Basic Information

Name [ICD-11: FA20]
Protein Number 54
Molecule Number 819

Active subnetwork

Terpenoid-protein target Activity Association

ID Uniport Pref_name Gene name value unit type
TKC118419 O00329 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform None 4 nM IC50
TKC118419 O00329 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform None 9 nM IC50
TKC118419 O00329 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform None 9 nM IC50
TKC118419 O00329 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform None 5.5 nM Kd
TKC050429 O14920 Inhibitor of nuclear factor kappa-B kinase subunit beta None 2620 nM IC50
TKC077819 O14920 Inhibitor of nuclear factor kappa-B kinase subunit beta None 4240 nM IC50
TKC118419 O14920 Inhibitor of nuclear factor kappa-B kinase subunit beta None 96 % Activity
TKC118419 O75116 Rho-associated protein kinase 2 None 99 % Activity
TKC076129 P00915 Carbonic anhydrase 1 None 8010 nM Ki
TKC104783 P00915 Carbonic anhydrase 1 None 2210 nM Ki
TKC105780 P00915 Carbonic anhydrase 1 None 1470 nM Ki
TKC076129 P00918 Carbonic anhydrase 2 None 6130 nM Ki
TKC104783 P00918 Carbonic anhydrase 2 None 1280 nM Ki
TKC105780 P00918 Carbonic anhydrase 2 None 970 nM Ki
TKC112756 P00918 Carbonic anhydrase 2 None >10000 nM IC50
TKC051021 P01375 Tumor necrosis factor None 9 nM Kd
TKC051029 P01375 Tumor necrosis factor None 9 nM Kd
TKC055869 P01375 Tumor necrosis factor None 10880 nM IC50
TKC063751 P01375 Tumor necrosis factor None 19 nM Kd
TKC064986 P01375 Tumor necrosis factor None 3 nM Kd
TKC075769 P01375 Tumor necrosis factor None 376 nM Potency
TKC101833 P01375 Tumor necrosis factor None 8 nM Kd
TKC145547 P01375 Tumor necrosis factor None 2 nM Kd
TKC148618 P01375 Tumor necrosis factor None 17 nM Kd
TKC151763 P01375 Tumor necrosis factor None 8 nM Kd
TKC151876 P01375 Tumor necrosis factor None 6 % Inhibition
TKC035272 P02768 Albumin None 2 10'5L/mol Ka
TKC053751 P02768 Albumin None 12000 nM Kd
TKC106240 P02768 Albumin None 93 % PPB
TKC107285 P02768 Albumin None 36 M-1.s-1 k_on
TKC123088 P02768 Albumin None 593 nM Kd
TKC149924 P02768 Albumin None 1 hr T1/2
TKC206884 P02768 Albumin None 50 % Activity
TKC206885 P02768 Albumin None 58 % Activity
TKC020117 P03956 Interstitial collagenase None 95 % Inhibition
TKC008187 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 30200 nM IC50
TKC023515 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 53 % Inhibition
TKC025574 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 52 % Inhibition
TKC026893 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 21 % Inhibition
TKC026895 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 61 % Inhibition
TKC057019 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 22300 nM IC50
TKC100777 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 30 % Inhibition
TKC101031 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 1500 nM IC50
TKC101538 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 39 % Inhibition
TKC101847 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 1000 nM IC50
TKC103703 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 40 % Inhibition
TKC137314 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 8400 nM IC50
TKC138471 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 21700 nM IC50
TKC017639 P04054 Phospholipase A2 None 95 % Activity
TKC017706 P04054 Phospholipase A2 None 5 % Activity
TKC045776 P04054 Phospholipase A2 None 1600 nM IC50
TKC045777 P04054 Phospholipase A2 None 3700 nM IC50
TKC045872 P04054 Phospholipase A2 None 44 % Activity
TKC046211 P04054 Phospholipase A2 None 3900 nM IC50
TKC046211 P04054 Phospholipase A2 None 13000 nM IC50
TKC055219 P04054 Phospholipase A2 None 2040 nM IC50
TKC055219 P04054 Phospholipase A2 None 2040 nM IC50
TKC077689 P04054 Phospholipase A2 None 3000 nM IC50
TKC105149 P04054 Phospholipase A2 None 8 % Activity
TKC106090 P04054 Phospholipase A2 None 95 % Activity
TKC106091 P04054 Phospholipase A2 None 90 % Activity
TKC106240 P04054 Phospholipase A2 None 5 % Activity
TKC109622 P04054 Phospholipase A2 None 10000 nM Kd
TKC110322 P04054 Phospholipase A2 None 67 % Inhibition
TKC110427 P04054 Phospholipase A2 None 13800 nM IC50
TKC112787 P04054 Phospholipase A2 None 40 % Activity
TKC115260 P04054 Phospholipase A2 None 55 % Inhibition
TKC146194 P04054 Phospholipase A2 None 5 % Activity
TKC151364 P04054 Phospholipase A2 None 30 % Activity
TKC152148 P04054 Phospholipase A2 None 47 % Inhibition
TKC206812 P04054 Phospholipase A2 None 35 % Activity
TKC206849 P04054 Phospholipase A2 None 80 % Activity
TKC206884 P04054 Phospholipase A2 None 150000 nM Kd
TKC013753 P04150 Glucocorticoid receptor None 5012 nM Potency
TKC019368 P04150 Glucocorticoid receptor None 10000 nM Potency
TKC021365 P04150 Glucocorticoid receptor None 5623 nM Potency
TKC021425 P04150 Glucocorticoid receptor None 5623 nM Potency
TKC023246 P04150 Glucocorticoid receptor None >3210 nM Ki
TKC023246 P04150 Glucocorticoid receptor None 2465 nM Ki
TKC030239 P04150 Glucocorticoid receptor None 30 nM Ki
TKC030239 P04150 Glucocorticoid receptor None 69 % Inhibition
TKC035272 P04150 Glucocorticoid receptor None 44668 nM Potency
TKC048937 P04150 Glucocorticoid receptor None 56 % Inhibition
TKC063171 P04150 Glucocorticoid receptor None 56 % Inhibition
TKC074866 P04150 Glucocorticoid receptor None 25119 nM Potency
TKC075769 P04150 Glucocorticoid receptor None 562 nM Potency
TKC081853 P04150 Glucocorticoid receptor None 84 % Activity
TKC087664 P04150 Glucocorticoid receptor None 4 nM Potency
TKC087988 P04150 Glucocorticoid receptor None 1995 nM Potency
TKC092297 P04150 Glucocorticoid receptor None 794 nM Potency
TKC096011 P04150 Glucocorticoid receptor None 1 nM Ki
TKC106250 P04150 Glucocorticoid receptor None 298700 nM EC50
TKC106877 P04150 Glucocorticoid receptor None 2465 nM Ki
TKC106878 P04150 Glucocorticoid receptor None >2465 nM Ki
TKC106878 P04150 Glucocorticoid receptor None 3210 nM Ki
TKC106879 P04150 Glucocorticoid receptor None 3210 nM Ki
TKC107086 P04150 Glucocorticoid receptor None 8913 nM Potency
TKC109619 P04150 Glucocorticoid receptor None 298700 nM EC50
TKC111727 P04150 Glucocorticoid receptor None 17884 nM Ki
TKC114511 P04150 Glucocorticoid receptor None 252 nM Ki
TKC115268 P04150 Glucocorticoid receptor None 50119 nM Potency
TKC122884 P04150 Glucocorticoid receptor None 11220 nM Potency
TKC134780 P04150 Glucocorticoid receptor None 4 nM Potency
TKC136411 P04150 Glucocorticoid receptor None 1 nM Potency
TKC183618 P04150 Glucocorticoid receptor None 70 % Activity
TKC206652 P04150 Glucocorticoid receptor None 355 nM Potency
TKC206672 P04150 Glucocorticoid receptor None 50119 nM Potency
TKC206688 P04150 Glucocorticoid receptor None 501 nM Potency
TKC206690 P04150 Glucocorticoid receptor None 28184 nM Potency
