Basic Information

Name [ICD-11: BA00-BE2Z]
Protein Number 36
Molecule Number 462

Active subnetwork

Terpenoid-protein target Activity Association

ID Uniport Pref_name Gene name value unit type
TKC001786 O43353 Receptor-interacting serine/threonine-protein kinase 2 None 7034 nM IC50
TKC041149 O43353 Receptor-interacting serine/threonine-protein kinase 2 None >49751 nM IC50
TKC041436 O43353 Receptor-interacting serine/threonine-protein kinase 2 None >49791 nM IC50
TKC041460 O43353 Receptor-interacting serine/threonine-protein kinase 2 None >49756 nM IC50
TKC078094 O43353 Receptor-interacting serine/threonine-protein kinase 2 None >49729 nM IC50
TKC082378 O43353 Receptor-interacting serine/threonine-protein kinase 2 None 1188 nM IC50
TKC090566 O43353 Receptor-interacting serine/threonine-protein kinase 2 None >49751 nM IC50
TKC113063 O43353 Receptor-interacting serine/threonine-protein kinase 2 None 2654 nM IC50
TKC135702 O43353 Receptor-interacting serine/threonine-protein kinase 2 None >49761 nM IC50
TKC159332 O43353 Receptor-interacting serine/threonine-protein kinase 2 None 3095 nM IC50
TKC206362 O43353 Receptor-interacting serine/threonine-protein kinase 2 None 2296 nM IC50
TKC001732 O43451 Maltase-glucoamylase, intestinal None 17 % Inhibition
TKC001930 O43451 Maltase-glucoamylase, intestinal None 17 % Inhibition
TKC028968 O43451 Maltase-glucoamylase, intestinal None 78 % Inhibition
TKC045338 O43451 Maltase-glucoamylase, intestinal None 89 % Inhibition
TKC045339 O43451 Maltase-glucoamylase, intestinal None 27 % Inhibition
TKC078822 O43451 Maltase-glucoamylase, intestinal None 100000 nM IC50
TKC078823 O43451 Maltase-glucoamylase, intestinal None 11000 nM IC50
TKC078824 O43451 Maltase-glucoamylase, intestinal None 36000 nM IC50
TKC078825 O43451 Maltase-glucoamylase, intestinal None 25000 nM IC50
TKC078826 O43451 Maltase-glucoamylase, intestinal None 28000 nM IC50
TKC028037 O76074 cGMP-specific 3',5'-cyclic phosphodiesterase None -7 % Inhibition
TKC104905 O76074 cGMP-specific 3',5'-cyclic phosphodiesterase None 3810 nM IC50
TKC151761 P00519 Tyrosine-protein kinase ABL1 None >10000 nM IC50
TKC200866 P00519 Tyrosine-protein kinase ABL1 None >10000 nM IC50
TKC055903 P00734 Prothrombin None 4 nM IC50
TKC055903 P00734 Prothrombin None 50 nM IC50
TKC064786 P00734 Prothrombin None 130 nM IC50
TKC064787 P00734 Prothrombin None 70 nM IC50
TKC101989 P00734 Prothrombin None 4000 nM IC50
TKC106074 P00734 Prothrombin None >50000 nM IC50
TKC106074 P00734 Prothrombin None >50000 nM IC50
TKC122980 P00734 Prothrombin None 9200 nM IC50
TKC139119 P00734 Prothrombin None 90 nM IC50
TKC141433 P00734 Prothrombin None 18 nM IC50
TKC056231 P00797 Renin None >2046000 nM IC50
TKC061915 P00797 Renin None >2117000 nM IC50
TKC061947 P00797 Renin None >1990000 nM IC50
TKC088747 P00797 Renin None >1663000 nM IC50
TKC008187 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 30200 nM IC50
TKC023515 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 53 % Inhibition
TKC025574 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 52 % Inhibition
TKC026893 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 21 % Inhibition
TKC026895 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 61 % Inhibition
TKC057019 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 22300 nM IC50
TKC100777 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 30 % Inhibition
TKC101031 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 1500 nM IC50
TKC101538 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 39 % Inhibition
TKC101847 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 1000 nM IC50
TKC103703 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 40 % Inhibition
TKC137314 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 8400 nM IC50
TKC138471 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 21700 nM IC50
TKC017639 P04054 Phospholipase A2 None 95 % Activity
