Terpenoid ID | TKC206765 | |
Cell line | 0 | |
Protein target | 13 | |
DiseaseNCIT | 0 | |
ORDO | 0 | |
ICD | 18 |
ID | Cell Line | Synonyms | Value | Unit | Type | NCIt | ORDO |
---|---|---|---|---|---|---|---|
TKC206765 | MCF7 | 5.0 | nM | EC50 | C4194 | ||
TKC206765 | HepG2 | 28184.0 | nM | Potency | C3728 | Orphanet_449 |
ID | Uniport | Pref_name | Gene name | value | unit | type |
---|---|---|---|---|---|---|
TKC206765 | P04062 | Lysosomal acid glucosylceramidase | GBA1 | 4467 | nM | Potency |
TKC206765 | Q9NUW8 | Tyrosyl-DNA phosphodiesterase 1 | TDP1 | 5805 | nM | Potency |
TKC206765 | P43220 | Glucagon-like peptide 1 receptor | GLP1R | 15849 | nM | Potency |
TKC206765 | O75164 | Lysine-specific demethylase 4A | KDM4A | 89125 | nM | Potency |
TKC206765 | Q9UNA4 | DNA polymerase iota | POLI | 89125 | nM | Potency |
TKC206765 | O75496 | Geminin | GMNN | 29093 | nM | Potency |
TKC206765 | O94782 | Ubiquitin carboxyl-terminal hydrolase 1 | USP1 | 7080 | nM | Potency |
TKC206765 | P39748 | Flap endonuclease 1 | FEN1 | 112202 | nM | Potency |
TKC206765 | Q92731 | Estrogen receptor beta | ESR2 | 18000000 | M-1 | Ka |
TKC206765 | P02545 | Prelamin-A/C | LMNA | 25119 | nM | Potency |
TKC206765 | P0DTE4 | UDP-glucuronosyltransferase 2A1 | UGT2A1 | 105 | pm/min/mg | Activity |
TKC206765 | P22309 | UDP-glucuronosyltransferase 1A1 | UGT1A1 | 0 | pm/min/mg | Activity |
TKC206765 | P22310 | UDP-glucuronosyltransferase 1A4 | UGT1A4 | 32 | pm/min/mg | Activity |
TKC206765 | P54855 | UDP-glucuronosyltransferase 2B15 | UGT2B15 | 2 | pm/min/mg | Activity |
TKC206765 | Q9HAW9 | UDP-glucuronosyltransferase 1A8 | UGT1A8 | 33 | pm/min/mg | Activity |
TKC206765 | P16662 | UDP-glucuronosyltransferase 2B7 | UGT2B7 | 5 | total picomoles | Activity |
TKC206765 | P04278 | Sex hormone-binding globulin | SHBG | 1 | nM | Kd |
TKC206765 | P08185 | Corticosteroid-binding globulin | SERPINA6 | 10000 | nM | Ki |
TKC206765 | P56937 | 3-keto-steroid reductase/17-beta-hydroxysteroid dehydrogenase 7 | HSD17B7 | 5 | % | Inhibition |
TKC206765 | O09028 | Gamma-aminobutyric acid receptor subunit pi | Gabrp | 1867 | nM | IC50 |
TKC206765 | Q8TDU6 | G-protein coupled bile acid receptor 1 | GPBAR1 | 7010 | nM | EC50 |
TKC206765 | P06133 | UDP-glucuronosyltransferase 2B4 | UGT2B4 | 12 | total picomoles | Activity |
TKC206765 | O75795 | UDP-glucuronosyltransferase 2B17 | UGT2B17 | 0 | pm/min/mg | Activity |
Uniport ID | Uniport Name | ICD-11 |
---|---|---|
P43220 | GLP1R_HUMAN | Cardiovascular disease [ICD-11: BA00-BE2Z] |
P43220 | GLP1R_HUMAN | Obesity [ICD-11: 5B80-5B81] |
P43220 | GLP1R_HUMAN | Type 2 diabetes mellitus [ICD-11: 5A11] |
P43220 | GLP1R_HUMAN | Type-1/2 diabete [ICD-11: 5A10-5A11] |
P43220 | GLP1R_HUMAN | Acute diabete complication [ICD-11: 5A2Y] |
P43220 | GLP1R_HUMAN | Diabetes mellitus [ICD-11: 5A10] |
P43220 | GLP1R_HUMAN | Dyspepsia [ICD-11: MD92] |
P43220 | GLP1R_HUMAN | Irritable bowel syndrome [ICD-11: DD91] |
P43220 | GLP1R_HUMAN | Intracranial injury [ICD-11: NA07] |
P43220 | GLP1R_HUMAN | Non-alcoholic fatty liver disease [ICD-11: DB92] |
O94782 | UBP1_HUMAN | Solid tumour/cancer [ICD-11: 2A00-2F9Z] |
Q92731 | ESR2_HUMAN | Breast cancer [ICD-11: 2C60-2C6Y] |
Q92731 | ESR2_HUMAN | Cushing syndrome [ICD-11: 5A70] |
Q92731 | ESR2_HUMAN | Menopausal disorder [ICD-11: GA30] |
Q92731 | ESR2_HUMAN | Vasomotor/allergic rhinitis [ICD-11: CA08] |
Q92731 | ESR2_HUMAN | Hepatitis virus infection [ICD-11: 1E50-1E51] |
Q92731 | ESR2_HUMAN | Hyper-lipoproteinaemia [ICD-11: 5C80] |
Q92731 | ESR2_HUMAN | Prostate cancer [ICD-11: 2C82] |
Q92731 | ESR2_HUMAN | Alzheimer disease [ICD-11: 8A20] |
Q92731 | ESR2_HUMAN | Indeterminate colitis [ICD-11: DD72] |
Q92731 | ESR2_HUMAN | Prostate hyperplasia [ICD-11: GA90] |
Q92731 | ESR2_HUMAN | Sepsis [ICD-11: 1G40-1G41] |
Q92731 | ESR2_HUMAN | Irregularities [ICD-11: N.A.] |
Q92731 | ESR2_HUMAN | Trematode disease [ICD-11: 1F8Y] |
Q92731 | ESR2_HUMAN | Low bone mass disorder [ICD-11: FB83] |
Q92731 | ESR2_HUMAN | Thrombocytopenia [ICD-11: 3B64] |
Q92731 | ESR2_HUMAN | Solid tumour/cancer [ICD-11: 2A00-2F9Z] |
Q92731 | ESR2_HUMAN | Herpes simplex infection [ICD-11: 1F00] |
Q92731 | ESR2_HUMAN | Postoperative inflammation [ICD-11: 1A00-CA43] |
P22309 | UD11_HUMAN | Inborn porphyrin/heme metabolism error [ICD-11: 5C58] |
P08185 | CBG_HUMAN | Asthma [ICD-11: CA23] |
P08185 | CBG_HUMAN | Postoperative inflammation [ICD-11: 1A00-CA43] |
P08185 | CBG_HUMAN | Respiratory system disease [ICD-11: CB40-CB7Z] |
P08185 | CBG_HUMAN | Retinopathy [ICD-11: 9B71] |
Q8TDU6 | GPBAR_HUMAN | Type 2 diabetes mellitus [ICD-11: 5A11] |
Q8TDU6 | GPBAR_HUMAN | Hepatic fibrosis/cirrhosis [ICD-11: DB93] |
Q8TDU6 | GPBAR_HUMAN | Metabolic disorder [ICD-11: 5C50-5D2Z] |