Basic Information

Name	[ICD-11: MG30-MG3Z]
Protein Number	54
Molecule Number	1023

Active subnetwork

Terpenoid-protein target Activity Association

ID	Uniport	Pref_name	Gene name	value	unit	type
TKC117625	O14763	Tumor necrosis factor receptor superfamily member 10B	None	2800	nM	EC50
TKC011555	O75762	Transient receptor potential cation channel subfamily A member 1	None	130	nM	EC50
TKC019467	O75762	Transient receptor potential cation channel subfamily A member 1	None	70	%	Inhibition
TKC019475	O75762	Transient receptor potential cation channel subfamily A member 1	None	70	%	Inhibition
TKC019507	O75762	Transient receptor potential cation channel subfamily A member 1	None	19700	nM	EC50
TKC020479	O75762	Transient receptor potential cation channel subfamily A member 1	None	6000	nM	EC50
TKC020479	O75762	Transient receptor potential cation channel subfamily A member 1	None	6000	nM	EC50
TKC020479	O75762	Transient receptor potential cation channel subfamily A member 1	None	60256	nM	EC50
TKC020491	O75762	Transient receptor potential cation channel subfamily A member 1	None	7000	nM	EC50
TKC020491	O75762	Transient receptor potential cation channel subfamily A member 1	None	17000	nM	EC50
TKC020943	O75762	Transient receptor potential cation channel subfamily A member 1	None	41000	nM	EC50
TKC022809	O75762	Transient receptor potential cation channel subfamily A member 1	None	300000	nM	IC50
TKC022931	O75762	Transient receptor potential cation channel subfamily A member 1	None	400000	nM	IC50
TKC031476	O75762	Transient receptor potential cation channel subfamily A member 1	None	59	nM	EC50
TKC039202	O75762	Transient receptor potential cation channel subfamily A member 1	None	590	nM	EC50
TKC085168	O75762	Transient receptor potential cation channel subfamily A member 1	None	96000	nM	EC50
TKC086929	O75762	Transient receptor potential cation channel subfamily A member 1	None	28400	nM	EC50
TKC086929	O75762	Transient receptor potential cation channel subfamily A member 1	None	31623	nM	EC50
TKC133551	O75762	Transient receptor potential cation channel subfamily A member 1	None	33000	nM	EC50
TKC013753	P03372	Estrogen receptor	None	8913	nM	Potency
TKC019072	P03372	Estrogen receptor	None	78	%	Activity
TKC022931	P03372	Estrogen receptor	None	1995	nM	Potency
TKC022961	P03372	Estrogen receptor	None	54	%	Activity
TKC028029	P03372	Estrogen receptor	None	0	%	Activity
TKC028034	P03372	Estrogen receptor	None	<0	%	Activity
TKC028037	P03372	Estrogen receptor	None	1	%	Activity
TKC028038	P03372	Estrogen receptor	None	<0	%	Activity
TKC028041	P03372	Estrogen receptor	None	<0	%	Activity
TKC034016	P03372	Estrogen receptor	None	51	%	Activity
TKC034337	P03372	Estrogen receptor	None	2800000	nM	IC50
TKC034640	P03372	Estrogen receptor	None	>1000000	nM	Ki
TKC035208	P03372	Estrogen receptor	None	39	%	Activity
TKC035272	P03372	Estrogen receptor	None	2551	nM	IC50
TKC035462	P03372	Estrogen receptor	None	42	%	Activity
TKC066169	P03372	Estrogen receptor	None	39811	nM	Potency
TKC075769	P03372	Estrogen receptor	None	251	nM	Potency
TKC079320	P03372	Estrogen receptor	None	<0	%	Activity
TKC079321	P03372	Estrogen receptor	None	<0	%	Activity
TKC087664	P03372	Estrogen receptor	None	3162	nM	Potency
TKC087988	P03372	Estrogen receptor	None	631	nM	Potency
TKC087991	P03372	Estrogen receptor	None	4467	nM	Potency
TKC092297	P03372	Estrogen receptor	None	15849	nM	Potency
TKC092348	P03372	Estrogen receptor	None	8913	nM	Potency
TKC096012	P03372	Estrogen receptor	None	126	nM	Potency
TKC100644	P03372	Estrogen receptor	None	31623	nM	Potency
TKC101365	P03372	Estrogen receptor	None	12570	nM	EC50
TKC102448	P03372	Estrogen receptor	None	2550	nM	EC50
TKC107086	P03372	Estrogen receptor	None	8913	nM	Potency
TKC107735	P03372	Estrogen receptor	None	50119	nM	Potency
TKC111727	P03372	Estrogen receptor	None	0	nM	Ki
TKC111738	P03372	Estrogen receptor	None	1	nM	EC50
TKC111738	P03372	Estrogen receptor	None	166	nM	IC50
TKC111738	P03372	Estrogen receptor	None	210	nM	IC50
TKC111738	P03372	Estrogen receptor	None	96	nM	IC50
TKC112923	P03372	Estrogen receptor	None	26	nM	EC50
TKC115268	P03372	Estrogen receptor	None	15849	nM	Potency
TKC129821	P03372	Estrogen receptor	None	70	%	Activity
TKC151345	P03372	Estrogen receptor	None	35	%	Activity
TKC151713	P03372	Estrogen receptor	None	40	%	Activity
TKC151765	P03372	Estrogen receptor	None	81	%	Activity
TKC206549	P03372	Estrogen receptor	None	3548	nM	Potency
TKC206608	P03372	Estrogen receptor	None	8170	nM	EC50
TKC206652	P03372	Estrogen receptor	None	112	nM	Potency
TKC206725	P03372	Estrogen receptor	None	8	nM	Ki
TKC206726	P03372	Estrogen receptor	None	72	nM	EC50
TKC206759	P03372	Estrogen receptor	None	>10000	nM	IC50
TKC206759	P03372	Estrogen receptor	None	>10000	nM	IC50
TKC206760	P03372	Estrogen receptor	None	25119	nM	Potency
TKC206764	P03372	Estrogen receptor	None	0	%	RBA
TKC206770	P03372	Estrogen receptor	None	5012	nM	Potency
TKC206779	P03372	Estrogen receptor	None	6310	nM	Potency
TKC206812	P03372	Estrogen receptor	None	62000	nM	IC50
TKC206812	P03372	Estrogen receptor	None	39811	nM	Potency
TKC206816	P03372	Estrogen receptor	None	>1000	nM	IC50
TKC206816	P03372	Estrogen receptor	None	>1000	nM	IC50
TKC008187	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	30200	nM	IC50
TKC023515	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	53	%	Inhibition
TKC025574	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	52	%	Inhibition
TKC026893	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	21	%	Inhibition
TKC026895	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	61	%	Inhibition
TKC057019	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	22300	nM	IC50
TKC100777	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	30	%	Inhibition
TKC101031	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	1500	nM	IC50
TKC101538	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	39	%	Inhibition
TKC101847	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	1000	nM	IC50
TKC103703	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	40	%	Inhibition
TKC137314	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	8400	nM	IC50
TKC138471	P04035	3-hydroxy-3-methylglutaryl-coenzyme A reductase	None	21700	nM	IC50
TKC010405	P06276	Cholinesterase	None	175800	nM	IC50
TKC010478	P06276	Cholinesterase	None	25000	nM	IC50
TKC010538	P06276	Cholinesterase	None	21100	nM	IC50
TKC010825	P06276	Cholinesterase	None	98100	nM	IC50
TKC012269	P06276	Cholinesterase	None	6	%	Inhibition
TKC026451	P06276	Cholinesterase	None	80	%	Inhibition
TKC026505	P06276	Cholinesterase	None	83	%	Inhibition
TKC050924	P06276	Cholinesterase	None	>4780	nM	Ki
TKC051021	P06276	Cholinesterase	None	>200000	nM	IC50
TKC051031	P06276	Cholinesterase	None	>200000	nM	IC50
TKC051032	P06276	Cholinesterase	None	>200000	nM	IC50
TKC051042	P06276	Cholinesterase	None	>200000	nM	IC50
TKC056997	P06276	Cholinesterase	None	>200000	nM	IC50
