
TKC205544	P11387	DNA topoisomerase 1	None	30000	nM	IC50
TKC205878	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC207002	P11387	DNA topoisomerase 1	None	>250000	nM	IC50
TKC031920	P11388	DNA topoisomerase 2-alpha	None	18600	nM	IC50
TKC048122	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC048308	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC048324	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC048330	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC048341	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC049417	P11388	DNA topoisomerase 2-alpha	None	25000	nM	IC50
TKC049501	P11388	DNA topoisomerase 2-alpha	None	8900	nM	IC50
TKC049788	P11388	DNA topoisomerase 2-alpha	None	17600	nM	IC50
TKC054931	P11388	DNA topoisomerase 2-alpha	None	42600	nM	IC50
TKC054932	P11388	DNA topoisomerase 2-alpha	None	75700	nM	IC50
TKC055381	P11388	DNA topoisomerase 2-alpha	None	4600	nM	IC50
TKC056419	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC056423	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC056425	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC056427	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC056430	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC058767	P11388	DNA topoisomerase 2-alpha	None	17500	nM	IC50
TKC058891	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC058895	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC058897	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC058919	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC058921	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC058935	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC058949	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC058950	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC058953	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC058979	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059000	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059030	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059045	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059148	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059149	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059160	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059165	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059317	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059337	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059344	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059345	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059425	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC059947	P11388	DNA topoisomerase 2-alpha	None	38700	nM	IC50
TKC060891	P11388	DNA topoisomerase 2-alpha	None	4	%	Inhibition
TKC060913	P11388	DNA topoisomerase 2-alpha	None	37500	nM	IC50
TKC072969	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC072970	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC081646	P11388	DNA topoisomerase 2-alpha	None	67300	nM	IC50
TKC096715	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC100727	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC103324	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC105545	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC122884	P11388	DNA topoisomerase 2-alpha	None	>500000	nM	IC50
TKC122982	P11388	DNA topoisomerase 2-alpha	None	>500000	nM	IC50
TKC137826	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC137841	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC138033	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC138054	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC142897	P11388	DNA topoisomerase 2-alpha	None	>33	%	Inhibition
TKC143022	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC143033	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC143055	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC143114	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC143115	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC145932	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC146257	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC147779	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC147805	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC148618	P11388	DNA topoisomerase 2-alpha	None	17000	nM	IC50
TKC148944	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC152742	P11388	DNA topoisomerase 2-alpha	None	38600	nM	IC50
TKC152772	P11388	DNA topoisomerase 2-alpha	None	10400	nM	IC50
TKC173262	P11388	DNA topoisomerase 2-alpha	None	50400	nM	IC50
TKC205878	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC206913	P11388	DNA topoisomerase 2-alpha	None	>500000	nM	IC50
TKC207002	P11388	DNA topoisomerase 2-alpha	None	>250000	nM	IC50
TKC000075	P11473	Vitamin D3 receptor	None	70795	nM	Potency
TKC002371	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC005454	P11473	Vitamin D3 receptor	None	7080	nM	Potency
TKC008359	P11473	Vitamin D3 receptor	None	28184	nM	Potency
TKC011412	P11473	Vitamin D3 receptor	None	19953	nM	Potency
TKC013736	P11473	Vitamin D3 receptor	None	11220	nM	Potency
TKC013755	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC013760	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC014568	P11473	Vitamin D3 receptor	None	63096	nM	Potency
TKC016371	P11473	Vitamin D3 receptor	None	56234	nM	Potency
TKC017379	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC020031	P11473	Vitamin D3 receptor	None	100000	nM	Potency
TKC020117	P11473	Vitamin D3 receptor	None	56234	nM	Potency
TKC027192	P11473	Vitamin D3 receptor	None	35481	nM	Potency
TKC030239	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC032619	P11473	Vitamin D3 receptor	None	31623	nM	Potency
TKC032913	P11473	Vitamin D3 receptor	None	70795	nM	Potency
TKC034083	P11473	Vitamin D3 receptor	None	39811	nM	Potency
TKC034760	P11473	Vitamin D3 receptor	None	35481	nM	Potency
TKC035208	P11473	Vitamin D3 receptor	None	39811	nM	Potency
TKC035272	P11473	Vitamin D3 receptor	None	6310	nM	Potency
TKC037521	P11473	Vitamin D3 receptor	None	79433	nM	Potency
TKC038268	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC038273	P11473	Vitamin D3 receptor	None	56234	nM	Potency
TKC038706	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC041160	P11473	Vitamin D3 receptor	None	79433	nM	Potency
TKC043519	P11473	Vitamin D3 receptor	None	79433	nM	Potency
TKC053095	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC053227	P11473	Vitamin D3 receptor	None	14125	nM	Potency
TKC053825	P11473	Vitamin D3 receptor	None	35481	nM	Potency
TKC055219	P11473	Vitamin D3 receptor	None	100000	nM	Potency
TKC057133	P11473	Vitamin D3 receptor	None	39811	nM	Potency
TKC062321	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC062327	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC062332	P11473	Vitamin D3 receptor	None	70795	nM	Potency
TKC062333	P11473	Vitamin D3 receptor	None	39811	nM	Potency
TKC062669	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC066096	P11473	Vitamin D3 receptor	None	28184	nM	Potency
TKC066169	P11473	Vitamin D3 receptor	None	7943	nM	Potency
TKC073833	P11473	Vitamin D3 receptor	None	56234	nM	Potency
TKC073873	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC074866	P11473	Vitamin D3 receptor	None	1	nM	Potency
TKC075769	P11473	Vitamin D3 receptor	None	562	nM	Potency
TKC082279	P11473	Vitamin D3 receptor	None	70795	nM	Potency
TKC082378	P11473	Vitamin D3 receptor	None	25119	nM	Potency
TKC083025	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC086929	P11473	Vitamin D3 receptor	None	39811	nM	Potency
TKC087533	P11473	Vitamin D3 receptor	None	56234	nM	Potency
TKC087664	P11473	Vitamin D3 receptor	None	100000	nM	Potency
TKC087988	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC091895	P11473	Vitamin D3 receptor	None	79433	nM	Potency
TKC092297	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC092348	P11473	Vitamin D3 receptor	None	39811	nM	Potency
TKC093161	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC095442	P11473	Vitamin D3 receptor	None	39811	nM	Potency
TKC095452	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC096012	P11473	Vitamin D3 receptor	None	31623	nM	Potency
TKC097937	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC098345	P11473	Vitamin D3 receptor	None	28184	nM	Potency
TKC098704	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC099703	P11473	Vitamin D3 receptor	None	39811	nM	Potency
TKC100636	P11473	Vitamin D3 receptor	None	3981	nM	Potency
TKC100644	P11473	Vitamin D3 receptor	None	35481	nM	Potency
TKC100701	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC101052	P11473	Vitamin D3 receptor	None	56234	nM	Potency
TKC101598	P11473	Vitamin D3 receptor	None	56234	nM	Potency
TKC102204	P11473	Vitamin D3 receptor	None	28184	nM	Potency
TKC102407	P11473	Vitamin D3 receptor	None	15849	nM	Potency
TKC102540	P11473	Vitamin D3 receptor	None	35481	nM	Potency
TKC102593	P11473	Vitamin D3 receptor	None	7080	nM	Potency
TKC102939	P11473	Vitamin D3 receptor	None	63096	nM	Potency
TKC103023	P11473	Vitamin D3 receptor	None	28184	nM	Potency
TKC103159	P11473	Vitamin D3 receptor	None	100000	nM	Potency
TKC103257	P11473	Vitamin D3 receptor	None	3162	nM	Potency
TKC103542	P11473	Vitamin D3 receptor	None	28184	nM	Potency
TKC103736	P11473	Vitamin D3 receptor	None	3548	nM	Potency
TKC104404	P11473	Vitamin D3 receptor	None	28184	nM	Potency
TKC104960	P11473	Vitamin D3 receptor	None	79433	nM	Potency
TKC104961	P11473	Vitamin D3 receptor	None	35481	nM	Potency
TKC105153	P11473	Vitamin D3 receptor	None	7943	nM	Potency
TKC105295	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC105424	P11473	Vitamin D3 receptor	None	19953	nM	Potency
TKC105932	P11473	Vitamin D3 receptor	None	63096	nM	Potency
TKC106240	P11473	Vitamin D3 receptor	None	>50000	nM	IC50
TKC106250	P11473	Vitamin D3 receptor	None	>50000	nM	IC50
TKC106301	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC106364	P11473	Vitamin D3 receptor	None	7080	nM	Potency
TKC106367	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC106426	P11473	Vitamin D3 receptor	None	14125	nM	Potency
TKC107086	P11473	Vitamin D3 receptor	None	31623	nM	Potency
TKC107332	P11473	Vitamin D3 receptor	None	19953	nM	Potency
TKC107625	P11473	Vitamin D3 receptor	None	56234	nM	Potency
TKC107627	P11473	Vitamin D3 receptor	None	35481	nM	Potency
TKC107735	P11473	Vitamin D3 receptor	None	17783	nM	Potency
TKC107775	P11473	Vitamin D3 receptor	None	100000	nM	Potency
TKC107830	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC109619	P11473	Vitamin D3 receptor	None	>50000	nM	IC50
TKC109849	P11473	Vitamin D3 receptor	None	>100000	nM	IC50
TKC109996	P11473	Vitamin D3 receptor	None	100000	nM	Potency
TKC111464	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC112754	P11473	Vitamin D3 receptor	None	79433	nM	Potency
TKC112759	P11473	Vitamin D3 receptor	None	70795	nM	Potency
TKC112784	P11473	Vitamin D3 receptor	None	19953	nM	Potency
TKC112785	P11473	Vitamin D3 receptor	None	>40100	nM	IC50
TKC112787	P11473	Vitamin D3 receptor	None	>14500	nM	IC50
TKC112792	P11473	Vitamin D3 receptor	None	28184	nM	Potency
TKC112906	P11473	Vitamin D3 receptor	None	25119	nM	Potency
TKC113063	P11473	Vitamin D3 receptor	None	5805	nM	Potency
TKC113146	P11473	Vitamin D3 receptor	None	39811	nM	Potency
TKC113150	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC113161	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC113663	P11473	Vitamin D3 receptor	None	35481	nM	Potency
TKC114511	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC114568	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC114819	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC115268	P11473	Vitamin D3 receptor	None	0	nM	EC50
TKC115284	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC115284	P11473	Vitamin D3 receptor	None	>2408	uM	Activity
TKC118419	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC122884	P11473	Vitamin D3 receptor	None	35481	nM	Potency
TKC122892	P11473	Vitamin D3 receptor	None	0	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	2	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	1	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	0.08	nM	IC50
TKC122892	P11473	Vitamin D3 receptor	None	7.7	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	0.7	nM	IC50
TKC122892	P11473	Vitamin D3 receptor	None	0.8	nM	IC50
TKC122892	P11473	Vitamin D3 receptor	None	322	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	0.06	nM	IC50
TKC122892	P11473	Vitamin D3 receptor	None	0.35	nM	IC50
TKC122892	P11473	Vitamin D3 receptor	None	3.9	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	10	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	0.3	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	0.16	nM	IC50
TKC122892	P11473	Vitamin D3 receptor	None	0.065	nM	Kd
TKC122892	P11473	Vitamin D3 receptor	None	9	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	0.5	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	0.555	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	1	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	13	nM	IC50
TKC122892	P11473	Vitamin D3 receptor	None	1.24	nM	IC50
TKC122892	P11473	Vitamin D3 receptor	None	0.04	nM	IC50
TKC122892	P11473	Vitamin D3 receptor	None	>0.900000	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	3	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	0.026	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	7.7	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	15	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	1.6	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	0.0953	nM	IC50
TKC122892	P11473	Vitamin D3 receptor	None	0.011	nM	EC50
TKC122892	P11473	Vitamin D3 receptor	None	24	nM	Kd
TKC134702	P11473	Vitamin D3 receptor	None	31623	nM	Potency
TKC136931	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC143885	P11473	Vitamin D3 receptor	None	79433	nM	Potency
TKC147290	P11473	Vitamin D3 receptor	None	25119	nM	Potency
TKC147303	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC148601	P11473	Vitamin D3 receptor	None	35481	nM	Potency
TKC149827	P11473	Vitamin D3 receptor	None	14125	nM	Potency
TKC151237	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC151571	P11473	Vitamin D3 receptor	None	22387	nM	Potency
TKC151609	P11473	Vitamin D3 receptor	None	79433	nM	Potency
TKC151675	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC151758	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC151784	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC151885	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC174441	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC205788	P11473	Vitamin D3 receptor	None	0	nM	ED50
TKC205791	P11473	Vitamin D3 receptor	None	1	nM	IC50
TKC205796	P11473	Vitamin D3 receptor	None	631	nM	Potency
TKC205798	P11473	Vitamin D3 receptor	None	11	%	Activity
TKC206385	P11473	Vitamin D3 receptor	None	>44	uM	Activity
TKC206544	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC206652	P11473	Vitamin D3 receptor	None	562	nM	Potency
TKC206669	P11473	Vitamin D3 receptor	None	>50000	nM	IC50
TKC206672	P11473	Vitamin D3 receptor	None	>50000	nM	IC50
TKC206758	P11473	Vitamin D3 receptor	None	56234	nM	Potency
TKC206760	P11473	Vitamin D3 receptor	None	8913	nM	Potency
TKC206760	P11473	Vitamin D3 receptor	None	6	%	Activity
TKC206760	P11473	Vitamin D3 receptor	None	330	nM	Kd
TKC206761	P11473	Vitamin D3 receptor	None	>15100	nM	IC50
TKC206780	P11473	Vitamin D3 receptor	None	89125	nM	Potency
TKC206812	P11473	Vitamin D3 receptor	None	44668	nM	Potency
TKC206812	P11473	Vitamin D3 receptor	None	2000	nM	IC50
TKC206816	P11473	Vitamin D3 receptor	None	15849	nM	Potency
