Basic Information

Name [ICD-11: 2A00]
Protein Number 39
Molecule Number 682

Active subnetwork

Terpenoid-protein target Activity Association

ID Uniport Pref_name Gene name value unit type
TKC005454 O14746 Telomerase reverse transcriptase None 75 % Inhibition
TKC014568 O14746 Telomerase reverse transcriptase None 65 % Inhibition
TKC035208 O14746 Telomerase reverse transcriptase None 65000 nM IC50
TKC066096 O14746 Telomerase reverse transcriptase None 780 nM IC50
TKC134702 O14746 Telomerase reverse transcriptase None 4000 nM IC50
TKC007127 P00533 Epidermal growth factor receptor None 19 % Inhibition
TKC025462 P00533 Epidermal growth factor receptor None >200 ug.mL-1 IC50
TKC025466 P00533 Epidermal growth factor receptor None >200 ug.mL-1 IC50
TKC025475 P00533 Epidermal growth factor receptor None 197 ug.mL-1 IC50
TKC071640 P00533 Epidermal growth factor receptor None >20000 nM IC50
TKC076041 P00533 Epidermal growth factor receptor None 75 % Inhibition
TKC077689 P00533 Epidermal growth factor receptor None >20000 nM IC50
TKC106319 P00533 Epidermal growth factor receptor None 56 nM IC50
TKC108557 P00533 Epidermal growth factor receptor None 0.82 nM Kd
TKC151761 P00533 Epidermal growth factor receptor None >10000 nM IC50
TKC200866 P00533 Epidermal growth factor receptor None >10000 nM IC50
TKC013753 P03372 Estrogen receptor None 8913 nM Potency
TKC019072 P03372 Estrogen receptor None 78 % Activity
TKC022931 P03372 Estrogen receptor None 1995 nM Potency
TKC022961 P03372 Estrogen receptor None 54 % Activity
TKC028029 P03372 Estrogen receptor None 0 % Activity
TKC028034 P03372 Estrogen receptor None <0 % Activity
TKC028037 P03372 Estrogen receptor None 1 % Activity
TKC028038 P03372 Estrogen receptor None <0 % Activity
TKC028041 P03372 Estrogen receptor None <0 % Activity
TKC034016 P03372 Estrogen receptor None 51 % Activity
TKC034337 P03372 Estrogen receptor None 2800000 nM IC50
TKC034640 P03372 Estrogen receptor None >1000000 nM Ki
TKC035208 P03372 Estrogen receptor None 39 % Activity
TKC035272 P03372 Estrogen receptor None 2551 nM IC50
TKC035462 P03372 Estrogen receptor None 42 % Activity
TKC066169 P03372 Estrogen receptor None 39811 nM Potency
TKC075769 P03372 Estrogen receptor None 251 nM Potency
TKC079320 P03372 Estrogen receptor None <0 % Activity
TKC079321 P03372 Estrogen receptor None <0 % Activity
TKC087664 P03372 Estrogen receptor None 3162 nM Potency
TKC087988 P03372 Estrogen receptor None 631 nM Potency
TKC087991 P03372 Estrogen receptor None 4467 nM Potency
TKC092297 P03372 Estrogen receptor None 15849 nM Potency
TKC092348 P03372 Estrogen receptor None 8913 nM Potency
TKC096012 P03372 Estrogen receptor None 126 nM Potency
TKC100644 P03372 Estrogen receptor None 31623 nM Potency
TKC101365 P03372 Estrogen receptor None 12570 nM EC50
TKC102448 P03372 Estrogen receptor None 2550 nM EC50
TKC107086 P03372 Estrogen receptor None 8913 nM Potency
TKC107735 P03372 Estrogen receptor None 50119 nM Potency
TKC111727 P03372 Estrogen receptor None 0 nM Ki
TKC111738 P03372 Estrogen receptor None 1 nM EC50
TKC111738 P03372 Estrogen receptor None 166 nM IC50
TKC111738 P03372 Estrogen receptor None 210 nM IC50
TKC111738 P03372 Estrogen receptor None 96 nM IC50
TKC112923 P03372 Estrogen receptor None 26 nM EC50
TKC115268 P03372 Estrogen receptor None 15849 nM Potency
TKC129821 P03372 Estrogen receptor None 70 % Activity
TKC151345 P03372 Estrogen receptor None 35 % Activity
TKC151713 P03372 Estrogen receptor None 40 % Activity
TKC151765 P03372 Estrogen receptor None 81 % Activity
TKC206549 P03372 Estrogen receptor None 3548 nM Potency
TKC206608 P03372 Estrogen receptor None 8170 nM EC50
TKC206652 P03372 Estrogen receptor None 112 nM Potency
TKC206725 P03372 Estrogen receptor None 8 nM Ki
TKC206726 P03372 Estrogen receptor None 72 nM EC50
TKC206759 P03372 Estrogen receptor None >10000 nM IC50
TKC206759 P03372 Estrogen receptor None >10000 nM IC50
TKC206760 P03372 Estrogen receptor None 25119 nM Potency
TKC206764 P03372 Estrogen receptor None 0 % RBA
TKC206770 P03372 Estrogen receptor None 5012 nM Potency
TKC206779 P03372 Estrogen receptor None 6310 nM Potency
TKC206812 P03372 Estrogen receptor None 62000 nM IC50
TKC206812 P03372 Estrogen receptor None 39811 nM Potency
TKC206816 P03372 Estrogen receptor None >1000 nM IC50
TKC206816 P03372 Estrogen receptor None >1000 nM IC50
TKC020117 P03956 Interstitial collagenase None 95 % Inhibition
TKC025462 P04626 Receptor tyrosine-protein kinase erbB-2 None >200 ug.mL-1 IC50
TKC025466 P04626 Receptor tyrosine-protein kinase erbB-2 None >200 ug.mL-1 IC50
TKC025475 P04626 Receptor tyrosine-protein kinase erbB-2 None 125 ug.mL-1 IC50
TKC026211 P04626 Receptor tyrosine-protein kinase erbB-2 None 6 ug.mL-1 IC50
TKC026214 P04626 Receptor tyrosine-protein kinase erbB-2 None 8 ug.mL-1 IC50
TKC026217 P04626 Receptor tyrosine-protein kinase erbB-2 None 4 ug.mL-1 IC50
TKC026229 P04626 Receptor tyrosine-protein kinase erbB-2 None 8 ug.mL-1 IC50
TKC012971 P04637 Cellular tumor antigen p53 None 15849 nM Potency
TKC013753 P04637 Cellular tumor antigen p53 None 13 nM Potency
TKC014568 P04637 Cellular tumor antigen p53 None 2512 nM Potency
TKC016418 P04637 Cellular tumor antigen p53 None 15849 nM Potency
TKC018710 P04637 Cellular tumor antigen p53 None 5 nM Potency
TKC020116 P04637 Cellular tumor antigen p53 None 1585 nM Potency
TKC020117 P04637 Cellular tumor antigen p53 None 12589 nM Potency
TKC020732 P04637 Cellular tumor antigen p53 None 3162 nM Potency
TKC022945 P04637 Cellular tumor antigen p53 None 10000 nM Potency
TKC032619 P04637 Cellular tumor antigen p53 None 15849 nM Potency
TKC034083 P04637 Cellular tumor antigen p53 None 31623 nM Potency
TKC035272 P04637 Cellular tumor antigen p53 None 12589 nM Potency
TKC039869 P04637 Cellular tumor antigen p53 None 25119 nM Potency
TKC052854 P04637 Cellular tumor antigen p53 None 25119 nM Potency
TKC062321 P04637 Cellular tumor antigen p53 None 10000 nM Potency