TKC056998	P06276	Cholinesterase	None	>200000	nM	IC50
TKC057020	P06276	Cholinesterase	None	156270	nM	IC50
TKC061148	P06276	Cholinesterase	None	>30000	nM	IC50
TKC062012	P06276	Cholinesterase	None	>30000	nM	IC50
TKC062026	P06276	Cholinesterase	None	>30000	nM	IC50
TKC062075	P06276	Cholinesterase	None	>30000	nM	IC50
TKC063185	P06276	Cholinesterase	None	>30000	nM	IC50
TKC064964	P06276	Cholinesterase	None	188360	nM	IC50
TKC064991	P06276	Cholinesterase	None	>200000	nM	IC50
TKC095827	P06276	Cholinesterase	None	>30000	nM	IC50
TKC107319	P06276	Cholinesterase	None	>100000	nM	Ki
TKC109307	P06276	Cholinesterase	None	23780	nM	IC50
TKC109315	P06276	Cholinesterase	None	1600	nM	Ki
TKC109320	P06276	Cholinesterase	None	18200	nM	IC50
TKC109322	P06276	Cholinesterase	None	17990	nM	IC50
TKC109330	P06276	Cholinesterase	None	16200	nM	Ki
TKC109348	P06276	Cholinesterase	None	26300	nM	Ki
TKC109381	P06276	Cholinesterase	None	2100	nM	IC50
TKC109383	P06276	Cholinesterase	None	600	nM	IC50
TKC109488	P06276	Cholinesterase	None	61500	nM	IC50
TKC112739	P06276	Cholinesterase	None	164670	nM	IC50
TKC112743	P06276	Cholinesterase	None	20870	nM	IC50
TKC112909	P06276	Cholinesterase	None	102660	nM	IC50
TKC114538	P06276	Cholinesterase	None	8600	nM	Ki
TKC114548	P06276	Cholinesterase	None	500	nM	IC50
TKC114549	P06276	Cholinesterase	None	7500	nM	Ki
TKC114554	P06276	Cholinesterase	None	3250	nM	Ki
TKC114561	P06276	Cholinesterase	None	4840	nM	IC50
TKC114562	P06276	Cholinesterase	None	3400	nM	Ki
TKC114777	P06276	Cholinesterase	None	3650	nM	IC50
TKC115315	P06276	Cholinesterase	None	550	ug.mL-1	IC50
TKC116871	P06276	Cholinesterase	None	142450	nM	IC50
TKC139191	P06276	Cholinesterase	None	>30000	nM	IC50
TKC141633	P06276	Cholinesterase	None	>200000	nM	IC50
TKC142015	P06276	Cholinesterase	None	>200000	nM	IC50
TKC144380	P06276	Cholinesterase	None	1370	nM	IC50
TKC144901	P06276	Cholinesterase	None	>30000	nM	IC50
TKC144904	P06276	Cholinesterase	None	>30000	nM	IC50
TKC145173	P06276	Cholinesterase	None	>200000	nM	IC50
TKC145183	P06276	Cholinesterase	None	>200000	nM	IC50
TKC147230	P06276	Cholinesterase	None	>200000	nM	IC50
TKC147240	P06276	Cholinesterase	None	>200000	nM	IC50
TKC148618	P06276	Cholinesterase	None	>200000	nM	IC50
TKC168054	P06276	Cholinesterase	None	420	nM	IC50
TKC174459	P06276	Cholinesterase	None	>200000	nM	IC50
TKC206328	P06276	Cholinesterase	None	>10000	nM	IC50
TKC206329	P06276	Cholinesterase	None	>10000	nM	IC50
TKC206750	P06276	Cholinesterase	None	506	ug.mL-1	IC50
TKC206759	P06276	Cholinesterase	None	53500	nM	IC50
TKC206770	P06276	Cholinesterase	None	1550	nM	IC50
TKC046324	P06493	Cyclin-dependent kinase 1	None	>100000	nM	IC50
TKC117541	P06493	Cyclin-dependent kinase 1	None	34	%	Activity
TKC024886	P08069	Insulin-like growth factor 1 receptor	None	11800	nM	IC50
TKC025690	P08069	Insulin-like growth factor 1 receptor	None	3310	nM	IC50
TKC115259	P08069	Insulin-like growth factor 1 receptor	None	3160	nM	IC50
TKC115261	P08069	Insulin-like growth factor 1 receptor	None	2420	nM	IC50
TKC115272	P08069	Insulin-like growth factor 1 receptor	None	>100000	nM	IC50
TKC115273	P08069	Insulin-like growth factor 1 receptor	None	2300	nM	IC50
TKC152148	P08069	Insulin-like growth factor 1 receptor	None	2770	nM	IC50
TKC152157	P08069	Insulin-like growth factor 1 receptor	None	2460	nM	IC50
TKC174547	P08069	Insulin-like growth factor 1 receptor	None	>100000	nM	IC50
TKC000192	P08575	Receptor-type tyrosine-protein phosphatase C	None	>19000	nM	IC50
TKC005454	P08575	Receptor-type tyrosine-protein phosphatase C	None	41400	nM	IC50
TKC031060	P08575	Receptor-type tyrosine-protein phosphatase C	None	10000	nM	IC50
TKC045915	P08575	Receptor-type tyrosine-protein phosphatase C	None	>30000	nM	IC50
TKC045916	P08575	Receptor-type tyrosine-protein phosphatase C	None	>27000	nM	IC50
TKC077689	P08575	Receptor-type tyrosine-protein phosphatase C	None	1000	nM	IC50
TKC096804	P08575	Receptor-type tyrosine-protein phosphatase C	None	1200	nM	IC50
TKC105683	P08575	Receptor-type tyrosine-protein phosphatase C	None	9000	nM	IC50
TKC106945	P08575	Receptor-type tyrosine-protein phosphatase C	None	>16000	nM	IC50
TKC156704	P08575	Receptor-type tyrosine-protein phosphatase C	None	>16000	nM	IC50
TKC191566	P08575	Receptor-type tyrosine-protein phosphatase C	None	>19000	nM	IC50
TKC151523	P08908	5-hydroxytryptamine receptor 1A	None	>100000	nM	Ki
TKC205544	P08908	5-hydroxytryptamine receptor 1A	None	4500	nM	Ki
TKC205544	P08908	5-hydroxytryptamine receptor 1A	None	1500	nM	Ki
TKC205544	P08908	5-hydroxytryptamine receptor 1A	None	642	nM	Ki
TKC205544	P08908	5-hydroxytryptamine receptor 1A	None	1258.92	nM	Ki
TKC206544	P08908	5-hydroxytryptamine receptor 1A	None	>10000	nM	Ki
TKC206549	P08908	5-hydroxytryptamine receptor 1A	None	30	pM well-1	cAMP
TKC112785	P08912	Muscarinic acetylcholine receptor M5	None	>10000	nM	Ki
TKC206544	P08912	Muscarinic acetylcholine receptor M5	None	>10000	nM	Ki
TKC100416	P08913	Alpha-2A adrenergic receptor	None	31623	nM	Kd
TKC205544	P08913	Alpha-2A adrenergic receptor	None	0	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	0	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	0.32	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	132	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	2.7	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	3.6	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	0.43	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	3.76	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	0.71	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	1.2	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	7.94	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	2.5	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	3.5	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	170	nM	IC50
TKC205544	P08913	Alpha-2A adrenergic receptor	None	8	nM	IC50
TKC205544	P08913	Alpha-2A adrenergic receptor	None	7.5	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	1.8	nM	Ki
TKC205544	P08913	Alpha-2A adrenergic receptor	None	8.5	nM	EC50
TKC205544	P08913	Alpha-2A adrenergic receptor	None	3.67	nM	IC50
TKC205806	P08913	Alpha-2A adrenergic receptor	None	8	nM	Ki
TKC020117	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	-67	%	Inhibition
TKC024485	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>50000	nM	IC50
TKC024587	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	600	nM	IC50
TKC024956	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	18000	nM	IC50
TKC024992	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	450	nM	IC50
TKC024993	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	14000	nM	IC50
TKC025965	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>150000	nM	IC50
TKC026303	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	4600	nM	IC50
TKC026309	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	680	nM	IC50
TKC027255	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>67	%	Activity