TKC017706 P04054 Phospholipase A2 None 5 % Activity
TKC045776 P04054 Phospholipase A2 None 1600 nM IC50
TKC045777 P04054 Phospholipase A2 None 3700 nM IC50
TKC045872 P04054 Phospholipase A2 None 44 % Activity
TKC046211 P04054 Phospholipase A2 None 3900 nM IC50
TKC046211 P04054 Phospholipase A2 None 13000 nM IC50
TKC055219 P04054 Phospholipase A2 None 2040 nM IC50
TKC055219 P04054 Phospholipase A2 None 2040 nM IC50
TKC077689 P04054 Phospholipase A2 None 3000 nM IC50
TKC105149 P04054 Phospholipase A2 None 8 % Activity
TKC106090 P04054 Phospholipase A2 None 95 % Activity
TKC106091 P04054 Phospholipase A2 None 90 % Activity
TKC106240 P04054 Phospholipase A2 None 5 % Activity
TKC109622 P04054 Phospholipase A2 None 10000 nM Kd
TKC110322 P04054 Phospholipase A2 None 67 % Inhibition
TKC110427 P04054 Phospholipase A2 None 13800 nM IC50
TKC112787 P04054 Phospholipase A2 None 40 % Activity
TKC115260 P04054 Phospholipase A2 None 55 % Inhibition
TKC146194 P04054 Phospholipase A2 None 5 % Activity
TKC151364 P04054 Phospholipase A2 None 30 % Activity
TKC152148 P04054 Phospholipase A2 None 47 % Inhibition
TKC206812 P04054 Phospholipase A2 None 35 % Activity
TKC206849 P04054 Phospholipase A2 None 80 % Activity
TKC206884 P04054 Phospholipase A2 None 150000 nM Kd
TKC151761 P05106 Integrin beta-3 None 34 nM IC50
TKC200866 P05106 Integrin beta-3 None 34 nM IC50
TKC026717 P06239 Tyrosine-protein kinase Lck None 80 ug.mL-1 IC50
TKC046110 P06239 Tyrosine-protein kinase Lck None 45 % Activity
TKC105249 P06239 Tyrosine-protein kinase Lck None 92 ug.mL-1 IC50
TKC111609 P06239 Tyrosine-protein kinase Lck None 47 % Activity
TKC111658 P06239 Tyrosine-protein kinase Lck None 42 % Activity
TKC118419 P06239 Tyrosine-protein kinase Lck None 95 % Inhibition
TKC032962 P07550 Beta-2 adrenergic receptor None 32643 nM Potency
TKC087533 P07550 Beta-2 adrenergic receptor None 631 nM Potency
TKC095493 P07550 Beta-2 adrenergic receptor None 28184 nM Potency
TKC109493 P07550 Beta-2 adrenergic receptor None 6513 nM Potency
TKC151237 P07550 Beta-2 adrenergic receptor None 28184 nM Potency
TKC206544 P08172 Muscarinic acetylcholine receptor M2 None >10000 nM Ki
TKC030239 P08235 Mineralocorticoid receptor None 2.9 nM EC50
TKC030239 P08235 Mineralocorticoid receptor None 0.5 nM Kd
TKC114511 P08235 Mineralocorticoid receptor None 1880 nM IC50
TKC206688 P08235 Mineralocorticoid receptor None 1 nM Kd
TKC206812 P08235 Mineralocorticoid receptor None 39 nM Ki
TKC206816 P08235 Mineralocorticoid receptor None 0 nM Kd
TKC206816 P08235 Mineralocorticoid receptor None 14 nM IC50
TKC206816 P08235 Mineralocorticoid receptor None 14 nM IC50
TKC206816 P08235 Mineralocorticoid receptor None 14 nM IC50
TKC206816 P08235 Mineralocorticoid receptor None 14 nM IC50
TKC206816 P08235 Mineralocorticoid receptor None >14 nM IC50
TKC020712 P08581 Hepatocyte growth factor receptor None >20000 nM IC50
TKC024886 P08581 Hepatocyte growth factor receptor None 3120 nM IC50
TKC025690 P08581 Hepatocyte growth factor receptor None >100000 nM IC50
TKC033871 P08581 Hepatocyte growth factor receptor None 50000 nM IC50
TKC082039 P08581 Hepatocyte growth factor receptor None 5500 nM IC50
TKC115259 P08581 Hepatocyte growth factor receptor None 34000 nM IC50
TKC115261 P08581 Hepatocyte growth factor receptor None 47600 nM IC50
TKC115272 P08581 Hepatocyte growth factor receptor None >100000 nM IC50
TKC115273 P08581 Hepatocyte growth factor receptor None 27500 nM IC50
TKC152148 P08581 Hepatocyte growth factor receptor None 78000 nM IC50
TKC152157 P08581 Hepatocyte growth factor receptor None 71500 nM IC50
TKC174547 P08581 Hepatocyte growth factor receptor None >100000 nM IC50
TKC020117 P09917 Polyunsaturated fatty acid 5-lipoxygenase None -67 % Inhibition
TKC024485 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >50000 nM IC50
TKC024587 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 600 nM IC50
TKC024956 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 18000 nM IC50