TKC206876	P11473	Vitamin D3 receptor	None	79433	nM	Potency
TKC206884	P11473	Vitamin D3 receptor	None	50119	nM	Potency
TKC206884	P11473	Vitamin D3 receptor	None	>150000	nM	EC50
TKC206901	P11473	Vitamin D3 receptor	None	31623	nM	Potency
TKC206902	P11473	Vitamin D3 receptor	None	35481	nM	Potency
TKC206960	P11473	Vitamin D3 receptor	None	17783	nM	Potency
TKC026583	P11802	Cyclin-dependent kinase 4	None	9	ug.mL-1	IC50
TKC113582	P11802	Cyclin-dependent kinase 4	None	10	ug.mL-1	IC50
TKC011761	P12931	Proto-oncogene tyrosine-protein kinase Src	None	61	%	Inhibition
TKC024886	P12931	Proto-oncogene tyrosine-protein kinase Src	None	8620	nM	IC50
TKC025690	P12931	Proto-oncogene tyrosine-protein kinase Src	None	19700	nM	IC50
TKC115259	P12931	Proto-oncogene tyrosine-protein kinase Src	None	2400	nM	IC50
TKC115261	P12931	Proto-oncogene tyrosine-protein kinase Src	None	2240	nM	IC50
TKC115272	P12931	Proto-oncogene tyrosine-protein kinase Src	None	>100000	nM	IC50
TKC115273	P12931	Proto-oncogene tyrosine-protein kinase Src	None	1480	nM	IC50
TKC135974	P12931	Proto-oncogene tyrosine-protein kinase Src	None	35800	nM	IC50
TKC151761	P12931	Proto-oncogene tyrosine-protein kinase Src	None	>10000	nM	IC50
TKC152148	P12931	Proto-oncogene tyrosine-protein kinase Src	None	1910	nM	IC50
TKC152157	P12931	Proto-oncogene tyrosine-protein kinase Src	None	2170	nM	IC50
TKC174547	P12931	Proto-oncogene tyrosine-protein kinase Src	None	>100000	nM	IC50
TKC200866	P12931	Proto-oncogene tyrosine-protein kinase Src	None	>10000	nM	IC50
TKC050174	P13726	Tissue factor	None	10	nM	IC50
TKC060193	P13726	Tissue factor	None	16	nM	IC50
TKC060801	P13726	Tissue factor	None	0	nM	IC50
TKC060880	P13726	Tissue factor	None	0	nM	IC50
TKC071640	P13726	Tissue factor	None	0	nM	IC50
TKC077689	P13726	Tissue factor	None	5	nM	IC50
TKC107399	P13726	Tissue factor	None	11	nM	IC50
TKC123023	P13726	Tissue factor	None	0	nM	IC50
TKC123078	P13726	Tissue factor	None	0	nM	IC50
TKC139000	P13726	Tissue factor	None	1	nM	IC50
TKC142381	P13726	Tissue factor	None	0	nM	IC50
TKC146780	P13726	Tissue factor	None	0	nM	IC50
TKC147930	P13726	Tissue factor	None	6	nM	IC50
TKC206115	P13726	Tissue factor	None	1	nM	IC50
TKC055345	P14174	Macrophage migration inhibitory factor	None	35200	nM	IC50
TKC058241	P14174	Macrophage migration inhibitory factor	None	17500	nM	IC50
TKC061683	P14174	Macrophage migration inhibitory factor	None	85300	nM	IC50
TKC151638	P14174	Macrophage migration inhibitory factor	None	6000	nM	IC50
TKC151638	P14174	Macrophage migration inhibitory factor	None	6400	nM	IC50
TKC151638	P14174	Macrophage migration inhibitory factor	None	6400	nM	IC50
TKC001229	P14324	Farnesyl pyrophosphate synthase	None	13300	nM	IC50
TKC001231	P14324	Farnesyl pyrophosphate synthase	None	18700	nM	IC50
TKC001233	P14324	Farnesyl pyrophosphate synthase	None	230	nM	IC50
TKC011411	P14324	Farnesyl pyrophosphate synthase	None	7800	nM	IC50
TKC011412	P14324	Farnesyl pyrophosphate synthase	None	20000	nM	IC50
TKC013844	P14324	Farnesyl pyrophosphate synthase	None	>100000	nM	IC50
TKC019382	P14324	Farnesyl pyrophosphate synthase	None	4400	nM	Km
TKC071323	P14324	Farnesyl pyrophosphate synthase	None	>10000	nM	IC50
TKC071323	P14324	Farnesyl pyrophosphate synthase	None	>10000	nM	IC50
TKC074868	P14324	Farnesyl pyrophosphate synthase	None	4400	nM	Km
TKC104488	P14324	Farnesyl pyrophosphate synthase	None	473	nM	IC50
TKC205544	P14416	D(2) dopamine receptor	None	687	nM	Ki
TKC205544	P14416	D(2) dopamine receptor	None	280	nM	Ki
TKC205544	P14416	D(2) dopamine receptor	None	398.1	nM	Ki
TKC206544	P14416	D(2) dopamine receptor	None	>10000	nM	Ki
TKC035272	P14618	Pyruvate kinase PKM	None	31623	nM	Potency
TKC037410	P14618	Pyruvate kinase PKM	None	6	nM	EC50
TKC039332	P14618	Pyruvate kinase PKM	None	25119	nM	Potency
TKC100416	P14618	Pyruvate kinase PKM	None	13	nM	Potency
TKC151609	P14618	Pyruvate kinase PKM	None	11220	nM	Potency
TKC206901	P14618	Pyruvate kinase PKM	None	2	nM	Potency
TKC020117	P14780	Matrix metalloproteinase-9	None	99	%	Inhibition
TKC023429	P14780	Matrix metalloproteinase-9	None	1	ug.mL-1	IC50
TKC037777	P14780	Matrix metalloproteinase-9	None	6	ug.mL-1	IC50
TKC039471	P14780	Matrix metalloproteinase-9	None	6	ug.mL-1	IC50
TKC006896	P14902	Indoleamine 2,3-dioxygenase 1	None	7700	nM	IC50
TKC014575	P14902	Indoleamine 2,3-dioxygenase 1	None	4680	nM	IC50
TKC024473	P14902	Indoleamine 2,3-dioxygenase 1	None	10000	nM	IC50
TKC024474	P14902	Indoleamine 2,3-dioxygenase 1	None	11000	nM	IC50
TKC104241	P14902	Indoleamine 2,3-dioxygenase 1	None	0	nM	EC50
TKC011761	P15056	Serine/threonine-protein kinase B-raf	None	-7	%	Inhibition
TKC065182	P15559	NAD(P)H dehydrogenase [quinone] 1	None	>20	ug ml-1	CD
TKC071640	P15559	NAD(P)H dehydrogenase [quinone] 1	None	>20	ug ml-1	CD
TKC105886	P15559	NAD(P)H dehydrogenase [quinone] 1	None	>20	ug ml-1	CD
TKC123088	P15559	NAD(P)H dehydrogenase [quinone] 1	None	>20	ug ml-1	CD
TKC138780	P15559	NAD(P)H dehydrogenase [quinone] 1	None	>20	ug ml-1	CD
TKC000192	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	>19000	nM	IC50
TKC002550	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	9300	nM	IC50
TKC005454	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	55700	nM	IC50
TKC008778	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	7400	nM	IC50
TKC013306	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	<50	%	Inhibition
TKC026891	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	<50	%	Inhibition
TKC030269	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	45900	nM	IC50
TKC030508	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	15700	nM	IC50
TKC031060	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	100000	nM	IC50
TKC037481	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	26800	nM	IC50
TKC043218	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	36700	nM	IC50
TKC043220	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	62000	nM	IC50
TKC045915	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	9600	nM	IC50
TKC045916	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	21500	nM	IC50
TKC055829	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	5100	nM	IC50
TKC056482	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	2400	nM	IC50
TKC056482	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	3330	nM	IC50
TKC056482	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	6700	nM	IC50
TKC060880	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	5630	nM	IC50
TKC063247	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	>20000	nM	IC50
TKC066096	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	18800	nM	IC50
TKC077689	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	1600	nM	IC50
TKC077689	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	4230	nM	IC50
TKC077689	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	5.5	nM	IC50
TKC077689	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	5460	nM	IC50
TKC077689	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	5460	nM	IC50
TKC077689	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	>120000	nM	IC50
TKC077689	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	5460	nM	IC50
TKC077689	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	7860	nM	IC50
TKC077689	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	5000	nM	IC50
TKC077689	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	6420	nM	IC50
TKC077689	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	10550	nM	IC50
TKC077689	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	3400	nM	IC50
TKC088678	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	>20000	nM	IC50
TKC089416	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	160	nM	IC50
TKC096804	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	800	nM	IC50
TKC105683	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	3700	nM	IC50
TKC106945	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	>16000	nM	IC50
TKC112796	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	<50	%	Inhibition
TKC116328	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	<50	%	Inhibition
TKC116342	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	<50	%	Inhibition
TKC131482	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	35090	nM	IC50
TKC139322	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	11310	nM	IC50
TKC139366	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	9450	nM	IC50
TKC141805	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	>20000	nM	IC50
TKC142814	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	>20000	nM	IC50
TKC146774	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	19470	nM	IC50
TKC149652	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	3000	nM	IC50
TKC150004	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	<50	%	Inhibition
TKC150706	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	>20000	nM	IC50
TKC156704	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	>16000	nM	IC50
TKC191566	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	>19000	nM	IC50
TKC206409	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	>100000	nM	IC50
TKC206760	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	20450	nM	IC50
TKC206840	P17706	Tyrosine-protein phosphatase non-receptor type 2	None	<50	%	Inhibition
TKC075756	P17948	Vascular endothelial growth factor receptor 1	None	1001	nM	Ki
TKC012971	P19838	Nuclear factor NF-kappa-B p105 subunit	None	10	nM	Potency
TKC016414	P19838	Nuclear factor NF-kappa-B p105 subunit	None	49600	nM	IC50
TKC030239	P19838	Nuclear factor NF-kappa-B p105 subunit	None	14	nM	Potency
TKC035272	P19838	Nuclear factor NF-kappa-B p105 subunit	None	44668	nM	Potency
TKC092297	P19838	Nuclear factor NF-kappa-B p105 subunit	None	6310	nM	Potency
TKC100644	P19838	Nuclear factor NF-kappa-B p105 subunit	None	44668	nM	Potency
TKC101618	P19838	Nuclear factor NF-kappa-B p105 subunit	None	6310	nM	Potency
TKC103149	P19838	Nuclear factor NF-kappa-B p105 subunit	None	11220	nM	Potency
TKC104071	P19838	Nuclear factor NF-kappa-B p105 subunit	None	100	nM	Potency
TKC105037	P19838	Nuclear factor NF-kappa-B p105 subunit	None	178	nM	Potency
TKC106232	P19838	Nuclear factor NF-kappa-B p105 subunit	None	14125	nM	Potency
TKC106426	P19838	Nuclear factor NF-kappa-B p105 subunit	None	3981	nM	Potency
TKC107086	P19838	Nuclear factor NF-kappa-B p105 subunit	None	19953	nM	Potency
TKC111738	P19838	Nuclear factor NF-kappa-B p105 subunit	None	3981	nM	Potency
TKC151571	P19838	Nuclear factor NF-kappa-B p105 subunit	None	10000	nM	Potency
TKC206453	P19838	Nuclear factor NF-kappa-B p105 subunit	None	1000	nM	Potency
TKC206688	P19838	Nuclear factor NF-kappa-B p105 subunit	None	20	nM	Potency
TKC206754	P19838	Nuclear factor NF-kappa-B p105 subunit	None	1585	nM	Potency
TKC206760	P19838	Nuclear factor NF-kappa-B p105 subunit	None	50119	nM	Potency
TKC206770	P19838	Nuclear factor NF-kappa-B p105 subunit	None	31623	nM	Potency
TKC206812	P19838	Nuclear factor NF-kappa-B p105 subunit	None	50119	nM	Potency
TKC206901	P19838	Nuclear factor NF-kappa-B p105 subunit	None	141	nM	Potency
TKC039202	P21453	Sphingosine 1-phosphate receptor 1	None	4962	nM	IC50
TKC096012	P21453	Sphingosine 1-phosphate receptor 1	None	34120	nM	EC50
TKC096012	P21453	Sphingosine 1-phosphate receptor 1	None	>95100	nM	EC50
TKC096012	P21453	Sphingosine 1-phosphate receptor 1	None	25400	nM	EC50
TKC005454	P22303	Acetylcholinesterase	None	>6410	nM	Ki
TKC008149	P22303	Acetylcholinesterase	None	0	ug	Activity
TKC010478	P22303	Acetylcholinesterase	None	14500	nM	IC50
TKC010538	P22303	Acetylcholinesterase	None	22800	nM	IC50
TKC011270	P22303	Acetylcholinesterase	None	>10	ug	Activity
TKC012269	P22303	Acetylcholinesterase	None	>22	%	Inhibition
TKC014568	P22303	Acetylcholinesterase	None	>50000	nM	IC50
TKC014568	P22303	Acetylcholinesterase	None	>100000	nM	Ki
TKC025887	P22303	Acetylcholinesterase	None	2500	nM	IC50
TKC026245	P22303	Acetylcholinesterase	None	10	ug	MIC
TKC026257	P22303	Acetylcholinesterase	None	1	ug	MIC
TKC039110	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC039119	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC039122	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC048637	P22303	Acetylcholinesterase	None	29	%	Inhibition
TKC050924	P22303	Acetylcholinesterase	None	10670	nM	IC50
TKC051021	P22303	Acetylcholinesterase	None	22630	nM	IC50
TKC051031	P22303	Acetylcholinesterase	None	18350	nM	IC50
TKC051032	P22303	Acetylcholinesterase	None	30260	nM	IC50
TKC051042	P22303	Acetylcholinesterase	None	17140	nM	IC50
TKC056997	P22303	Acetylcholinesterase	None	16270	nM	IC50
TKC056998	P22303	Acetylcholinesterase	None	25080	nM	IC50
TKC057020	P22303	Acetylcholinesterase	None	31030	nM	IC50
TKC061148	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC062012	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC062026	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC062075	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC063185	P22303	Acetylcholinesterase	None	9980	nM	IC50
TKC064964	P22303	Acetylcholinesterase	None	25910	nM	IC50
TKC064991	P22303	Acetylcholinesterase	None	9400	nM	IC50
TKC068847	P22303	Acetylcholinesterase	None	34	%	Inhibition
TKC083115	P22303	Acetylcholinesterase	None	26	%	Inhibition
TKC092147	P22303	Acetylcholinesterase	None	>10	ug	MIC
TKC092148	P22303	Acetylcholinesterase	None	1	ug	MIC
TKC092149	P22303	Acetylcholinesterase	None	1	ug	MIC
TKC092150	P22303	Acetylcholinesterase	None	10	ug	MIC
TKC092151	P22303	Acetylcholinesterase	None	1	ug	MIC
TKC092152	P22303	Acetylcholinesterase	None	>10	ug	MIC
TKC092153	P22303	Acetylcholinesterase	None	>10	ug	MIC
TKC092154	P22303	Acetylcholinesterase	None	>10	ug	MIC
TKC092155	P22303	Acetylcholinesterase	None	10	ug	MIC
TKC092156	P22303	Acetylcholinesterase	None	>10	ug	MIC
TKC092182	P22303	Acetylcholinesterase	None	>10	ug	MIC
TKC095827	P22303	Acetylcholinesterase	None	910	nM	IC50
TKC101947	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC103473	P22303	Acetylcholinesterase	None	10	ug	Activity
TKC107319	P22303	Acetylcholinesterase	None	>100000	nM	Ki
TKC108605	P22303	Acetylcholinesterase	None	10	ug	Activity
TKC109315	P22303	Acetylcholinesterase	None	5754	nM	IC50
TKC109320	P22303	Acetylcholinesterase	None	181970	nM	IC50
TKC109322	P22303	Acetylcholinesterase	None	229087	nM	IC50
TKC109330	P22303	Acetylcholinesterase	None	77625	nM	IC50
TKC109347	P22303	Acetylcholinesterase	None	33113	nM	IC50
TKC109348	P22303	Acetylcholinesterase	None	61660	nM	IC50
TKC109364	P22303	Acetylcholinesterase	None	15849	nM	IC50
TKC109367	P22303	Acetylcholinesterase	None	30200	nM	IC50
TKC109381	P22303	Acetylcholinesterase	None	7079	nM	IC50
TKC109383	P22303	Acetylcholinesterase	None	9900	nM	IC50
TKC110247	P22303	Acetylcholinesterase	None	>10	ug.mL-1	IC50
TKC112463	P22303	Acetylcholinesterase	None	251189	nM	IC50
TKC112467	P22303	Acetylcholinesterase	None	83176	nM	IC50
TKC112468	P22303	Acetylcholinesterase	None	48978	nM	IC50
TKC112505	P22303	Acetylcholinesterase	None	42658	nM	IC50
TKC114542	P22303	Acetylcholinesterase	None	50119	nM	IC50
TKC114543	P22303	Acetylcholinesterase	None	70795	nM	IC50
TKC114548	P22303	Acetylcholinesterase	None	28000	nM	IC50
TKC114549	P22303	Acetylcholinesterase	None	69183	nM	IC50
TKC114551	P22303	Acetylcholinesterase	None	28840	nM	IC50
TKC114558	P22303	Acetylcholinesterase	None	6457	nM	IC50
TKC114561	P22303	Acetylcholinesterase	None	19498	nM	IC50
TKC114562	P22303	Acetylcholinesterase	None	6457	nM	IC50
TKC114777	P22303	Acetylcholinesterase	None	6166	nM	IC50
TKC119401	P22303	Acetylcholinesterase	None	26000	nM	IC50
TKC129743	P22303	Acetylcholinesterase	None	>10	ug	Activity
