| Terpenoid ID | TKC107681 |
|
| Chirality | TKC107682 | |
| Cell line | 0 | |
| Protein target | 1 | |
| DiseaseNCIT | 0 | |
| ORDO | 0 | |
| ICD | 8 |
| ID | Cell Line | Synonyms | Value | Unit | Type | NCIt | ORDO |
|---|---|---|---|---|---|---|---|
| TKC107681 | NCI-H460 | NCI.H460; H460; H-460; NCIH460; NCI-HUT-460; NCI-460 | 17.0 | % | Activity | C4450 | |
| TKC107681 | HFF | 700.0 | nM | CC50 |
| ID | Uniport | Pref_name | Gene name | value | unit | type |
|---|---|---|---|---|---|---|
| TKC107681 | P05023 | Sodium/potassium-transporting ATPase subunit alpha-1 | ATP1A1 | 5 | nM | IC50 |
| Uniport ID | Uniport Name | ICD-11 |
|---|---|---|
| P05023 | AT1A1_HUMAN | Cardiac arrhythmia [ICD-11: BC9Z] |
| P05023 | AT1A1_HUMAN | Chronic obstructive pulmonary disease [ICD-11: CA22] |
| P05023 | AT1A1_HUMAN | Corneal disease [ICD-11: 9A76-9A78] |
| P05023 | AT1A1_HUMAN | Heart failure [ICD-11: BD10-BD1Z] |
| P05023 | AT1A1_HUMAN | Hyperhidrosis [ICD-11: EE00] |
| P05023 | AT1A1_HUMAN | Malaria [ICD-11: 1F40-1F45] |
| P05023 | AT1A1_HUMAN | Supraventricular tachyarrhythmia [ICD-11: BC81] |
| P05023 | AT1A1_HUMAN | Solid tumour/cancer [ICD-11: 2A00-2F9Z] |