| Terpenoid ID | TKC001253 |
|
| Cell line | 0 | |
| Protein target | 1 | |
| DiseaseNCIT | 0 | |
| ORDO | 0 | |
| ICD | 2 |
| ID | Cell Line | Synonyms | Value | Unit | Type | NCIt | ORDO |
|---|---|---|---|---|---|---|---|
| TKC001253 | SK-MEL-1 | SK-Mel-1; SK Mel 1; SK-Mel 1; SK-Mel1; SKMEL-1; SkMEL-1; SKMEL1; SK 1 | 9600.0 | nM | IC50 | C3224 | |
| TKC001253 | HL-60 | HL 60; HL.60 HL60; Human Leukemia-60 | 4800.0 | nM | IC50 | C9154 | Orphanet_519 |
| TKC001253 | U-937 | U937; U 937 | 3000.0 | nM | IC50 | C8263 | Orphanet_514 |
| TKC001253 | MOLT-3 | Molt-3; MOLT 3; Molt 3; MOLT3; Molt3 | 1800.0 | nM | IC50 | C9142 | Orphanet_99861 |
| TKC001253 | HT-29 | HT 29; HT29 | 2500.0 | nM | IC50 | C4349 |
| ID | Uniport | Pref_name | Gene name | value | unit | type |
|---|---|---|---|---|---|---|
| TKC001253 | P68371 | Tubulin beta-4B chain | TUBB4B | 45 | % | Inhibition |
| TKC001253 | Q09472 | Histone acetyltransferase p300 | EP300 | 4850 | nM | IC50 |
| Uniport ID | Uniport Name | ICD-11 |
|---|---|---|
| Q09472 | EP300_HUMAN | Solid tumour/cancer [ICD-11: 2A00-2F9Z] |
| Q09472 | EP300_HUMAN | Prostate cancer [ICD-11: 2C82] |