TKC034201	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>200000	nM	IC50
TKC040026	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	72	%	Inhibition
TKC051154	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	2700	nM	IC50
TKC056482	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>64	%	Activity
TKC058811	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	42000	nM	IC50
TKC058812	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>93	%	Activity
TKC064374	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	42000	nM	IC50
TKC064407	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>72	%	Activity
TKC065375	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>70	%	Activity
TKC071640	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>60	%	Activity
TKC076350	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	100	%	Activity
TKC077689	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	100	%	Activity
TKC077703	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>86	%	Activity
TKC078194	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	31800	nM	IC50
TKC082039	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	48	%	Inhibition
TKC088678	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	24800	nM	IC50
TKC089448	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	35	%	Inhibition
TKC094647	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	97	%	Activity
TKC107943	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	2000	nM	IC50
TKC123028	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	30400	nM	IC50
TKC124303	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	750	nM	IC50
TKC133309	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>200000	nM	IC50
TKC133656	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	25100	nM	IC50
TKC134278	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>200000	nM	IC50
TKC139322	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>67	%	Activity
TKC139366	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	3000	nM	IC50
TKC141401	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	42000	nM	IC50
TKC141499	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	25700	nM	IC50
TKC141805	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>53	%	Activity
TKC142849	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>70	%	Activity
TKC142897	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	30600	nM	IC50
TKC142922	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>61	%	Activity
TKC143539	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	100	%	Activity
TKC145848	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	42000	nM	IC50
TKC145932	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>56	%	Activity
TKC145968	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	100	%	Activity
TKC146774	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>63	%	Activity
TKC149759	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>73	%	Activity
TKC150706	P09917	Polyunsaturated fatty acid 5-lipoxygenase	None	>62	%	Activity
TKC013304	P10145	Interleukin-8	None	74978	nM	Potency
TKC013753	P10145	Interleukin-8	None	422	nM	Potency
TKC018710	P10145	Interleukin-8	None	33492	nM	Potency
TKC066169	P10145	Interleukin-8	None	42163	nM	Potency
TKC075769	P10145	Interleukin-8	None	299	nM	Potency
TKC087664	P10145	Interleukin-8	None	37578	nM	Potency
TKC087991	P10145	Interleukin-8	None	422	nM	Potency
TKC092297	P10145	Interleukin-8	None	66824	nM	Potency
TKC104088	P10145	Interleukin-8	None	817	nM	IC50
TKC107086	P10145	Interleukin-8	None	66824	nM	Potency
TKC107735	P10145	Interleukin-8	None	66824	nM	Potency
TKC115268	P10145	Interleukin-8	None	66824	nM	Potency
TKC132609	P10145	Interleukin-8	None	7490	nM	IC50
TKC136411	P10145	Interleukin-8	None	74978	nM	Potency
TKC206759	P10145	Interleukin-8	None	74978	nM	Potency
TKC206760	P10145	Interleukin-8	None	74978	nM	Potency
TKC206770	P10145	Interleukin-8	None	74978	nM	Potency
TKC206812	P10145	Interleukin-8	None	66824	nM	Potency
TKC206816	P10145	Interleukin-8	None	74978	nM	Potency
TKC206884	P10145	Interleukin-8	None	74978	nM	Potency
TKC001669	P10275	Androgen receptor	None	260	nM	IC50
TKC006934	P10275	Androgen receptor	None	50119	nM	Potency
TKC013304	P10275	Androgen receptor	None	70795	nM	Potency
TKC019571	P10275	Androgen receptor	None	19953	nM	Potency
TKC021325	P10275	Androgen receptor	None	31623	nM	Potency
TKC021332	P10275	Androgen receptor	None	31623	nM	Potency
TKC023246	P10275	Androgen receptor	None	449	nM	IC50
TKC030239	P10275	Androgen receptor	None	14	nM	Potency
TKC035272	P10275	Androgen receptor	None	15849	nM	Potency
TKC056140	P10275	Androgen receptor	None	50	%	Activity
TKC066169	P10275	Androgen receptor	None	3981	nM	Potency
TKC074867	P10275	Androgen receptor	None	28184	nM	Potency
TKC075769	P10275	Androgen receptor	None	355	nM	Potency
TKC079001	P10275	Androgen receptor	None	1	nM	Potency
TKC096012	P10275	Androgen receptor	None	178	nM	Potency
TKC100644	P10275	Androgen receptor	None	35481	nM	Potency
TKC102407	P10275	Androgen receptor	None	44668	nM	Potency
TKC106878	P10275	Androgen receptor	None	238	nM	IC50
TKC107086	P10275	Androgen receptor	None	17783	nM	Potency
TKC107735	P10275	Androgen receptor	None	3981	nM	Potency
TKC111738	P10275	Androgen receptor	None	17783	nM	Potency
TKC112923	P10275	Androgen receptor	None	212	nM	IC50
TKC114095	P10275	Androgen receptor	None	1790	nM	IC50
TKC114511	P10275	Androgen receptor	None	315	nM	Ki
TKC115268	P10275	Androgen receptor	None	35481	nM	Potency
TKC115284	P10275	Androgen receptor	None	1	nM	Ki
TKC117154	P10275	Androgen receptor	None	580	nM	IC50
TKC120161	P10275	Androgen receptor	None	44668	nM	Potency
TKC122884	P10275	Androgen receptor	None	39811	nM	Potency
TKC122892	P10275	Androgen receptor	None	10000	nM	IC50
TKC134780	P10275	Androgen receptor	None	2	nM	Potency
TKC147240	P10275	Androgen receptor	None	50	%	Activity
TKC206652	P10275	Androgen receptor	None	50	nM	Potency
TKC206688	P10275	Androgen receptor	None	224	nM	Potency
TKC206690	P10275	Androgen receptor	None	36	nM	Potency
TKC206759	P10275	Androgen receptor	None	2	nM	Potency
TKC206759	P10275	Androgen receptor	None	3.9	nM	IC50
TKC206759	P10275	Androgen receptor	None	4.7	nM	IC50
TKC206759	P10275	Androgen receptor	None	4.2	nM	IC50
TKC206759	P10275	Androgen receptor	None	29	nM	Ki
TKC206759	P10275	Androgen receptor	None	1.1	nM	EC50
TKC206759	P10275	Androgen receptor	None	2.7	nM	IC50
TKC206759	P10275	Androgen receptor	None	2.7	nM	IC50
TKC206759	P10275	Androgen receptor	None	2.7	nM	IC50
TKC206759	P10275	Androgen receptor	None	30	nM	IC50
TKC206759	P10275	Androgen receptor	None	4.57	nM	IC50
TKC206770	P10275	Androgen receptor	None	224	nM	Potency
TKC206779	P10275	Androgen receptor	None	2	nM	Potency
TKC206812	P10275	Androgen receptor	None	220	nM	IC50
TKC206816	P10275	Androgen receptor	None	9	nM	Ki
TKC206816	P10275	Androgen receptor	None	8.5	nM	Ki