TKC206759 P04150 Glucocorticoid receptor None 1457 nM Ki
TKC206760 P04150 Glucocorticoid receptor None 39811 nM Potency
TKC206770 P04150 Glucocorticoid receptor None 2818 nM Potency
TKC206779 P04150 Glucocorticoid receptor None 23 nM Ki
TKC206812 P04150 Glucocorticoid receptor None 224 nM Ki
TKC206816 P04150 Glucocorticoid receptor None 31 nM Ki
TKC206816 P04150 Glucocorticoid receptor None 31 nM Ki
TKC206816 P04150 Glucocorticoid receptor None 31 nM Ki
TKC206816 P04150 Glucocorticoid receptor None 31 nM Ki
TKC206816 P04150 Glucocorticoid receptor None 31 nM Ki
TKC206816 P04150 Glucocorticoid receptor None >1000 nM IC50
TKC206816 P04150 Glucocorticoid receptor None >1000 nM IC50
TKC206816 P04150 Glucocorticoid receptor None 31 nM Ki
TKC066096 P04608 Protein Tat None >100000 nM IC50
TKC012127 P05412 Transcription factor AP-1 None 1500 nM IC50
TKC012492 P05412 Transcription factor AP-1 None 3 % Activity
TKC058501 P05412 Transcription factor AP-1 None 130 nM EC50
TKC079230 P05412 Transcription factor AP-1 None 5 % Activity
TKC079243 P05412 Transcription factor AP-1 None 3 % Activity
TKC102298 P05412 Transcription factor AP-1 None 71 nM IC50
TKC103273 P05412 Transcription factor AP-1 None 4000 nM IC50
TKC105096 P05412 Transcription factor AP-1 None 2 % Activity
TKC140438 P05412 Transcription factor AP-1 None 40 nM IC50
TKC143885 P05412 Transcription factor AP-1 None 30000 nM IC50
TKC143885 P05412 Transcription factor AP-1 None 130000 nM IC50
TKC146899 P05412 Transcription factor AP-1 None 32 nM IC50
TKC012929 P05771 Protein kinase C beta type None 2 nM Ki
TKC055602 P05771 Protein kinase C beta type None >150000 nM IC50
TKC075924 P05771 Protein kinase C beta type None 90 % Inhibition
TKC090435 P05771 Protein kinase C beta type None 0.2 nM Kd
TKC103074 P05771 Protein kinase C beta type None >150000 nM IC50
TKC104128 P05771 Protein kinase C beta type None >150000 nM IC50
TKC104703 P05771 Protein kinase C beta type None >150000 nM IC50
TKC105956 P05771 Protein kinase C beta type None 2 nM Ki
TKC123088 P05771 Protein kinase C beta type None >150000 nM IC50
TKC151276 P05771 Protein kinase C beta type None >150000 nM IC50
TKC151326 P05771 Protein kinase C beta type None 1 nM Kd
TKC151326 P05771 Protein kinase C beta type None 1.3 nM Kd
TKC151326 P05771 Protein kinase C beta type None 1.3 nM Kd
TKC151326 P05771 Protein kinase C beta type None 1.8 nM Ki
TKC151326 P05771 Protein kinase C beta type None 1.3 nM Kd
TKC151326 P05771 Protein kinase C beta type None 1.3 nM Kd
TKC152742 P05771 Protein kinase C beta type None >150000 nM IC50
TKC206051 P07858 Cathepsin B None 103500 nM IC50
TKC022234 P08246 Neutrophil elastase None >1 % Inhibition
TKC022237 P08246 Neutrophil elastase None 100000 nM IC50
TKC022245 P08246 Neutrophil elastase None 18000 nM IC50
TKC055903 P08246 Neutrophil elastase None >10000 nM IC50
TKC056482 P08246 Neutrophil elastase None 416 nM IC50
TKC093449 P08246 Neutrophil elastase None 100000 nM IC50
TKC093451 P08246 Neutrophil elastase None >40 % Inhibition
TKC104777 P08246 Neutrophil elastase None 1560 nM IC50
TKC020117 P08254 Stromelysin-1 None 98 % Inhibition
TKC042585 P08254 Stromelysin-1 None 300 nM MIC50
TKC042586 P08254 Stromelysin-1 None 300 nM MIC50
TKC042587 P08254 Stromelysin-1 None 300 nM MIC50
TKC020117 P09917 Polyunsaturated fatty acid 5-lipoxygenase None -67 % Inhibition
TKC024485 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >50000 nM IC50
TKC024587 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 600 nM IC50
TKC024956 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 18000 nM IC50
TKC024992 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 450 nM IC50
TKC024993 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 14000 nM IC50
TKC025965 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >150000 nM IC50
TKC026303 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 4600 nM IC50
TKC026309 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 680 nM IC50
TKC027255 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >67 % Activity
TKC034201 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >200000 nM IC50
TKC040026 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 72 % Inhibition
TKC051154 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 2700 nM IC50
TKC056482 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >64 % Activity
TKC058811 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 42000 nM IC50
TKC058812 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >93 % Activity
TKC064374 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 42000 nM IC50
TKC064407 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >72 % Activity
TKC065375 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >70 % Activity
TKC071640 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >60 % Activity
TKC076350 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 100 % Activity
TKC077689 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 100 % Activity
TKC077703 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >86 % Activity
TKC078194 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 31800 nM IC50
TKC082039 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 48 % Inhibition
TKC088678 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 24800 nM IC50
TKC089448 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 35 % Inhibition
TKC094647 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 97 % Activity
TKC107943 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 2000 nM IC50
TKC123028 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 30400 nM IC50
TKC124303 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 750 nM IC50
TKC133309 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >200000 nM IC50
TKC133656 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 25100 nM IC50
TKC134278 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >200000 nM IC50
TKC139322 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >67 % Activity
TKC139366 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 3000 nM IC50
TKC141401 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 42000 nM IC50
TKC141499 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 25700 nM IC50
TKC141805 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >53 % Activity
TKC142849 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >70 % Activity
TKC142897 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 30600 nM IC50
TKC142922 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >61 % Activity
TKC143539 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 100 % Activity
TKC145848 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 42000 nM IC50
TKC145932 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >56 % Activity
TKC145968 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 100 % Activity