TKC024992 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 450 nM IC50
TKC024993 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 14000 nM IC50
TKC025965 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >150000 nM IC50
TKC026303 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 4600 nM IC50
TKC026309 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 680 nM IC50
TKC027255 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >67 % Activity
TKC034201 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >200000 nM IC50
TKC040026 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 72 % Inhibition
TKC051154 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 2700 nM IC50
TKC056482 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >64 % Activity
TKC058811 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 42000 nM IC50
TKC058812 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >93 % Activity
TKC064374 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 42000 nM IC50
TKC064407 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >72 % Activity
TKC065375 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >70 % Activity
TKC071640 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >60 % Activity
TKC076350 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 100 % Activity
TKC077689 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 100 % Activity
TKC077703 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >86 % Activity
TKC078194 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 31800 nM IC50
TKC082039 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 48 % Inhibition
TKC088678 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 24800 nM IC50
TKC089448 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 35 % Inhibition
TKC094647 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 97 % Activity
TKC107943 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 2000 nM IC50
TKC123028 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 30400 nM IC50
TKC124303 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 750 nM IC50
TKC133309 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >200000 nM IC50
TKC133656 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 25100 nM IC50
TKC134278 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >200000 nM IC50
TKC139322 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >67 % Activity
TKC139366 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 3000 nM IC50
TKC141401 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 42000 nM IC50
TKC141499 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 25700 nM IC50
TKC141805 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >53 % Activity
TKC142849 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >70 % Activity
TKC142897 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 30600 nM IC50
TKC142922 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >61 % Activity
TKC143539 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 100 % Activity
TKC145848 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 42000 nM IC50
TKC145932 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >56 % Activity
TKC145968 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 100 % Activity
TKC146774 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >63 % Activity
TKC149759 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >73 % Activity
TKC150706 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >62 % Activity
TKC001669 P10275 Androgen receptor None 260 nM IC50
TKC006934 P10275 Androgen receptor None 50119 nM Potency
TKC013304 P10275 Androgen receptor None 70795 nM Potency
TKC019571 P10275 Androgen receptor None 19953 nM Potency
TKC021325 P10275 Androgen receptor None 31623 nM Potency
TKC021332 P10275 Androgen receptor None 31623 nM Potency
TKC023246 P10275 Androgen receptor None 449 nM IC50