TKC135978	P22303	Acetylcholinesterase	None	191100	nM	IC50
TKC139191	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC141633	P22303	Acetylcholinesterase	None	24040	nM	IC50
TKC142015	P22303	Acetylcholinesterase	None	21100	nM	IC50
TKC144380	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC144901	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC144904	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC145173	P22303	Acetylcholinesterase	None	22970	nM	IC50
TKC145183	P22303	Acetylcholinesterase	None	18350	nM	IC50
TKC147230	P22303	Acetylcholinesterase	None	22310	nM	IC50
TKC147240	P22303	Acetylcholinesterase	None	26780	nM	IC50
TKC148618	P22303	Acetylcholinesterase	None	21840	nM	IC50
TKC150909	P22303	Acetylcholinesterase	None	<10	ug.mL-1	IC50
TKC161356	P22303	Acetylcholinesterase	None	81500	nM	IC50
TKC168054	P22303	Acetylcholinesterase	None	1690	nM	IC50
TKC174459	P22303	Acetylcholinesterase	None	12260	nM	IC50
TKC205554	P22303	Acetylcholinesterase	None	1	ug	MIC
TKC205771	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC205772	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC206567	P22303	Acetylcholinesterase	None	1	ug	Activity
TKC207001	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC207197	P22303	Acetylcholinesterase	None	1	ug	MIC
TKC076129	P22748	Carbonic anhydrase 4	None	510	nM	Ki
TKC104783	P22748	Carbonic anhydrase 4	None	4360	nM	Ki
TKC105780	P22748	Carbonic anhydrase 4	None	2750	nM	Ki
TKC000611	P23219	Prostaglandin G/H synthase 1	None	40000	nM	IC50
TKC001618	P23219	Prostaglandin G/H synthase 1	None	34000	nM	IC50
TKC009896	P23219	Prostaglandin G/H synthase 1	None	791100	nM	IC50
TKC019819	P23219	Prostaglandin G/H synthase 1	None	48	%	Inhibition
TKC019859	P23219	Prostaglandin G/H synthase 1	None	54	%	Inhibition
TKC020491	P23219	Prostaglandin G/H synthase 1	None	4000	nM	IC50
TKC020796	P23219	Prostaglandin G/H synthase 1	None	30	%	Inhibition
TKC021940	P23219	Prostaglandin G/H synthase 1	None	40	%	Inhibition
TKC022833	P23219	Prostaglandin G/H synthase 1	None	43	%	Inhibition
TKC022834	P23219	Prostaglandin G/H synthase 1	None	43	%	Inhibition
TKC022961	P23219	Prostaglandin G/H synthase 1	None	44	%	Inhibition
TKC024587	P23219	Prostaglandin G/H synthase 1	None	3300	nM	IC50
TKC024587	P23219	Prostaglandin G/H synthase 1	None	3300	nM	IC50
TKC031258	P23219	Prostaglandin G/H synthase 1	None	3600	nM	IC50
TKC034201	P23219	Prostaglandin G/H synthase 1	None	>200000	nM	IC50
TKC034358	P23219	Prostaglandin G/H synthase 1	None	39000	nM	IC50
TKC034359	P23219	Prostaglandin G/H synthase 1	None	39000	nM	IC50
TKC036372	P23219	Prostaglandin G/H synthase 1	None	14000	nM	IC50
TKC037595	P23219	Prostaglandin G/H synthase 1	None	36000	nM	IC50
TKC043613	P23219	Prostaglandin G/H synthase 1	None	43000	nM	IC50
TKC049750	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC049818	P23219	Prostaglandin G/H synthase 1	None	44	ug	IC50
TKC054011	P23219	Prostaglandin G/H synthase 1	None	8800	nM	IC50
TKC054031	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC054081	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC054090	P23219	Prostaglandin G/H synthase 1	None	7500	nM	IC50
TKC054099	P23219	Prostaglandin G/H synthase 1	None	8800	nM	IC50
TKC054100	P23219	Prostaglandin G/H synthase 1	None	8900	nM	IC50
TKC054101	P23219	Prostaglandin G/H synthase 1	None	7600	nM	IC50
TKC054240	P23219	Prostaglandin G/H synthase 1	None	7800	nM	IC50
TKC054241	P23219	Prostaglandin G/H synthase 1	None	6300	nM	IC50
TKC056482	P23219	Prostaglandin G/H synthase 1	None	210000	nM	IC50
TKC060184	P23219	Prostaglandin G/H synthase 1	None	8300	nM	IC50
TKC060216	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC060284	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC060302	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC060303	P23219	Prostaglandin G/H synthase 1	None	7800	nM	IC50
TKC060304	P23219	Prostaglandin G/H synthase 1	None	8000	nM	IC50
TKC060399	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC060602	P23219	Prostaglandin G/H synthase 1	None	5900	nM	IC50
TKC066954	P23219	Prostaglandin G/H synthase 1	None	38	%	Inhibition
TKC068533	P23219	Prostaglandin G/H synthase 1	None	28000	nM	IC50
TKC071010	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC077689	P23219	Prostaglandin G/H synthase 1	None	380000	nM	IC50
TKC077689	P23219	Prostaglandin G/H synthase 1	None	380000	nM	IC50
TKC095276	P23219	Prostaglandin G/H synthase 1	None	48	%	Inhibition
TKC113936	P23219	Prostaglandin G/H synthase 1	None	65	%	Inhibition
TKC122543	P23219	Prostaglandin G/H synthase 1	None	35	%	Inhibition
TKC130084	P23219	Prostaglandin G/H synthase 1	None	39	%	Inhibition
TKC130119	P23219	Prostaglandin G/H synthase 1	None	33	%	Inhibition
TKC130577	P23219	Prostaglandin G/H synthase 1	None	<43	%	Inhibition
TKC130901	P23219	Prostaglandin G/H synthase 1	None	36	%	Inhibition
TKC133309	P23219	Prostaglandin G/H synthase 1	None	>200000	nM	IC50
TKC133517	P23219	Prostaglandin G/H synthase 1	None	1300	nM	IC50
TKC133656	P23219	Prostaglandin G/H synthase 1	None	>200000	nM	IC50
TKC134278	P23219	Prostaglandin G/H synthase 1	None	>200000	nM	IC50
TKC139036	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC140627	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC141365	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC143641	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC151113	P23219	Prostaglandin G/H synthase 1	None	116400	nM	IC50
TKC151284	P23219	Prostaglandin G/H synthase 1	None	51	%	Inhibition
TKC151765	P23219	Prostaglandin G/H synthase 1	None	48	%	Inhibition
TKC151792	P23219	Prostaglandin G/H synthase 1	None	14000	nM	IC50
TKC172853	P23219	Prostaglandin G/H synthase 1	None	43700	nM	IC50
TKC076129	P23280	Carbonic anhydrase 6	None	860	nM	Ki
TKC104783	P23280	Carbonic anhydrase 6	None	9780	nM	Ki
TKC105780	P23280	Carbonic anhydrase 6	None	6960	nM	Ki
TKC118419	P23443	Ribosomal protein S6 kinase beta-1	None	95	%	Activity
TKC032440	P24530	Endothelin receptor type B	None	50000	nM	IC50
TKC032443	P24530	Endothelin receptor type B	None	21000	nM	IC50
TKC118419	P24941	Cyclin-dependent kinase 2	None	95	%	Activity
TKC206292	P24941	Cyclin-dependent kinase 2	None	4800	nM	Kd
TKC110447	P25024	C-X-C chemokine receptor type 1	None	4500	nM	IC50
TKC119009	P25024	C-X-C chemokine receptor type 1	None	20000	nM	IC50
TKC119010	P25024	C-X-C chemokine receptor type 1	None	5500	nM	IC50
TKC205544	P25100	Alpha-1D adrenergic receptor	None	2	nM	Ki
TKC205544	P25100	Alpha-1D adrenergic receptor	None	158.48	nM	Ki
TKC205544	P25100	Alpha-1D adrenergic receptor	None	954.99	nM	Ki
TKC205544	P25100	Alpha-1D adrenergic receptor	None	289	nM	Ki
TKC032440	P25101	Endothelin-1 receptor	None	135000	nM	IC50
TKC032443	P25101	Endothelin-1 receptor	None	62000	nM	IC50
TKC007073	P25105	Platelet-activating factor receptor	None	5	uM	Binding affinity
TKC105026	P25105	Platelet-activating factor receptor	None	575	nM	IC50
TKC105028	P25105	Platelet-activating factor receptor	None	575	nM	IC50
TKC106540	P25105	Platelet-activating factor receptor	None	964	nM	Ki
TKC147486	P25105	Platelet-activating factor receptor	None	4	uM	Binding affinity
TKC147612	P25105	Platelet-activating factor receptor	None	5	uM	Binding affinity
TKC151784	P25105	Platelet-activating factor receptor	None	128	nM	IC50
TKC205457	P25105	Platelet-activating factor receptor	None	1259	nM	IC50
TKC022852	P26358	DNA (cytosine-5)-methyltransferase 1	None	2	uM	Activity
TKC022854	P26358	DNA (cytosine-5)-methyltransferase 1	None	55	uM	Activity
TKC055219	P26358	DNA (cytosine-5)-methyltransferase 1	None	5930	nM	IC50
TKC055219	P26358	DNA (cytosine-5)-methyltransferase 1	None	5930	nM	IC50
TKC118419	P27361	Mitogen-activated protein kinase 3	None	106	%	Activity
TKC206779	P27361	Mitogen-activated protein kinase 3	None	3157	nM	IC50
TKC118419	P27448	MAP/microtubule affinity-regulating kinase 3	None	85	%	Activity
TKC001930	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	31623	nM	Potency
TKC005139	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	4467	nM	Potency
TKC005313	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	6	nM	Potency
TKC005454	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	39811	nM	Potency
TKC008286	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	11220	nM	Potency
TKC009499	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	11220	nM	Potency
TKC011384	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	39811	nM	Potency
TKC011526	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	5	nM	Potency
TKC011921	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	39811	nM	Potency
TKC012929	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	891	nM	Potency
TKC013755	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	6	nM	Potency
TKC018288	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	7943	nM	Potency
TKC018339	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	35481	nM	Potency
TKC019571	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	891	nM	Potency
TKC019887	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	35481	nM	Potency
TKC020117	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	14125	nM	Potency
TKC020459	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	35481	nM	Potency
TKC020574	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	31623	nM	Potency
TKC021477	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	7943	nM	Potency
TKC022945	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	50	nM	Potency
TKC023619	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	31623	nM	Potency
TKC025405	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	15849	nM	Potency
TKC026870	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	3162	nM	Potency
TKC028718	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	11220	nM	Potency
TKC029307	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	47444	nM	Potency
TKC030478	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	18888	nM	Potency
TKC035029	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	398	nM	Potency
TKC035272	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	31623	nM	Potency
TKC035580	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	3	nM	Potency
TKC036999	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	31623	nM	Potency
TKC038473	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	447	nM	Potency
TKC039332	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	5012	nM	Potency
TKC040026	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	0	nM	Potency
TKC040829	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	316	nM	Potency
TKC052854	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	21192	nM	Potency
TKC053751	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	39811	nM	Potency
TKC055066	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	70795	nM	Potency
TKC056469	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	19953	nM	Potency
TKC056482	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	44668	nM	Potency
TKC057133	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	35481	nM	Potency
TKC062333	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	39811	nM	Potency
TKC063247	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	5	nM	Potency
TKC066332	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	31623	nM	Potency
TKC066411	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	5012	nM	Potency
TKC066631	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	2239	nM	Potency
TKC073833	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	3	nM	Potency
TKC075769	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	44668	nM	Potency
TKC076129	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	7080	nM	Potency
TKC077689	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	4467	nM	Potency
TKC080049	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	7943	nM	Potency
TKC080874	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	44668	nM	Potency
TKC085168	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	50	nM	Potency
TKC088230	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	2512	nM	Potency
TKC088231	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	31623	nM	Potency
TKC088678	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	316	nM	Potency
TKC090518	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	19953	nM	Potency
TKC092297	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	398	nM	Potency
TKC095442	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	2	nM	Potency
TKC095645	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	22387	nM	Potency
TKC097937	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	19953	nM	Potency
TKC097944	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	14125	nM	Potency
TKC100524	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	19953	nM	Potency
TKC100990	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	562	nM	Potency
TKC102657	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	29935	nM	Potency
TKC103150	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	31623	nM	Potency
TKC103159	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	50119	nM	Potency
TKC103538	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	4	nM	Potency
TKC104194	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	25119	nM	Potency
TKC105095	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	28184	nM	Potency
TKC105168	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	4	nM	Potency
TKC105226	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	11220	nM	Potency
TKC105356	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	39811	nM	Potency
TKC105357	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	35481	nM	Potency
TKC105378	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	355	nM	Potency
TKC105710	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	6310	nM	Potency
TKC105717	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	12589	nM	Potency
TKC106074	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	40	nM	Potency
TKC106147	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	1122	nM	Potency
TKC106537	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	19953	nM	Potency
TKC106682	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	20	nM	Potency
TKC107104	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	11220	nM	Potency
TKC107593	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	1259	nM	Potency
TKC107830	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	56	nM	Potency
TKC108060	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	44668	nM	Potency
TKC108363	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	11220	nM	Potency
TKC109484	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	3	nM	Potency
TKC109493	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	1337	nM	Potency
TKC110002	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	8913	nM	Potency
TKC112576	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	1413	nM	Potency
TKC112754	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	794	nM	Potency
TKC112784	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	3981	nM	Potency
TKC112813	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	7080	nM	Potency
TKC113063	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	28184	nM	Potency
TKC113150	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	1995	nM	Potency
TKC118131	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	44668	nM	Potency
TKC118419	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	44668	nM	Potency
TKC118895	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	14	nM	Potency