TKC206816	P10275	Androgen receptor	None	8.5	nM	Ki
TKC206816	P10275	Androgen receptor	None	8.5	nM	Ki
TKC206816	P10275	Androgen receptor	None	8.5	nM	Ki
TKC206816	P10275	Androgen receptor	None	37	nM	IC50
TKC206816	P10275	Androgen receptor	None	8.5	nM	Ki
TKC206816	P10275	Androgen receptor	None	35	nM	Ki
TKC206816	P10275	Androgen receptor	None	14	nM	IC50
TKC205544	P14416	D(2) dopamine receptor	None	687	nM	Ki
TKC205544	P14416	D(2) dopamine receptor	None	280	nM	Ki
TKC205544	P14416	D(2) dopamine receptor	None	398.1	nM	Ki
TKC206544	P14416	D(2) dopamine receptor	None	>10000	nM	Ki
TKC035272	P14618	Pyruvate kinase PKM	None	31623	nM	Potency
TKC037410	P14618	Pyruvate kinase PKM	None	6	nM	EC50
TKC039332	P14618	Pyruvate kinase PKM	None	25119	nM	Potency
TKC100416	P14618	Pyruvate kinase PKM	None	13	nM	Potency
TKC151609	P14618	Pyruvate kinase PKM	None	11220	nM	Potency
TKC206901	P14618	Pyruvate kinase PKM	None	2	nM	Potency
TKC013753	P15121	Aldo-keto reductase family 1 member B1	None	1100000	nM	Km
TKC035272	P15121	Aldo-keto reductase family 1 member B1	None	500	nM	Ki
TKC035273	P15121	Aldo-keto reductase family 1 member B1	None	1500	nM	Ki
TKC048308	P15121	Aldo-keto reductase family 1 member B1	None	>200000	nM	IC50
TKC048325	P15121	Aldo-keto reductase family 1 member B1	None	147300	nM	IC50
TKC048341	P15121	Aldo-keto reductase family 1 member B1	None	>200000	nM	IC50
TKC049175	P15121	Aldo-keto reductase family 1 member B1	None	25	ug.mL-1	IC50
TKC051021	P15121	Aldo-keto reductase family 1 member B1	None	>193500	nM	IC50
TKC051028	P15121	Aldo-keto reductase family 1 member B1	None	22800	nM	IC50
TKC051029	P15121	Aldo-keto reductase family 1 member B1	None	>193500	nM	IC50
TKC051032	P15121	Aldo-keto reductase family 1 member B1	None	>189400	nM	IC50
TKC055115	P15121	Aldo-keto reductase family 1 member B1	None	12000	ug.mL-1	IC50
TKC056482	P15121	Aldo-keto reductase family 1 member B1	None	41000	nM	IC50
TKC057931	P15121	Aldo-keto reductase family 1 member B1	None	6	/min	Kcat
TKC060859	P15121	Aldo-keto reductase family 1 member B1	None	25	ug.mL-1	IC50
TKC063401	P15121	Aldo-keto reductase family 1 member B1	None	25	ug.mL-1	IC50
TKC063402	P15121	Aldo-keto reductase family 1 member B1	None	25	ug.mL-1	IC50
TKC063751	P15121	Aldo-keto reductase family 1 member B1	None	>195300	nM	IC50
TKC077689	P15121	Aldo-keto reductase family 1 member B1	None	124000	nM	IC50
TKC081137	P15121	Aldo-keto reductase family 1 member B1	None	>193500	nM	IC50
TKC088678	P15121	Aldo-keto reductase family 1 member B1	None	280000	nM	IC50
TKC092322	P15121	Aldo-keto reductase family 1 member B1	None	400000	nM	Km
TKC101833	P15121	Aldo-keto reductase family 1 member B1	None	>193500	nM	IC50
TKC123088	P15121	Aldo-keto reductase family 1 member B1	None	11000	nM	IC50
TKC137747	P15121	Aldo-keto reductase family 1 member B1	None	>200000	nM	IC50
TKC137786	P15121	Aldo-keto reductase family 1 member B1	None	>200000	nM	IC50
TKC137982	P15121	Aldo-keto reductase family 1 member B1	None	>200000	nM	IC50
TKC138004	P15121	Aldo-keto reductase family 1 member B1	None	>200000	nM	IC50
TKC141585	P15121	Aldo-keto reductase family 1 member B1	None	>194400	nM	IC50
TKC142922	P15121	Aldo-keto reductase family 1 member B1	None	84000	nM	IC50
TKC145170	P15121	Aldo-keto reductase family 1 member B1	None	>199200	nM	IC50
TKC145534	P15121	Aldo-keto reductase family 1 member B1	None	>187900	nM	IC50
TKC145540	P15121	Aldo-keto reductase family 1 member B1	None	>174200	nM	IC50
TKC145547	P15121	Aldo-keto reductase family 1 member B1	None	>174700	nM	IC50
TKC146774	P15121	Aldo-keto reductase family 1 member B1	None	72000	nM	IC50
TKC150706	P15121	Aldo-keto reductase family 1 member B1	None	34000	nM	IC50
TKC151691	P15121	Aldo-keto reductase family 1 member B1	None	119200	nM	IC50
TKC151763	P15121	Aldo-keto reductase family 1 member B1	None	43800	nM	IC50
TKC151921	P15121	Aldo-keto reductase family 1 member B1	None	>194400	nM	IC50
TKC156642	P15121	Aldo-keto reductase family 1 member B1	None	>189400	nM	IC50
TKC206760	P15121	Aldo-keto reductase family 1 member B1	None	6900	nM	IC50
TKC207025	P15121	Aldo-keto reductase family 1 member B1	None	>183900	nM	IC50
TKC087988	P18089	Alpha-2B adrenergic receptor	None	3019	nM	Ki
TKC100416	P18089	Alpha-2B adrenergic receptor	None	32	nM	Kd
TKC205544	P18089	Alpha-2B adrenergic receptor	None	1	nM	Ki
TKC205544	P18089	Alpha-2B adrenergic receptor	None	1.18	nM	Ki
TKC205544	P18089	Alpha-2B adrenergic receptor	None	77	nM	Ki
TKC205544	P18089	Alpha-2B adrenergic receptor	None	4.59	nM	Ki
TKC205544	P18089	Alpha-2B adrenergic receptor	None	1.2	nM	Ki
TKC205544	P18089	Alpha-2B adrenergic receptor	None	1.99	nM	Ki
TKC205544	P18089	Alpha-2B adrenergic receptor	None	2	nM	Ki
TKC205544	P18089	Alpha-2B adrenergic receptor	None	4.6	nM	Ki
TKC205544	P18089	Alpha-2B adrenergic receptor	None	15	nM	Ki
TKC205544	P18089	Alpha-2B adrenergic receptor	None	1.2	nM	Ki
TKC205806	P18089	Alpha-2B adrenergic receptor	None	15	nM	Ki
TKC205544	P18825	Alpha-2C adrenergic receptor	None	1	nM	Ki
TKC205544	P18825	Alpha-2C adrenergic receptor	None	0.13	nM	Ki
TKC205544	P18825	Alpha-2C adrenergic receptor	None	0.78	nM	Ki
TKC205544	P18825	Alpha-2C adrenergic receptor	None	0.55	nM	Ki
TKC205544	P18825	Alpha-2C adrenergic receptor	None	0.25	nM	Ki
TKC205544	P18825	Alpha-2C adrenergic receptor	None	0.5	nM	Ki
TKC205544	P18825	Alpha-2C adrenergic receptor	None	2.3	nM	Ki
TKC205544	P18825	Alpha-2C adrenergic receptor	None	1.9	nM	Ki
TKC205544	P18825	Alpha-2C adrenergic receptor	None	0.8	nM	Ki
TKC205544	P18825	Alpha-2C adrenergic receptor	None	27.1	nM	IC50
TKC205806	P18825	Alpha-2C adrenergic receptor	None	5	nM	Ki
TKC027341	P21554	Cannabinoid receptor 1	None	714	nM	Ki
TKC027353	P21554	Cannabinoid receptor 1	None	1459	nM	Ki
TKC027353	P21554	Cannabinoid receptor 1	None	1259	nM	Ki
TKC027353	P21554	Cannabinoid receptor 1	None	4350	nM	Ki
TKC027353	P21554	Cannabinoid receptor 1	None	2400	nM	Ki
TKC027353	P21554	Cannabinoid receptor 1	None	4.37E+12	nM	Ki
TKC027356	P21554	Cannabinoid receptor 1	None	14710	nM	Ki
TKC027364	P21554	Cannabinoid receptor 1	None	760	nM	Ki
TKC027373	P21554	Cannabinoid receptor 1	None	13	nM	Ki
TKC027373	P21554	Cannabinoid receptor 1	None	308	nM	Ki
TKC027373	P21554	Cannabinoid receptor 1	None	3.09E+11	nM	Ki
TKC027397	P21554	Cannabinoid receptor 1	None	565	nM	EC50
TKC095132	P21554	Cannabinoid receptor 1	None	1	nM	EC50
TKC095132	P21554	Cannabinoid receptor 1	None	18.6	nM	Ki
TKC095197	P21554	Cannabinoid receptor 1	None	6	nM	Ki
TKC095197	P21554	Cannabinoid receptor 1	None	927	nM	EC50
TKC146116	P21554	Cannabinoid receptor 1	None	>1.0e+4	nM	Ki
TKC205544	P21554	Cannabinoid receptor 1	None	35	%	Inhibition
TKC005313	P21728	D(1A) dopamine receptor	None	517	nM	Potency
TKC035272	P21728	D(1A) dopamine receptor	None	12589	nM	Potency
TKC035984	P21728	D(1A) dopamine receptor	None	20	nM	Potency
TKC084630	P21728	D(1A) dopamine receptor	None	14125	nM	Potency