TKC075769 P04637 Cellular tumor antigen p53 None 159 nM Potency
TKC084075 P04637 Cellular tumor antigen p53 None 8 nM Potency
TKC091895 P04637 Cellular tumor antigen p53 None 50119 nM Potency
TKC092297 P04637 Cellular tumor antigen p53 None 15849 nM Potency
TKC095493 P04637 Cellular tumor antigen p53 None 3162 nM Potency
TKC100636 P04637 Cellular tumor antigen p53 None 1585 nM Potency
TKC100701 P04637 Cellular tumor antigen p53 None 10000 nM Potency
TKC101020 P04637 Cellular tumor antigen p53 None 12589 nM Potency
TKC101618 P04637 Cellular tumor antigen p53 None 12589 nM Potency
TKC102204 P04637 Cellular tumor antigen p53 None 31623 nM Potency
TKC102540 P04637 Cellular tumor antigen p53 None 31623 nM Potency
TKC103149 P04637 Cellular tumor antigen p53 None 12589 nM Potency
TKC103210 P04637 Cellular tumor antigen p53 None 40 nM Potency
TKC103257 P04637 Cellular tumor antigen p53 None 10000 nM Potency
TKC103736 P04637 Cellular tumor antigen p53 None 2512 nM Potency
TKC104070 P04637 Cellular tumor antigen p53 None 63 nM Potency
TKC104071 P04637 Cellular tumor antigen p53 None 50 nM Potency
TKC104072 P04637 Cellular tumor antigen p53 None 126 nM Potency
TKC104073 P04637 Cellular tumor antigen p53 None 63 nM Potency
TKC104114 P04637 Cellular tumor antigen p53 None 79 nM Potency
TKC105153 P04637 Cellular tumor antigen p53 None 5012 nM Potency
TKC105168 P04637 Cellular tumor antigen p53 None 12589 nM Potency
TKC105360 P04637 Cellular tumor antigen p53 None 15849 nM Potency
TKC105424 P04637 Cellular tumor antigen p53 None 25119 nM Potency
TKC105784 P04637 Cellular tumor antigen p53 None 25119 nM Potency
TKC105891 P04637 Cellular tumor antigen p53 None 10000 nM Potency
TKC106232 P04637 Cellular tumor antigen p53 None 15849 nM Potency
TKC107086 P04637 Cellular tumor antigen p53 None 12589 nM Potency
TKC107104 P04637 Cellular tumor antigen p53 None 12589 nM Potency
TKC107201 P04637 Cellular tumor antigen p53 None 19953 nM Potency
TKC107332 P04637 Cellular tumor antigen p53 None 10000 nM Potency
TKC107525 P04637 Cellular tumor antigen p53 None 31623 nM Potency
TKC107627 P04637 Cellular tumor antigen p53 None 25119 nM Potency
TKC107818 P04637 Cellular tumor antigen p53 None 12589 nM Potency
TKC108536 P04637 Cellular tumor antigen p53 None 5 nM Potency
TKC108732 P04637 Cellular tumor antigen p53 None 19953 nM Potency
TKC109484 P04637 Cellular tumor antigen p53 None 20 nM Potency
TKC109519 P04637 Cellular tumor antigen p53 None 10000 nM Potency
TKC109561 P04637 Cellular tumor antigen p53 None 159 nM Potency
TKC109569 P04637 Cellular tumor antigen p53 None 32 nM Potency
TKC110010 P04637 Cellular tumor antigen p53 None 56234 nM Potency
TKC112576 P04637 Cellular tumor antigen p53 None 50 nM Potency
TKC112784 P04637 Cellular tumor antigen p53 None 31623 nM Potency
TKC112792 P04637 Cellular tumor antigen p53 None 25119 nM Potency
TKC115268 P04637 Cellular tumor antigen p53 None 70795 nM Potency
TKC117625 P04637 Cellular tumor antigen p53 None 3162 nM Potency
TKC117993 P04637 Cellular tumor antigen p53 None 501 nM Potency
TKC117994 P04637 Cellular tumor antigen p53 None 40 nM Potency
TKC118006 P04637 Cellular tumor antigen p53 None 100 nM Potency
TKC118895 P04637 Cellular tumor antigen p53 None 31623 nM Potency
TKC132609 P04637 Cellular tumor antigen p53 None 11220 nM Potency
TKC134635 P04637 Cellular tumor antigen p53 None 56234 nM Potency
TKC138777 P04637 Cellular tumor antigen p53 None 15849 nM Potency
TKC140757 P04637 Cellular tumor antigen p53 None 31623 nM Potency
TKC147290 P04637 Cellular tumor antigen p53 None 12589 nM Potency
TKC148482 P04637 Cellular tumor antigen p53 None 19953 nM Potency
TKC149827 P04637 Cellular tumor antigen p53 None 1000 nM Potency
TKC150706 P04637 Cellular tumor antigen p53 None 31623 nM Potency
TKC151237 P04637 Cellular tumor antigen p53 None 35481 nM Potency
TKC151303 P04637 Cellular tumor antigen p53 None 31623 nM Potency
TKC151571 P04637 Cellular tumor antigen p53 None 6310 nM Potency
TKC151758 P04637 Cellular tumor antigen p53 None 19953 nM Potency
TKC173955 P04637 Cellular tumor antigen p53 None 31623 nM Potency
TKC206652 P04637 Cellular tumor antigen p53 None 32 nM Potency
TKC206657 P04637 Cellular tumor antigen p53 None 8 nM Potency
TKC206760 P04637 Cellular tumor antigen p53 None 31623 nM Potency
TKC206760 P04637 Cellular tumor antigen p53 None 15000 nM Kd
TKC206812 P04637 Cellular tumor antigen p53 None 31623 nM Potency
TKC206872 P04637 Cellular tumor antigen p53 None 631 nM Potency
TKC206889 P04637 Cellular tumor antigen p53 None 501 nM Potency
TKC206901 P04637 Cellular tumor antigen p53 None 2512 nM Potency
TKC022945 P05067 Amyloid-beta precursor protein None 23109 nM Potency
TKC027272 P05067 Amyloid-beta precursor protein None >300000 nM EC50
TKC027273 P05067 Amyloid-beta precursor protein None 65400 nM EC50
TKC050321 P05067 Amyloid-beta precursor protein None 100 % Activity
TKC050560 P05067 Amyloid-beta precursor protein None 0 % Inhibition
TKC051308 P05067 Amyloid-beta precursor protein None 0 % Inhibition
TKC059731 P05067 Amyloid-beta precursor protein None 39 % Activity
TKC060461 P05067 Amyloid-beta precursor protein None 65 % Activity
TKC077689 P05067 Amyloid-beta precursor protein None 100 % Activity
TKC102625 P05067 Amyloid-beta precursor protein None 0 % Inhibition
TKC111348 P05067 Amyloid-beta precursor protein None 17 % Activity
TKC113610 P05067 Amyloid-beta precursor protein None 20 % Activity
TKC113764 P05067 Amyloid-beta precursor protein None 71900 nM IC50
TKC113765 P05067 Amyloid-beta precursor protein None 28000 nM IC50
TKC113766 P05067 Amyloid-beta precursor protein None 34300 nM IC50
TKC113767 P05067 Amyloid-beta precursor protein None 55 % Inhibition
TKC113768 P05067 Amyloid-beta precursor protein None 43500 nM IC50
TKC113769 P05067 Amyloid-beta precursor protein None 1200 nM IC50
TKC118380 P05067 Amyloid-beta precursor protein None 13400 nM IC50
TKC118381 P05067 Amyloid-beta precursor protein None 10100 nM IC50