TKC118911	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	112	nM	Potency
TKC130327	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	251	nM	Potency
TKC130342	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	17783	nM	Potency
TKC133919	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	1585	nM	Potency
TKC141805	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	39811	nM	Potency
TKC150625	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	9466	nM	Potency
TKC150706	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	11220	nM	Potency
TKC151293	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	8913	nM	Potency
TKC151326	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	13	nM	Potency
TKC151609	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	39811	nM	Potency
TKC164433	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	9466	nM	Potency
TKC169452	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	2239	nM	Potency
TKC169457	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	2239	nM	Potency
TKC174441	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	8437	nM	Potency
TKC202992	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	3	nM	Potency
TKC206113	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	1778	nM	Potency
TKC206177	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	2511886	nM	Potency
TKC206657	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	501	nM	Potency
TKC206760	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	39811	nM	Potency
TKC206764	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	12589254	nM	Potency
TKC206779	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	79	nM	Potency
TKC206872	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	200	nM	Potency
TKC207103	P27695	DNA-(apurinic or apyrimidinic site) endonuclease	None	22	nM	Potency
TKC005313	P28482	Mitogen-activated protein kinase 1	None	25119	nM	Potency
TKC008529	P28482	Mitogen-activated protein kinase 1	None	126	nM	Potency
TKC013736	P28482	Mitogen-activated protein kinase 1	None	6310	nM	Potency
TKC019571	P28482	Mitogen-activated protein kinase 1	None	32	nM	Potency
TKC021977	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC022811	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC022814	P28482	Mitogen-activated protein kinase 1	None	28184	nM	Potency
TKC022945	P28482	Mitogen-activated protein kinase 1	None	5012	nM	Potency
TKC035272	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC035580	P28482	Mitogen-activated protein kinase 1	None	17783	nM	Potency
TKC038273	P28482	Mitogen-activated protein kinase 1	None	31623	nM	Potency
TKC039202	P28482	Mitogen-activated protein kinase 1	None	10000	nM	Potency
TKC054329	P28482	Mitogen-activated protein kinase 1	None	19953	nM	Potency
TKC060863	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC084630	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC087664	P28482	Mitogen-activated protein kinase 1	None	32	nM	Potency
TKC087988	P28482	Mitogen-activated protein kinase 1	None	462	nM	IC50
TKC092297	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC096011	P28482	Mitogen-activated protein kinase 1	None	3162	nM	Potency
TKC096012	P28482	Mitogen-activated protein kinase 1	None	576	nM	IC50
TKC100675	P28482	Mitogen-activated protein kinase 1	None	7943	nM	Potency
TKC101618	P28482	Mitogen-activated protein kinase 1	None	7943	nM	Potency
TKC102941	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC103150	P28482	Mitogen-activated protein kinase 1	None	3548	nM	Potency
TKC103257	P28482	Mitogen-activated protein kinase 1	None	14125	nM	Potency
TKC103736	P28482	Mitogen-activated protein kinase 1	None	15849	nM	Potency
TKC104091	P28482	Mitogen-activated protein kinase 1	None	5012	nM	Potency
TKC104194	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC105033	P28482	Mitogen-activated protein kinase 1	None	1259	nM	Potency
TKC105034	P28482	Mitogen-activated protein kinase 1	None	1259	nM	Potency
TKC105037	P28482	Mitogen-activated protein kinase 1	None	501	nM	Potency
TKC105210	P28482	Mitogen-activated protein kinase 1	None	6310	nM	Potency
TKC105295	P28482	Mitogen-activated protein kinase 1	None	126	nM	Potency
TKC105891	P28482	Mitogen-activated protein kinase 1	None	19953	nM	Potency
TKC106074	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC106212	P28482	Mitogen-activated protein kinase 1	None	282	nM	Potency
TKC106422	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC107086	P28482	Mitogen-activated protein kinase 1	None	31623	nM	Potency
TKC107201	P28482	Mitogen-activated protein kinase 1	None	22387	nM	Potency
TKC107525	P28482	Mitogen-activated protein kinase 1	None	31623	nM	Potency
TKC107627	P28482	Mitogen-activated protein kinase 1	None	15849	nM	Potency
TKC108295	P28482	Mitogen-activated protein kinase 1	None	12589	nM	Potency
TKC108473	P28482	Mitogen-activated protein kinase 1	None	11220	nM	Potency
TKC108555	P28482	Mitogen-activated protein kinase 1	None	10000	nM	Potency
TKC108732	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC112745	P28482	Mitogen-activated protein kinase 1	None	31623	nM	Potency
TKC112747	P28482	Mitogen-activated protein kinase 1	None	126	nM	Potency
TKC112759	P28482	Mitogen-activated protein kinase 1	None	31623	nM	Potency
TKC112784	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC113125	P28482	Mitogen-activated protein kinase 1	None	22387	nM	Potency
TKC114819	P28482	Mitogen-activated protein kinase 1	None	19953	nM	Potency
TKC118419	P28482	Mitogen-activated protein kinase 1	None	90	%	Activity
TKC122892	P28482	Mitogen-activated protein kinase 1	None	25119	nM	Potency
TKC134702	P28482	Mitogen-activated protein kinase 1	None	31623	nM	Potency
TKC135961	P28482	Mitogen-activated protein kinase 1	None	5012	nM	Potency
TKC136852	P28482	Mitogen-activated protein kinase 1	None	1413	nM	Potency
TKC140757	P28482	Mitogen-activated protein kinase 1	None	28184	nM	Potency
TKC148482	P28482	Mitogen-activated protein kinase 1	None	159	nM	Potency
TKC149827	P28482	Mitogen-activated protein kinase 1	None	19953	nM	Potency
TKC151571	P28482	Mitogen-activated protein kinase 1	None	3981	nM	Potency
TKC151758	P28482	Mitogen-activated protein kinase 1	None	31623	nM	Potency
TKC206688	P28482	Mitogen-activated protein kinase 1	None	3162	nM	Potency
TKC206760	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC206770	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC206781	P28482	Mitogen-activated protein kinase 1	None	39811	nM	Potency
TKC206812	P28482	Mitogen-activated protein kinase 1	None	31623	nM	Potency
TKC206816	P28482	Mitogen-activated protein kinase 1	None	14125	nM	Potency
TKC206901	P28482	Mitogen-activated protein kinase 1	None	7943	nM	Potency
TKC207103	P28482	Mitogen-activated protein kinase 1	None	25119	nM	Potency
TKC112785	P29317	Ephrin type-A receptor 2	None	48978	nM	IC50
TKC206760	P29317	Ephrin type-A receptor 2	None	50000	nM	IC50
TKC012269	P30304	M-phase inducer phosphatase 1	None	>20	ug.mL-1	IC50
TKC045754	P30304	M-phase inducer phosphatase 1	None	9400	nM	IC50
TKC045754	P30304	M-phase inducer phosphatase 1	None	35000	nM	IC50
TKC045754	P30304	M-phase inducer phosphatase 1	None	9400	nM	IC50
TKC045754	P30304	M-phase inducer phosphatase 1	None	9400	nM	IC50
TKC045754	P30304	M-phase inducer phosphatase 1	None	9400	nM	IC50
TKC045754	P30304	M-phase inducer phosphatase 1	None	9400	nM	IC50
TKC046478	P30304	M-phase inducer phosphatase 1	None	8400	nM	IC50
TKC072047	P30304	M-phase inducer phosphatase 1	None	5100	nM	IC50
TKC072048	P30304	M-phase inducer phosphatase 1	None	15000	nM	IC50
TKC094559	P30304	M-phase inducer phosphatase 1	None	7800	nM	IC50
TKC103390	P30304	M-phase inducer phosphatase 1	None	13000	nM	IC50
TKC115268	P30304	M-phase inducer phosphatase 1	None	890	nM	IC50
TKC164952	P30304	M-phase inducer phosphatase 1	None	5900	nM	IC50
TKC205544	P30304	M-phase inducer phosphatase 1	None	22300	nM	IC50
TKC013306	P30305	M-phase inducer phosphatase 2	None	<50	%	Inhibition
TKC026600	P30305	M-phase inducer phosphatase 2	None	92000	nM	IC50
TKC026891	P30305	M-phase inducer phosphatase 2	None	<50	%	Inhibition
TKC045754	P30305	M-phase inducer phosphatase 2	None	87000	nM	IC50
TKC072048	P30305	M-phase inducer phosphatase 2	None	19000	nM	IC50
TKC077689	P30305	M-phase inducer phosphatase 2	None	980	nM	IC50
TKC096012	P30305	M-phase inducer phosphatase 2	None	>50000	nM	IC50
TKC103390	P30305	M-phase inducer phosphatase 2	None	18000	nM	IC50
TKC112796	P30305	M-phase inducer phosphatase 2	None	<50	%	Inhibition
TKC116328	P30305	M-phase inducer phosphatase 2	None	<50	%	Inhibition
TKC116342	P30305	M-phase inducer phosphatase 2	None	<50	%	Inhibition
TKC131482	P30305	M-phase inducer phosphatase 2	None	23230	nM	IC50
TKC150004	P30305	M-phase inducer phosphatase 2	None	<50	%	Inhibition
TKC206840	P30305	M-phase inducer phosphatase 2	None	<50	%	Inhibition
TKC024886	P30530	Tyrosine-protein kinase receptor UFO	None	13100	nM	IC50
TKC025690	P30530	Tyrosine-protein kinase receptor UFO	None	14700	nM	IC50
TKC115259	P30530	Tyrosine-protein kinase receptor UFO	None	21900	nM	IC50
TKC115261	P30530	Tyrosine-protein kinase receptor UFO	None	14700	nM	IC50
TKC115272	P30530	Tyrosine-protein kinase receptor UFO	None	>100000	nM	IC50
TKC115273	P30530	Tyrosine-protein kinase receptor UFO	None	20200	nM	IC50
TKC152148	P30530	Tyrosine-protein kinase receptor UFO	None	16900	nM	IC50
TKC152157	P30530	Tyrosine-protein kinase receptor UFO	None	32600	nM	IC50
TKC174547	P30530	Tyrosine-protein kinase receptor UFO	None	>100000	nM	IC50
TKC111727	P31645	Sodium-dependent serotonin transporter	None	5491	nM	Ki
TKC111738	P31645	Sodium-dependent serotonin transporter	None	2816	nM	Ki
TKC205544	P31645	Sodium-dependent serotonin transporter	None	1000	nM	Ki
TKC011761	P31749	RAC-alpha serine/threonine-protein kinase	None	54	%	Inhibition
TKC016414	P31749	RAC-alpha serine/threonine-protein kinase	None	36	%	Activity
TKC024886	P31749	RAC-alpha serine/threonine-protein kinase	None	48400	nM	IC50
TKC025690	P31749	RAC-alpha serine/threonine-protein kinase	None	>100000	nM	IC50
TKC044763	P31749	RAC-alpha serine/threonine-protein kinase	None	100	%	Inhibition
TKC115259	P31749	RAC-alpha serine/threonine-protein kinase	None	>100000	nM	IC50
TKC115261	P31749	RAC-alpha serine/threonine-protein kinase	None	>100000	nM	IC50
TKC115272	P31749	RAC-alpha serine/threonine-protein kinase	None	>100000	nM	IC50
TKC115273	P31749	RAC-alpha serine/threonine-protein kinase	None	>100000	nM	IC50
TKC118419	P31749	RAC-alpha serine/threonine-protein kinase	None	96	%	Inhibition
TKC152148	P31749	RAC-alpha serine/threonine-protein kinase	None	>100000	nM	IC50
TKC152157	P31749	RAC-alpha serine/threonine-protein kinase	None	>100000	nM	IC50
TKC174547	P31749	RAC-alpha serine/threonine-protein kinase	None	>100000	nM	IC50
TKC206776	P31749	RAC-alpha serine/threonine-protein kinase	None	3	uM	Activity
TKC146515	P32302	C-X-C chemokine receptor type 5	None	9456	nM	IC50
TKC011412	P35222	Catenin beta-1	None	5213	nM	IC50
TKC037534	P35228	Nitric oxide synthase, inducible	None	99	%	Inhibition
TKC060880	P35228	Nitric oxide synthase, inducible	None	37000	nM	IC50
TKC077689	P35228	Nitric oxide synthase, inducible	None	>40000	nM	IC50
TKC206319	P35228	Nitric oxide synthase, inducible	None	100	%	Inhibition
TKC008359	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC010020	P35354	Prostaglandin G/H synthase 2	None	61	%	Inhibition
TKC010022	P35354	Prostaglandin G/H synthase 2	None	55	%	Inhibition
TKC010023	P35354	Prostaglandin G/H synthase 2	None	57	%	Inhibition
TKC010024	P35354	Prostaglandin G/H synthase 2	None	42	%	Inhibition
TKC010025	P35354	Prostaglandin G/H synthase 2	None	78	%	Inhibition
TKC010026	P35354	Prostaglandin G/H synthase 2	None	17	%	Inhibition
TKC011599	P35354	Prostaglandin G/H synthase 2	None	64	%	Inhibition
TKC012919	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC012941	P35354	Prostaglandin G/H synthase 2	None	8500	nM	IC50
TKC012956	P35354	Prostaglandin G/H synthase 2	None	2200	nM	IC50
TKC012962	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC015443	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC015459	P35354	Prostaglandin G/H synthase 2	None	2200	nM	IC50
TKC015537	P35354	Prostaglandin G/H synthase 2	None	0	%	Inhibition
TKC016794	P35354	Prostaglandin G/H synthase 2	None	40	nM	IC50
TKC019436	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC019466	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC019819	P35354	Prostaglandin G/H synthase 2	None	35	%	Inhibition
TKC019859	P35354	Prostaglandin G/H synthase 2	None	<33	%	Inhibition
TKC020479	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC020796	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC021940	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC022833	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC022834	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC022961	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC026245	P35354	Prostaglandin G/H synthase 2	None	2300	nM	IC50
TKC027200	P35354	Prostaglandin G/H synthase 2	None	700	nM	IC50
TKC028143	P35354	Prostaglandin G/H synthase 2	None	100	%	Inhibition
TKC031202	P35354	Prostaglandin G/H synthase 2	None	3800	nM	IC50
TKC031223	P35354	Prostaglandin G/H synthase 2	None	45	%	Inhibition
TKC032234	P35354	Prostaglandin G/H synthase 2	None	400	nM	IC50
TKC035208	P35354	Prostaglandin G/H synthase 2	None	7	uM	IC60
TKC037534	P35354	Prostaglandin G/H synthase 2	None	97	%	Inhibition
TKC038330	P35354	Prostaglandin G/H synthase 2	None	2900	nM	IC50
TKC041884	P35354	Prostaglandin G/H synthase 2	None	18000	nM	IC50
TKC043993	P35354	Prostaglandin G/H synthase 2	None	98	%	Inhibition
TKC045188	P35354	Prostaglandin G/H synthase 2	None	98	%	Inhibition
TKC048282	P35354	Prostaglandin G/H synthase 2	None	370	nM	IC50
TKC049750	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC049818	P35354	Prostaglandin G/H synthase 2	None	5	ug	IC50
TKC051154	P35354	Prostaglandin G/H synthase 2	None	>61	%	Activity
TKC054011	P35354	Prostaglandin G/H synthase 2	None	9000	nM	IC50
TKC054031	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC054081	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC054090	P35354	Prostaglandin G/H synthase 2	None	8900	nM	IC50
TKC054099	P35354	Prostaglandin G/H synthase 2	None	7800	nM	IC50
TKC054100	P35354	Prostaglandin G/H synthase 2	None	7900	nM	IC50
TKC054101	P35354	Prostaglandin G/H synthase 2	None	8800	nM	IC50
TKC054240	P35354	Prostaglandin G/H synthase 2	None	6700	nM	IC50
TKC054241	P35354	Prostaglandin G/H synthase 2	None	6100	nM	IC50
TKC056482	P35354	Prostaglandin G/H synthase 2	None	40000	nM	IC50
TKC056482	P35354	Prostaglandin G/H synthase 2	None	86000	nM	IC50
TKC056482	P35354	Prostaglandin G/H synthase 2	None	130000	nM	IC50
TKC057308	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC058811	P35354	Prostaglandin G/H synthase 2	None	>85	%	Activity
TKC058812	P35354	Prostaglandin G/H synthase 2	None	>78	%	Activity
TKC060184	P35354	Prostaglandin G/H synthase 2	None	8500	nM	IC50
TKC060216	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC060284	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC060302	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC060303	P35354	Prostaglandin G/H synthase 2	None	7200	nM	IC50
TKC060304	P35354	Prostaglandin G/H synthase 2	None	7600	nM	IC50
TKC060399	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC060602	P35354	Prostaglandin G/H synthase 2	None	6700	nM	IC50
TKC061939	P35354	Prostaglandin G/H synthase 2	None	>10000	nM	IC50
TKC061968	P35354	Prostaglandin G/H synthase 2	None	>10000	nM	IC50
TKC061969	P35354	Prostaglandin G/H synthase 2	None	>10000	nM	IC50