TKC092297	P21728	D(1A) dopamine receptor	None	2909	nM	Potency
TKC205544	P21728	D(1A) dopamine receptor	None	2909	nM	Potency
TKC205544	P21728	D(1A) dopamine receptor	None	>10000	nM	Ki
TKC206544	P21728	D(1A) dopamine receptor	None	>10000	nM	Ki
TKC206622	P21728	D(1A) dopamine receptor	None	231	nM	Potency
TKC206690	P21728	D(1A) dopamine receptor	None	26	nM	Potency
TKC206777	P21728	D(1A) dopamine receptor	None	23109	nM	Potency
TKC206816	P21728	D(1A) dopamine receptor	None	14125	nM	Potency
TKC005454	P22303	Acetylcholinesterase	None	>6410	nM	Ki
TKC008149	P22303	Acetylcholinesterase	None	0	ug	Activity
TKC010478	P22303	Acetylcholinesterase	None	14500	nM	IC50
TKC010538	P22303	Acetylcholinesterase	None	22800	nM	IC50
TKC011270	P22303	Acetylcholinesterase	None	>10	ug	Activity
TKC012269	P22303	Acetylcholinesterase	None	>22	%	Inhibition
TKC014568	P22303	Acetylcholinesterase	None	>50000	nM	IC50
TKC014568	P22303	Acetylcholinesterase	None	>100000	nM	Ki
TKC025887	P22303	Acetylcholinesterase	None	2500	nM	IC50
TKC026245	P22303	Acetylcholinesterase	None	10	ug	MIC
TKC026257	P22303	Acetylcholinesterase	None	1	ug	MIC
TKC039110	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC039119	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC039122	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC048637	P22303	Acetylcholinesterase	None	29	%	Inhibition
TKC050924	P22303	Acetylcholinesterase	None	10670	nM	IC50
TKC051021	P22303	Acetylcholinesterase	None	22630	nM	IC50
TKC051031	P22303	Acetylcholinesterase	None	18350	nM	IC50
TKC051032	P22303	Acetylcholinesterase	None	30260	nM	IC50
TKC051042	P22303	Acetylcholinesterase	None	17140	nM	IC50
TKC056997	P22303	Acetylcholinesterase	None	16270	nM	IC50
TKC056998	P22303	Acetylcholinesterase	None	25080	nM	IC50
TKC057020	P22303	Acetylcholinesterase	None	31030	nM	IC50
TKC061148	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC062012	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC062026	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC062075	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC063185	P22303	Acetylcholinesterase	None	9980	nM	IC50
TKC064964	P22303	Acetylcholinesterase	None	25910	nM	IC50
TKC064991	P22303	Acetylcholinesterase	None	9400	nM	IC50
TKC068847	P22303	Acetylcholinesterase	None	34	%	Inhibition
TKC083115	P22303	Acetylcholinesterase	None	26	%	Inhibition
TKC092147	P22303	Acetylcholinesterase	None	>10	ug	MIC
TKC092148	P22303	Acetylcholinesterase	None	1	ug	MIC
TKC092149	P22303	Acetylcholinesterase	None	1	ug	MIC
TKC092150	P22303	Acetylcholinesterase	None	10	ug	MIC
TKC092151	P22303	Acetylcholinesterase	None	1	ug	MIC
TKC092152	P22303	Acetylcholinesterase	None	>10	ug	MIC
TKC092153	P22303	Acetylcholinesterase	None	>10	ug	MIC
TKC092154	P22303	Acetylcholinesterase	None	>10	ug	MIC
TKC092155	P22303	Acetylcholinesterase	None	10	ug	MIC
TKC092156	P22303	Acetylcholinesterase	None	>10	ug	MIC
TKC092182	P22303	Acetylcholinesterase	None	>10	ug	MIC
TKC095827	P22303	Acetylcholinesterase	None	910	nM	IC50
TKC101947	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC103473	P22303	Acetylcholinesterase	None	10	ug	Activity
TKC107319	P22303	Acetylcholinesterase	None	>100000	nM	Ki
TKC108605	P22303	Acetylcholinesterase	None	10	ug	Activity
TKC109315	P22303	Acetylcholinesterase	None	5754	nM	IC50
TKC109320	P22303	Acetylcholinesterase	None	181970	nM	IC50
TKC109322	P22303	Acetylcholinesterase	None	229087	nM	IC50
TKC109330	P22303	Acetylcholinesterase	None	77625	nM	IC50
TKC109347	P22303	Acetylcholinesterase	None	33113	nM	IC50
TKC109348	P22303	Acetylcholinesterase	None	61660	nM	IC50
TKC109364	P22303	Acetylcholinesterase	None	15849	nM	IC50
TKC109367	P22303	Acetylcholinesterase	None	30200	nM	IC50
TKC109381	P22303	Acetylcholinesterase	None	7079	nM	IC50
TKC109383	P22303	Acetylcholinesterase	None	9900	nM	IC50
TKC110247	P22303	Acetylcholinesterase	None	>10	ug.mL-1	IC50
TKC112463	P22303	Acetylcholinesterase	None	251189	nM	IC50
TKC112467	P22303	Acetylcholinesterase	None	83176	nM	IC50
TKC112468	P22303	Acetylcholinesterase	None	48978	nM	IC50
TKC112505	P22303	Acetylcholinesterase	None	42658	nM	IC50
TKC114542	P22303	Acetylcholinesterase	None	50119	nM	IC50
TKC114543	P22303	Acetylcholinesterase	None	70795	nM	IC50
TKC114548	P22303	Acetylcholinesterase	None	28000	nM	IC50
TKC114549	P22303	Acetylcholinesterase	None	69183	nM	IC50
TKC114551	P22303	Acetylcholinesterase	None	28840	nM	IC50
TKC114558	P22303	Acetylcholinesterase	None	6457	nM	IC50
TKC114561	P22303	Acetylcholinesterase	None	19498	nM	IC50
TKC114562	P22303	Acetylcholinesterase	None	6457	nM	IC50
TKC114777	P22303	Acetylcholinesterase	None	6166	nM	IC50
TKC119401	P22303	Acetylcholinesterase	None	26000	nM	IC50
TKC129743	P22303	Acetylcholinesterase	None	>10	ug	Activity
TKC135978	P22303	Acetylcholinesterase	None	191100	nM	IC50
TKC139191	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC141633	P22303	Acetylcholinesterase	None	24040	nM	IC50
TKC142015	P22303	Acetylcholinesterase	None	21100	nM	IC50
TKC144380	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC144901	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC144904	P22303	Acetylcholinesterase	None	>30000	nM	IC50
TKC145173	P22303	Acetylcholinesterase	None	22970	nM	IC50
TKC145183	P22303	Acetylcholinesterase	None	18350	nM	IC50
TKC147230	P22303	Acetylcholinesterase	None	22310	nM	IC50
TKC147240	P22303	Acetylcholinesterase	None	26780	nM	IC50
TKC148618	P22303	Acetylcholinesterase	None	21840	nM	IC50
TKC150909	P22303	Acetylcholinesterase	None	<10	ug.mL-1	IC50
TKC161356	P22303	Acetylcholinesterase	None	81500	nM	IC50
TKC168054	P22303	Acetylcholinesterase	None	1690	nM	IC50
TKC174459	P22303	Acetylcholinesterase	None	12260	nM	IC50
TKC205554	P22303	Acetylcholinesterase	None	1	ug	MIC
TKC205771	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC205772	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC206567	P22303	Acetylcholinesterase	None	1	ug	Activity
TKC207001	P22303	Acetylcholinesterase	None	4	ug	MIC
TKC207197	P22303	Acetylcholinesterase	None	1	ug	MIC
TKC000611	P23219	Prostaglandin G/H synthase 1	None	40000	nM	IC50
TKC001618	P23219	Prostaglandin G/H synthase 1	None	34000	nM	IC50
TKC009896	P23219	Prostaglandin G/H synthase 1	None	791100	nM	IC50
TKC019819	P23219	Prostaglandin G/H synthase 1	None	48	%	Inhibition
TKC019859	P23219	Prostaglandin G/H synthase 1	None	54	%	Inhibition
TKC020491	P23219	Prostaglandin G/H synthase 1	None	4000	nM	IC50
TKC020796	P23219	Prostaglandin G/H synthase 1	None	30	%	Inhibition
TKC021940	P23219	Prostaglandin G/H synthase 1	None	40	%	Inhibition
TKC022833	P23219	Prostaglandin G/H synthase 1	None	43	%	Inhibition
TKC022834	P23219	Prostaglandin G/H synthase 1	None	43	%	Inhibition
TKC022961	P23219	Prostaglandin G/H synthase 1	None	44	%	Inhibition
TKC024587	P23219	Prostaglandin G/H synthase 1	None	3300	nM	IC50
TKC024587	P23219	Prostaglandin G/H synthase 1	None	3300	nM	IC50