TKC030239 P10275 Androgen receptor None 14 nM Potency
TKC035272 P10275 Androgen receptor None 15849 nM Potency
TKC056140 P10275 Androgen receptor None 50 % Activity
TKC066169 P10275 Androgen receptor None 3981 nM Potency
TKC074867 P10275 Androgen receptor None 28184 nM Potency
TKC075769 P10275 Androgen receptor None 355 nM Potency
TKC079001 P10275 Androgen receptor None 1 nM Potency
TKC096012 P10275 Androgen receptor None 178 nM Potency
TKC100644 P10275 Androgen receptor None 35481 nM Potency
TKC102407 P10275 Androgen receptor None 44668 nM Potency
TKC106878 P10275 Androgen receptor None 238 nM IC50
TKC107086 P10275 Androgen receptor None 17783 nM Potency
TKC107735 P10275 Androgen receptor None 3981 nM Potency
TKC111738 P10275 Androgen receptor None 17783 nM Potency
TKC112923 P10275 Androgen receptor None 212 nM IC50
TKC114095 P10275 Androgen receptor None 1790 nM IC50
TKC114511 P10275 Androgen receptor None 315 nM Ki
TKC115268 P10275 Androgen receptor None 35481 nM Potency
TKC115284 P10275 Androgen receptor None 1 nM Ki
TKC117154 P10275 Androgen receptor None 580 nM IC50
TKC120161 P10275 Androgen receptor None 44668 nM Potency
TKC122884 P10275 Androgen receptor None 39811 nM Potency
TKC122892 P10275 Androgen receptor None 10000 nM IC50
TKC134780 P10275 Androgen receptor None 2 nM Potency
TKC147240 P10275 Androgen receptor None 50 % Activity
TKC206652 P10275 Androgen receptor None 50 nM Potency
TKC206688 P10275 Androgen receptor None 224 nM Potency
TKC206690 P10275 Androgen receptor None 36 nM Potency
TKC206759 P10275 Androgen receptor None 2 nM Potency
TKC206759 P10275 Androgen receptor None 3.9 nM IC50
TKC206759 P10275 Androgen receptor None 4.7 nM IC50
TKC206759 P10275 Androgen receptor None 4.2 nM IC50
TKC206759 P10275 Androgen receptor None 29 nM Ki
TKC206759 P10275 Androgen receptor None 1.1 nM EC50
TKC206759 P10275 Androgen receptor None 2.7 nM IC50
TKC206759 P10275 Androgen receptor None 2.7 nM IC50
TKC206759 P10275 Androgen receptor None 2.7 nM IC50
TKC206759 P10275 Androgen receptor None 30 nM IC50
TKC206759 P10275 Androgen receptor None 4.57 nM IC50
TKC206770 P10275 Androgen receptor None 224 nM Potency
TKC206779 P10275 Androgen receptor None 2 nM Potency
TKC206812 P10275 Androgen receptor None 220 nM IC50
TKC206816 P10275 Androgen receptor None 9 nM Ki
TKC206816 P10275 Androgen receptor None 8.5 nM Ki
TKC206816 P10275 Androgen receptor None 8.5 nM Ki
TKC206816 P10275 Androgen receptor None 8.5 nM Ki
TKC206816 P10275 Androgen receptor None 8.5 nM Ki
TKC206816 P10275 Androgen receptor None 37 nM IC50
TKC206816 P10275 Androgen receptor None 8.5 nM Ki
TKC206816 P10275 Androgen receptor None 35 nM Ki
TKC206816 P10275 Androgen receptor None 14 nM IC50
TKC066096 P11413 Glucose-6-phosphate 1-dehydrogenase None >80000 nM IC50
TKC109495 P11413 Glucose-6-phosphate 1-dehydrogenase None 15800 nM IC50
TKC109970 P11413 Glucose-6-phosphate 1-dehydrogenase None 6300 nM IC50
TKC109998 P11413 Glucose-6-phosphate 1-dehydrogenase None 31600 nM IC50
TKC110077 P11413 Glucose-6-phosphate 1-dehydrogenase None 5300 nM IC50
TKC112485 P11413 Glucose-6-phosphate 1-dehydrogenase None >200000 nM IC50
TKC112754 P11413 Glucose-6-phosphate 1-dehydrogenase None 6200 nM Ki
TKC112754 P11413 Glucose-6-phosphate 1-dehydrogenase None 24900 nM IC50
TKC113159 P11413 Glucose-6-phosphate 1-dehydrogenase None 81400 nM IC50
TKC151885 P11413 Glucose-6-phosphate 1-dehydrogenase None >80000 nM IC50
TKC206687 P11413 Glucose-6-phosphate 1-dehydrogenase None 900 nM IC50
TKC206754 P11413 Glucose-6-phosphate 1-dehydrogenase None 3000 nM Ki
TKC206754 P11413 Glucose-6-phosphate 1-dehydrogenase None >200000 nM IC50
TKC206758 P11413 Glucose-6-phosphate 1-dehydrogenase None >200000 nM IC50
TKC206777 P11413 Glucose-6-phosphate 1-dehydrogenase None 4300 nM IC50
TKC206899 P11413 Glucose-6-phosphate 1-dehydrogenase None 5200 nM IC50
TKC002411 P11597 Cholesteryl ester transfer protein None 196000 nM IC50