TKC064374	P35354	Prostaglandin G/H synthase 2	None	>73	%	Activity
TKC064407	P35354	Prostaglandin G/H synthase 2	None	>78	%	Activity
TKC065375	P35354	Prostaglandin G/H synthase 2	None	>70	%	Activity
TKC066954	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC070952	P35354	Prostaglandin G/H synthase 2	None	>100000	nM	IC50
TKC071010	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC071640	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC076350	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC077689	P35354	Prostaglandin G/H synthase 2	None	40000	nM	IC50
TKC077689	P35354	Prostaglandin G/H synthase 2	None	295000	nM	IC50
TKC077689	P35354	Prostaglandin G/H synthase 2	None	295000	nM	IC50
TKC077689	P35354	Prostaglandin G/H synthase 2	None	87000	nM	IC50
TKC077703	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC078194	P35354	Prostaglandin G/H synthase 2	None	>74	%	Activity
TKC085168	P35354	Prostaglandin G/H synthase 2	None	<60	%	Inhibition
TKC088678	P35354	Prostaglandin G/H synthase 2	None	>72	%	Activity
TKC095276	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC095567	P35354	Prostaglandin G/H synthase 2	None	>10000	nM	IC50
TKC110247	P35354	Prostaglandin G/H synthase 2	None	>10	ug.mL-1	IC50
TKC113936	P35354	Prostaglandin G/H synthase 2	None	60	%	Inhibition
TKC122543	P35354	Prostaglandin G/H synthase 2	None	30	%	Inhibition
TKC123028	P35354	Prostaglandin G/H synthase 2	None	>72	%	Activity
TKC129152	P35354	Prostaglandin G/H synthase 2	None	>100000	nM	IC50
TKC130084	P35354	Prostaglandin G/H synthase 2	None	37	%	Inhibition
TKC130119	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC130223	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC130577	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC130901	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC135264	P35354	Prostaglandin G/H synthase 2	None	400	nM	IC50
TKC135559	P35354	Prostaglandin G/H synthase 2	None	4600	nM	IC50
TKC139036	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC139322	P35354	Prostaglandin G/H synthase 2	None	>82	%	Activity
TKC139366	P35354	Prostaglandin G/H synthase 2	None	40000	nM	IC50
TKC140627	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC141365	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC141401	P35354	Prostaglandin G/H synthase 2	None	>75	%	Activity
TKC141499	P35354	Prostaglandin G/H synthase 2	None	>87	%	Activity
TKC141601	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC141602	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC141622	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC141805	P35354	Prostaglandin G/H synthase 2	None	40000	nM	IC50
TKC142150	P35354	Prostaglandin G/H synthase 2	None	450000	nM	IC50
TKC142203	P35354	Prostaglandin G/H synthase 2	None	>10000	nM	IC50
TKC142208	P35354	Prostaglandin G/H synthase 2	None	>10000	nM	IC50
TKC142849	P35354	Prostaglandin G/H synthase 2	None	>69	%	Activity
TKC142897	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC142922	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC143527	P35354	Prostaglandin G/H synthase 2	None	97	%	Inhibition
TKC143539	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC143641	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC145295	P35354	Prostaglandin G/H synthase 2	None	22	%	Inhibition
TKC145848	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC145932	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC145968	P35354	Prostaglandin G/H synthase 2	None	>94	%	Activity
TKC146116	P35354	Prostaglandin G/H synthase 2	None	>5.0e+4	nM	IC50
TKC146774	P35354	Prostaglandin G/H synthase 2	None	>78	%	Activity
TKC146857	P35354	Prostaglandin G/H synthase 2	None	600	nM	IC50
TKC149251	P35354	Prostaglandin G/H synthase 2	None	1100	nM	IC50
TKC149759	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC149924	P35354	Prostaglandin G/H synthase 2	None	800	nM	IC50
TKC149926	P35354	Prostaglandin G/H synthase 2	None	800	nM	IC50
TKC150635	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC150706	P35354	Prostaglandin G/H synthase 2	None	>76	%	Activity
TKC150907	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC151280	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC151284	P35354	Prostaglandin G/H synthase 2	None	33	%	Inhibition
TKC151765	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC152742	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC152813	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC156345	P35354	Prostaglandin G/H synthase 2	None	25	%	Inhibition
TKC156572	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC156716	P35354	Prostaglandin G/H synthase 2	None	2200	nM	IC50
TKC170277	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC172853	P35354	Prostaglandin G/H synthase 2	None	4700	nM	IC50
TKC174442	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC205509	P35354	Prostaglandin G/H synthase 2	None	540000	nM	IC50
TKC205699	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC205700	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC206319	P35354	Prostaglandin G/H synthase 2	None	99	%	Inhibition
TKC205544	P35462	D(3) dopamine receptor	None	2489	nM	Ki
TKC205544	P35462	D(3) dopamine receptor	None	3981.07	nM	Ki
TKC206544	P35462	D(3) dopamine receptor	None	>10000	nM	Ki
TKC206549	P35869	Aryl hydrocarbon receptor	None	17783	nM	Potency
TKC024886	P35968	Vascular endothelial growth factor receptor 2	None	4810	nM	IC50
TKC025690	P35968	Vascular endothelial growth factor receptor 2	None	3660	nM	IC50
TKC051154	P35968	Vascular endothelial growth factor receptor 2	None	40	%	Inhibition
TKC051155	P35968	Vascular endothelial growth factor receptor 2	None	46	%	Inhibition
TKC065375	P35968	Vascular endothelial growth factor receptor 2	None	0	%	Inhibition
TKC102689	P35968	Vascular endothelial growth factor receptor 2	None	0	%	Inhibition
TKC108267	P35968	Vascular endothelial growth factor receptor 2	None	0	%	Inhibition
TKC115259	P35968	Vascular endothelial growth factor receptor 2	None	4950	nM	IC50
TKC115261	P35968	Vascular endothelial growth factor receptor 2	None	4600	nM	IC50
TKC115272	P35968	Vascular endothelial growth factor receptor 2	None	>100000	nM	IC50
TKC115273	P35968	Vascular endothelial growth factor receptor 2	None	4850	nM	IC50
TKC146202	P35968	Vascular endothelial growth factor receptor 2	None	61	%	Inhibition
TKC152148	P35968	Vascular endothelial growth factor receptor 2	None	4350	nM	IC50
TKC152157	P35968	Vascular endothelial growth factor receptor 2	None	6010	nM	IC50
TKC174547	P35968	Vascular endothelial growth factor receptor 2	None	>100000	nM	IC50
TKC207124	P35968	Vascular endothelial growth factor receptor 2	None	40400	nM	IC50
TKC005728	P37231	Peroxisome proliferator-activated receptor gamma	None	>100000	nM	EC50
TKC005729	P37231	Peroxisome proliferator-activated receptor gamma	None	16700	nM	EC50
TKC013753	P37231	Peroxisome proliferator-activated receptor gamma	None	2818	nM	Potency
TKC021262	P37231	Peroxisome proliferator-activated receptor gamma	None	21700	nM	EC50
TKC035272	P37231	Peroxisome proliferator-activated receptor gamma	None	7943	nM	Potency
TKC066169	P37231	Peroxisome proliferator-activated receptor gamma	None	28184	nM	Potency
TKC075769	P37231	Peroxisome proliferator-activated receptor gamma	None	316	nM	Potency
TKC079000	P37231	Peroxisome proliferator-activated receptor gamma	None	50119	nM	Potency
TKC087664	P37231	Peroxisome proliferator-activated receptor gamma	None	44668	nM	Potency
TKC087991	P37231	Peroxisome proliferator-activated receptor gamma	None	3162	nM	Potency
TKC088230	P37231	Peroxisome proliferator-activated receptor gamma	None	44668	nM	Potency
TKC092297	P37231	Peroxisome proliferator-activated receptor gamma	None	15849	nM	Potency
TKC096012	P37231	Peroxisome proliferator-activated receptor gamma	None	316	nM	Potency
TKC100644	P37231	Peroxisome proliferator-activated receptor gamma	None	44668	nM	Potency
TKC102407	P37231	Peroxisome proliferator-activated receptor gamma	None	50119	nM	Potency
TKC107086	P37231	Peroxisome proliferator-activated receptor gamma	None	28184	nM	Potency
TKC107735	P37231	Peroxisome proliferator-activated receptor gamma	None	39811	nM	Potency
TKC108536	P37231	Peroxisome proliferator-activated receptor gamma	None	44668	nM	Potency
TKC110634	P37231	Peroxisome proliferator-activated receptor gamma	None	6400	nM	EC50
TKC110635	P37231	Peroxisome proliferator-activated receptor gamma	None	8200	nM	EC50
TKC111200	P37231	Peroxisome proliferator-activated receptor gamma	None	22300	nM	EC50
TKC111271	P37231	Peroxisome proliferator-activated receptor gamma	None	>50000	nM	EC50
TKC111272	P37231	Peroxisome proliferator-activated receptor gamma	None	18700	nM	EC50
TKC111273	P37231	Peroxisome proliferator-activated receptor gamma	None	>50000	nM	EC50
TKC111274	P37231	Peroxisome proliferator-activated receptor gamma	None	20600	nM	EC50
TKC111276	P37231	Peroxisome proliferator-activated receptor gamma	None	>50000	nM	EC50
TKC111284	P37231	Peroxisome proliferator-activated receptor gamma	None	>50000	nM	EC50
TKC111466	P37231	Peroxisome proliferator-activated receptor gamma	None	>50000	nM	EC50
TKC115268	P37231	Peroxisome proliferator-activated receptor gamma	None	44668	nM	Potency
TKC170559	P37231	Peroxisome proliferator-activated receptor gamma	None	1000	nM	EC50
TKC206549	P37231	Peroxisome proliferator-activated receptor gamma	None	126	nM	Potency
TKC206652	P37231	Peroxisome proliferator-activated receptor gamma	None	316	nM	Potency
TKC206672	P37231	Peroxisome proliferator-activated receptor gamma	None	31623	nM	Potency
TKC206759	P37231	Peroxisome proliferator-activated receptor gamma	None	12589	nM	Potency
TKC206760	P37231	Peroxisome proliferator-activated receptor gamma	None	17783	nM	Potency
TKC206812	P37231	Peroxisome proliferator-activated receptor gamma	None	27000	nM	IC50
TKC206812	P37231	Peroxisome proliferator-activated receptor gamma	None	50119	nM	Potency
TKC206816	P37231	Peroxisome proliferator-activated receptor gamma	None	39811	nM	Potency
TKC003060	P40763	Signal transducer and activator of transcription 3	None	>50000	nM	IC50
TKC005454	P40763	Signal transducer and activator of transcription 3	None	4600	nM	IC50
TKC016414	P40763	Signal transducer and activator of transcription 3	None	>10000	nM	EC50
TKC020636	P40763	Signal transducer and activator of transcription 3	None	6900	nM	IC50
TKC020796	P40763	Signal transducer and activator of transcription 3	None	22900	nM	IC50
TKC020867	P40763	Signal transducer and activator of transcription 3	None	26	%	Inhibition
TKC020868	P40763	Signal transducer and activator of transcription 3	None	31	%	Inhibition
TKC020869	P40763	Signal transducer and activator of transcription 3	None	49	%	Inhibition
TKC022393	P40763	Signal transducer and activator of transcription 3	None	89500	nM	IC50
TKC022771	P40763	Signal transducer and activator of transcription 3	None	>100000	nM	IC50
TKC028367	P40763	Signal transducer and activator of transcription 3	None	4100	nM	IC50
TKC030728	P40763	Signal transducer and activator of transcription 3	None	2	%	Inhibition
TKC033506	P40763	Signal transducer and activator of transcription 3	None	2400	nM	IC50
TKC033507	P40763	Signal transducer and activator of transcription 3	None	2300	nM	IC50
TKC036334	P40763	Signal transducer and activator of transcription 3	None	4	%	Inhibition
TKC038766	P40763	Signal transducer and activator of transcription 3	None	1	%	Inhibition
TKC039282	P40763	Signal transducer and activator of transcription 3	None	2	%	Inhibition
TKC042554	P40763	Signal transducer and activator of transcription 3	None	6300	nM	IC50
TKC042556	P40763	Signal transducer and activator of transcription 3	None	110000	nM	IC50
TKC044507	P40763	Signal transducer and activator of transcription 3	None	4	%	Inhibition
TKC044595	P40763	Signal transducer and activator of transcription 3	None	4	%	Inhibition
TKC044621	P40763	Signal transducer and activator of transcription 3	None	3	%	Inhibition
TKC044669	P40763	Signal transducer and activator of transcription 3	None	4	%	Inhibition
TKC047957	P40763	Signal transducer and activator of transcription 3	None	17100	nM	IC50
TKC047959	P40763	Signal transducer and activator of transcription 3	None	>30000	nM	IC50
TKC047961	P40763	Signal transducer and activator of transcription 3	None	>30000	nM	IC50
TKC048029	P40763	Signal transducer and activator of transcription 3	None	270	nM	IC50
TKC048030	P40763	Signal transducer and activator of transcription 3	None	19200	nM	IC50
TKC048031	P40763	Signal transducer and activator of transcription 3	None	590	nM	IC50
TKC051029	P40763	Signal transducer and activator of transcription 3	None	60000	nM	MIC
TKC060882	P40763	Signal transducer and activator of transcription 3	None	>25000	nM	IC50
TKC075769	P40763	Signal transducer and activator of transcription 3	None	1862	nM	IC50
TKC077689	P40763	Signal transducer and activator of transcription 3	None	>50000	nM	IC50
TKC078334	P40763	Signal transducer and activator of transcription 3	None	>50000	nM	IC50
TKC087623	P40763	Signal transducer and activator of transcription 3	None	>100000	nM	IC50
TKC087625	P40763	Signal transducer and activator of transcription 3	None	7000	nM	IC50
TKC093311	P40763	Signal transducer and activator of transcription 3	None	>50000	nM	IC50
TKC100739	P40763	Signal transducer and activator of transcription 3	None	>50000	nM	IC50
TKC101161	P40763	Signal transducer and activator of transcription 3	None	>50000	nM	IC50
TKC103159	P40763	Signal transducer and activator of transcription 3	None	3000	nM	IC50
TKC103189	P40763	Signal transducer and activator of transcription 3	None	32500	nM	IC50
TKC103191	P40763	Signal transducer and activator of transcription 3	None	24800	nM	IC50
TKC105152	P40763	Signal transducer and activator of transcription 3	None	>50000	nM	IC50
TKC107659	P40763	Signal transducer and activator of transcription 3	None	4	%	Inhibition
TKC108773	P40763	Signal transducer and activator of transcription 3	None	>50000	nM	IC50
TKC112576	P40763	Signal transducer and activator of transcription 3	None	1154	nM	IC50
TKC134761	P40763	Signal transducer and activator of transcription 3	None	48	%	Inhibition
TKC135961	P40763	Signal transducer and activator of transcription 3	None	73000	nM	IC50
TKC135978	P40763	Signal transducer and activator of transcription 3	None	14210	nM	IC50
TKC136653	P40763	Signal transducer and activator of transcription 3	None	2	%	Inhibition
TKC148207	P40763	Signal transducer and activator of transcription 3	None	15840	nM	IC50
TKC149924	P40763	Signal transducer and activator of transcription 3	None	74	%	Inhibition
TKC151284	P40763	Signal transducer and activator of transcription 3	None	14000	nM	IC50
TKC156528	P40763	Signal transducer and activator of transcription 3	None	>30000	nM	IC50
TKC206318	P40763	Signal transducer and activator of transcription 3	None	12200	nM	IC50
TKC206468	P40763	Signal transducer and activator of transcription 3	None	46	%	Inhibition
TKC206627	P40763	Signal transducer and activator of transcription 3	None	>100000	nM	IC50
TKC206646	P40763	Signal transducer and activator of transcription 3	None	67000	nM	IC50
TKC206652	P40763	Signal transducer and activator of transcription 3	None	700	nM	IC50
TKC025058	P42336	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	None	100	nM	IC50
TKC118380	P42336	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	None	1	nM	IC50
TKC118419	P42336	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	None	1	nM	IC50
TKC118419	P42336	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	None	12	nM	IC50
TKC118419	P42336	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	None	17.6	nM	IC50