TKC031258	P23219	Prostaglandin G/H synthase 1	None	3600	nM	IC50
TKC034201	P23219	Prostaglandin G/H synthase 1	None	>200000	nM	IC50
TKC034358	P23219	Prostaglandin G/H synthase 1	None	39000	nM	IC50
TKC034359	P23219	Prostaglandin G/H synthase 1	None	39000	nM	IC50
TKC036372	P23219	Prostaglandin G/H synthase 1	None	14000	nM	IC50
TKC037595	P23219	Prostaglandin G/H synthase 1	None	36000	nM	IC50
TKC043613	P23219	Prostaglandin G/H synthase 1	None	43000	nM	IC50
TKC049750	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC049818	P23219	Prostaglandin G/H synthase 1	None	44	ug	IC50
TKC054011	P23219	Prostaglandin G/H synthase 1	None	8800	nM	IC50
TKC054031	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC054081	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC054090	P23219	Prostaglandin G/H synthase 1	None	7500	nM	IC50
TKC054099	P23219	Prostaglandin G/H synthase 1	None	8800	nM	IC50
TKC054100	P23219	Prostaglandin G/H synthase 1	None	8900	nM	IC50
TKC054101	P23219	Prostaglandin G/H synthase 1	None	7600	nM	IC50
TKC054240	P23219	Prostaglandin G/H synthase 1	None	7800	nM	IC50
TKC054241	P23219	Prostaglandin G/H synthase 1	None	6300	nM	IC50
TKC056482	P23219	Prostaglandin G/H synthase 1	None	210000	nM	IC50
TKC060184	P23219	Prostaglandin G/H synthase 1	None	8300	nM	IC50
TKC060216	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC060284	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC060302	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC060303	P23219	Prostaglandin G/H synthase 1	None	7800	nM	IC50
TKC060304	P23219	Prostaglandin G/H synthase 1	None	8000	nM	IC50
TKC060399	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC060602	P23219	Prostaglandin G/H synthase 1	None	5900	nM	IC50
TKC066954	P23219	Prostaglandin G/H synthase 1	None	38	%	Inhibition
TKC068533	P23219	Prostaglandin G/H synthase 1	None	28000	nM	IC50
TKC071010	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC077689	P23219	Prostaglandin G/H synthase 1	None	380000	nM	IC50
TKC077689	P23219	Prostaglandin G/H synthase 1	None	380000	nM	IC50
TKC095276	P23219	Prostaglandin G/H synthase 1	None	48	%	Inhibition
TKC113936	P23219	Prostaglandin G/H synthase 1	None	65	%	Inhibition
TKC122543	P23219	Prostaglandin G/H synthase 1	None	35	%	Inhibition
TKC130084	P23219	Prostaglandin G/H synthase 1	None	39	%	Inhibition
TKC130119	P23219	Prostaglandin G/H synthase 1	None	33	%	Inhibition
TKC130577	P23219	Prostaglandin G/H synthase 1	None	<43	%	Inhibition
TKC130901	P23219	Prostaglandin G/H synthase 1	None	36	%	Inhibition
TKC133309	P23219	Prostaglandin G/H synthase 1	None	>200000	nM	IC50
TKC133517	P23219	Prostaglandin G/H synthase 1	None	1300	nM	IC50
TKC133656	P23219	Prostaglandin G/H synthase 1	None	>200000	nM	IC50
TKC134278	P23219	Prostaglandin G/H synthase 1	None	>200000	nM	IC50
TKC139036	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC140627	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC141365	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC143641	P23219	Prostaglandin G/H synthase 1	None	>50000	nM	IC50
TKC151113	P23219	Prostaglandin G/H synthase 1	None	116400	nM	IC50
TKC151284	P23219	Prostaglandin G/H synthase 1	None	51	%	Inhibition
TKC151765	P23219	Prostaglandin G/H synthase 1	None	48	%	Inhibition
TKC151792	P23219	Prostaglandin G/H synthase 1	None	14000	nM	IC50
TKC172853	P23219	Prostaglandin G/H synthase 1	None	43700	nM	IC50
TKC205544	P23975	Sodium-dependent noradrenaline transporter	None	>20000	nM	IC50
TKC000660	P25021	Histamine H2 receptor	None	>10000	nM	Ki
TKC110447	P25024	C-X-C chemokine receptor type 1	None	4500	nM	IC50
TKC119009	P25024	C-X-C chemokine receptor type 1	None	20000	nM	IC50
TKC119010	P25024	C-X-C chemokine receptor type 1	None	5500	nM	IC50
TKC205544	P25100	Alpha-1D adrenergic receptor	None	2	nM	Ki
TKC205544	P25100	Alpha-1D adrenergic receptor	None	158.48	nM	Ki
TKC205544	P25100	Alpha-1D adrenergic receptor	None	954.99	nM	Ki
TKC205544	P25100	Alpha-1D adrenergic receptor	None	289	nM	Ki
TKC205544	P28222	5-hydroxytryptamine receptor 1B	None	5	nM	Ki
TKC205544	P28222	5-hydroxytryptamine receptor 1B	None	16	nM	Ki
TKC205544	P28222	5-hydroxytryptamine receptor 1B	None	39.81	nM	Ki
TKC205544	P28222	5-hydroxytryptamine receptor 1B	None	158.48	nM	Ki
TKC206544	P28222	5-hydroxytryptamine receptor 1B	None	>10000	nM	Ki
TKC205544	P28335	5-hydroxytryptamine receptor 2C	None	>10000	nM	Ki
TKC205544	P28335	5-hydroxytryptamine receptor 2C	None	1690	nM	Ki
TKC205544	P28335	5-hydroxytryptamine receptor 2C	None	645.65	nM	Ki
TKC205544	P28335	5-hydroxytryptamine receptor 2C	None	1000	nM	Ki
TKC206781	P28335	5-hydroxytryptamine receptor 2C	None	2	nM	Ki
TKC111727	P31645	Sodium-dependent serotonin transporter	None	5491	nM	Ki
TKC111738	P31645	Sodium-dependent serotonin transporter	None	2816	nM	Ki
TKC205544	P31645	Sodium-dependent serotonin transporter	None	1000	nM	Ki
TKC027341	P34972	Cannabinoid receptor 2	None	257	nM	Ki
TKC027353	P34972	Cannabinoid receptor 2	None	372	nM	Ki
TKC027353	P34972	Cannabinoid receptor 2	None	229	nM	Ki
TKC027353	P34972	Cannabinoid receptor 2	None	2860	nM	Ki
TKC027353	P34972	Cannabinoid receptor 2	None	10000	nM	Ki
TKC027353	P34972	Cannabinoid receptor 2	None	2.88E+12	nM	Ki
TKC027356	P34972	Cannabinoid receptor 2	None	574	nM	Ki
TKC027364	P34972	Cannabinoid receptor 2	None	153	nM	Ki
TKC027373	P34972	Cannabinoid receptor 2	None	16	nM	Ki
TKC027373	P34972	Cannabinoid receptor 2	None	126	nM	Ki
TKC027373	P34972	Cannabinoid receptor 2	None	96	nM	Ki
TKC027373	P34972	Cannabinoid receptor 2	None	95499258602	nM	Ki
TKC027397	P34972	Cannabinoid receptor 2	None	4780	nM	EC50
TKC095132	P34972	Cannabinoid receptor 2	None	0	nM	Ki
TKC095132	P34972	Cannabinoid receptor 2	None	150	nM	Ki
TKC095132	P34972	Cannabinoid receptor 2	None	0.251189	nM	EC50
TKC095197	P34972	Cannabinoid receptor 2	None	171	nM	Ki
TKC146115	P34972	Cannabinoid receptor 2	None	150	nM	Ki
TKC205544	P34972	Cannabinoid receptor 2	None	20	%	Inhibition
TKC037534	P35228	Nitric oxide synthase, inducible	None	99	%	Inhibition
TKC060880	P35228	Nitric oxide synthase, inducible	None	37000	nM	IC50
TKC077689	P35228	Nitric oxide synthase, inducible	None	>40000	nM	IC50
TKC206319	P35228	Nitric oxide synthase, inducible	None	100	%	Inhibition
TKC013725	P35348	Alpha-1A adrenergic receptor	None	13	nM	IC50
TKC100416	P35348	Alpha-1A adrenergic receptor	None	32	nM	Kd
TKC205544	P35348	Alpha-1A adrenergic receptor	None	398	nM	Kd
TKC205544	P35348	Alpha-1A adrenergic receptor	None	148	nM	Kd
TKC205544	P35348	Alpha-1A adrenergic receptor	None	770	nM	Ki
TKC205544	P35348	Alpha-1A adrenergic receptor	None	199.52	nM	Ki
TKC205544	P35348	Alpha-1A adrenergic receptor	None	3162.28	nM	Ki
TKC205544	P35348	Alpha-1A adrenergic receptor	None	1057	nM	Ki
TKC206544	P35348	Alpha-1A adrenergic receptor	None	>10000	nM	Ki
TKC008359	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC010020	P35354	Prostaglandin G/H synthase 2	None	61	%	Inhibition