TKC026245 P11597 Cholesteryl ester transfer protein None 25000 nM IC50
TKC026309 P11597 Cholesteryl ester transfer protein None 6000 nM IC50
TKC026600 P11597 Cholesteryl ester transfer protein None 100000 nM IC50
TKC027200 P11597 Cholesteryl ester transfer protein None 5000 nM IC50
TKC027200 P11597 Cholesteryl ester transfer protein None 5200 nM IC50
TKC027201 P11597 Cholesteryl ester transfer protein None 1000 nM IC50
TKC027201 P11597 Cholesteryl ester transfer protein None 5200 nM IC50
TKC056482 P11597 Cholesteryl ester transfer protein None 46600 nM IC50
TKC077689 P11597 Cholesteryl ester transfer protein None 10 % Inhibition
TKC094496 P11597 Cholesteryl ester transfer protein None 46000 nM IC50
TKC097288 P11597 Cholesteryl ester transfer protein None 600 nM IC50
TKC106450 P11597 Cholesteryl ester transfer protein None 5200 nM IC50
TKC123088 P11597 Cholesteryl ester transfer protein None 31 % Inhibition
TKC019954 P12821 Angiotensin-converting enzyme None 15 % Inhibition
TKC039868 P12821 Angiotensin-converting enzyme None 17 % Inhibition
TKC011761 P12931 Proto-oncogene tyrosine-protein kinase Src None 61 % Inhibition
TKC024886 P12931 Proto-oncogene tyrosine-protein kinase Src None 8620 nM IC50
TKC025690 P12931 Proto-oncogene tyrosine-protein kinase Src None 19700 nM IC50
TKC115259 P12931 Proto-oncogene tyrosine-protein kinase Src None 2400 nM IC50
TKC115261 P12931 Proto-oncogene tyrosine-protein kinase Src None 2240 nM IC50
TKC115272 P12931 Proto-oncogene tyrosine-protein kinase Src None >100000 nM IC50
TKC115273 P12931 Proto-oncogene tyrosine-protein kinase Src None 1480 nM IC50
TKC135974 P12931 Proto-oncogene tyrosine-protein kinase Src None 35800 nM IC50
TKC151761 P12931 Proto-oncogene tyrosine-protein kinase Src None >10000 nM IC50
TKC152148 P12931 Proto-oncogene tyrosine-protein kinase Src None 1910 nM IC50
TKC152157 P12931 Proto-oncogene tyrosine-protein kinase Src None 2170 nM IC50
TKC174547 P12931 Proto-oncogene tyrosine-protein kinase Src None >100000 nM IC50
TKC200866 P12931 Proto-oncogene tyrosine-protein kinase Src None >10000 nM IC50
TKC096804 P13866 Sodium/glucose cotransporter 1 None <25 % Inhibition
TKC205544 P14416 D(2) dopamine receptor None 687 nM Ki
TKC205544 P14416 D(2) dopamine receptor None 280 nM Ki
TKC205544 P14416 D(2) dopamine receptor None 398.1 nM Ki
TKC206544 P14416 D(2) dopamine receptor None >10000 nM Ki
TKC039202 P21453 Sphingosine 1-phosphate receptor 1 None 4962 nM IC50
TKC096012 P21453 Sphingosine 1-phosphate receptor 1 None 34120 nM EC50
TKC096012 P21453 Sphingosine 1-phosphate receptor 1 None >95100 nM EC50
TKC096012 P21453 Sphingosine 1-phosphate receptor 1 None 25400 nM EC50
TKC032440 P24530 Endothelin receptor type B None 50000 nM IC50
TKC032443 P24530 Endothelin receptor type B None 21000 nM IC50
TKC032440 P25101 Endothelin-1 receptor None 135000 nM IC50
TKC032443 P25101 Endothelin-1 receptor None 62000 nM IC50
TKC054329 P25929 Neuropeptide Y receptor type 1 None >35000 nM IC50
TKC205544 P28223 5-hydroxytryptamine receptor 2A None >10000 nM Ki
TKC205544 P28223 5-hydroxytryptamine receptor 2A None 252 nM Ki
TKC205544 P28223 5-hydroxytryptamine receptor 2A None 288.4 nM Ki
TKC205544 P28223 5-hydroxytryptamine receptor 2A None 1000 nM Ki
TKC206781 P28223 5-hydroxytryptamine receptor 2A None 1.4 nM Ki
TKC096804 P31639 Sodium/glucose cotransporter 2 None 50 % Inhibition
TKC011761 P31749 RAC-alpha serine/threonine-protein kinase None 54 % Inhibition
TKC016414 P31749 RAC-alpha serine/threonine-protein kinase None 36 % Activity
TKC024886 P31749 RAC-alpha serine/threonine-protein kinase None 48400 nM IC50
TKC025690 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC044763 P31749 RAC-alpha serine/threonine-protein kinase None 100 % Inhibition
TKC115259 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC115261 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC115272 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC115273 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC118419 P31749 RAC-alpha serine/threonine-protein kinase None 96 % Inhibition