TKC118419	P42336	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	None	120	nM	Ki
TKC118419	P42336	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	None	12	nM	IC50
TKC118419	P42336	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	None	12	nM	IC50
TKC118419	P42336	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	None	13	nM	IC50
TKC118419	P42336	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	None	1	nM	IC50
TKC118419	P42336	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	None	5.4	nM	Kd
TKC118419	P42338	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	None	8	nM	Kd
TKC118419	P42338	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	None	7.6	nM	Kd
TKC118419	P42338	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	None	10	nM	IC50
TKC118419	P42338	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	None	15	nM	IC50
TKC118419	P42338	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	None	14	nM	IC50
TKC022945	P42345	Serine/threonine-protein kinase mTOR	None	4645	nM	Potency
TKC032619	P42345	Serine/threonine-protein kinase mTOR	None	2931	nM	Potency
TKC035272	P42345	Serine/threonine-protein kinase mTOR	None	2612	nM	Potency
TKC035984	P42345	Serine/threonine-protein kinase mTOR	None	4	nM	Potency
TKC084630	P42345	Serine/threonine-protein kinase mTOR	None	3690	nM	Potency
TKC087988	P42345	Serine/threonine-protein kinase mTOR	None	4645	nM	Potency
TKC092297	P42345	Serine/threonine-protein kinase mTOR	None	13092	nM	Potency
TKC118419	P42345	Serine/threonine-protein kinase mTOR	None	40	nM	IC50
TKC118419	P42345	Serine/threonine-protein kinase mTOR	None	9200	nM	Kd
TKC205544	P42345	Serine/threonine-protein kinase mTOR	None	14689	nM	Potency
TKC206622	P42345	Serine/threonine-protein kinase mTOR	None	23281	nM	Potency
TKC206688	P42345	Serine/threonine-protein kinase mTOR	None	16482	nM	Potency
TKC036497	P42574	Caspase-3	None	200000	nM	IC50
TKC096499	P42574	Caspase-3	None	50000	nM	IC50
TKC205544	P43119	Prostacyclin receptor	None	8	%	Inhibition
TKC108557	P43405	Tyrosine-protein kinase SYK	None	0.2	nM	IC50
TKC021977	P45983	Mitogen-activated protein kinase 8	None	51	%	Inhibition
TKC118419	P45983	Mitogen-activated protein kinase 8	None	84	%	Activity
TKC130761	P45983	Mitogen-activated protein kinase 8	None	66	%	Inhibition
TKC118419	P45984	Mitogen-activated protein kinase 9	None	83	%	Activity
TKC112367	P46531	Neurogenic locus notch homolog protein 1	None	300	nM	IC50
TKC112399	P46531	Neurogenic locus notch homolog protein 1	None	2400	nM	IC50
TKC117085	P46531	Neurogenic locus notch homolog protein 1	None	17300	nM	IC50
TKC118351	P46531	Neurogenic locus notch homolog protein 1	None	400	nM	IC50
TKC118354	P46531	Neurogenic locus notch homolog protein 1	None	2000	nM	IC50
TKC118356	P46531	Neurogenic locus notch homolog protein 1	None	300	nM	IC50
TKC118360	P46531	Neurogenic locus notch homolog protein 1	None	700	nM	IC50
TKC206738	P46531	Neurogenic locus notch homolog protein 1	None	800	nM	IC50
TKC013186	P47989	Xanthine dehydrogenase/oxidase	None	1	%	Inhibition
TKC013187	P47989	Xanthine dehydrogenase/oxidase	None	0	%	Inhibition
TKC013189	P47989	Xanthine dehydrogenase/oxidase	None	1	%	Inhibition
TKC013192	P47989	Xanthine dehydrogenase/oxidase	None	8	%	Inhibition
TKC013193	P47989	Xanthine dehydrogenase/oxidase	None	-5	%	Inhibition
TKC013194	P47989	Xanthine dehydrogenase/oxidase	None	-1	%	Inhibition
TKC013195	P47989	Xanthine dehydrogenase/oxidase	None	-2	%	Inhibition
TKC013196	P47989	Xanthine dehydrogenase/oxidase	None	-7	%	Inhibition
TKC013229	P47989	Xanthine dehydrogenase/oxidase	None	5	%	Inhibition
TKC013255	P47989	Xanthine dehydrogenase/oxidase	None	1	%	Inhibition
TKC013256	P47989	Xanthine dehydrogenase/oxidase	None	0	%	Inhibition
TKC013260	P47989	Xanthine dehydrogenase/oxidase	None	2	%	Inhibition
TKC055544	P47989	Xanthine dehydrogenase/oxidase	None	97300	nM	IC50
TKC066955	P47989	Xanthine dehydrogenase/oxidase	None	150400	nM	IC50
TKC094167	P47989	Xanthine dehydrogenase/oxidase	None	79880	nM	IC50
TKC011761	P48443	Retinoic acid receptor RXR-gamma	None	42000	nM	EC50
TKC013755	P48443	Retinoic acid receptor RXR-gamma	None	4	nM	IC50
TKC013755	P48443	Retinoic acid receptor RXR-gamma	None	219	nM	EC50
TKC013755	P48443	Retinoic acid receptor RXR-gamma	None	4.3	nM	EC50
TKC013755	P48443	Retinoic acid receptor RXR-gamma	None	14	nM	Ki
TKC013755	P48443	Retinoic acid receptor RXR-gamma	None	140	nM	EC50
TKC013755	P48443	Retinoic acid receptor RXR-gamma	None	11	nM	Ki
TKC013755	P48443	Retinoic acid receptor RXR-gamma	None	14	nM	Kd
TKC013755	P48443	Retinoic acid receptor RXR-gamma	None	30	nM	Kd
TKC013755	P48443	Retinoic acid receptor RXR-gamma	None	14	nM	Kd
TKC013755	P48443	Retinoic acid receptor RXR-gamma	None	140	nM	EC50
TKC013755	P48443	Retinoic acid receptor RXR-gamma	None	16	nM	Kd
TKC013755	P48443	Retinoic acid receptor RXR-gamma	None	27	nM	Ki
TKC092297	P48443	Retinoic acid receptor RXR-gamma	None	>6000	nM	Ki
TKC096012	P48443	Retinoic acid receptor RXR-gamma	None	1100	nM	EC50
TKC096012	P48443	Retinoic acid receptor RXR-gamma	None	350	nM	IC50
TKC096012	P48443	Retinoic acid receptor RXR-gamma	None	288	nM	Ki
TKC096012	P48443	Retinoic acid receptor RXR-gamma	None	2	nM	EC50
TKC096012	P48443	Retinoic acid receptor RXR-gamma	None	1100	nM	EC50
TKC096012	P48443	Retinoic acid receptor RXR-gamma	None	120	nM	Ki
TKC096012	P48443	Retinoic acid receptor RXR-gamma	None	>0.001000	nM	Kd
TKC096012	P48443	Retinoic acid receptor RXR-gamma	None	1.4	nM	Ki
TKC096012	P48443	Retinoic acid receptor RXR-gamma	None	306	nM	Kd
TKC096012	P48443	Retinoic acid receptor RXR-gamma	None	1100	nM	EC50
TKC122848	P48443	Retinoic acid receptor RXR-gamma	None	33000	nM	EC50
TKC136411	P48443	Retinoic acid receptor RXR-gamma	None	43000	nM	EC50
TKC025058	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	1000	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	5	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	19	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	55	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	55000	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	89	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	5	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	15	nM	Kd
TKC025129	P49137	MAP kinase-activated protein kinase 2	None	20000	nM	IC50
TKC026722	P49137	MAP kinase-activated protein kinase 2	None	9600	nM	IC50
TKC045646	P49137	MAP kinase-activated protein kinase 2	None	90000	nM	IC50
TKC045794	P49137	MAP kinase-activated protein kinase 2	None	90000	nM	IC50
TKC045994	P49137	MAP kinase-activated protein kinase 2	None	90000	nM	IC50
TKC045996	P49137	MAP kinase-activated protein kinase 2	None	90000	nM	IC50
TKC118419	P49137	MAP kinase-activated protein kinase 2	None	102	%	Inhibition
TKC087988	P49327	Fatty acid synthase	None	>40	%	Inhibition
TKC011761	P49841	Glycogen synthase kinase-3 beta	None	20	%	Inhibition
TKC046098	P49841	Glycogen synthase kinase-3 beta	None	794	nM	IC50
TKC046099	P49841	Glycogen synthase kinase-3 beta	None	2300	nM	IC50
TKC046324	P49841	Glycogen synthase kinase-3 beta	None	4500	nM	IC50
TKC046324	P49841	Glycogen synthase kinase-3 beta	None	1900	nM	IC50
TKC118419	P49841	Glycogen synthase kinase-3 beta	None	65	%	Activity
TKC146056	P49841	Glycogen synthase kinase-3 beta	None	3000	nM	IC50
TKC113582	P50281	Matrix metalloproteinase-14	None	19	ug.mL-1	IC50
TKC034760	P50579	Methionine aminopeptidase 2	None	1	nM	IC50
TKC039945	P50579	Methionine aminopeptidase 2	None	0	nM	IC50
TKC039946	P50579	Methionine aminopeptidase 2	None	4	nM	IC50
TKC039948	P50579	Methionine aminopeptidase 2	None	6	nM	IC50
TKC039950	P50579	Methionine aminopeptidase 2	None	0.4	nM	IC50
TKC074337	P50579	Methionine aminopeptidase 2	None	1	nM	IC50
TKC074337	P50579	Methionine aminopeptidase 2	None	1	nM	Ki
TKC074337	P50579	Methionine aminopeptidase 2	None	1050	nM	IC50
TKC074337	P50579	Methionine aminopeptidase 2	None	1	nM	IC50
TKC074337	P50579	Methionine aminopeptidase 2	None	1320	nM	IC50
TKC074338	P50579	Methionine aminopeptidase 2	None	1	nM	IC50
TKC074338	P50579	Methionine aminopeptidase 2	None	275	nM	IC50
TKC074339	P50579	Methionine aminopeptidase 2	None	1	nM	IC50
TKC089659	P50579	Methionine aminopeptidase 2	None	0.4	nM	IC50
TKC101244	P50579	Methionine aminopeptidase 2	None	8	nM	IC50
TKC104441	P50579	Methionine aminopeptidase 2	None	1	nM	IC50
TKC104442	P50579	Methionine aminopeptidase 2	None	4	%	Activity
TKC146326	P50579	Methionine aminopeptidase 2	None	9	%	Inhibition
TKC013304	P51449	Nuclear receptor ROR-gamma	None	66824	nM	Potency
TKC013753	P51449	Nuclear receptor ROR-gamma	None	29849	nM	Potency
TKC013755	P51449	Nuclear receptor ROR-gamma	None	14000	nM	EC50
TKC021977	P51449	Nuclear receptor ROR-gamma	None	42163	nM	Potency
TKC022931	P51449	Nuclear receptor ROR-gamma	None	84	nM	Potency
TKC056482	P51449	Nuclear receptor ROR-gamma	None	130	nM	IC50
TKC066169	P51449	Nuclear receptor ROR-gamma	None	33492	nM	Potency
TKC075769	P51449	Nuclear receptor ROR-gamma	None	1980	nM	IC50
TKC075769	P51449	Nuclear receptor ROR-gamma	None	109	nM	Kd
TKC075769	P51449	Nuclear receptor ROR-gamma	None	2000	nM	IC50
TKC083807	P51449	Nuclear receptor ROR-gamma	None	10591	nM	Potency
TKC087664	P51449	Nuclear receptor ROR-gamma	None	47308	nM	Potency
TKC087991	P51449	Nuclear receptor ROR-gamma	None	21132	nM	Potency
TKC088230	P51449	Nuclear receptor ROR-gamma	None	1333	nM	Potency
TKC088231	P51449	Nuclear receptor ROR-gamma	None	23710	nM	Potency
TKC092297	P51449	Nuclear receptor ROR-gamma	None	26603	nM	Potency
TKC096012	P51449	Nuclear receptor ROR-gamma	None	200	nM	IC50
TKC096012	P51449	Nuclear receptor ROR-gamma	None	18000	nM	EC50
TKC097944	P51449	Nuclear receptor ROR-gamma	None	4216	nM	Potency
TKC102407	P51449	Nuclear receptor ROR-gamma	None	21132	nM	Potency
TKC107086	P51449	Nuclear receptor ROR-gamma	None	3758	nM	Potency
TKC115268	P51449	Nuclear receptor ROR-gamma	None	37578	nM	Potency
TKC118648	P51449	Nuclear receptor ROR-gamma	None	80	nM	EC50
TKC118652	P51449	Nuclear receptor ROR-gamma	None	110	nM	EC50
TKC118929	P51449	Nuclear receptor ROR-gamma	None	10	nM	Ki
TKC118938	P51449	Nuclear receptor ROR-gamma	None	10	nM	Ki
TKC122884	P51449	Nuclear receptor ROR-gamma	None	20	nM	EC50
TKC136411	P51449	Nuclear receptor ROR-gamma	None	37578	nM	Potency
TKC151274	P51449	Nuclear receptor ROR-gamma	None	60	nM	Potency
TKC206457	P51449	Nuclear receptor ROR-gamma	None	20	nM	EC50
TKC206457	P51449	Nuclear receptor ROR-gamma	None	20	nM	EC50
TKC206457	P51449	Nuclear receptor ROR-gamma	None	20	nM	EC50
TKC206458	P51449	Nuclear receptor ROR-gamma	None	20	nM	EC50
TKC206459	P51449	Nuclear receptor ROR-gamma	None	7	degrees C	T
TKC206672	P51449	Nuclear receptor ROR-gamma	None	42163	nM	Potency
TKC206688	P51449	Nuclear receptor ROR-gamma	None	23710	nM	Potency
TKC206759	P51449	Nuclear receptor ROR-gamma	None	26603	nM	Potency
TKC206760	P51449	Nuclear receptor ROR-gamma	None	74978	nM	Potency
TKC206770	P51449	Nuclear receptor ROR-gamma	None	33492	nM	Potency
TKC206812	P51449	Nuclear receptor ROR-gamma	None	47308	nM	Potency
TKC206816	P51449	Nuclear receptor ROR-gamma	None	8413	nM	Potency
TKC206915	P51449	Nuclear receptor ROR-gamma	None	10	nM	Ki
TKC046294	P51681	C-C chemokine receptor type 5	None	40000	nM	IC50
TKC046601	P51681	C-C chemokine receptor type 5	None	32000	nM	IC50
TKC054684	P51681	C-C chemokine receptor type 5	None	5100	nM	Ki
TKC054723	P51681	C-C chemokine receptor type 5	None	30000	nM	Ki
TKC137374	P51681	C-C chemokine receptor type 5	None	9000	nM	IC50
TKC027726	P52732	Kinesin-like protein KIF11	None	3500	nM	IC50
TKC035272	P52732	Kinesin-like protein KIF11	None	10800	nM	IC50
TKC035272	P52732	Kinesin-like protein KIF11	None	25000	nM	IC50
TKC108557	P52732	Kinesin-like protein KIF11	None	0.3	nM	IC50
TKC001786	P53350	Serine/threonine-protein kinase PLK1	None	23778	nM	Potency
TKC005454	P53350	Serine/threonine-protein kinase PLK1	None	26680	nM	Potency
TKC011384	P53350	Serine/threonine-protein kinase PLK1	None	18888	nM	Potency
TKC014568	P53350	Serine/threonine-protein kinase PLK1	None	26680	nM	Potency
TKC016277	P53350	Serine/threonine-protein kinase PLK1	None	29935	nM	Potency
TKC018288	P53350	Serine/threonine-protein kinase PLK1	None	13371	nM	Potency
TKC020967	P53350	Serine/threonine-protein kinase PLK1	None	2180	nM	IC50
TKC020987	P53350	Serine/threonine-protein kinase PLK1	None	23778	nM	Potency
TKC024886	P53350	Serine/threonine-protein kinase PLK1	None	21700	nM	IC50
TKC025690	P53350	Serine/threonine-protein kinase PLK1	None	>100000	nM	IC50
TKC037521	P53350	Serine/threonine-protein kinase PLK1	None	18888	nM	Potency
TKC040032	P53350	Serine/threonine-protein kinase PLK1	None	29935	nM	Potency
TKC055219	P53350	Serine/threonine-protein kinase PLK1	None	13371	nM	Potency
TKC055869	P53350	Serine/threonine-protein kinase PLK1	None	33588	nM	Potency
TKC066096	P53350	Serine/threonine-protein kinase PLK1	None	2119	nM	Potency
TKC066411	P53350	Serine/threonine-protein kinase PLK1	None	2994	nM	Potency
TKC077689	P53350	Serine/threonine-protein kinase PLK1	None	26680	nM	Potency
TKC082378	P53350	Serine/threonine-protein kinase PLK1	None	15003	nM	Potency
TKC087988	P53350	Serine/threonine-protein kinase PLK1	None	26680	nM	Potency
TKC088678	P53350	Serine/threonine-protein kinase PLK1	None	37686	nM	Potency
TKC091895	P53350	Serine/threonine-protein kinase PLK1	None	26680	nM	Potency
TKC098704	P53350	Serine/threonine-protein kinase PLK1	None	26680	nM	Potency
TKC101726	P53350	Serine/threonine-protein kinase PLK1	None	26680	nM	Potency
TKC104088	P53350	Serine/threonine-protein kinase PLK1	None	33588	nM	Potency
TKC107557	P53350	Serine/threonine-protein kinase PLK1	None	26680	nM	Potency
TKC112826	P53350	Serine/threonine-protein kinase PLK1	None	33588	nM	Potency
TKC115259	P53350	Serine/threonine-protein kinase PLK1	None	>100000	nM	IC50
TKC115261	P53350	Serine/threonine-protein kinase PLK1	None	>100000	nM	IC50
TKC115272	P53350	Serine/threonine-protein kinase PLK1	None	>100000	nM	IC50
TKC115273	P53350	Serine/threonine-protein kinase PLK1	None	100000	nM	IC50
TKC118419	P53350	Serine/threonine-protein kinase PLK1	None	6	nM	IC50
TKC118419	P53350	Serine/threonine-protein kinase PLK1	None	1500	nM	Ki
TKC118419	P53350	Serine/threonine-protein kinase PLK1	None	24	nM	IC50
TKC141147	P53350	Serine/threonine-protein kinase PLK1	None	13371	nM	Potency
TKC150277	P53350	Serine/threonine-protein kinase PLK1	None	23778	nM	Potency
TKC151609	P53350	Serine/threonine-protein kinase PLK1	None	23778	nM	Potency
TKC151885	P53350	Serine/threonine-protein kinase PLK1	None	6702	nM	Potency
TKC151902	P53350	Serine/threonine-protein kinase PLK1	None	26680	nM	Potency
TKC151910	P53350	Serine/threonine-protein kinase PLK1	None	18888	nM	Potency
TKC152148	P53350	Serine/threonine-protein kinase PLK1	None	>100000	nM	IC50
TKC152157	P53350	Serine/threonine-protein kinase PLK1	None	>100000	nM	IC50
TKC159332	P53350	Serine/threonine-protein kinase PLK1	None	21192	nM	Potency
TKC171689	P53350	Serine/threonine-protein kinase PLK1	None	23778	nM	Potency
TKC174547	P53350	Serine/threonine-protein kinase PLK1	None	>100000	nM	IC50
TKC206362	P53350	Serine/threonine-protein kinase PLK1	None	13371	nM	Potency
TKC206589	P53350	Serine/threonine-protein kinase PLK1	None	29935	nM	Potency
TKC206760	P53350	Serine/threonine-protein kinase PLK1	None	21192	nM	Potency
TKC007963	P55072	Transitional endoplasmic reticulum ATPase	None	>100000	nM	IC50
TKC035272	P55072	Transitional endoplasmic reticulum ATPase	None	5386	nM	IC50
TKC038988	P55072	Transitional endoplasmic reticulum ATPase	None	>100000	nM	IC50
TKC113058	P55072	Transitional endoplasmic reticulum ATPase	None	22000	nM	IC50
TKC016794	P55085	Proteinase-activated receptor 2	None	14	nM	IC50