TKC010022	P35354	Prostaglandin G/H synthase 2	None	55	%	Inhibition
TKC010023	P35354	Prostaglandin G/H synthase 2	None	57	%	Inhibition
TKC010024	P35354	Prostaglandin G/H synthase 2	None	42	%	Inhibition
TKC010025	P35354	Prostaglandin G/H synthase 2	None	78	%	Inhibition
TKC010026	P35354	Prostaglandin G/H synthase 2	None	17	%	Inhibition
TKC011599	P35354	Prostaglandin G/H synthase 2	None	64	%	Inhibition
TKC012919	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC012941	P35354	Prostaglandin G/H synthase 2	None	8500	nM	IC50
TKC012956	P35354	Prostaglandin G/H synthase 2	None	2200	nM	IC50
TKC012962	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC015443	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC015459	P35354	Prostaglandin G/H synthase 2	None	2200	nM	IC50
TKC015537	P35354	Prostaglandin G/H synthase 2	None	0	%	Inhibition
TKC016794	P35354	Prostaglandin G/H synthase 2	None	40	nM	IC50
TKC019436	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC019466	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC019819	P35354	Prostaglandin G/H synthase 2	None	35	%	Inhibition
TKC019859	P35354	Prostaglandin G/H synthase 2	None	<33	%	Inhibition
TKC020479	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC020796	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC021940	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC022833	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC022834	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC022961	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC026245	P35354	Prostaglandin G/H synthase 2	None	2300	nM	IC50
TKC027200	P35354	Prostaglandin G/H synthase 2	None	700	nM	IC50
TKC028143	P35354	Prostaglandin G/H synthase 2	None	100	%	Inhibition
TKC031202	P35354	Prostaglandin G/H synthase 2	None	3800	nM	IC50
TKC031223	P35354	Prostaglandin G/H synthase 2	None	45	%	Inhibition
TKC032234	P35354	Prostaglandin G/H synthase 2	None	400	nM	IC50
TKC035208	P35354	Prostaglandin G/H synthase 2	None	7	uM	IC60
TKC037534	P35354	Prostaglandin G/H synthase 2	None	97	%	Inhibition
TKC038330	P35354	Prostaglandin G/H synthase 2	None	2900	nM	IC50
TKC041884	P35354	Prostaglandin G/H synthase 2	None	18000	nM	IC50
TKC043993	P35354	Prostaglandin G/H synthase 2	None	98	%	Inhibition
TKC045188	P35354	Prostaglandin G/H synthase 2	None	98	%	Inhibition
TKC048282	P35354	Prostaglandin G/H synthase 2	None	370	nM	IC50
TKC049750	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC049818	P35354	Prostaglandin G/H synthase 2	None	5	ug	IC50
TKC051154	P35354	Prostaglandin G/H synthase 2	None	>61	%	Activity
TKC054011	P35354	Prostaglandin G/H synthase 2	None	9000	nM	IC50
TKC054031	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC054081	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC054090	P35354	Prostaglandin G/H synthase 2	None	8900	nM	IC50
TKC054099	P35354	Prostaglandin G/H synthase 2	None	7800	nM	IC50
TKC054100	P35354	Prostaglandin G/H synthase 2	None	7900	nM	IC50
TKC054101	P35354	Prostaglandin G/H synthase 2	None	8800	nM	IC50
TKC054240	P35354	Prostaglandin G/H synthase 2	None	6700	nM	IC50
TKC054241	P35354	Prostaglandin G/H synthase 2	None	6100	nM	IC50
TKC056482	P35354	Prostaglandin G/H synthase 2	None	40000	nM	IC50
TKC056482	P35354	Prostaglandin G/H synthase 2	None	86000	nM	IC50
TKC056482	P35354	Prostaglandin G/H synthase 2	None	130000	nM	IC50
TKC057308	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC058811	P35354	Prostaglandin G/H synthase 2	None	>85	%	Activity
TKC058812	P35354	Prostaglandin G/H synthase 2	None	>78	%	Activity
TKC060184	P35354	Prostaglandin G/H synthase 2	None	8500	nM	IC50
TKC060216	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC060284	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC060302	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC060303	P35354	Prostaglandin G/H synthase 2	None	7200	nM	IC50
TKC060304	P35354	Prostaglandin G/H synthase 2	None	7600	nM	IC50
TKC060399	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC060602	P35354	Prostaglandin G/H synthase 2	None	6700	nM	IC50
TKC061939	P35354	Prostaglandin G/H synthase 2	None	>10000	nM	IC50
TKC061968	P35354	Prostaglandin G/H synthase 2	None	>10000	nM	IC50
TKC061969	P35354	Prostaglandin G/H synthase 2	None	>10000	nM	IC50
TKC064374	P35354	Prostaglandin G/H synthase 2	None	>73	%	Activity
TKC064407	P35354	Prostaglandin G/H synthase 2	None	>78	%	Activity
TKC065375	P35354	Prostaglandin G/H synthase 2	None	>70	%	Activity
TKC066954	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC070952	P35354	Prostaglandin G/H synthase 2	None	>100000	nM	IC50
TKC071010	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC071640	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC076350	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC077689	P35354	Prostaglandin G/H synthase 2	None	40000	nM	IC50
TKC077689	P35354	Prostaglandin G/H synthase 2	None	295000	nM	IC50
TKC077689	P35354	Prostaglandin G/H synthase 2	None	295000	nM	IC50
TKC077689	P35354	Prostaglandin G/H synthase 2	None	87000	nM	IC50
TKC077703	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC078194	P35354	Prostaglandin G/H synthase 2	None	>74	%	Activity
TKC085168	P35354	Prostaglandin G/H synthase 2	None	<60	%	Inhibition
TKC088678	P35354	Prostaglandin G/H synthase 2	None	>72	%	Activity
TKC095276	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC095567	P35354	Prostaglandin G/H synthase 2	None	>10000	nM	IC50
TKC110247	P35354	Prostaglandin G/H synthase 2	None	>10	ug.mL-1	IC50
TKC113936	P35354	Prostaglandin G/H synthase 2	None	60	%	Inhibition
TKC122543	P35354	Prostaglandin G/H synthase 2	None	30	%	Inhibition
TKC123028	P35354	Prostaglandin G/H synthase 2	None	>72	%	Activity
TKC129152	P35354	Prostaglandin G/H synthase 2	None	>100000	nM	IC50
TKC130084	P35354	Prostaglandin G/H synthase 2	None	37	%	Inhibition
TKC130119	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC130223	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC130577	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC130901	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC135264	P35354	Prostaglandin G/H synthase 2	None	400	nM	IC50
TKC135559	P35354	Prostaglandin G/H synthase 2	None	4600	nM	IC50
TKC139036	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC139322	P35354	Prostaglandin G/H synthase 2	None	>82	%	Activity
TKC139366	P35354	Prostaglandin G/H synthase 2	None	40000	nM	IC50
TKC140627	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC141365	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC141401	P35354	Prostaglandin G/H synthase 2	None	>75	%	Activity
TKC141499	P35354	Prostaglandin G/H synthase 2	None	>87	%	Activity
TKC141601	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC141602	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC141622	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC141805	P35354	Prostaglandin G/H synthase 2	None	40000	nM	IC50