TKC118419 P05067 Amyloid-beta precursor protein None 231 nM Potency
TKC123071 P05067 Amyloid-beta precursor protein None 20 % Activity
TKC150909 P05067 Amyloid-beta precursor protein None 0 % Activity
TKC152398 P05067 Amyloid-beta precursor protein None 100000 nM IC50
TKC179988 P05067 Amyloid-beta precursor protein None 8 hr TIME
TKC206799 P05067 Amyloid-beta precursor protein None 95900 nM IC50
TKC012929 P05771 Protein kinase C beta type None 2 nM Ki
TKC055602 P05771 Protein kinase C beta type None >150000 nM IC50
TKC075924 P05771 Protein kinase C beta type None 90 % Inhibition
TKC090435 P05771 Protein kinase C beta type None 0.2 nM Kd
TKC103074 P05771 Protein kinase C beta type None >150000 nM IC50
TKC104128 P05771 Protein kinase C beta type None >150000 nM IC50
TKC104703 P05771 Protein kinase C beta type None >150000 nM IC50
TKC105956 P05771 Protein kinase C beta type None 2 nM Ki
TKC123088 P05771 Protein kinase C beta type None >150000 nM IC50
TKC151276 P05771 Protein kinase C beta type None >150000 nM IC50
TKC151326 P05771 Protein kinase C beta type None 1 nM Kd
TKC151326 P05771 Protein kinase C beta type None 1.3 nM Kd
TKC151326 P05771 Protein kinase C beta type None 1.3 nM Kd
TKC151326 P05771 Protein kinase C beta type None 1.8 nM Ki
TKC151326 P05771 Protein kinase C beta type None 1.3 nM Kd
TKC151326 P05771 Protein kinase C beta type None 1.3 nM Kd
TKC152742 P05771 Protein kinase C beta type None >150000 nM IC50
TKC206051 P07858 Cathepsin B None 103500 nM IC50
TKC009193 P08253 72 kDa type IV collagenase None 33260 nM IC50
TKC020117 P08253 72 kDa type IV collagenase None 90 % Inhibition
TKC023429 P08253 72 kDa type IV collagenase None 0 ug.mL-1 IC50
TKC020712 P08581 Hepatocyte growth factor receptor None >20000 nM IC50
TKC024886 P08581 Hepatocyte growth factor receptor None 3120 nM IC50
TKC025690 P08581 Hepatocyte growth factor receptor None >100000 nM IC50
TKC033871 P08581 Hepatocyte growth factor receptor None 50000 nM IC50
TKC082039 P08581 Hepatocyte growth factor receptor None 5500 nM IC50
TKC115259 P08581 Hepatocyte growth factor receptor None 34000 nM IC50
TKC115261 P08581 Hepatocyte growth factor receptor None 47600 nM IC50
TKC115272 P08581 Hepatocyte growth factor receptor None >100000 nM IC50
TKC115273 P08581 Hepatocyte growth factor receptor None 27500 nM IC50
TKC152148 P08581 Hepatocyte growth factor receptor None 78000 nM IC50
TKC152157 P08581 Hepatocyte growth factor receptor None 71500 nM IC50
TKC174547 P08581 Hepatocyte growth factor receptor None >100000 nM IC50
TKC014892 P11387 DNA topoisomerase 1 None 3 ug.mL-1 MIC
TKC014893 P11387 DNA topoisomerase 1 None 13 ug.mL-1 MIC
TKC017201 P11387 DNA topoisomerase 1 None 13 ug.mL-1 MIC
TKC048122 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC048308 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC048324 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC048330 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC048341 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC049414 P11387 DNA topoisomerase 1 None 25000 nM IC50
TKC049417 P11387 DNA topoisomerase 1 None 55000 nM IC50
TKC056419 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC056423 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC056425 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC056427 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC056430 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC058891 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC058895 P11387 DNA topoisomerase 1 None 48600 nM IC50
TKC058897 P11387 DNA topoisomerase 1 None 45100 nM IC50
TKC058919 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC058921 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC058935 P11387 DNA topoisomerase 1 None 109300 nM IC50
TKC058949 P11387 DNA topoisomerase 1 None 250000 nM IC50
TKC058950 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC058953 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC058979 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC059000 P11387 DNA topoisomerase 1 None 53700 nM IC50
TKC059030 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC059045 P11387 DNA topoisomerase 1 None 131700 nM IC50
TKC059148 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC059149 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC059160 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC059165 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC059317 P11387 DNA topoisomerase 1 None 250000 nM IC50
TKC059337 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC059344 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC059345 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC059425 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC072969 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC072970 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC096715 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC100727 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC103324 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC105545 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC137826 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC137841 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC138033 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC138054 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC143022 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC143033 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC143055 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC143114 P11387 DNA topoisomerase 1 None 250000 nM IC50
TKC143115 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC145932 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC146257 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC147779 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC147805 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC148618 P11387 DNA topoisomerase 1 None 106000 nM IC50