TKC146774 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >63 % Activity
TKC149759 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >73 % Activity
TKC150706 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >62 % Activity
TKC087988 P0DMS8 Adenosine receptor A3 None 2357 nM Ki
TKC096012 P0DMS8 Adenosine receptor A3 None 2982 nM Ki
TKC205544 P0DMS8 Adenosine receptor A3 None 95 nM IC50
TKC206779 P0DMS8 Adenosine receptor A3 None 2674 nM Ki
TKC066096 P11413 Glucose-6-phosphate 1-dehydrogenase None >80000 nM IC50
TKC109495 P11413 Glucose-6-phosphate 1-dehydrogenase None 15800 nM IC50
TKC109970 P11413 Glucose-6-phosphate 1-dehydrogenase None 6300 nM IC50
TKC109998 P11413 Glucose-6-phosphate 1-dehydrogenase None 31600 nM IC50
TKC110077 P11413 Glucose-6-phosphate 1-dehydrogenase None 5300 nM IC50
TKC112485 P11413 Glucose-6-phosphate 1-dehydrogenase None >200000 nM IC50
TKC112754 P11413 Glucose-6-phosphate 1-dehydrogenase None 6200 nM Ki
TKC112754 P11413 Glucose-6-phosphate 1-dehydrogenase None 24900 nM IC50
TKC113159 P11413 Glucose-6-phosphate 1-dehydrogenase None 81400 nM IC50
TKC151885 P11413 Glucose-6-phosphate 1-dehydrogenase None >80000 nM IC50
TKC206687 P11413 Glucose-6-phosphate 1-dehydrogenase None 900 nM IC50
TKC206754 P11413 Glucose-6-phosphate 1-dehydrogenase None 3000 nM Ki
TKC206754 P11413 Glucose-6-phosphate 1-dehydrogenase None >200000 nM IC50
TKC206758 P11413 Glucose-6-phosphate 1-dehydrogenase None >200000 nM IC50
TKC206777 P11413 Glucose-6-phosphate 1-dehydrogenase None 4300 nM IC50
TKC206899 P11413 Glucose-6-phosphate 1-dehydrogenase None 5200 nM IC50
TKC020114 P14679 Tyrosinase None 2300 nM IC50
TKC020116 P14679 Tyrosinase None <1000000 nM IC50
TKC020117 P14679 Tyrosinase None 8980 nM IC50
TKC020119 P14679 Tyrosinase None 1150 nM IC50
TKC020458 P14679 Tyrosinase None 50000 nM IC50
TKC048730 P14679 Tyrosinase None 54640 nM IC50
TKC051754 P14679 Tyrosinase None 13950 nM IC50
TKC051758 P14679 Tyrosinase None 48920 nM IC50
TKC051808 P14679 Tyrosinase None 92250 nM IC50
TKC051810 P14679 Tyrosinase None 102390 nM IC50
TKC062678 P14679 Tyrosinase None 85010 nM IC50
TKC122980 P14679 Tyrosinase None 14 % Inhibition
TKC151523 P14679 Tyrosinase None 4 % Inhibition
TKC152829 P14679 Tyrosinase None -2 % Inhibition
TKC205699 P14679 Tyrosinase None 1600 nM IC50
TKC205700 P14679 Tyrosinase None 1600 nM IC50
TKC206231 P14679 Tyrosinase None >50000 nM IC50
TKC206436 P14679 Tyrosinase None >50000 nM IC50
TKC206456 P14679 Tyrosinase None >50000 nM IC50
TKC207074 P14679 Tyrosinase None >50000 nM IC50
TKC020117 P14780 Matrix metalloproteinase-9 None 99 % Inhibition
TKC023429 P14780 Matrix metalloproteinase-9 None 1 ug.mL-1 IC50
TKC037777 P14780 Matrix metalloproteinase-9 None 6 ug.mL-1 IC50
TKC039471 P14780 Matrix metalloproteinase-9 None 6 ug.mL-1 IC50
TKC013753 P15121 Aldo-keto reductase family 1 member B1 None 1100000 nM Km
TKC035272 P15121 Aldo-keto reductase family 1 member B1 None 500 nM Ki
TKC035273 P15121 Aldo-keto reductase family 1 member B1 None 1500 nM Ki
TKC048308 P15121 Aldo-keto reductase family 1 member B1 None >200000 nM IC50
TKC048325 P15121 Aldo-keto reductase family 1 member B1 None 147300 nM IC50
TKC048341 P15121 Aldo-keto reductase family 1 member B1 None >200000 nM IC50
TKC049175 P15121 Aldo-keto reductase family 1 member B1 None 25 ug.mL-1 IC50
TKC051021 P15121 Aldo-keto reductase family 1 member B1 None >193500 nM IC50
TKC051028 P15121 Aldo-keto reductase family 1 member B1 None 22800 nM IC50
TKC051029 P15121 Aldo-keto reductase family 1 member B1 None >193500 nM IC50
TKC051032 P15121 Aldo-keto reductase family 1 member B1 None >189400 nM IC50
TKC055115 P15121 Aldo-keto reductase family 1 member B1 None 12000 ug.mL-1 IC50
TKC056482 P15121 Aldo-keto reductase family 1 member B1 None 41000 nM IC50
TKC057931 P15121 Aldo-keto reductase family 1 member B1 None 6 /min Kcat
TKC060859 P15121 Aldo-keto reductase family 1 member B1 None 25 ug.mL-1 IC50
TKC063401 P15121 Aldo-keto reductase family 1 member B1 None 25 ug.mL-1 IC50
TKC063402 P15121 Aldo-keto reductase family 1 member B1 None 25 ug.mL-1 IC50
TKC063751 P15121 Aldo-keto reductase family 1 member B1 None >195300 nM IC50
TKC077689 P15121 Aldo-keto reductase family 1 member B1 None 124000 nM IC50
TKC081137 P15121 Aldo-keto reductase family 1 member B1 None >193500 nM IC50
TKC088678 P15121 Aldo-keto reductase family 1 member B1 None 280000 nM IC50
TKC092322 P15121 Aldo-keto reductase family 1 member B1 None 400000 nM Km
TKC101833 P15121 Aldo-keto reductase family 1 member B1 None >193500 nM IC50
TKC123088 P15121 Aldo-keto reductase family 1 member B1 None 11000 nM IC50
TKC137747 P15121 Aldo-keto reductase family 1 member B1 None >200000 nM IC50
TKC137786 P15121 Aldo-keto reductase family 1 member B1 None >200000 nM IC50
TKC137982 P15121 Aldo-keto reductase family 1 member B1 None >200000 nM IC50
TKC138004 P15121 Aldo-keto reductase family 1 member B1 None >200000 nM IC50
TKC141585 P15121 Aldo-keto reductase family 1 member B1 None >194400 nM IC50
TKC142922 P15121 Aldo-keto reductase family 1 member B1 None 84000 nM IC50
TKC145170 P15121 Aldo-keto reductase family 1 member B1 None >199200 nM IC50
TKC145534 P15121 Aldo-keto reductase family 1 member B1 None >187900 nM IC50
TKC145540 P15121 Aldo-keto reductase family 1 member B1 None >174200 nM IC50
TKC145547 P15121 Aldo-keto reductase family 1 member B1 None >174700 nM IC50
TKC146774 P15121 Aldo-keto reductase family 1 member B1 None 72000 nM IC50
TKC150706 P15121 Aldo-keto reductase family 1 member B1 None 34000 nM IC50
TKC151691 P15121 Aldo-keto reductase family 1 member B1 None 119200 nM IC50
TKC151763 P15121 Aldo-keto reductase family 1 member B1 None 43800 nM IC50
TKC151921 P15121 Aldo-keto reductase family 1 member B1 None >194400 nM IC50
TKC156642 P15121 Aldo-keto reductase family 1 member B1 None >189400 nM IC50
TKC206760 P15121 Aldo-keto reductase family 1 member B1 None 6900 nM IC50
TKC207025 P15121 Aldo-keto reductase family 1 member B1 None >183900 nM IC50
TKC039202 P21453 Sphingosine 1-phosphate receptor 1 None 4962 nM IC50
TKC096012 P21453 Sphingosine 1-phosphate receptor 1 None 34120 nM EC50
TKC096012 P21453 Sphingosine 1-phosphate receptor 1 None >95100 nM EC50
TKC096012 P21453 Sphingosine 1-phosphate receptor 1 None 25400 nM EC50
TKC020117 P22894 Neutrophil collagenase None 100 % Inhibition
TKC000611 P23219 Prostaglandin G/H synthase 1 None 40000 nM IC50
TKC001618 P23219 Prostaglandin G/H synthase 1 None 34000 nM IC50
TKC009896 P23219 Prostaglandin G/H synthase 1 None 791100 nM IC50
TKC019819 P23219 Prostaglandin G/H synthase 1 None 48 % Inhibition
TKC019859 P23219 Prostaglandin G/H synthase 1 None 54 % Inhibition
TKC020491 P23219 Prostaglandin G/H synthase 1 None 4000 nM IC50
TKC020796 P23219 Prostaglandin G/H synthase 1 None 30 % Inhibition