TKC152148 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC152157 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC174547 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC206776 P31749 RAC-alpha serine/threonine-protein kinase None 3 uM Activity
TKC037534 P35228 Nitric oxide synthase, inducible None 99 % Inhibition
TKC060880 P35228 Nitric oxide synthase, inducible None 37000 nM IC50
TKC077689 P35228 Nitric oxide synthase, inducible None >40000 nM IC50
TKC206319 P35228 Nitric oxide synthase, inducible None 100 % Inhibition
TKC024886 P35968 Vascular endothelial growth factor receptor 2 None 4810 nM IC50
TKC025690 P35968 Vascular endothelial growth factor receptor 2 None 3660 nM IC50
TKC051154 P35968 Vascular endothelial growth factor receptor 2 None 40 % Inhibition
TKC051155 P35968 Vascular endothelial growth factor receptor 2 None 46 % Inhibition
TKC065375 P35968 Vascular endothelial growth factor receptor 2 None 0 % Inhibition
TKC102689 P35968 Vascular endothelial growth factor receptor 2 None 0 % Inhibition
TKC108267 P35968 Vascular endothelial growth factor receptor 2 None 0 % Inhibition
TKC115259 P35968 Vascular endothelial growth factor receptor 2 None 4950 nM IC50
TKC115261 P35968 Vascular endothelial growth factor receptor 2 None 4600 nM IC50
TKC115272 P35968 Vascular endothelial growth factor receptor 2 None >100000 nM IC50
TKC115273 P35968 Vascular endothelial growth factor receptor 2 None 4850 nM IC50
TKC146202 P35968 Vascular endothelial growth factor receptor 2 None 61 % Inhibition
TKC152148 P35968 Vascular endothelial growth factor receptor 2 None 4350 nM IC50
TKC152157 P35968 Vascular endothelial growth factor receptor 2 None 6010 nM IC50
TKC174547 P35968 Vascular endothelial growth factor receptor 2 None >100000 nM IC50
TKC207124 P35968 Vascular endothelial growth factor receptor 2 None 40400 nM IC50
TKC146780 P37288 Vasopressin V1a receptor None 2325 nM EC50
TKC001786 P43220 Glucagon-like peptide 1 receptor None 1778 nM Potency
TKC002371 P43220 Glucagon-like peptide 1 receptor None 891 nM Potency
TKC002916 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC004286 P43220 Glucagon-like peptide 1 receptor None 11220 nM Potency
TKC005139 P43220 Glucagon-like peptide 1 receptor None 8913 nM Potency
TKC005308 P43220 Glucagon-like peptide 1 receptor None 1995 nM Potency
TKC005454 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC005842 P43220 Glucagon-like peptide 1 receptor None 8913 nM Potency
TKC008286 P43220 Glucagon-like peptide 1 receptor None 2818 nM Potency
TKC011526 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC012100 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC012116 P43220 Glucagon-like peptide 1 receptor None 7080 nM Potency
TKC013322 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC014761 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC014800 P43220 Glucagon-like peptide 1 receptor None 3548 nM Potency
TKC014807 P43220 Glucagon-like peptide 1 receptor None 11220 nM Potency
TKC016277 P43220 Glucagon-like peptide 1 receptor None 15849 nM Potency
TKC016338 P43220 Glucagon-like peptide 1 receptor None 25119 nM Potency
TKC016371 P43220 Glucagon-like peptide 1 receptor None 5623 nM Potency
TKC016544 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC018288 P43220 Glucagon-like peptide 1 receptor None 11220 nM Potency
TKC020117 P43220 Glucagon-like peptide 1 receptor None 2239 nM Potency
TKC022811 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC022814 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC022818 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC022945 P43220 Glucagon-like peptide 1 receptor None 1778 nM Potency
TKC028040 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC030034 P43220 Glucagon-like peptide 1 receptor None 7080 nM Potency