TKC205544 P11387 DNA topoisomerase 1 None 30000 nM IC50
TKC205878 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC207002 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC026583 P11802 Cyclin-dependent kinase 4 None 9 ug.mL-1 IC50
TKC113582 P11802 Cyclin-dependent kinase 4 None 10 ug.mL-1 IC50
TKC011761 P12931 Proto-oncogene tyrosine-protein kinase Src None 61 % Inhibition
TKC024886 P12931 Proto-oncogene tyrosine-protein kinase Src None 8620 nM IC50
TKC025690 P12931 Proto-oncogene tyrosine-protein kinase Src None 19700 nM IC50
TKC115259 P12931 Proto-oncogene tyrosine-protein kinase Src None 2400 nM IC50
TKC115261 P12931 Proto-oncogene tyrosine-protein kinase Src None 2240 nM IC50
TKC115272 P12931 Proto-oncogene tyrosine-protein kinase Src None >100000 nM IC50
TKC115273 P12931 Proto-oncogene tyrosine-protein kinase Src None 1480 nM IC50
TKC135974 P12931 Proto-oncogene tyrosine-protein kinase Src None 35800 nM IC50
TKC151761 P12931 Proto-oncogene tyrosine-protein kinase Src None >10000 nM IC50
TKC152148 P12931 Proto-oncogene tyrosine-protein kinase Src None 1910 nM IC50
TKC152157 P12931 Proto-oncogene tyrosine-protein kinase Src None 2170 nM IC50
TKC174547 P12931 Proto-oncogene tyrosine-protein kinase Src None >100000 nM IC50
TKC200866 P12931 Proto-oncogene tyrosine-protein kinase Src None >10000 nM IC50
TKC205544 P14416 D(2) dopamine receptor None 687 nM Ki
TKC205544 P14416 D(2) dopamine receptor None 280 nM Ki
TKC205544 P14416 D(2) dopamine receptor None 398.1 nM Ki
TKC206544 P14416 D(2) dopamine receptor None >10000 nM Ki
TKC020117 P14780 Matrix metalloproteinase-9 None 99 % Inhibition
TKC023429 P14780 Matrix metalloproteinase-9 None 1 ug.mL-1 IC50
TKC037777 P14780 Matrix metalloproteinase-9 None 6 ug.mL-1 IC50
TKC039471 P14780 Matrix metalloproteinase-9 None 6 ug.mL-1 IC50
TKC006896 P14902 Indoleamine 2,3-dioxygenase 1 None 7700 nM IC50
TKC014575 P14902 Indoleamine 2,3-dioxygenase 1 None 4680 nM IC50
TKC024473 P14902 Indoleamine 2,3-dioxygenase 1 None 10000 nM IC50
TKC024474 P14902 Indoleamine 2,3-dioxygenase 1 None 11000 nM IC50
TKC104241 P14902 Indoleamine 2,3-dioxygenase 1 None 0 nM EC50
TKC118419 P24941 Cyclin-dependent kinase 2 None 95 % Activity
TKC206292 P24941 Cyclin-dependent kinase 2 None 4800 nM Kd
TKC022852 P26358 DNA (cytosine-5)-methyltransferase 1 None 2 uM Activity
TKC022854 P26358 DNA (cytosine-5)-methyltransferase 1 None 55 uM Activity
TKC055219 P26358 DNA (cytosine-5)-methyltransferase 1 None 5930 nM IC50
TKC055219 P26358 DNA (cytosine-5)-methyltransferase 1 None 5930 nM IC50
TKC001930 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 31623 nM Potency
TKC005139 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 4467 nM Potency
TKC005313 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 6 nM Potency
TKC005454 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 39811 nM Potency
TKC008286 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 11220 nM Potency
TKC009499 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 11220 nM Potency
TKC011384 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 39811 nM Potency
TKC011526 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 5 nM Potency
TKC011921 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 39811 nM Potency
TKC012929 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 891 nM Potency
TKC013755 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 6 nM Potency
TKC018288 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 7943 nM Potency
TKC018339 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 35481 nM Potency
TKC019571 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 891 nM Potency
TKC019887 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 35481 nM Potency
TKC020117 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 14125 nM Potency
TKC020459 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 35481 nM Potency
TKC020574 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 31623 nM Potency
TKC021477 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 7943 nM Potency
TKC022945 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 50 nM Potency
TKC023619 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 31623 nM Potency
TKC025405 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 15849 nM Potency
TKC026870 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 3162 nM Potency
TKC028718 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 11220 nM Potency
TKC029307 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 47444 nM Potency
TKC030478 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 18888 nM Potency
TKC035029 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 398 nM Potency
TKC035272 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 31623 nM Potency
TKC035580 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 3 nM Potency
TKC036999 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 31623 nM Potency
TKC038473 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 447 nM Potency
TKC039332 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 5012 nM Potency
TKC040026 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 0 nM Potency
TKC040829 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 316 nM Potency
TKC052854 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 21192 nM Potency
TKC053751 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 39811 nM Potency
TKC055066 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 70795 nM Potency
TKC056469 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 19953 nM Potency
TKC056482 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 44668 nM Potency
TKC057133 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 35481 nM Potency
TKC062333 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 39811 nM Potency
TKC063247 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 5 nM Potency
TKC066332 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 31623 nM Potency