TKC021940 P23219 Prostaglandin G/H synthase 1 None 40 % Inhibition
TKC022833 P23219 Prostaglandin G/H synthase 1 None 43 % Inhibition
TKC022834 P23219 Prostaglandin G/H synthase 1 None 43 % Inhibition
TKC022961 P23219 Prostaglandin G/H synthase 1 None 44 % Inhibition
TKC024587 P23219 Prostaglandin G/H synthase 1 None 3300 nM IC50
TKC024587 P23219 Prostaglandin G/H synthase 1 None 3300 nM IC50
TKC031258 P23219 Prostaglandin G/H synthase 1 None 3600 nM IC50
TKC034201 P23219 Prostaglandin G/H synthase 1 None >200000 nM IC50
TKC034358 P23219 Prostaglandin G/H synthase 1 None 39000 nM IC50
TKC034359 P23219 Prostaglandin G/H synthase 1 None 39000 nM IC50
TKC036372 P23219 Prostaglandin G/H synthase 1 None 14000 nM IC50
TKC037595 P23219 Prostaglandin G/H synthase 1 None 36000 nM IC50
TKC043613 P23219 Prostaglandin G/H synthase 1 None 43000 nM IC50
TKC049750 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC049818 P23219 Prostaglandin G/H synthase 1 None 44 ug IC50
TKC054011 P23219 Prostaglandin G/H synthase 1 None 8800 nM IC50
TKC054031 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC054081 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC054090 P23219 Prostaglandin G/H synthase 1 None 7500 nM IC50
TKC054099 P23219 Prostaglandin G/H synthase 1 None 8800 nM IC50
TKC054100 P23219 Prostaglandin G/H synthase 1 None 8900 nM IC50
TKC054101 P23219 Prostaglandin G/H synthase 1 None 7600 nM IC50
TKC054240 P23219 Prostaglandin G/H synthase 1 None 7800 nM IC50
TKC054241 P23219 Prostaglandin G/H synthase 1 None 6300 nM IC50
TKC056482 P23219 Prostaglandin G/H synthase 1 None 210000 nM IC50
TKC060184 P23219 Prostaglandin G/H synthase 1 None 8300 nM IC50
TKC060216 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC060284 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC060302 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC060303 P23219 Prostaglandin G/H synthase 1 None 7800 nM IC50
TKC060304 P23219 Prostaglandin G/H synthase 1 None 8000 nM IC50
TKC060399 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC060602 P23219 Prostaglandin G/H synthase 1 None 5900 nM IC50
TKC066954 P23219 Prostaglandin G/H synthase 1 None 38 % Inhibition
TKC068533 P23219 Prostaglandin G/H synthase 1 None 28000 nM IC50
TKC071010 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC077689 P23219 Prostaglandin G/H synthase 1 None 380000 nM IC50
TKC077689 P23219 Prostaglandin G/H synthase 1 None 380000 nM IC50
TKC095276 P23219 Prostaglandin G/H synthase 1 None 48 % Inhibition
TKC113936 P23219 Prostaglandin G/H synthase 1 None 65 % Inhibition
TKC122543 P23219 Prostaglandin G/H synthase 1 None 35 % Inhibition
TKC130084 P23219 Prostaglandin G/H synthase 1 None 39 % Inhibition
TKC130119 P23219 Prostaglandin G/H synthase 1 None 33 % Inhibition
TKC130577 P23219 Prostaglandin G/H synthase 1 None <43 % Inhibition
TKC130901 P23219 Prostaglandin G/H synthase 1 None 36 % Inhibition
TKC133309 P23219 Prostaglandin G/H synthase 1 None >200000 nM IC50
TKC133517 P23219 Prostaglandin G/H synthase 1 None 1300 nM IC50
TKC133656 P23219 Prostaglandin G/H synthase 1 None >200000 nM IC50
TKC134278 P23219 Prostaglandin G/H synthase 1 None >200000 nM IC50
TKC139036 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC140627 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC141365 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC143641 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC151113 P23219 Prostaglandin G/H synthase 1 None 116400 nM IC50
TKC151284 P23219 Prostaglandin G/H synthase 1 None 51 % Inhibition
TKC151765 P23219 Prostaglandin G/H synthase 1 None 48 % Inhibition
TKC151792 P23219 Prostaglandin G/H synthase 1 None 14000 nM IC50
TKC172853 P23219 Prostaglandin G/H synthase 1 None 43700 nM IC50
TKC005313 P28482 Mitogen-activated protein kinase 1 None 25119 nM Potency
TKC008529 P28482 Mitogen-activated protein kinase 1 None 126 nM Potency
TKC013736 P28482 Mitogen-activated protein kinase 1 None 6310 nM Potency
TKC019571 P28482 Mitogen-activated protein kinase 1 None 32 nM Potency
TKC021977 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC022811 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC022814 P28482 Mitogen-activated protein kinase 1 None 28184 nM Potency
TKC022945 P28482 Mitogen-activated protein kinase 1 None 5012 nM Potency
TKC035272 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC035580 P28482 Mitogen-activated protein kinase 1 None 17783 nM Potency
TKC038273 P28482 Mitogen-activated protein kinase 1 None 31623 nM Potency
TKC039202 P28482 Mitogen-activated protein kinase 1 None 10000 nM Potency
TKC054329 P28482 Mitogen-activated protein kinase 1 None 19953 nM Potency
TKC060863 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC084630 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC087664 P28482 Mitogen-activated protein kinase 1 None 32 nM Potency
TKC087988 P28482 Mitogen-activated protein kinase 1 None 462 nM IC50
TKC092297 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC096011 P28482 Mitogen-activated protein kinase 1 None 3162 nM Potency
TKC096012 P28482 Mitogen-activated protein kinase 1 None 576 nM IC50
TKC100675 P28482 Mitogen-activated protein kinase 1 None 7943 nM Potency
TKC101618 P28482 Mitogen-activated protein kinase 1 None 7943 nM Potency
TKC102941 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC103150 P28482 Mitogen-activated protein kinase 1 None 3548 nM Potency
TKC103257 P28482 Mitogen-activated protein kinase 1 None 14125 nM Potency
TKC103736 P28482 Mitogen-activated protein kinase 1 None 15849 nM Potency
TKC104091 P28482 Mitogen-activated protein kinase 1 None 5012 nM Potency
TKC104194 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC105033 P28482 Mitogen-activated protein kinase 1 None 1259 nM Potency
TKC105034 P28482 Mitogen-activated protein kinase 1 None 1259 nM Potency
TKC105037 P28482 Mitogen-activated protein kinase 1 None 501 nM Potency
TKC105210 P28482 Mitogen-activated protein kinase 1 None 6310 nM Potency
TKC105295 P28482 Mitogen-activated protein kinase 1 None 126 nM Potency
TKC105891 P28482 Mitogen-activated protein kinase 1 None 19953 nM Potency
TKC106074 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC106212 P28482 Mitogen-activated protein kinase 1 None 282 nM Potency
TKC106422 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC107086 P28482 Mitogen-activated protein kinase 1 None 31623 nM Potency
TKC107201 P28482 Mitogen-activated protein kinase 1 None 22387 nM Potency
TKC107525 P28482 Mitogen-activated protein kinase 1 None 31623 nM Potency
TKC107627 P28482 Mitogen-activated protein kinase 1 None 15849 nM Potency
TKC108295 P28482 Mitogen-activated protein kinase 1 None 12589 nM Potency
TKC108473 P28482 Mitogen-activated protein kinase 1 None 11220 nM Potency