TKC031180 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC031572 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC032913 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC035580 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC037521 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC038268 P43220 Glucagon-like peptide 1 receptor None 355 nM Potency
TKC038273 P43220 Glucagon-like peptide 1 receptor None 4467 nM Potency
TKC039202 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC039542 P43220 Glucagon-like peptide 1 receptor None 1585 nM Potency
TKC043354 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC043518 P43220 Glucagon-like peptide 1 receptor None 11220 nM Potency
TKC048922 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC053815 P43220 Glucagon-like peptide 1 receptor None 5623 nM Potency
TKC060099 P43220 Glucagon-like peptide 1 receptor None 1000 nM Potency
TKC060929 P43220 Glucagon-like peptide 1 receptor None 3548 nM Potency
TKC062669 P43220 Glucagon-like peptide 1 receptor None 3548 nM Potency
TKC062670 P43220 Glucagon-like peptide 1 receptor None 1000 nM Potency
TKC064576 P43220 Glucagon-like peptide 1 receptor None 5012 nM Potency
TKC066096 P43220 Glucagon-like peptide 1 receptor None 1000 nM Potency
TKC066411 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC073833 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC073873 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC076529 P43220 Glucagon-like peptide 1 receptor None 6310 nM Potency
TKC082378 P43220 Glucagon-like peptide 1 receptor None 1122 nM Potency
TKC092297 P43220 Glucagon-like peptide 1 receptor None 8913 nM Potency
TKC092591 P43220 Glucagon-like peptide 1 receptor None 562 nM Potency
TKC093162 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC095265 P43220 Glucagon-like peptide 1 receptor None 3981 nM Potency
TKC095493 P43220 Glucagon-like peptide 1 receptor None 6310 nM Potency
TKC098290 P43220 Glucagon-like peptide 1 receptor None 1000 nM Potency
TKC098410 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC099065 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC101432 P43220 Glucagon-like peptide 1 receptor None 11220 nM Potency
TKC103159 P43220 Glucagon-like peptide 1 receptor None 31623 nM Potency
TKC103380 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC103381 P43220 Glucagon-like peptide 1 receptor None 14125 nM Potency
TKC103725 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC104414 P43220 Glucagon-like peptide 1 receptor None 14125 nM Potency
TKC104558 P43220 Glucagon-like peptide 1 receptor None 11220 nM Potency
TKC105932 P43220 Glucagon-like peptide 1 receptor None 19953 nM Potency
TKC107499 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC107557 P43220 Glucagon-like peptide 1 receptor None 15849 nM Potency
TKC107625 P43220 Glucagon-like peptide 1 receptor None 7080 nM Potency
TKC108316 P43220 Glucagon-like peptide 1 receptor None 11220 nM Potency
TKC111738 P43220 Glucagon-like peptide 1 receptor None 1778 nM Potency
TKC112759 P43220 Glucagon-like peptide 1 receptor None 8913 nM Potency
TKC112909 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC112910 P43220 Glucagon-like peptide 1 receptor None 11220 nM Potency
TKC112925 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC113150 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC117617 P43220 Glucagon-like peptide 1 receptor None 891 nM Potency
TKC117638 P43220 Glucagon-like peptide 1 receptor None 501 nM Potency
TKC117993 P43220 Glucagon-like peptide 1 receptor None 1000 nM Potency
TKC118131 P43220 Glucagon-like peptide 1 receptor None 501 nM Potency
TKC123088 P43220 Glucagon-like peptide 1 receptor None 3162 nM Potency
TKC129193 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC132374 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC132609 P43220 Glucagon-like peptide 1 receptor None 8913 nM Potency