TKC066411 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 5012 nM Potency
TKC066631 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 2239 nM Potency
TKC073833 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 3 nM Potency
TKC075769 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 44668 nM Potency
TKC076129 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 7080 nM Potency
TKC077689 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 4467 nM Potency
TKC080049 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 7943 nM Potency
TKC080874 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 44668 nM Potency
TKC085168 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 50 nM Potency
TKC088230 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 2512 nM Potency
TKC088231 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 31623 nM Potency
TKC088678 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 316 nM Potency
TKC090518 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 19953 nM Potency
TKC092297 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 398 nM Potency
TKC095442 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 2 nM Potency
TKC095645 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 22387 nM Potency
TKC097937 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 19953 nM Potency
TKC097944 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 14125 nM Potency
TKC100524 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 19953 nM Potency
TKC100990 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 562 nM Potency
TKC102657 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 29935 nM Potency
TKC103150 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 31623 nM Potency
TKC103159 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 50119 nM Potency
TKC103538 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 4 nM Potency
TKC104194 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 25119 nM Potency
TKC105095 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 28184 nM Potency
TKC105168 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 4 nM Potency
TKC105226 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 11220 nM Potency
TKC105356 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 39811 nM Potency
TKC105357 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 35481 nM Potency
TKC105378 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 355 nM Potency
TKC105710 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 6310 nM Potency
TKC105717 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 12589 nM Potency
TKC106074 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 40 nM Potency
TKC106147 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 1122 nM Potency
TKC106537 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 19953 nM Potency
TKC106682 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 20 nM Potency
TKC107104 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 11220 nM Potency
TKC107593 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 1259 nM Potency
TKC107830 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 56 nM Potency
TKC108060 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 44668 nM Potency
TKC108363 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 11220 nM Potency
TKC109484 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 3 nM Potency
TKC109493 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 1337 nM Potency
TKC110002 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 8913 nM Potency
TKC112576 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 1413 nM Potency
TKC112754 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 794 nM Potency
TKC112784 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 3981 nM Potency
TKC112813 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 7080 nM Potency
TKC113063 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 28184 nM Potency
TKC113150 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 1995 nM Potency
TKC118131 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 44668 nM Potency
TKC118419 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 44668 nM Potency
TKC118895 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 14 nM Potency
TKC118911 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 112 nM Potency
TKC130327 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 251 nM Potency
TKC130342 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 17783 nM Potency
TKC133919 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 1585 nM Potency
TKC141805 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 39811 nM Potency
TKC150625 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 9466 nM Potency
TKC150706 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 11220 nM Potency
TKC151293 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 8913 nM Potency
TKC151326 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 13 nM Potency
TKC151609 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 39811 nM Potency
TKC164433 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 9466 nM Potency
TKC169452 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 2239 nM Potency
TKC169457 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 2239 nM Potency
TKC174441 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 8437 nM Potency
TKC202992 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 3 nM Potency
TKC206113 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 1778 nM Potency
TKC206177 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 2511886 nM Potency
TKC206657 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 501 nM Potency
TKC206760 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 39811 nM Potency
TKC206764 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 12589254 nM Potency