TKC108555 P28482 Mitogen-activated protein kinase 1 None 10000 nM Potency
TKC108732 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC112745 P28482 Mitogen-activated protein kinase 1 None 31623 nM Potency
TKC112747 P28482 Mitogen-activated protein kinase 1 None 126 nM Potency
TKC112759 P28482 Mitogen-activated protein kinase 1 None 31623 nM Potency
TKC112784 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC113125 P28482 Mitogen-activated protein kinase 1 None 22387 nM Potency
TKC114819 P28482 Mitogen-activated protein kinase 1 None 19953 nM Potency
TKC118419 P28482 Mitogen-activated protein kinase 1 None 90 % Activity
TKC122892 P28482 Mitogen-activated protein kinase 1 None 25119 nM Potency
TKC134702 P28482 Mitogen-activated protein kinase 1 None 31623 nM Potency
TKC135961 P28482 Mitogen-activated protein kinase 1 None 5012 nM Potency
TKC136852 P28482 Mitogen-activated protein kinase 1 None 1413 nM Potency
TKC140757 P28482 Mitogen-activated protein kinase 1 None 28184 nM Potency
TKC148482 P28482 Mitogen-activated protein kinase 1 None 159 nM Potency
TKC149827 P28482 Mitogen-activated protein kinase 1 None 19953 nM Potency
TKC151571 P28482 Mitogen-activated protein kinase 1 None 3981 nM Potency
TKC151758 P28482 Mitogen-activated protein kinase 1 None 31623 nM Potency
TKC206688 P28482 Mitogen-activated protein kinase 1 None 3162 nM Potency
TKC206760 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC206770 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC206781 P28482 Mitogen-activated protein kinase 1 None 39811 nM Potency
TKC206812 P28482 Mitogen-activated protein kinase 1 None 31623 nM Potency
TKC206816 P28482 Mitogen-activated protein kinase 1 None 14125 nM Potency
TKC206901 P28482 Mitogen-activated protein kinase 1 None 7943 nM Potency
TKC207103 P28482 Mitogen-activated protein kinase 1 None 25119 nM Potency
TKC020967 P29466 Caspase-1 None 1080 nM IC50
TKC035272 P29466 Caspase-1 None 12589 nM Potency
TKC035272 P29466 Caspase-1 None 1230 nM IC50
TKC036497 P29466 Caspase-1 None 100000 nM IC50
TKC042585 P29466 Caspase-1 None 30000 nM MIC50
TKC042586 P29466 Caspase-1 None 30000 nM MIC50
TKC042587 P29466 Caspase-1 None 30000 nM MIC50
TKC096499 P29466 Caspase-1 None 90000 nM IC50
TKC149924 P29466 Caspase-1 None 4 /s Kinact
TKC027341 P34972 Cannabinoid receptor 2 None 257 nM Ki
TKC027353 P34972 Cannabinoid receptor 2 None 372 nM Ki
TKC027353 P34972 Cannabinoid receptor 2 None 229 nM Ki
TKC027353 P34972 Cannabinoid receptor 2 None 2860 nM Ki
TKC027353 P34972 Cannabinoid receptor 2 None 10000 nM Ki
TKC027353 P34972 Cannabinoid receptor 2 None 2.88E+12 nM Ki
TKC027356 P34972 Cannabinoid receptor 2 None 574 nM Ki
TKC027364 P34972 Cannabinoid receptor 2 None 153 nM Ki
TKC027373 P34972 Cannabinoid receptor 2 None 16 nM Ki
TKC027373 P34972 Cannabinoid receptor 2 None 126 nM Ki
TKC027373 P34972 Cannabinoid receptor 2 None 96 nM Ki
TKC027373 P34972 Cannabinoid receptor 2 None 95499258602 nM Ki
TKC027397 P34972 Cannabinoid receptor 2 None 4780 nM EC50
TKC095132 P34972 Cannabinoid receptor 2 None 0 nM Ki
TKC095132 P34972 Cannabinoid receptor 2 None 150 nM Ki
TKC095132 P34972 Cannabinoid receptor 2 None 0.251189 nM EC50
TKC095197 P34972 Cannabinoid receptor 2 None 171 nM Ki
TKC146115 P34972 Cannabinoid receptor 2 None 150 nM Ki
TKC205544 P34972 Cannabinoid receptor 2 None 20 % Inhibition
TKC037534 P35228 Nitric oxide synthase, inducible None 99 % Inhibition
TKC060880 P35228 Nitric oxide synthase, inducible None 37000 nM IC50
TKC077689 P35228 Nitric oxide synthase, inducible None >40000 nM IC50
TKC206319 P35228 Nitric oxide synthase, inducible None 100 % Inhibition
TKC008359 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC010020 P35354 Prostaglandin G/H synthase 2 None 61 % Inhibition
TKC010022 P35354 Prostaglandin G/H synthase 2 None 55 % Inhibition
TKC010023 P35354 Prostaglandin G/H synthase 2 None 57 % Inhibition
TKC010024 P35354 Prostaglandin G/H synthase 2 None 42 % Inhibition
TKC010025 P35354 Prostaglandin G/H synthase 2 None 78 % Inhibition
TKC010026 P35354 Prostaglandin G/H synthase 2 None 17 % Inhibition
TKC011599 P35354 Prostaglandin G/H synthase 2 None 64 % Inhibition
TKC012919 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC012941 P35354 Prostaglandin G/H synthase 2 None 8500 nM IC50
TKC012956 P35354 Prostaglandin G/H synthase 2 None 2200 nM IC50
TKC012962 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC015443 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC015459 P35354 Prostaglandin G/H synthase 2 None 2200 nM IC50
TKC015537 P35354 Prostaglandin G/H synthase 2 None 0 % Inhibition
TKC016794 P35354 Prostaglandin G/H synthase 2 None 40 nM IC50
TKC019436 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC019466 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC019819 P35354 Prostaglandin G/H synthase 2 None 35 % Inhibition
TKC019859 P35354 Prostaglandin G/H synthase 2 None <33 % Inhibition
TKC020479 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC020796 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC021940 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC022833 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC022834 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC022961 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC026245 P35354 Prostaglandin G/H synthase 2 None 2300 nM IC50
TKC027200 P35354 Prostaglandin G/H synthase 2 None 700 nM IC50
TKC028143 P35354 Prostaglandin G/H synthase 2 None 100 % Inhibition
TKC031202 P35354 Prostaglandin G/H synthase 2 None 3800 nM IC50
TKC031223 P35354 Prostaglandin G/H synthase 2 None 45 % Inhibition
TKC032234 P35354 Prostaglandin G/H synthase 2 None 400 nM IC50
TKC035208 P35354 Prostaglandin G/H synthase 2 None 7 uM IC60
TKC037534 P35354 Prostaglandin G/H synthase 2 None 97 % Inhibition
TKC038330 P35354 Prostaglandin G/H synthase 2 None 2900 nM IC50
TKC041884 P35354 Prostaglandin G/H synthase 2 None 18000 nM IC50
TKC043993 P35354 Prostaglandin G/H synthase 2 None 98 % Inhibition
TKC045188 P35354 Prostaglandin G/H synthase 2 None 98 % Inhibition
TKC048282 P35354 Prostaglandin G/H synthase 2 None 370 nM IC50
TKC049750 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC049818 P35354 Prostaglandin G/H synthase 2 None 5 ug IC50
TKC051154 P35354 Prostaglandin G/H synthase 2 None >61 % Activity
TKC054011 P35354 Prostaglandin G/H synthase 2 None 9000 nM IC50
TKC054031 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC054081 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC054090 P35354 Prostaglandin G/H synthase 2 None 8900 nM IC50
TKC054099 P35354 Prostaglandin G/H synthase 2 None 7800 nM IC50
TKC054100 P35354 Prostaglandin G/H synthase 2 None 7900 nM IC50
TKC054101 P35354 Prostaglandin G/H synthase 2 None 8800 nM IC50
TKC054240 P35354 Prostaglandin G/H synthase 2 None 6700 nM IC50