TKC020117	P56524	Histone deacetylase 4	None	>20000	nM	Ki
TKC020117	P56524	Histone deacetylase 4	None	3.32	nM	Ki
TKC021620	P60568	Interleukin-2	None	3	nM	Kd
TKC116180	P60568	Interleukin-2	None	0	nM	Kd
TKC205544	P61073	C-X-C chemokine receptor type 4	None	21	%	Inhibition
TKC011412	P78417	Glutathione S-transferase omega-1	None	62000	nM	IC50
TKC095638	P78417	Glutathione S-transferase omega-1	None	4000	nM	IC50
TKC095669	P78417	Glutathione S-transferase omega-1	None	2000	nM	IC50
TKC206672	P78417	Glutathione S-transferase omega-1	None	1020000	nM	IC50
TKC118419	P78527	DNA-dependent protein kinase catalytic subunit	None	120	nM	Ki
TKC118419	P78527	DNA-dependent protein kinase catalytic subunit	None	120	nM	Ki
TKC020117	Q00987	E3 ubiquitin-protein ligase Mdm2	None	3580	nM	IC50
TKC035272	Q00987	E3 ubiquitin-protein ligase Mdm2	None	>25000	nM	Ki
TKC038273	Q00987	E3 ubiquitin-protein ligase Mdm2	None	7680	nM	EC50
TKC076529	Q00987	E3 ubiquitin-protein ligase Mdm2	None	11620	nM	EC50
TKC134702	Q00987	E3 ubiquitin-protein ligase Mdm2	None	420	nM	EC50
TKC134744	Q00987	E3 ubiquitin-protein ligase Mdm2	None	590	nM	EC50
TKC024886	Q02750	Dual specificity mitogen-activated protein kinase kinase 1	None	>100000	nM	IC50
TKC025690	Q02750	Dual specificity mitogen-activated protein kinase kinase 1	None	>100000	nM	IC50
TKC115259	Q02750	Dual specificity mitogen-activated protein kinase kinase 1	None	>100000	nM	IC50
TKC115261	Q02750	Dual specificity mitogen-activated protein kinase kinase 1	None	>100000	nM	IC50
TKC115272	Q02750	Dual specificity mitogen-activated protein kinase kinase 1	None	>100000	nM	IC50
TKC115273	Q02750	Dual specificity mitogen-activated protein kinase kinase 1	None	>100000	nM	IC50
TKC118419	Q02750	Dual specificity mitogen-activated protein kinase kinase 1	None	63	%	Activity
TKC152148	Q02750	Dual specificity mitogen-activated protein kinase kinase 1	None	48900	nM	IC50
TKC152157	Q02750	Dual specificity mitogen-activated protein kinase kinase 1	None	>100000	nM	IC50
TKC174547	Q02750	Dual specificity mitogen-activated protein kinase kinase 1	None	>100000	nM	IC50
TKC011761	Q05397	Focal adhesion kinase 1	None	67	%	Inhibition
TKC024886	Q05397	Focal adhesion kinase 1	None	4560	nM	IC50
TKC025690	Q05397	Focal adhesion kinase 1	None	7780	nM	IC50
TKC115259	Q05397	Focal adhesion kinase 1	None	16900	nM	IC50
TKC115261	Q05397	Focal adhesion kinase 1	None	9920	nM	IC50
TKC115272	Q05397	Focal adhesion kinase 1	None	>100000	nM	IC50
TKC115273	Q05397	Focal adhesion kinase 1	None	10700	nM	IC50
TKC152148	Q05397	Focal adhesion kinase 1	None	13200	nM	IC50
TKC152157	Q05397	Focal adhesion kinase 1	None	9630	nM	IC50
TKC174547	Q05397	Focal adhesion kinase 1	None	>100000	nM	IC50
TKC110249	Q05513	Protein kinase C zeta type	None	530	nM	IC50
TKC113327	Q05513	Protein kinase C zeta type	None	110	nM	IC50
TKC113657	Q05513	Protein kinase C zeta type	None	1590	nM	IC50
TKC118419	Q05513	Protein kinase C zeta type	None	84	%	Activity
TKC152603	Q05513	Protein kinase C zeta type	None	1210	nM	IC50
TKC005454	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	22500	nM	IC50
TKC013306	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	<50	%	Inhibition
TKC014568	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	2570	nM	IC50
TKC026891	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	<50	%	Inhibition
TKC031060	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	29000	nM	IC50
TKC063400	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	61600	nM	IC50
TKC066096	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	3300	nM	IC50
TKC077689	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	11620	nM	IC50
TKC077689	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	>120000	nM	IC50
TKC088678	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	9600	nM	IC50
TKC112796	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	<50	%	Inhibition
TKC116328	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	<50	%	Inhibition
TKC116342	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	<50	%	Inhibition
TKC131482	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	<50	%	Inhibition
TKC146774	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	>40000	nM	IC50
TKC150004	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	<50	%	Inhibition
TKC206840	Q06124	Tyrosine-protein phosphatase non-receptor type 11	None	<50	%	Inhibition
TKC206758	Q06278	Aldehyde oxidase	None	>100000	nM	IC50
TKC014568	Q06609	DNA repair protein RAD51 homolog 1	None	85000	nM	IC50
TKC105224	Q06609	DNA repair protein RAD51 homolog 1	None	85000	nM	IC50
TKC008684	Q07817	Bcl-2-like protein 1	None	380000	nM	IC50
TKC035272	Q07817	Bcl-2-like protein 1	None	310	nM	Ki
TKC035272	Q07817	Bcl-2-like protein 1	None	2720	nM	IC50
TKC035272	Q07817	Bcl-2-like protein 1	None	480	nM	IC50
TKC035272	Q07817	Bcl-2-like protein 1	None	1000	nM	Ki
TKC035272	Q07817	Bcl-2-like protein 1	None	620	nM	Ki
TKC035272	Q07817	Bcl-2-like protein 1	None	480	nM	Ki
TKC035272	Q07817	Bcl-2-like protein 1	None	640	nM	Ki
TKC035272	Q07817	Bcl-2-like protein 1	None	1710	nM	Kd
TKC035272	Q07817	Bcl-2-like protein 1	None	310	nM	Ki
TKC035272	Q07817	Bcl-2-like protein 1	None	1400	nM	Ki
TKC035272	Q07817	Bcl-2-like protein 1	None	480	nM	Ki
TKC035272	Q07817	Bcl-2-like protein 1	None	500	nM	IC50
TKC035272	Q07817	Bcl-2-like protein 1	None	480	nM	Ki
TKC039229	Q07817	Bcl-2-like protein 1	None	40000	nM	Ki
TKC039229	Q07817	Bcl-2-like protein 1	None	10800	nM	Ki
TKC039229	Q07817	Bcl-2-like protein 1	None	2600	nM	Ki
TKC050432	Q07817	Bcl-2-like protein 1	None	>100000	nM	Ki
TKC078259	Q07817	Bcl-2-like protein 1	None	7600	nM	Ki
TKC078261	Q07817	Bcl-2-like protein 1	None	5300	nM	Ki
TKC081833	Q07817	Bcl-2-like protein 1	None	>100000	nM	Ki
TKC083390	Q07817	Bcl-2-like protein 1	None	>100000	nM	Ki
TKC105178	Q07817	Bcl-2-like protein 1	None	100000	nM	Ki
TKC105179	Q07817	Bcl-2-like protein 1	None	2300	nM	Ki
TKC129211	Q07817	Bcl-2-like protein 1	None	400000	nM	IC50
TKC134945	Q07817	Bcl-2-like protein 1	None	8300	nM	Ki
TKC134945	Q07817	Bcl-2-like protein 1	None	2600	nM	Ki
TKC143158	Q07817	Bcl-2-like protein 1	None	>100000	nM	Ki
TKC143159	Q07817	Bcl-2-like protein 1	None	>100000	nM	Ki
TKC143166	Q07817	Bcl-2-like protein 1	None	17800	nM	Ki
TKC143167	Q07817	Bcl-2-like protein 1	None	>100000	nM	Ki
TKC143168	Q07817	Bcl-2-like protein 1	None	7200	nM	Ki
TKC151761	Q07817	Bcl-2-like protein 1	None	>10000	nM	GI50
TKC156346	Q07817	Bcl-2-like protein 1	None	14100	nM	Ki
TKC156347	Q07817	Bcl-2-like protein 1	None	>100000	nM	Ki
TKC156348	Q07817	Bcl-2-like protein 1	None	>100000	nM	Ki
TKC200866	Q07817	Bcl-2-like protein 1	None	>10000	nM	GI50
TKC028446	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	11400	nM	IC50
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	1356	nM	IC50
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	162	nM	Ki
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	180	nM	Ki
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	280	nM	Ki
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	310	nM	Ki
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	640	nM	Ki
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	180	nM	Ki
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	180	nM	Ki
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	200	nM	Ki
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	6543	nM	Ki
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	2324	nM	Kd
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	190	nM	Ki
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	2650	nM	Kd
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	190	nM	Ki
TKC035272	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	180	nM	Ki
TKC039229	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	12900	nM	Ki
TKC105178	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	14400	nM	Ki
TKC105179	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	4200	nM	Ki
TKC134945	Q07820	Induced myeloid leukemia cell differentiation protein Mcl-1	None	8600	nM	Ki
TKC021262	Q07869	Peroxisome proliferator-activated receptor alpha	None	19500	nM	EC50
TKC021666	Q07869	Peroxisome proliferator-activated receptor alpha	None	28	%	Activity
TKC021674	Q07869	Peroxisome proliferator-activated receptor alpha	None	25	%	Activity
TKC035272	Q07869	Peroxisome proliferator-activated receptor alpha	None	15849	nM	Potency
TKC056482	Q07869	Peroxisome proliferator-activated receptor alpha	None	259	%	Activity
TKC057132	Q07869	Peroxisome proliferator-activated receptor alpha	None	12589	nM	Potency
TKC088526	Q07869	Peroxisome proliferator-activated receptor alpha	None	12	%	Activity
TKC100644	Q07869	Peroxisome proliferator-activated receptor alpha	None	8913	nM	Potency
TKC108536	Q07869	Peroxisome proliferator-activated receptor alpha	None	50119	nM	Potency
TKC110634	Q07869	Peroxisome proliferator-activated receptor alpha	None	309	%	Activity
TKC110635	Q07869	Peroxisome proliferator-activated receptor alpha	None	289	%	Activity
TKC170559	Q07869	Peroxisome proliferator-activated receptor alpha	None	1000	nM	EC50
TKC171329	Q07869	Peroxisome proliferator-activated receptor alpha	None	184	nM	EC50
TKC206812	Q07869	Peroxisome proliferator-activated receptor alpha	None	>20000	nM	IC50
TKC001253	Q09472	Histone acetyltransferase p300	None	4850	nM	IC50
TKC078955	Q09472	Histone acetyltransferase p300	None	5000	nM	IC50
TKC116815	Q09472	Histone acetyltransferase p300	None	3300	nM	IC50
TKC151761	Q12866	Tyrosine-protein kinase Mer	None	4900	nM	IC50
TKC200866	Q12866	Tyrosine-protein kinase Mer	None	4900	nM	IC50
TKC016189	Q13315	Serine-protein kinase ATM	None	19953	nM	Potency
TKC016371	Q13315	Serine-protein kinase ATM	None	25119	nM	Potency
TKC029307	Q13315	Serine-protein kinase ATM	None	39811	nM	Potency
TKC039202	Q13315	Serine-protein kinase ATM	None	3548	nM	Potency
TKC063474	Q13315	Serine-protein kinase ATM	None	35481	nM	Potency
TKC066411	Q13315	Serine-protein kinase ATM	None	31623	nM	Potency
TKC103159	Q13315	Serine-protein kinase ATM	None	19953	nM	Potency
TKC150598	Q13315	Serine-protein kinase ATM	None	39811	nM	Potency
TKC151609	Q13315	Serine-protein kinase ATM	None	39811	nM	Potency
TKC174441	Q13315	Serine-protein kinase ATM	None	412	nM	Potency
TKC109622	Q13822	Ectonucleotide pyrophosphatase/phosphodiesterase family member 2	None	10300	nM	IC50
TKC118419	Q15118	Pyruvate dehydrogenase	None	88	%	Inhibition
TKC118419	Q15139	Serine/threonine-protein kinase D1	None	92	%	Activity
TKC005475	Q15910	Histone-lysine N-methyltransferase EZH2	None	9600	nM	IC50
TKC014568	Q15910	Histone-lysine N-methyltransferase EZH2	None	8900	nM	IC50
TKC087988	Q16539	Mitogen-activated protein kinase 14	None	2529	nM	IC50
TKC118419	Q16539	Mitogen-activated protein kinase 14	None	86	%	Inhibition
TKC005454	Q16665	Hypoxia-inducible factor 1-alpha	None	1360	nM	IC50
TKC005475	Q16665	Hypoxia-inducible factor 1-alpha	None	7340	nM	IC50
TKC010010	Q16665	Hypoxia-inducible factor 1-alpha	None	>20000	nM	IC50
TKC011921	Q16665	Hypoxia-inducible factor 1-alpha	None	1995	nM	Potency
TKC012261	Q16665	Hypoxia-inducible factor 1-alpha	None	280	nM	IC50
TKC012262	Q16665	Hypoxia-inducible factor 1-alpha	None	3180	nM	IC50
TKC012971	Q16665	Hypoxia-inducible factor 1-alpha	None	25119	nM	Potency
TKC014568	Q16665	Hypoxia-inducible factor 1-alpha	None	8510	nM	IC50
TKC017189	Q16665	Hypoxia-inducible factor 1-alpha	None	10600	nM	IC50
TKC017192	Q16665	Hypoxia-inducible factor 1-alpha	None	1700	nM	IC50
TKC017193	Q16665	Hypoxia-inducible factor 1-alpha	None	2300	nM	IC50
TKC020116	Q16665	Hypoxia-inducible factor 1-alpha	None	501	nM	Potency
TKC022945	Q16665	Hypoxia-inducible factor 1-alpha	None	2512	nM	Potency
TKC023570	Q16665	Hypoxia-inducible factor 1-alpha	None	15800	nM	IC50
TKC030239	Q16665	Hypoxia-inducible factor 1-alpha	None	200	nM	Potency
TKC035272	Q16665	Hypoxia-inducible factor 1-alpha	None	10000	nM	Potency
TKC037547	Q16665	Hypoxia-inducible factor 1-alpha	None	10	%	Activity
TKC038977	Q16665	Hypoxia-inducible factor 1-alpha	None	820	nM	IC50
TKC045710	Q16665	Hypoxia-inducible factor 1-alpha	None	500	nM	IC50
TKC045931	Q16665	Hypoxia-inducible factor 1-alpha	None	2900	nM	IC50
TKC045946	Q16665	Hypoxia-inducible factor 1-alpha	None	2900	nM	IC50
TKC047694	Q16665	Hypoxia-inducible factor 1-alpha	None	63	nM	IC50
TKC047695	Q16665	Hypoxia-inducible factor 1-alpha	None	68	nM	IC50
TKC056482	Q16665	Hypoxia-inducible factor 1-alpha	None	>100000	nM	IC50
TKC056482	Q16665	Hypoxia-inducible factor 1-alpha	None	>100000	nM	IC50
TKC062172	Q16665	Hypoxia-inducible factor 1-alpha	None	15000	nM	IC50
TKC062175	Q16665	Hypoxia-inducible factor 1-alpha	None	20000	nM	IC50
TKC062182	Q16665	Hypoxia-inducible factor 1-alpha	None	20000	nM	IC50
TKC062192	Q16665	Hypoxia-inducible factor 1-alpha	None	20000	nM	IC50
TKC062193	Q16665	Hypoxia-inducible factor 1-alpha	None	>30000	nM	IC50
TKC065782	Q16665	Hypoxia-inducible factor 1-alpha	None	>30000	nM	IC50
TKC081893	Q16665	Hypoxia-inducible factor 1-alpha	None	400	nM	IC50
TKC092297	Q16665	Hypoxia-inducible factor 1-alpha	None	39811	nM	Potency
TKC094057	Q16665	Hypoxia-inducible factor 1-alpha	None	>30000	nM	IC50
TKC094058	Q16665	Hypoxia-inducible factor 1-alpha	None	>20000	nM	IC50
TKC095493	Q16665	Hypoxia-inducible factor 1-alpha	None	3162	nM	Potency
TKC096011	Q16665	Hypoxia-inducible factor 1-alpha	None	1	nM	Potency
TKC096012	Q16665	Hypoxia-inducible factor 1-alpha	None	251	nM	Potency
TKC100416	Q16665	Hypoxia-inducible factor 1-alpha	None	25119	nM	Potency
TKC100643	Q16665	Hypoxia-inducible factor 1-alpha	None	12589	nM	Potency
TKC100990	Q16665	Hypoxia-inducible factor 1-alpha	None	159	nM	Potency
TKC101618	Q16665	Hypoxia-inducible factor 1-alpha	None	15849	nM	Potency
TKC102145	Q16665	Hypoxia-inducible factor 1-alpha	None	1259	nM	Potency
TKC102589	Q16665	Hypoxia-inducible factor 1-alpha	None	8000	nM	EC50
TKC103149	Q16665	Hypoxia-inducible factor 1-alpha	None	31623	nM	Potency
TKC103159	Q16665	Hypoxia-inducible factor 1-alpha	None	270	nM	IC50
TKC103433	Q16665	Hypoxia-inducible factor 1-alpha	None	>30000	nM	IC50
TKC103494	Q16665	Hypoxia-inducible factor 1-alpha	None	79	nM	Potency
TKC103496	Q16665	Hypoxia-inducible factor 1-alpha	None	20	nM	Potency
TKC104070	Q16665	Hypoxia-inducible factor 1-alpha	None	40	nM	Potency
TKC104071	Q16665	Hypoxia-inducible factor 1-alpha	None	100	nM	Potency
TKC104114	Q16665	Hypoxia-inducible factor 1-alpha	None	126	nM	Potency
TKC104664	Q16665	Hypoxia-inducible factor 1-alpha	None	794	nM	Potency
TKC105037	Q16665	Hypoxia-inducible factor 1-alpha	None	794	nM	Potency
TKC105510	Q16665	Hypoxia-inducible factor 1-alpha	None	6000	nM	EC50
TKC105710	Q16665	Hypoxia-inducible factor 1-alpha	None	12589	nM	Potency
TKC106426	Q16665	Hypoxia-inducible factor 1-alpha	None	1000	nM	Potency
TKC106576	Q16665	Hypoxia-inducible factor 1-alpha	None	13000	nM	EC50
TKC107086	Q16665	Hypoxia-inducible factor 1-alpha	None	19953	nM	Potency
TKC109561	Q16665	Hypoxia-inducible factor 1-alpha	None	251	nM	Potency
TKC110002	Q16665	Hypoxia-inducible factor 1-alpha	None	63	nM	Potency
TKC110007	Q16665	Hypoxia-inducible factor 1-alpha	None	7943	nM	Potency
TKC111738	Q16665	Hypoxia-inducible factor 1-alpha	None	16	nM	Potency
TKC112789	Q16665	Hypoxia-inducible factor 1-alpha	None	1000	nM	Potency
TKC112906	Q16665	Hypoxia-inducible factor 1-alpha	None	5012	nM	Potency
TKC114819	Q16665	Hypoxia-inducible factor 1-alpha	None	12589	nM	Potency
TKC117993	Q16665	Hypoxia-inducible factor 1-alpha	None	2000	nM	EC50
TKC117997	Q16665	Hypoxia-inducible factor 1-alpha	None	40	nM	EC50
TKC118004	Q16665	Hypoxia-inducible factor 1-alpha	None	2512	nM	Potency
TKC118012	Q16665	Hypoxia-inducible factor 1-alpha	None	600	nM	EC50