TKC206779 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 79 nM Potency
TKC206872 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 200 nM Potency
TKC207103 P27695 DNA-(apurinic or apyrimidinic site) endonuclease None 22 nM Potency
TKC112785 P29317 Ephrin type-A receptor 2 None 48978 nM IC50
TKC206760 P29317 Ephrin type-A receptor 2 None 50000 nM IC50
TKC011761 P31749 RAC-alpha serine/threonine-protein kinase None 54 % Inhibition
TKC016414 P31749 RAC-alpha serine/threonine-protein kinase None 36 % Activity
TKC024886 P31749 RAC-alpha serine/threonine-protein kinase None 48400 nM IC50
TKC025690 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC044763 P31749 RAC-alpha serine/threonine-protein kinase None 100 % Inhibition
TKC115259 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC115261 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC115272 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC115273 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC118419 P31749 RAC-alpha serine/threonine-protein kinase None 96 % Inhibition
TKC152148 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC152157 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC174547 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC206776 P31749 RAC-alpha serine/threonine-protein kinase None 3 uM Activity
TKC205544 P35462 D(3) dopamine receptor None 2489 nM Ki
TKC205544 P35462 D(3) dopamine receptor None 3981.07 nM Ki
TKC206544 P35462 D(3) dopamine receptor None >10000 nM Ki
TKC206549 P35869 Aryl hydrocarbon receptor None 17783 nM Potency
TKC024886 P35968 Vascular endothelial growth factor receptor 2 None 4810 nM IC50
TKC025690 P35968 Vascular endothelial growth factor receptor 2 None 3660 nM IC50
TKC051154 P35968 Vascular endothelial growth factor receptor 2 None 40 % Inhibition
TKC051155 P35968 Vascular endothelial growth factor receptor 2 None 46 % Inhibition
TKC065375 P35968 Vascular endothelial growth factor receptor 2 None 0 % Inhibition
TKC102689 P35968 Vascular endothelial growth factor receptor 2 None 0 % Inhibition
TKC108267 P35968 Vascular endothelial growth factor receptor 2 None 0 % Inhibition
TKC115259 P35968 Vascular endothelial growth factor receptor 2 None 4950 nM IC50
TKC115261 P35968 Vascular endothelial growth factor receptor 2 None 4600 nM IC50
TKC115272 P35968 Vascular endothelial growth factor receptor 2 None >100000 nM IC50
TKC115273 P35968 Vascular endothelial growth factor receptor 2 None 4850 nM IC50
TKC146202 P35968 Vascular endothelial growth factor receptor 2 None 61 % Inhibition
TKC152148 P35968 Vascular endothelial growth factor receptor 2 None 4350 nM IC50
TKC152157 P35968 Vascular endothelial growth factor receptor 2 None 6010 nM IC50
TKC174547 P35968 Vascular endothelial growth factor receptor 2 None >100000 nM IC50
TKC207124 P35968 Vascular endothelial growth factor receptor 2 None 40400 nM IC50
TKC003060 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC005454 P40763 Signal transducer and activator of transcription 3 None 4600 nM IC50
TKC016414 P40763 Signal transducer and activator of transcription 3 None >10000 nM EC50
TKC020636 P40763 Signal transducer and activator of transcription 3 None 6900 nM IC50
TKC020796 P40763 Signal transducer and activator of transcription 3 None 22900 nM IC50
TKC020867 P40763 Signal transducer and activator of transcription 3 None 26 % Inhibition
TKC020868 P40763 Signal transducer and activator of transcription 3 None 31 % Inhibition
TKC020869 P40763 Signal transducer and activator of transcription 3 None 49 % Inhibition
TKC022393 P40763 Signal transducer and activator of transcription 3 None 89500 nM IC50
TKC022771 P40763 Signal transducer and activator of transcription 3 None >100000 nM IC50
TKC028367 P40763 Signal transducer and activator of transcription 3 None 4100 nM IC50
TKC030728 P40763 Signal transducer and activator of transcription 3 None 2 % Inhibition
TKC033506 P40763 Signal transducer and activator of transcription 3 None 2400 nM IC50
TKC033507 P40763 Signal transducer and activator of transcription 3 None 2300 nM IC50
TKC036334 P40763 Signal transducer and activator of transcription 3 None 4 % Inhibition
TKC038766 P40763 Signal transducer and activator of transcription 3 None 1 % Inhibition
TKC039282 P40763 Signal transducer and activator of transcription 3 None 2 % Inhibition
TKC042554 P40763 Signal transducer and activator of transcription 3 None 6300 nM IC50
TKC042556 P40763 Signal transducer and activator of transcription 3 None 110000 nM IC50
TKC044507 P40763 Signal transducer and activator of transcription 3 None 4 % Inhibition
TKC044595 P40763 Signal transducer and activator of transcription 3 None 4 % Inhibition
TKC044621 P40763 Signal transducer and activator of transcription 3 None 3 % Inhibition
TKC044669 P40763 Signal transducer and activator of transcription 3 None 4 % Inhibition
TKC047957 P40763 Signal transducer and activator of transcription 3 None 17100 nM IC50
TKC047959 P40763 Signal transducer and activator of transcription 3 None >30000 nM IC50
TKC047961 P40763 Signal transducer and activator of transcription 3 None >30000 nM IC50
TKC048029 P40763 Signal transducer and activator of transcription 3 None 270 nM IC50
TKC048030 P40763 Signal transducer and activator of transcription 3 None 19200 nM IC50
TKC048031 P40763 Signal transducer and activator of transcription 3 None 590 nM IC50
TKC051029 P40763 Signal transducer and activator of transcription 3 None 60000 nM MIC
TKC060882 P40763 Signal transducer and activator of transcription 3 None >25000 nM IC50
TKC075769 P40763 Signal transducer and activator of transcription 3 None 1862 nM IC50
TKC077689 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC078334 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC087623 P40763 Signal transducer and activator of transcription 3 None >100000 nM IC50
TKC087625 P40763 Signal transducer and activator of transcription 3 None 7000 nM IC50