TKC054241 P35354 Prostaglandin G/H synthase 2 None 6100 nM IC50
TKC056482 P35354 Prostaglandin G/H synthase 2 None 40000 nM IC50
TKC056482 P35354 Prostaglandin G/H synthase 2 None 86000 nM IC50
TKC056482 P35354 Prostaglandin G/H synthase 2 None 130000 nM IC50
TKC057308 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC058811 P35354 Prostaglandin G/H synthase 2 None >85 % Activity
TKC058812 P35354 Prostaglandin G/H synthase 2 None >78 % Activity
TKC060184 P35354 Prostaglandin G/H synthase 2 None 8500 nM IC50
TKC060216 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC060284 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC060302 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC060303 P35354 Prostaglandin G/H synthase 2 None 7200 nM IC50
TKC060304 P35354 Prostaglandin G/H synthase 2 None 7600 nM IC50
TKC060399 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC060602 P35354 Prostaglandin G/H synthase 2 None 6700 nM IC50
TKC061939 P35354 Prostaglandin G/H synthase 2 None >10000 nM IC50
TKC061968 P35354 Prostaglandin G/H synthase 2 None >10000 nM IC50
TKC061969 P35354 Prostaglandin G/H synthase 2 None >10000 nM IC50
TKC064374 P35354 Prostaglandin G/H synthase 2 None >73 % Activity
TKC064407 P35354 Prostaglandin G/H synthase 2 None >78 % Activity
TKC065375 P35354 Prostaglandin G/H synthase 2 None >70 % Activity
TKC066954 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC070952 P35354 Prostaglandin G/H synthase 2 None >100000 nM IC50
TKC071010 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC071640 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC076350 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC077689 P35354 Prostaglandin G/H synthase 2 None 40000 nM IC50
TKC077689 P35354 Prostaglandin G/H synthase 2 None 295000 nM IC50
TKC077689 P35354 Prostaglandin G/H synthase 2 None 295000 nM IC50
TKC077689 P35354 Prostaglandin G/H synthase 2 None 87000 nM IC50
TKC077703 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC078194 P35354 Prostaglandin G/H synthase 2 None >74 % Activity
TKC085168 P35354 Prostaglandin G/H synthase 2 None <60 % Inhibition
TKC088678 P35354 Prostaglandin G/H synthase 2 None >72 % Activity
TKC095276 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC095567 P35354 Prostaglandin G/H synthase 2 None >10000 nM IC50
TKC110247 P35354 Prostaglandin G/H synthase 2 None >10 ug.mL-1 IC50
TKC113936 P35354 Prostaglandin G/H synthase 2 None 60 % Inhibition
TKC122543 P35354 Prostaglandin G/H synthase 2 None 30 % Inhibition
TKC123028 P35354 Prostaglandin G/H synthase 2 None >72 % Activity
TKC129152 P35354 Prostaglandin G/H synthase 2 None >100000 nM IC50
TKC130084 P35354 Prostaglandin G/H synthase 2 None 37 % Inhibition
TKC130119 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC130223 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC130577 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC130901 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC135264 P35354 Prostaglandin G/H synthase 2 None 400 nM IC50
TKC135559 P35354 Prostaglandin G/H synthase 2 None 4600 nM IC50
TKC139036 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC139322 P35354 Prostaglandin G/H synthase 2 None >82 % Activity
TKC139366 P35354 Prostaglandin G/H synthase 2 None 40000 nM IC50
TKC140627 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC141365 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC141401 P35354 Prostaglandin G/H synthase 2 None >75 % Activity
TKC141499 P35354 Prostaglandin G/H synthase 2 None >87 % Activity
TKC141601 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC141602 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC141622 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC141805 P35354 Prostaglandin G/H synthase 2 None 40000 nM IC50
TKC142150 P35354 Prostaglandin G/H synthase 2 None 450000 nM IC50
TKC142203 P35354 Prostaglandin G/H synthase 2 None >10000 nM IC50
TKC142208 P35354 Prostaglandin G/H synthase 2 None >10000 nM IC50
TKC142849 P35354 Prostaglandin G/H synthase 2 None >69 % Activity
TKC142897 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC142922 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC143527 P35354 Prostaglandin G/H synthase 2 None 97 % Inhibition
TKC143539 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC143641 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC145295 P35354 Prostaglandin G/H synthase 2 None 22 % Inhibition
TKC145848 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC145932 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC145968 P35354 Prostaglandin G/H synthase 2 None >94 % Activity
TKC146116 P35354 Prostaglandin G/H synthase 2 None >5.0e+4 nM IC50
TKC146774 P35354 Prostaglandin G/H synthase 2 None >78 % Activity
TKC146857 P35354 Prostaglandin G/H synthase 2 None 600 nM IC50
TKC149251 P35354 Prostaglandin G/H synthase 2 None 1100 nM IC50
TKC149759 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC149924 P35354 Prostaglandin G/H synthase 2 None 800 nM IC50
TKC149926 P35354 Prostaglandin G/H synthase 2 None 800 nM IC50
TKC150635 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC150706 P35354 Prostaglandin G/H synthase 2 None >76 % Activity
TKC150907 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC151280 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC151284 P35354 Prostaglandin G/H synthase 2 None 33 % Inhibition
TKC151765 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC152742 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC152813 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC156345 P35354 Prostaglandin G/H synthase 2 None 25 % Inhibition
TKC156572 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC156716 P35354 Prostaglandin G/H synthase 2 None 2200 nM IC50
TKC170277 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC172853 P35354 Prostaglandin G/H synthase 2 None 4700 nM IC50
TKC174442 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC205509 P35354 Prostaglandin G/H synthase 2 None 540000 nM IC50
TKC205699 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC205700 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC206319 P35354 Prostaglandin G/H synthase 2 None 99 % Inhibition
TKC205544 P35367 Histamine H1 receptor None 30 % Inhibition
TKC206544 P35367 Histamine H1 receptor None >10000 nM Ki
TKC002194 P41143 Delta-type opioid receptor None 2830 nM Ke
TKC005708 P41143 Delta-type opioid receptor None >10000 nM Ki
TKC045774 P41143 Delta-type opioid receptor None >64582 nM EC50
TKC093001 P41143 Delta-type opioid receptor None 10000 nM Ki
TKC093006 P41143 Delta-type opioid receptor None 6690 nM Ki
TKC093006 P41143 Delta-type opioid receptor None 6690 nM Ki
TKC093010 P41143 Delta-type opioid receptor None 1017 nM Ki
TKC093012 P41143 Delta-type opioid receptor None 2840 nM Ki