TKC118131	Q16665	Hypoxia-inducible factor 1-alpha	None	126	nM	Potency
TKC134897	Q16665	Hypoxia-inducible factor 1-alpha	None	3400	nM	IC50
TKC137120	Q16665	Hypoxia-inducible factor 1-alpha	None	200	nM	IC50
TKC137126	Q16665	Hypoxia-inducible factor 1-alpha	None	2400	nM	IC50
TKC137243	Q16665	Hypoxia-inducible factor 1-alpha	None	200	nM	IC50
TKC144475	Q16665	Hypoxia-inducible factor 1-alpha	None	25000	nM	IC50
TKC151571	Q16665	Hypoxia-inducible factor 1-alpha	None	7943	nM	Potency
TKC205806	Q16665	Hypoxia-inducible factor 1-alpha	None	5012	nM	Potency
TKC206042	Q16665	Hypoxia-inducible factor 1-alpha	None	6310	nM	Potency
TKC206395	Q16665	Hypoxia-inducible factor 1-alpha	None	12589	nM	Potency
TKC206453	Q16665	Hypoxia-inducible factor 1-alpha	None	25119	nM	Potency
TKC206617	Q16665	Hypoxia-inducible factor 1-alpha	None	12700	nM	IC50
TKC206688	Q16665	Hypoxia-inducible factor 1-alpha	None	63	nM	Potency
TKC206726	Q16665	Hypoxia-inducible factor 1-alpha	None	79	nM	Potency
TKC206760	Q16665	Hypoxia-inducible factor 1-alpha	None	50119	nM	Potency
TKC206780	Q16665	Hypoxia-inducible factor 1-alpha	None	3981	nM	Potency
TKC206812	Q16665	Hypoxia-inducible factor 1-alpha	None	79433	nM	Potency
TKC206816	Q16665	Hypoxia-inducible factor 1-alpha	None	12589	nM	Potency
TKC206872	Q16665	Hypoxia-inducible factor 1-alpha	None	1000	nM	Potency
TKC206889	Q16665	Hypoxia-inducible factor 1-alpha	None	501	nM	Potency
TKC206890	Q16665	Hypoxia-inducible factor 1-alpha	None	20	nM	EC50
TKC206901	Q16665	Hypoxia-inducible factor 1-alpha	None	159	nM	Potency
TKC076129	Q16790	Carbonic anhydrase 9	None	980	nM	Ki
TKC105649	Q16881	Thioredoxin reductase 1, cytoplasmic	None	280	nM	Ki
TKC019571	Q7Z2W7	Transient receptor potential cation channel subfamily M member 8	None	100	uM	Activity
TKC074866	Q7Z2W7	Transient receptor potential cation channel subfamily M member 8	None	5900000	nM	EC50
TKC085168	Q7Z2W7	Transient receptor potential cation channel subfamily M member 8	None	10100	nM	EC50
TKC086929	Q7Z2W7	Transient receptor potential cation channel subfamily M member 8	None	3000	nM	EC50
TKC023246	Q92731	Estrogen receptor beta	None	>10000	nM	IC50
TKC028029	Q92731	Estrogen receptor beta	None	<1	%	Activity
TKC028037	Q92731	Estrogen receptor beta	None	10	%	Activity
TKC035272	Q92731	Estrogen receptor beta	None	>50000	nM	IC50
TKC100932	Q92731	Estrogen receptor beta	None	25300	nM	EC50
TKC101365	Q92731	Estrogen receptor beta	None	17690	nM	EC50
TKC102448	Q92731	Estrogen receptor beta	None	4680	nM	EC50
TKC106878	Q92731	Estrogen receptor beta	None	>10000	nM	IC50
TKC110673	Q92731	Estrogen receptor beta	None	2.78E+11	M-1	Ka
TKC111721	Q92731	Estrogen receptor beta	None	1520000000	M-1	Ka
TKC111727	Q92731	Estrogen receptor beta	None	614000000	M-1	Ka
TKC111727	Q92731	Estrogen receptor beta	None	0	nM	EC50
TKC111738	Q92731	Estrogen receptor beta	None	2	nM	EC50
TKC111738	Q92731	Estrogen receptor beta	None	4	%	RSA
TKC111738	Q92731	Estrogen receptor beta	None	26	nM	IC50
TKC111738	Q92731	Estrogen receptor beta	None	540	nM	IC50
TKC111738	Q92731	Estrogen receptor beta	None	8	nM	EC50
TKC112923	Q92731	Estrogen receptor beta	None	6	nM	EC50
TKC206608	Q92731	Estrogen receptor beta	None	4280	nM	EC50
TKC206725	Q92731	Estrogen receptor beta	None	24	nM	Ki
TKC206726	Q92731	Estrogen receptor beta	None	11	nM	EC50
TKC206759	Q92731	Estrogen receptor beta	None	>10000	nM	IC50
TKC206759	Q92731	Estrogen receptor beta	None	>10000	nM	IC50
TKC206764	Q92731	Estrogen receptor beta	None	1	%	RBA
TKC206765	Q92731	Estrogen receptor beta	None	18000000	M-1	Ka
TKC206769	Q92731	Estrogen receptor beta	None	27000000	M-1	Ka
TKC206812	Q92731	Estrogen receptor beta	None	>5000	nM	IC50
TKC206816	Q92731	Estrogen receptor beta	None	1000000	nM	IC50
TKC020117	Q92769	Histone deacetylase 2	None	15	nM	Ki
TKC035272	Q92843	Bcl-2-like protein 2	None	17700	nM	Ki
TKC046098	Q93009	Ubiquitin carboxyl-terminal hydrolase 7	None	2700	nM	IC50
TKC046099	Q93009	Ubiquitin carboxyl-terminal hydrolase 7	None	3500	nM	IC50
TKC056482	Q93009	Ubiquitin carboxyl-terminal hydrolase 7	None	7000	nM	IC50
TKC048132	Q96EB6	NAD-dependent protein deacetylase sirtuin-1	None	28	%	Activity
TKC048343	Q96EB6	NAD-dependent protein deacetylase sirtuin-1	None	88	%	Activity
TKC048346	Q96EB6	NAD-dependent protein deacetylase sirtuin-1	None	8	%	Activity
TKC024886	Q96GD4	Aurora kinase B	None	3890	nM	IC50
TKC025690	Q96GD4	Aurora kinase B	None	>100000	nM	IC50
TKC115259	Q96GD4	Aurora kinase B	None	38100	nM	IC50
TKC115261	Q96GD4	Aurora kinase B	None	>100000	nM	IC50
TKC115272	Q96GD4	Aurora kinase B	None	>100000	nM	IC50
TKC115273	Q96GD4	Aurora kinase B	None	>100000	nM	IC50
TKC118419	Q96GD4	Aurora kinase B	None	83	%	Activity
TKC152148	Q96GD4	Aurora kinase B	None	25100	nM	IC50
TKC152157	Q96GD4	Aurora kinase B	None	>100000	nM	IC50
TKC174547	Q96GD4	Aurora kinase B	None	>100000	nM	IC50
TKC005139	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	89125	nM	Potency
TKC005313	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	25	nM	Potency
TKC005454	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	7080	nM	Potency
TKC008359	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	19953	nM	Potency
TKC008623	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	31623	nM	Potency
TKC011412	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	3548	nM	Potency
TKC011921	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	6310	nM	Potency
TKC013263	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	25119	nM	Potency
TKC013738	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	14125	nM	Potency
TKC013755	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	22387	nM	Potency
TKC013760	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	25119	nM	Potency
TKC014568	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	3162	nM	Potency
TKC017379	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	14125	nM	Potency
TKC020117	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	11220	nM	Potency
TKC027192	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	14125	nM	Potency
TKC032619	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	7943	nM	Potency
TKC034640	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	44668	nM	Potency
TKC034641	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	44668	nM	Potency
TKC034760	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	22387	nM	Potency
TKC035272	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	35481	nM	Potency
TKC035984	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	3981	nM	Potency
TKC038273	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	3162	nM	Potency
TKC038756	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	12589	nM	Potency
TKC039202	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	79433	nM	Potency
TKC040032	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	22387	nM	Potency
TKC053751	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	24	nM	Potency
TKC055219	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	79433	nM	Potency
TKC083025	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	19953	nM	Potency
TKC083534	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	25119	nM	Potency
TKC084630	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	50119	nM	Potency
TKC087533	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	31623	nM	Potency
TKC087988	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	17783	nM	Potency
TKC092297	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	12589	nM	Potency
TKC092348	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	19953	nM	Potency
TKC093115	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	1000	nM	Potency
TKC095442	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	7943	nM	Potency
TKC096012	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	23778	nM	Potency
TKC099703	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	3548	nM	Potency
TKC100416	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	37686	nM	Potency
TKC103150	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	10000	nM	Potency
TKC103542	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	2818	nM	Potency
TKC105022	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	15849	nM	Potency
TKC105356	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	355	nM	Potency
TKC106013	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	100000	nM	Potency
TKC106026	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	631	nM	Potency
TKC106301	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	22	nM	Potency
TKC106364	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	7080	nM	Potency
TKC106426	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	8913	nM	Potency
TKC109998	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	891	nM	Potency
TKC110002	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	22	nM	Potency
TKC110162	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	3548	nM	Potency
TKC112576	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	10000	nM	Potency
TKC112754	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	22	nM	Potency
TKC112906	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	8913	nM	Potency
TKC114511	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	22	nM	Potency
TKC115268	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	3162	nM	Potency
TKC115284	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	22387	nM	Potency
TKC116870	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	316	nM	Potency
TKC117216	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	3162	nM	Potency
TKC118131	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	10000	nM	Potency
TKC118419	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	6310	nM	Potency
TKC122892	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	28184	nM	Potency
TKC130092	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	17783	nM	Potency
TKC134702	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	11220	nM	Potency
TKC140412	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	89125	nM	Potency
TKC146423	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	17783	nM	Potency
TKC151237	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	6310	nM	Potency
TKC151303	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	794	nM	Potency
TKC151609	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	11220	nM	Potency
TKC151885	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	891	nM	Potency
TKC151902	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	14125	nM	Potency
TKC197340	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	28184	nM	Potency
TKC205544	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	21192	nM	Potency
TKC205806	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	7943	nM	Potency
TKC206113	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	8913	nM	Potency
TKC206544	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	17783	nM	Potency
TKC206622	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	7943	nM	Potency
TKC206660	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	4467	nM	Potency
TKC206688	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	447	nM	Potency
TKC206689	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	10000	nM	Potency
TKC206690	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	11220	nM	Potency
TKC206758	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	25	nM	Potency
TKC206777	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	22	nM	Potency
TKC206779	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	38	nM	Potency
TKC206781	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	89125	nM	Potency
TKC206784	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	56234	nM	Potency
TKC206816	Q96KQ7	Histone-lysine N-methyltransferase EHMT2	None	1259	nM	Potency
TKC149924	Q96P20	NACHT, LRR and PYD domains-containing protein 3	None	26	%	Inhibition
TKC026309	Q99814	Endothelial PAS domain-containing protein 1	None	3300	nM	EC50
TKC035150	Q99814	Endothelial PAS domain-containing protein 1	None	10800	nM	IC50
TKC045708	Q99814	Endothelial PAS domain-containing protein 1	None	4200	nM	EC50
TKC045868	Q99814	Endothelial PAS domain-containing protein 1	None	1200	nM	EC50
TKC046523	Q99814	Endothelial PAS domain-containing protein 1	None	>100000	nM	EC50
TKC100652	Q99814	Endothelial PAS domain-containing protein 1	None	3400	nM	EC50
TKC101122	Q99814	Endothelial PAS domain-containing protein 1	None	6200	nM	EC50
TKC103124	Q99814	Endothelial PAS domain-containing protein 1	None	148900	nM	EC50
TKC104992	Q99814	Endothelial PAS domain-containing protein 1	None	107500	nM	EC50
TKC105151	Q99814	Endothelial PAS domain-containing protein 1	None	183300	nM	EC50
TKC118419	Q99814	Endothelial PAS domain-containing protein 1	None	3930	nM	IC50
TKC143885	Q99814	Endothelial PAS domain-containing protein 1	None	14400	nM	IC50
TKC165028	Q99814	Endothelial PAS domain-containing protein 1	None	11800	nM	EC50
TKC115268	Q99835	Smoothened homolog	None	36	%	Activity
TKC115284	Q99835	Smoothened homolog	None	28	%	Activity
TKC206385	Q99835	Smoothened homolog	None	70	%	Activity
TKC118419	Q9BUB5	MAP kinase-interacting serine/threonine-protein kinase 1	None	81	%	Activity
TKC020117	Q9BY41	Histone deacetylase 8	None	178	nM	Ki
TKC020117	Q9BY41	Histone deacetylase 8	None	105	nM	Ki
TKC056482	Q9GZT9	Egl nine homolog 1	None	>50000	nM	EC50
TKC077689	Q9GZT9	Egl nine homolog 1	None	>50000	nM	EC50
TKC088678	Q9GZT9	Egl nine homolog 1	None	>50000	nM	EC50
TKC123088	Q9GZT9	Egl nine homolog 1	None	>50000	nM	EC50
TKC118419	Q9HBH9	MAP kinase-interacting serine/threonine-protein kinase 2	None	97	%	Activity
TKC066096	Q9NR96	Toll-like receptor 9	None	3015	nM	IC50
TKC076529	Q9NR96	Toll-like receptor 9	None	>49739	nM	IC50
TKC076529	Q9NR96	Toll-like receptor 9	None	>49739	nM	IC50
TKC082378	Q9NR96	Toll-like receptor 9	None	7929	nM	IC50
TKC082378	Q9NR96	Toll-like receptor 9	None	7929	nM	IC50
TKC020967	Q9NYY3	Serine/threonine-protein kinase PLK2	None	14720	nM	IC50
TKC118419	Q9NYY3	Serine/threonine-protein kinase PLK2	None	2800	nM	Ki
TKC118419	Q9P1W9	Serine/threonine-protein kinase pim-2	None	83	%	Activity
TKC014593	Q9UBN7	Histone deacetylase 6	None	80000	nM	IC50
TKC020117	Q9UBN7	Histone deacetylase 6	None	>2500	nM	Ki
TKC076129	Q9ULX7	Carbonic anhydrase 14	None	1470	nM	Ki
TKC011761	Q9UM73	ALK tyrosine kinase receptor	None	18	%	Inhibition
TKC024886	Q9UM73	ALK tyrosine kinase receptor	None	2190	nM	IC50
TKC025690	Q9UM73	ALK tyrosine kinase receptor	None	3380	nM	IC50
TKC115259	Q9UM73	ALK tyrosine kinase receptor	None	9330	nM	IC50
TKC115261	Q9UM73	ALK tyrosine kinase receptor	None	4160	nM	IC50
TKC115272	Q9UM73	ALK tyrosine kinase receptor	None	>100000	nM	IC50
TKC115273	Q9UM73	ALK tyrosine kinase receptor	None	4360	nM	IC50
TKC152148	Q9UM73	ALK tyrosine kinase receptor	None	7550	nM	IC50
TKC152157	Q9UM73	ALK tyrosine kinase receptor	None	4730	nM	IC50
TKC174547	Q9UM73	ALK tyrosine kinase receptor	None	>100000	nM	IC50
TKC118419	Q9UQB9	Aurora kinase C	None	69	%	Activity
TKC104905	Q9Y233	cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A	None	>20000	nM	IC50
TKC112754	Q9Y6A2	Cholesterol 24-hydroxylase	None	56	%	Activity
TKC112826	Q9Y6A2	Cholesterol 24-hydroxylase	None	53	%	Activity
TKC112827	Q9Y6A2	Cholesterol 24-hydroxylase	None	30	%	Activity
TKC113159	Q9Y6A2	Cholesterol 24-hydroxylase	None	32	%	Activity
TKC119202	Q9Y6A2	Cholesterol 24-hydroxylase	None	50	nM	Kd
TKC122884	Q9Y6A2	Cholesterol 24-hydroxylase	None	670	nM	Kd
TKC206783	Q9Y6A2	Cholesterol 24-hydroxylase	None	2500	nM	Ki