TKC093311 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC100739 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC101161 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC103159 P40763 Signal transducer and activator of transcription 3 None 3000 nM IC50
TKC103189 P40763 Signal transducer and activator of transcription 3 None 32500 nM IC50
TKC103191 P40763 Signal transducer and activator of transcription 3 None 24800 nM IC50
TKC105152 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC107659 P40763 Signal transducer and activator of transcription 3 None 4 % Inhibition
TKC108773 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC112576 P40763 Signal transducer and activator of transcription 3 None 1154 nM IC50
TKC134761 P40763 Signal transducer and activator of transcription 3 None 48 % Inhibition
TKC135961 P40763 Signal transducer and activator of transcription 3 None 73000 nM IC50
TKC135978 P40763 Signal transducer and activator of transcription 3 None 14210 nM IC50
TKC136653 P40763 Signal transducer and activator of transcription 3 None 2 % Inhibition
TKC148207 P40763 Signal transducer and activator of transcription 3 None 15840 nM IC50
TKC149924 P40763 Signal transducer and activator of transcription 3 None 74 % Inhibition
TKC151284 P40763 Signal transducer and activator of transcription 3 None 14000 nM IC50
TKC156528 P40763 Signal transducer and activator of transcription 3 None >30000 nM IC50
TKC206318 P40763 Signal transducer and activator of transcription 3 None 12200 nM IC50
TKC206468 P40763 Signal transducer and activator of transcription 3 None 46 % Inhibition
TKC206627 P40763 Signal transducer and activator of transcription 3 None >100000 nM IC50
TKC206646 P40763 Signal transducer and activator of transcription 3 None 67000 nM IC50
TKC206652 P40763 Signal transducer and activator of transcription 3 None 700 nM IC50
TKC036497 P42574 Caspase-3 None 200000 nM IC50
TKC096499 P42574 Caspase-3 None 50000 nM IC50
TKC025058 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 1000 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 5 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 19 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 55 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 55000 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 89 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 5 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 15 nM Kd
TKC087988 P49327 Fatty acid synthase None >40 % Inhibition
TKC046324 P49840 Glycogen synthase kinase-3 alpha None 1600 nM IC50
TKC011761 P49841 Glycogen synthase kinase-3 beta None 20 % Inhibition
TKC046098 P49841 Glycogen synthase kinase-3 beta None 794 nM IC50
TKC046099 P49841 Glycogen synthase kinase-3 beta None 2300 nM IC50
TKC046324 P49841 Glycogen synthase kinase-3 beta None 4500 nM IC50
TKC046324 P49841 Glycogen synthase kinase-3 beta None 1900 nM IC50
TKC118419 P49841 Glycogen synthase kinase-3 beta None 65 % Activity
TKC146056 P49841 Glycogen synthase kinase-3 beta None 3000 nM IC50
TKC021620 P60568 Interleukin-2 None 3 nM Kd
TKC116180 P60568 Interleukin-2 None 0 nM Kd
TKC151761 Q12866 Tyrosine-protein kinase Mer None 4900 nM IC50
TKC200866 Q12866 Tyrosine-protein kinase Mer None 4900 nM IC50
TKC016189 Q13315 Serine-protein kinase ATM None 19953 nM Potency
TKC016371 Q13315 Serine-protein kinase ATM None 25119 nM Potency
TKC029307 Q13315 Serine-protein kinase ATM None 39811 nM Potency
TKC039202 Q13315 Serine-protein kinase ATM None 3548 nM Potency
TKC063474 Q13315 Serine-protein kinase ATM None 35481 nM Potency
TKC066411 Q13315 Serine-protein kinase ATM None 31623 nM Potency
TKC103159 Q13315 Serine-protein kinase ATM None 19953 nM Potency
TKC150598 Q13315 Serine-protein kinase ATM None 39811 nM Potency
TKC151609 Q13315 Serine-protein kinase ATM None 39811 nM Potency
TKC174441 Q13315 Serine-protein kinase ATM None 412 nM Potency
TKC005475 Q15910 Histone-lysine N-methyltransferase EZH2 None 9600 nM IC50
TKC014568 Q15910 Histone-lysine N-methyltransferase EZH2 None 8900 nM IC50
TKC005454 Q16665 Hypoxia-inducible factor 1-alpha None 1360 nM IC50
TKC005475 Q16665 Hypoxia-inducible factor 1-alpha None 7340 nM IC50
TKC010010 Q16665 Hypoxia-inducible factor 1-alpha None >20000 nM IC50
TKC011921 Q16665 Hypoxia-inducible factor 1-alpha None 1995 nM Potency
TKC012261 Q16665 Hypoxia-inducible factor 1-alpha None 280 nM IC50
TKC012262 Q16665 Hypoxia-inducible factor 1-alpha None 3180 nM IC50
TKC012971 Q16665 Hypoxia-inducible factor 1-alpha None 25119 nM Potency
TKC014568 Q16665 Hypoxia-inducible factor 1-alpha None 8510 nM IC50
TKC017189 Q16665 Hypoxia-inducible factor 1-alpha None 10600 nM IC50
TKC017192 Q16665 Hypoxia-inducible factor 1-alpha None 1700 nM IC50
TKC017193 Q16665 Hypoxia-inducible factor 1-alpha None 2300 nM IC50
TKC020116 Q16665 Hypoxia-inducible factor 1-alpha None 501 nM Potency
TKC022945 Q16665 Hypoxia-inducible factor 1-alpha None 2512 nM Potency
TKC023570 Q16665 Hypoxia-inducible factor 1-alpha None 15800 nM IC50
TKC030239 Q16665 Hypoxia-inducible factor 1-alpha None 200 nM Potency
TKC035272 Q16665 Hypoxia-inducible factor 1-alpha None 10000 nM Potency
TKC037547 Q16665 Hypoxia-inducible factor 1-alpha None 10 % Activity
TKC038977 Q16665 Hypoxia-inducible factor 1-alpha None 820 nM IC50
TKC045710 Q16665 Hypoxia-inducible factor 1-alpha None 500 nM IC50
TKC045931 Q16665 Hypoxia-inducible factor 1-alpha None 2900 nM IC50
TKC045946 Q16665 Hypoxia-inducible factor 1-alpha None 2900 nM IC50
TKC047694 Q16665 Hypoxia-inducible factor 1-alpha None 63 nM IC50
TKC047695 Q16665 Hypoxia-inducible factor 1-alpha None 68 nM IC50
TKC056482 Q16665 Hypoxia-inducible factor 1-alpha None >100000 nM IC50
TKC056482 Q16665 Hypoxia-inducible factor 1-alpha None >100000 nM IC50
TKC062172 Q16665 Hypoxia-inducible factor 1-alpha None 15000 nM IC50
TKC062175 Q16665 Hypoxia-inducible factor 1-alpha None 20000 nM IC50
TKC062182 Q16665 Hypoxia-inducible factor 1-alpha None 20000 nM IC50