TKC101289 P41143 Delta-type opioid receptor None >5000 nM Ki
TKC101290 P41143 Delta-type opioid receptor None >5000 nM Ki
TKC104953 P41143 Delta-type opioid receptor None 964 nM Ke
TKC105684 P41143 Delta-type opioid receptor None >10000 nM Ki
TKC105685 P41143 Delta-type opioid receptor None >10000 nM Ki
TKC109881 P41143 Delta-type opioid receptor None >92466 nM EC50
TKC109881 P41143 Delta-type opioid receptor None >92466 nM EC50
TKC156630 P41143 Delta-type opioid receptor None >10000 nM Ki
TKC206544 P41143 Delta-type opioid receptor None 3990 nM Ki
TKC206544 P41143 Delta-type opioid receptor None >10000 nM Ki
TKC206544 P41143 Delta-type opioid receptor None 5790 nM Ki
TKC206544 P41143 Delta-type opioid receptor None 5790 nM Ki
TKC206544 P41143 Delta-type opioid receptor None >10000 nM Ki
TKC206544 P41143 Delta-type opioid receptor None >10000 nM Ki
TKC206544 P41143 Delta-type opioid receptor None >10000 nM Ki
TKC206544 P41143 Delta-type opioid receptor None >10000 nM Ki
TKC025058 P42336 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform None 100 nM IC50
TKC118380 P42336 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform None 1 nM IC50
TKC118419 P42336 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform None 1 nM IC50
TKC118419 P42336 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform None 12 nM IC50
TKC118419 P42336 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform None 17.6 nM IC50
TKC118419 P42336 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform None 120 nM Ki
TKC118419 P42336 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform None 12 nM IC50
TKC118419 P42336 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform None 12 nM IC50
TKC118419 P42336 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform None 13 nM IC50
TKC118419 P42336 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform None 1 nM IC50
TKC118419 P42336 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform None 5.4 nM Kd
TKC108557 P43405 Tyrosine-protein kinase SYK None 0.2 nM IC50
TKC025058 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 1000 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 5 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 19 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 55 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 55000 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 89 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 5 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 15 nM Kd
TKC013304 P51449 Nuclear receptor ROR-gamma None 66824 nM Potency
TKC013753 P51449 Nuclear receptor ROR-gamma None 29849 nM Potency
TKC013755 P51449 Nuclear receptor ROR-gamma None 14000 nM EC50
TKC021977 P51449 Nuclear receptor ROR-gamma None 42163 nM Potency
TKC022931 P51449 Nuclear receptor ROR-gamma None 84 nM Potency
TKC056482 P51449 Nuclear receptor ROR-gamma None 130 nM IC50
TKC066169 P51449 Nuclear receptor ROR-gamma None 33492 nM Potency
TKC075769 P51449 Nuclear receptor ROR-gamma None 1980 nM IC50
TKC075769 P51449 Nuclear receptor ROR-gamma None 109 nM Kd
TKC075769 P51449 Nuclear receptor ROR-gamma None 2000 nM IC50
TKC083807 P51449 Nuclear receptor ROR-gamma None 10591 nM Potency
TKC087664 P51449 Nuclear receptor ROR-gamma None 47308 nM Potency
TKC087991 P51449 Nuclear receptor ROR-gamma None 21132 nM Potency
TKC088230 P51449 Nuclear receptor ROR-gamma None 1333 nM Potency
TKC088231 P51449 Nuclear receptor ROR-gamma None 23710 nM Potency
TKC092297 P51449 Nuclear receptor ROR-gamma None 26603 nM Potency
TKC096012 P51449 Nuclear receptor ROR-gamma None 200 nM IC50
TKC096012 P51449 Nuclear receptor ROR-gamma None 18000 nM EC50
TKC097944 P51449 Nuclear receptor ROR-gamma None 4216 nM Potency
TKC102407 P51449 Nuclear receptor ROR-gamma None 21132 nM Potency
TKC107086 P51449 Nuclear receptor ROR-gamma None 3758 nM Potency
TKC115268 P51449 Nuclear receptor ROR-gamma None 37578 nM Potency
TKC118648 P51449 Nuclear receptor ROR-gamma None 80 nM EC50
TKC118652 P51449 Nuclear receptor ROR-gamma None 110 nM EC50
TKC118929 P51449 Nuclear receptor ROR-gamma None 10 nM Ki
TKC118938 P51449 Nuclear receptor ROR-gamma None 10 nM Ki
TKC122884 P51449 Nuclear receptor ROR-gamma None 20 nM EC50
TKC136411 P51449 Nuclear receptor ROR-gamma None 37578 nM Potency
TKC151274 P51449 Nuclear receptor ROR-gamma None 60 nM Potency
TKC206457 P51449 Nuclear receptor ROR-gamma None 20 nM EC50
TKC206457 P51449 Nuclear receptor ROR-gamma None 20 nM EC50
TKC206457 P51449 Nuclear receptor ROR-gamma None 20 nM EC50
TKC206458 P51449 Nuclear receptor ROR-gamma None 20 nM EC50
TKC206459 P51449 Nuclear receptor ROR-gamma None 7 degrees C T
TKC206672 P51449 Nuclear receptor ROR-gamma None 42163 nM Potency
TKC206688 P51449 Nuclear receptor ROR-gamma None 23710 nM Potency
TKC206759 P51449 Nuclear receptor ROR-gamma None 26603 nM Potency
TKC206760 P51449 Nuclear receptor ROR-gamma None 74978 nM Potency
TKC206770 P51449 Nuclear receptor ROR-gamma None 33492 nM Potency
TKC206812 P51449 Nuclear receptor ROR-gamma None 47308 nM Potency
TKC206816 P51449 Nuclear receptor ROR-gamma None 8413 nM Potency
TKC206915 P51449 Nuclear receptor ROR-gamma None 10 nM Ki
TKC046294 P51681 C-C chemokine receptor type 5 None 40000 nM IC50
TKC046601 P51681 C-C chemokine receptor type 5 None 32000 nM IC50
TKC054684 P51681 C-C chemokine receptor type 5 None 5100 nM Ki
TKC054723 P51681 C-C chemokine receptor type 5 None 30000 nM Ki
TKC137374 P51681 C-C chemokine receptor type 5 None 9000 nM IC50
TKC009486 P52333 Tyrosine-protein kinase JAK3 None >100 nM IC50
TKC009499 P52333 Tyrosine-protein kinase JAK3 None >100 nM IC50
TKC011761 P52333 Tyrosine-protein kinase JAK3 None 100 nM IC50
TKC031094 P52333 Tyrosine-protein kinase JAK3 None >25 % Inhibition
TKC107626 P52333 Tyrosine-protein kinase JAK3 None 25 % Inhibition
TKC120591 P52333 Tyrosine-protein kinase JAK3 None >100 nM IC50
TKC120592 P52333 Tyrosine-protein kinase JAK3 None >100 nM IC50
TKC120593 P52333 Tyrosine-protein kinase JAK3 None >100 nM IC50
TKC134702 P52333 Tyrosine-protein kinase JAK3 None 25 % Inhibition
TKC151713 P52333 Tyrosine-protein kinase JAK3 None 25 % Inhibition
TKC118419 P53778 Mitogen-activated protein kinase 12 None 75 % Inhibition
TKC021620 P60568 Interleukin-2 None 3 nM Kd
TKC116180 P60568 Interleukin-2 None 0 nM Kd
TKC038192 Q02127 Dihydroorotate dehydrogenase None 3 % Inhibition
TKC039868 Q02127 Dihydroorotate dehydrogenase None 0 % Inhibition
TKC043742 Q02127 Dihydroorotate dehydrogenase None 0 % Inhibition
TKC079733 Q02127 Dihydroorotate dehydrogenase None 28 % Inhibition
TKC136181 Q02127 Dihydroorotate dehydrogenase None 12 % Inhibition
TKC028446 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 11400 nM IC50
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 1356 nM IC50