TKC134702 P43220 Glucagon-like peptide 1 receptor None 2512 nM Potency
TKC134744 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC135702 P43220 Glucagon-like peptide 1 receptor None 3548 nM Potency
TKC136632 P43220 Glucagon-like peptide 1 receptor None 19953 nM Potency
TKC138780 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC139094 P43220 Glucagon-like peptide 1 receptor None 14125 nM Potency
TKC143885 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC150277 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC150326 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC151609 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC156644 P43220 Glucagon-like peptide 1 receptor None 22387 nM Potency
TKC159332 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC169163 P43220 Glucagon-like peptide 1 receptor None 10000 nM Potency
TKC173955 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC174441 P43220 Glucagon-like peptide 1 receptor None 31623 nM Potency
TKC197335 P43220 Glucagon-like peptide 1 receptor None 316 nM Potency
TKC197337 P43220 Glucagon-like peptide 1 receptor None 316 nM Potency
TKC206362 P43220 Glucagon-like peptide 1 receptor None 3981 nM Potency
TKC206549 P43220 Glucagon-like peptide 1 receptor None 1259 nM Potency
TKC206657 P43220 Glucagon-like peptide 1 receptor None 7943 nM Potency
TKC206660 P43220 Glucagon-like peptide 1 receptor None 1122 nM Potency
TKC206754 P43220 Glucagon-like peptide 1 receptor None 11220 nM Potency
TKC206758 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC206765 P43220 Glucagon-like peptide 1 receptor None 15849 nM Potency
TKC206766 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC206767 P43220 Glucagon-like peptide 1 receptor None 28184 nM Potency
TKC206771 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC206780 P43220 Glucagon-like peptide 1 receptor None 12589 nM Potency
TKC206816 P43220 Glucagon-like peptide 1 receptor None 25119 nM Potency
TKC206872 P43220 Glucagon-like peptide 1 receptor None 501 nM Potency
TKC206876 P43220 Glucagon-like peptide 1 receptor None 5012 nM Potency
TKC206889 P43220 Glucagon-like peptide 1 receptor None 1000 nM Potency
TKC025058 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 1000 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 5 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 19 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 55 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 55000 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 89 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 5 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 15 nM Kd
TKC118419 P53778 Mitogen-activated protein kinase 12 None 75 % Inhibition
TKC021262 Q07869 Peroxisome proliferator-activated receptor alpha None 19500 nM EC50
TKC021666 Q07869 Peroxisome proliferator-activated receptor alpha None 28 % Activity
TKC021674 Q07869 Peroxisome proliferator-activated receptor alpha None 25 % Activity
TKC035272 Q07869 Peroxisome proliferator-activated receptor alpha None 15849 nM Potency
TKC056482 Q07869 Peroxisome proliferator-activated receptor alpha None 259 % Activity
TKC057132 Q07869 Peroxisome proliferator-activated receptor alpha None 12589 nM Potency
TKC088526 Q07869 Peroxisome proliferator-activated receptor alpha None 12 % Activity
TKC100644 Q07869 Peroxisome proliferator-activated receptor alpha None 8913 nM Potency
TKC108536 Q07869 Peroxisome proliferator-activated receptor alpha None 50119 nM Potency
TKC110634 Q07869 Peroxisome proliferator-activated receptor alpha None 309 % Activity
TKC110635 Q07869 Peroxisome proliferator-activated receptor alpha None 289 % Activity
TKC170559 Q07869 Peroxisome proliferator-activated receptor alpha None 1000 nM EC50
TKC171329 Q07869 Peroxisome proliferator-activated receptor alpha None 184 nM EC50
TKC206812 Q07869 Peroxisome proliferator-activated receptor alpha None >20000 nM IC50