TKC062192 Q16665 Hypoxia-inducible factor 1-alpha None 20000 nM IC50
TKC062193 Q16665 Hypoxia-inducible factor 1-alpha None >30000 nM IC50
TKC065782 Q16665 Hypoxia-inducible factor 1-alpha None >30000 nM IC50
TKC081893 Q16665 Hypoxia-inducible factor 1-alpha None 400 nM IC50
TKC092297 Q16665 Hypoxia-inducible factor 1-alpha None 39811 nM Potency
TKC094057 Q16665 Hypoxia-inducible factor 1-alpha None >30000 nM IC50
TKC094058 Q16665 Hypoxia-inducible factor 1-alpha None >20000 nM IC50
TKC095493 Q16665 Hypoxia-inducible factor 1-alpha None 3162 nM Potency
TKC096011 Q16665 Hypoxia-inducible factor 1-alpha None 1 nM Potency
TKC096012 Q16665 Hypoxia-inducible factor 1-alpha None 251 nM Potency
TKC100416 Q16665 Hypoxia-inducible factor 1-alpha None 25119 nM Potency
TKC100643 Q16665 Hypoxia-inducible factor 1-alpha None 12589 nM Potency
TKC100990 Q16665 Hypoxia-inducible factor 1-alpha None 159 nM Potency
TKC101618 Q16665 Hypoxia-inducible factor 1-alpha None 15849 nM Potency
TKC102145 Q16665 Hypoxia-inducible factor 1-alpha None 1259 nM Potency
TKC102589 Q16665 Hypoxia-inducible factor 1-alpha None 8000 nM EC50
TKC103149 Q16665 Hypoxia-inducible factor 1-alpha None 31623 nM Potency
TKC103159 Q16665 Hypoxia-inducible factor 1-alpha None 270 nM IC50
TKC103433 Q16665 Hypoxia-inducible factor 1-alpha None >30000 nM IC50
TKC103494 Q16665 Hypoxia-inducible factor 1-alpha None 79 nM Potency
TKC103496 Q16665 Hypoxia-inducible factor 1-alpha None 20 nM Potency
TKC104070 Q16665 Hypoxia-inducible factor 1-alpha None 40 nM Potency
TKC104071 Q16665 Hypoxia-inducible factor 1-alpha None 100 nM Potency
TKC104114 Q16665 Hypoxia-inducible factor 1-alpha None 126 nM Potency
TKC104664 Q16665 Hypoxia-inducible factor 1-alpha None 794 nM Potency
TKC105037 Q16665 Hypoxia-inducible factor 1-alpha None 794 nM Potency
TKC105510 Q16665 Hypoxia-inducible factor 1-alpha None 6000 nM EC50
TKC105710 Q16665 Hypoxia-inducible factor 1-alpha None 12589 nM Potency
TKC106426 Q16665 Hypoxia-inducible factor 1-alpha None 1000 nM Potency
TKC106576 Q16665 Hypoxia-inducible factor 1-alpha None 13000 nM EC50
TKC107086 Q16665 Hypoxia-inducible factor 1-alpha None 19953 nM Potency
TKC109561 Q16665 Hypoxia-inducible factor 1-alpha None 251 nM Potency
TKC110002 Q16665 Hypoxia-inducible factor 1-alpha None 63 nM Potency
TKC110007 Q16665 Hypoxia-inducible factor 1-alpha None 7943 nM Potency
TKC111738 Q16665 Hypoxia-inducible factor 1-alpha None 16 nM Potency
TKC112789 Q16665 Hypoxia-inducible factor 1-alpha None 1000 nM Potency
TKC112906 Q16665 Hypoxia-inducible factor 1-alpha None 5012 nM Potency
TKC114819 Q16665 Hypoxia-inducible factor 1-alpha None 12589 nM Potency
TKC117993 Q16665 Hypoxia-inducible factor 1-alpha None 2000 nM EC50
TKC117997 Q16665 Hypoxia-inducible factor 1-alpha None 40 nM EC50
TKC118004 Q16665 Hypoxia-inducible factor 1-alpha None 2512 nM Potency
TKC118012 Q16665 Hypoxia-inducible factor 1-alpha None 600 nM EC50
TKC118131 Q16665 Hypoxia-inducible factor 1-alpha None 126 nM Potency
TKC134897 Q16665 Hypoxia-inducible factor 1-alpha None 3400 nM IC50
TKC137120 Q16665 Hypoxia-inducible factor 1-alpha None 200 nM IC50
TKC137126 Q16665 Hypoxia-inducible factor 1-alpha None 2400 nM IC50
TKC137243 Q16665 Hypoxia-inducible factor 1-alpha None 200 nM IC50
TKC144475 Q16665 Hypoxia-inducible factor 1-alpha None 25000 nM IC50
TKC151571 Q16665 Hypoxia-inducible factor 1-alpha None 7943 nM Potency
TKC205806 Q16665 Hypoxia-inducible factor 1-alpha None 5012 nM Potency
TKC206042 Q16665 Hypoxia-inducible factor 1-alpha None 6310 nM Potency
TKC206395 Q16665 Hypoxia-inducible factor 1-alpha None 12589 nM Potency
TKC206453 Q16665 Hypoxia-inducible factor 1-alpha None 25119 nM Potency
TKC206617 Q16665 Hypoxia-inducible factor 1-alpha None 12700 nM IC50
TKC206688 Q16665 Hypoxia-inducible factor 1-alpha None 63 nM Potency
TKC206726 Q16665 Hypoxia-inducible factor 1-alpha None 79 nM Potency
TKC206760 Q16665 Hypoxia-inducible factor 1-alpha None 50119 nM Potency
TKC206780 Q16665 Hypoxia-inducible factor 1-alpha None 3981 nM Potency
TKC206812 Q16665 Hypoxia-inducible factor 1-alpha None 79433 nM Potency
TKC206816 Q16665 Hypoxia-inducible factor 1-alpha None 12589 nM Potency
TKC206872 Q16665 Hypoxia-inducible factor 1-alpha None 1000 nM Potency
TKC206889 Q16665 Hypoxia-inducible factor 1-alpha None 501 nM Potency
TKC206890 Q16665 Hypoxia-inducible factor 1-alpha None 20 nM EC50
TKC206901 Q16665 Hypoxia-inducible factor 1-alpha None 159 nM Potency
TKC026309 Q99814 Endothelial PAS domain-containing protein 1 None 3300 nM EC50
TKC035150 Q99814 Endothelial PAS domain-containing protein 1 None 10800 nM IC50
TKC045708 Q99814 Endothelial PAS domain-containing protein 1 None 4200 nM EC50
TKC045868 Q99814 Endothelial PAS domain-containing protein 1 None 1200 nM EC50
TKC046523 Q99814 Endothelial PAS domain-containing protein 1 None >100000 nM EC50
TKC100652 Q99814 Endothelial PAS domain-containing protein 1 None 3400 nM EC50
TKC101122 Q99814 Endothelial PAS domain-containing protein 1 None 6200 nM EC50
TKC103124 Q99814 Endothelial PAS domain-containing protein 1 None 148900 nM EC50
TKC104992 Q99814 Endothelial PAS domain-containing protein 1 None 107500 nM EC50
TKC105151 Q99814 Endothelial PAS domain-containing protein 1 None 183300 nM EC50
TKC118419 Q99814 Endothelial PAS domain-containing protein 1 None 3930 nM IC50
TKC143885 Q99814 Endothelial PAS domain-containing protein 1 None 14400 nM IC50
TKC165028 Q99814 Endothelial PAS domain-containing protein 1 None 11800 nM EC50
TKC115268 Q99835 Smoothened homolog None 36 % Activity
TKC115284 Q99835 Smoothened homolog None 28 % Activity
TKC206385 Q99835 Smoothened homolog None 70 % Activity
TKC066096 Q9NR96 Toll-like receptor 9 None 3015 nM IC50
TKC076529 Q9NR96 Toll-like receptor 9 None >49739 nM IC50
TKC076529 Q9NR96 Toll-like receptor 9 None >49739 nM IC50
TKC082378 Q9NR96 Toll-like receptor 9 None 7929 nM IC50
TKC082378 Q9NR96 Toll-like receptor 9 None 7929 nM IC50