Terpenoid ID | TKC034760 |
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Cell line | 2 | |
Protein target | 15 | |
DiseaseNCIT | 2 | |
ORDO | 0 | |
ICD | 39 |
ID | Cell Line | Synonyms | Value | Unit | Type | NCIt | ORDO |
---|---|---|---|---|---|---|---|
TKC034760 | A-431 | A431; A431/P | 5000 | nM | IC50 | C4819 | |
TKC034760 | L1210 | L 1210; L-1210; Leukemic 1210; Leukemia 1210; Leukemia L1210 | 8000 | nM | IC50 | C21604 |
ID | Uniport | Pref_name | Gene name | value | unit | type |
---|---|---|---|---|---|---|
TKC034760 | P00352 | Retinal dehydrogenase 1 | ALDH1A1 | 22387 | nM | Potency |
TKC034760 | P10636 | Microtubule-associated protein tau | MAPT | 17783 | nM | Potency |
TKC034760 | P11473 | Vitamin D3 receptor | VDR | 35481 | nM | Potency |
TKC034760 | Q9NUW8 | Tyrosyl-DNA phosphodiesterase 1 | TDP1 | 1884 | nM | Potency |
TKC034760 | Q16236 | Nuclear factor erythroid 2-related factor 2 | NFE2L2 | 13685 | nM | Potency |
TKC034760 | Q9UBT6 | DNA polymerase kappa | POLK | 39811 | nM | Potency |
TKC034760 | O42275 | Acetylcholinesterase | ache | -9 | % | Inhibition |
TKC034760 | P0DTD1 | Replicase polyprotein 1ab | rep | -2 | % | Inhibition |
TKC034760 | P81908 | Cholinesterase | BCHE | -3 | % | Inhibition |
TKC034760 | Q64133 | Amine oxidase [flavin-containing] A | Maoa | 0 | Activity | |
TKC034760 | Q8BW75 | Amine oxidase [flavin-containing] B | Maob | 0 | Activity | |
TKC034760 | Q96KQ7 | Histone-lysine N-methyltransferase EHMT2 | EHMT2 | 22387 | nM | Potency |
TKC034760 | O00255 | Menin | MEN1 | 39811 | nM | Potency |
TKC034760 | P02791 | Ferritin light chain | FTL | 39811 | nM | Potency |
TKC034760 | P25779 | Cruzipain | None | 10000 | nM | Potency |
TKC034760 | Q9F4F7 | 4'-phosphopantetheinyl transferase ffp | ffp | 39811 | nM | Potency |
TKC034760 | Q03181 | Peroxisome proliferator-activated receptor delta | PPARD | 50119 | nM | Potency |
TKC034760 | P0AE18 | Methionine aminopeptidase | map | >100000 | nM | IC50 |
TKC034760 | P50579 | Methionine aminopeptidase 2 | METAP2 | 1 | nM | IC50 |
TKC034760 | P53582 | Methionine aminopeptidase 1 | METAP1 | 0 | IC50 | |
TKC034760 | Q01662 | Methionine aminopeptidase 1 | MAP1 | >100000 | nM | IC50 |
Uniport ID | Uniport Name | ICD-11 | Disease |
---|---|---|---|
P10636 | TAU_HUMAN | ICD-11: 2A60 | leukaemia |
P10636 | TAU_HUMAN | ICD-11: 8A20 | disease |
P10636 | TAU_HUMAN | ICD-11: 6D71 | disorder |
P10636 | TAU_HUMAN | ICD-11: 8A01 | disorder |
P10636 | TAU_HUMAN | ICD-11: 8A00 | Parkinsonism |
P10636 | TAU_HUMAN | ICD-11: 8A04-8D87 | disease |
P10636 | TAU_HUMAN | ICD-11: 8A20-8A23 | disorder |
Q16236 | NF2L2_HUMAN | ICD-11: 8A03 | disorder |
Q16236 | NF2L2_HUMAN | ICD-11: 2C60-2C6Y | cancer |
Q16236 | NF2L2_HUMAN | ICD-11: 9C61 | Glaucoma |
Q16236 | NF2L2_HUMAN | ICD-11: 2C25 | cancer |
Q16236 | NF2L2_HUMAN | ICD-11: 9B75 | degeneration |
Q16236 | NF2L2_HUMAN | ICD-11: 2C30 | Melanoma |
Q16236 | NF2L2_HUMAN | ICD-11: 6E20-6E8Z | disorder |
Q16236 | NF2L2_HUMAN | ICD-11: BB01 | hypertension |
Q16236 | NF2L2_HUMAN | ICD-11: 8B01 | haemorrhage |
Q16236 | NF2L2_HUMAN | ICD-11: MF8Y | sympton |
Q16236 | NF2L2_HUMAN | ICD-11: DB92 | disease |
Q16236 | NF2L2_HUMAN | ICD-11: 5C5A | deficiency |
Q16236 | NF2L2_HUMAN | ICD-11: 8B60 | disease |
Q16236 | NF2L2_HUMAN | ICD-11: 8A40 | sclerosis |
Q96KQ7 | EHMT2_HUMAN | ICD-11: 2C60-2C6Y | cancer |
Q96KQ7 | EHMT2_HUMAN | ICD-11: 1A00-CA43 | inflammation |
Q96KQ7 | EHMT2_HUMAN | ICD-11: 2A00-2F9Z | tumour/cancer |
P25779 | CYSP_TRYCR | ICD-11: 1F90 | infestation |
P25779 | CYSP_TRYCR | ICD-11: 1F40-1F45 | Malaria |
Q03181 | PPARD_HUMAN | ICD-11: DB92 | disease |
Q03181 | PPARD_HUMAN | ICD-11: 5A11 | mellitus |
Q03181 | PPARD_HUMAN | ICD-11: DB96 | disease |
Q03181 | PPARD_HUMAN | ICD-11: 5C80 | Hyper-lipoproteinaemia |
Q03181 | PPARD_HUMAN | ICD-11: 5B80-5B81 | Obesity |
Q03181 | PPARD_HUMAN | ICD-11: 8A20 | disease |
Q03181 | PPARD_HUMAN | ICD-11: 5C80-5C81 | Dyslipidemia |
Q03181 | PPARD_HUMAN | ICD-11: 5C50-5D2Z | disorder |
Q03181 | PPARD_HUMAN | ICD-11: 5A10 | mellitus |
Q03181 | PPARD_HUMAN | ICD-11: 8A04-8D87 | disease |
P50579 | MAP2_HUMAN | ICD-11: 5B80-5B81 | Obesity |
P50579 | MAP2_HUMAN | ICD-11: 2A00-2F9Z | tumour/cancer |
P50579 | MAP2_HUMAN | ICD-11: 5A11 | mellitus |
P50579 | MAP2_HUMAN | ICD-11: 5A10 | mellitus |