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 162 nM Ki
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 180 nM Ki
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 280 nM Ki
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 310 nM Ki
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 640 nM Ki
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 180 nM Ki
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 180 nM Ki
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 200 nM Ki
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 6543 nM Ki
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 2324 nM Kd
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 190 nM Ki
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 2650 nM Kd
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 190 nM Ki
TKC035272 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 180 nM Ki
TKC039229 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 12900 nM Ki
TKC105178 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 14400 nM Ki
TKC105179 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 4200 nM Ki
TKC134945 Q07820 Induced myeloid leukemia cell differentiation protein Mcl-1 None 8600 nM Ki
TKC021262 Q07869 Peroxisome proliferator-activated receptor alpha None 19500 nM EC50
TKC021666 Q07869 Peroxisome proliferator-activated receptor alpha None 28 % Activity
TKC021674 Q07869 Peroxisome proliferator-activated receptor alpha None 25 % Activity
TKC035272 Q07869 Peroxisome proliferator-activated receptor alpha None 15849 nM Potency
TKC056482 Q07869 Peroxisome proliferator-activated receptor alpha None 259 % Activity
TKC057132 Q07869 Peroxisome proliferator-activated receptor alpha None 12589 nM Potency
TKC088526 Q07869 Peroxisome proliferator-activated receptor alpha None 12 % Activity
TKC100644 Q07869 Peroxisome proliferator-activated receptor alpha None 8913 nM Potency
TKC108536 Q07869 Peroxisome proliferator-activated receptor alpha None 50119 nM Potency
TKC110634 Q07869 Peroxisome proliferator-activated receptor alpha None 309 % Activity
TKC110635 Q07869 Peroxisome proliferator-activated receptor alpha None 289 % Activity
TKC170559 Q07869 Peroxisome proliferator-activated receptor alpha None 1000 nM EC50
TKC171329 Q07869 Peroxisome proliferator-activated receptor alpha None 184 nM EC50
TKC206812 Q07869 Peroxisome proliferator-activated receptor alpha None >20000 nM IC50
TKC051063 Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D None >20000 nM IC50
TKC104905 Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D None 245 nM IC50
TKC104906 Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D None 542 nM IC50
TKC146367 Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D None >20000 nM IC50
TKC109319 Q15125 3-beta-hydroxysteroid-Delta None 6800 nM IC50
TKC109355 Q15125 3-beta-hydroxysteroid-Delta None 600 nM IC50
TKC112505 Q15125 3-beta-hydroxysteroid-Delta None 400 nM IC50
TKC114545 Q15125 3-beta-hydroxysteroid-Delta None 600 nM IC50
TKC114551 Q15125 3-beta-hydroxysteroid-Delta None >20000 nM IC50
TKC206688 Q15125 3-beta-hydroxysteroid-Delta None >100000 nM Ki
TKC206759 Q15125 3-beta-hydroxysteroid-Delta None >100000 nM Ki
TKC206816 Q15125 3-beta-hydroxysteroid-Delta None >100000 nM Ki
TKC023254 Q15722 Leukotriene B4 receptor 1 None 44500 nM IC50
TKC118419 Q15759 Mitogen-activated protein kinase 11 None 74 % Inhibition
TKC087988 Q16539 Mitogen-activated protein kinase 14 None 2529 nM IC50
TKC118419 Q16539 Mitogen-activated protein kinase 14 None 86 % Inhibition
TKC105649 Q16881 Thioredoxin reductase 1, cytoplasmic None 280 nM Ki
TKC118419 Q8IW41 MAP kinase-activated protein kinase 5 None 69 % Activity
TKC013738 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 24 nM Ki
TKC013738 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 23 nM Ki
TKC013738 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 14 nM Ki
TKC013739 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 129 nM Ki
TKC023433 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 5000 nM IC50
TKC027364 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 1300 nM EC50
TKC027373 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 6200 nM EC50
TKC027397 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 6600 nM EC50
TKC033765 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 176 % Activity
TKC034016 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 94 % Activity
TKC036488 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 22 % Activity
TKC074866 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None >102 uM Activity
TKC090445 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 0 nM Ki
TKC092268 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 0 nM EC50
TKC092268 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 0.48 nM Ki
TKC092268 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 1.2 nM Ki
TKC092268 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 19 nM EC50
TKC092268 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 0.92 nM EC50
TKC098861 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 115 % Activity
TKC116435 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 1400 nM IC50
TKC122664 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 31 % Activity
TKC146124 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 45 % Activity
TKC151092 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 115 % Activity
TKC205687 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 1 nM Kd
TKC206945 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 6 nM Ki
TKC206945 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 4000 nM IC50
TKC206945 Q8NER1 Transient receptor potential cation channel subfamily V member 1 None 5.9 nM Ki
TKC048132 Q96EB6 NAD-dependent protein deacetylase sirtuin-1 None 28 % Activity
TKC048343 Q96EB6 NAD-dependent protein deacetylase sirtuin-1 None 88 % Activity
TKC048346 Q96EB6 NAD-dependent protein deacetylase sirtuin-1 None 8 % Activity
TKC030239 Q9UNQ0 Broad substrate specificity ATP-binding cassette transporter ABCG2 None 70 % Activity
TKC075756 Q9UNQ0 Broad substrate specificity ATP-binding cassette transporter ABCG2 None 9700 nM IC50
TKC111738 Q9UNQ0 Broad substrate specificity ATP-binding cassette transporter ABCG2 None 3000 nM IC50
TKC112787 Q9UNQ0 Broad substrate specificity ATP-binding cassette transporter ABCG2 None 20 % Activity
TKC112788 Q9UNQ0 Broad substrate specificity ATP-binding cassette transporter ABCG2 None 30 % Activity
TKC206758 Q9UNQ0 Broad substrate specificity ATP-binding cassette transporter ABCG2 None 50 % Activity
TKC206816 Q9UNQ0 Broad substrate specificity ATP-binding cassette transporter ABCG2 None 125893 nM IC50
TKC206849 Q9UNQ0 Broad substrate specificity ATP-binding cassette transporter ABCG2 None 70 % Activity