TKC142150	P35354	Prostaglandin G/H synthase 2	None	450000	nM	IC50
TKC142203	P35354	Prostaglandin G/H synthase 2	None	>10000	nM	IC50
TKC142208	P35354	Prostaglandin G/H synthase 2	None	>10000	nM	IC50
TKC142849	P35354	Prostaglandin G/H synthase 2	None	>69	%	Activity
TKC142897	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC142922	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC143527	P35354	Prostaglandin G/H synthase 2	None	97	%	Inhibition
TKC143539	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC143641	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC145295	P35354	Prostaglandin G/H synthase 2	None	22	%	Inhibition
TKC145848	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC145932	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC145968	P35354	Prostaglandin G/H synthase 2	None	>94	%	Activity
TKC146116	P35354	Prostaglandin G/H synthase 2	None	>5.0e+4	nM	IC50
TKC146774	P35354	Prostaglandin G/H synthase 2	None	>78	%	Activity
TKC146857	P35354	Prostaglandin G/H synthase 2	None	600	nM	IC50
TKC149251	P35354	Prostaglandin G/H synthase 2	None	1100	nM	IC50
TKC149759	P35354	Prostaglandin G/H synthase 2	None	100	%	Activity
TKC149924	P35354	Prostaglandin G/H synthase 2	None	800	nM	IC50
TKC149926	P35354	Prostaglandin G/H synthase 2	None	800	nM	IC50
TKC150635	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC150706	P35354	Prostaglandin G/H synthase 2	None	>76	%	Activity
TKC150907	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC151280	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC151284	P35354	Prostaglandin G/H synthase 2	None	33	%	Inhibition
TKC151765	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC152742	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC152813	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC156345	P35354	Prostaglandin G/H synthase 2	None	25	%	Inhibition
TKC156572	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC156716	P35354	Prostaglandin G/H synthase 2	None	2200	nM	IC50
TKC170277	P35354	Prostaglandin G/H synthase 2	None	>50000	nM	IC50
TKC172853	P35354	Prostaglandin G/H synthase 2	None	4700	nM	IC50
TKC174442	P35354	Prostaglandin G/H synthase 2	None	10000	nM	IC50
TKC205509	P35354	Prostaglandin G/H synthase 2	None	540000	nM	IC50
TKC205699	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC205700	P35354	Prostaglandin G/H synthase 2	None	<30	%	Inhibition
TKC206319	P35354	Prostaglandin G/H synthase 2	None	99	%	Inhibition
TKC205544	P35367	Histamine H1 receptor	None	30	%	Inhibition
TKC206544	P35367	Histamine H1 receptor	None	>10000	nM	Ki
TKC013725	P35368	Alpha-1B adrenergic receptor	None	215	nM	IC50
TKC205544	P35368	Alpha-1B adrenergic receptor	None	1	nM	Ki
TKC205544	P35368	Alpha-1B adrenergic receptor	None	158.48	nM	Ki
TKC205544	P35368	Alpha-1B adrenergic receptor	None	2398.83	nM	Ki
TKC205544	P35368	Alpha-1B adrenergic receptor	None	966	nM	Ki
TKC206544	P35368	Alpha-1B adrenergic receptor	None	>10000	nM	Ki
TKC002194	P35372	Mu-type opioid receptor	None	760	nM	Ke
TKC005708	P35372	Mu-type opioid receptor	None	>10000	nM	Ki
TKC093001	P35372	Mu-type opioid receptor	None	10000	nM	Ki
TKC093006	P35372	Mu-type opioid receptor	None	>1000	nM	Ki
TKC093006	P35372	Mu-type opioid receptor	None	>1000	nM	Ki
TKC093010	P35372	Mu-type opioid receptor	None	41	nM	Ki
TKC093012	P35372	Mu-type opioid receptor	None	390	nM	Ki
TKC101289	P35372	Mu-type opioid receptor	None	>5800	nM	Ki
TKC101290	P35372	Mu-type opioid receptor	None	777	nM	Ki
TKC104953	P35372	Mu-type opioid receptor	None	3650	nM	Ke
TKC105684	P35372	Mu-type opioid receptor	None	>10000	nM	Ki
TKC105685	P35372	Mu-type opioid receptor	None	>10000	nM	Ki
TKC109881	P35372	Mu-type opioid receptor	None	>92466	nM	EC50
TKC156630	P35372	Mu-type opioid receptor	None	>1900	nM	Ki
TKC206544	P35372	Mu-type opioid receptor	None	>0	%	Emax
TKC206544	P35372	Mu-type opioid receptor	None	>10000	nM	Ki
TKC206544	P35372	Mu-type opioid receptor	None	>10000	nM	Ki
TKC206544	P35372	Mu-type opioid receptor	None	4370	nM	Ki
TKC206544	P35372	Mu-type opioid receptor	None	>1000	nM	Ki
TKC206544	P35372	Mu-type opioid receptor	None	>10000	nM	Ki
TKC206544	P35372	Mu-type opioid receptor	None	2860	nM	EC50
TKC206544	P35372	Mu-type opioid receptor	None	1370	nM	Ki
TKC206544	P35372	Mu-type opioid receptor	None	>10000	nM	Ki
TKC002194	P41143	Delta-type opioid receptor	None	2830	nM	Ke
TKC005708	P41143	Delta-type opioid receptor	None	>10000	nM	Ki
TKC045774	P41143	Delta-type opioid receptor	None	>64582	nM	EC50
TKC093001	P41143	Delta-type opioid receptor	None	10000	nM	Ki
TKC093006	P41143	Delta-type opioid receptor	None	6690	nM	Ki
TKC093006	P41143	Delta-type opioid receptor	None	6690	nM	Ki
TKC093010	P41143	Delta-type opioid receptor	None	1017	nM	Ki
TKC093012	P41143	Delta-type opioid receptor	None	2840	nM	Ki
TKC101289	P41143	Delta-type opioid receptor	None	>5000	nM	Ki
TKC101290	P41143	Delta-type opioid receptor	None	>5000	nM	Ki
TKC104953	P41143	Delta-type opioid receptor	None	964	nM	Ke
TKC105684	P41143	Delta-type opioid receptor	None	>10000	nM	Ki
TKC105685	P41143	Delta-type opioid receptor	None	>10000	nM	Ki
TKC109881	P41143	Delta-type opioid receptor	None	>92466	nM	EC50
TKC109881	P41143	Delta-type opioid receptor	None	>92466	nM	EC50
TKC156630	P41143	Delta-type opioid receptor	None	>10000	nM	Ki
TKC206544	P41143	Delta-type opioid receptor	None	3990	nM	Ki
TKC206544	P41143	Delta-type opioid receptor	None	>10000	nM	Ki
TKC206544	P41143	Delta-type opioid receptor	None	5790	nM	Ki
TKC206544	P41143	Delta-type opioid receptor	None	5790	nM	Ki
TKC206544	P41143	Delta-type opioid receptor	None	>10000	nM	Ki
TKC206544	P41143	Delta-type opioid receptor	None	>10000	nM	Ki
TKC206544	P41143	Delta-type opioid receptor	None	>10000	nM	Ki
TKC206544	P41143	Delta-type opioid receptor	None	>10000	nM	Ki
TKC004780	P41145	Kappa-type opioid receptor	None	1	nM	Ki
TKC004780	P41145	Kappa-type opioid receptor	None	140	nM	Ki
TKC004780	P41145	Kappa-type opioid receptor	None	4.6	nM	Ki
TKC004780	P41145	Kappa-type opioid receptor	None	31.6	nM	Ki
TKC005708	P41145	Kappa-type opioid receptor	None	390	nM	Ki
TKC080736	P41145	Kappa-type opioid receptor	None	>2000	nM	EC50
TKC093001	P41145	Kappa-type opioid receptor	None	17	nM	Ki
TKC093006	P41145	Kappa-type opioid receptor	None	2	nM	Ki
TKC093006	P41145	Kappa-type opioid receptor	None	7.2	nM	Ki
TKC093006	P41145	Kappa-type opioid receptor	None	1.8	nM	Ki
TKC093008	P41145	Kappa-type opioid receptor	None	5	nM	Ki
TKC093010	P41145	Kappa-type opioid receptor	None	0	nM	EC50
TKC093011	P41145	Kappa-type opioid receptor	None	2	nM	Ki
TKC093012	P41145	Kappa-type opioid receptor	None	0	nM	EC50
TKC093013	P41145	Kappa-type opioid receptor	None	2	nM	Ki
TKC093014	P41145	Kappa-type opioid receptor	None	147	nM	Ki
TKC093016	P41145	Kappa-type opioid receptor	None	35	nM	Ki
TKC093018	P41145	Kappa-type opioid receptor	None	2	nM	Ki
TKC093019	P41145	Kappa-type opioid receptor	None	141	nM	Ki
TKC093021	P41145	Kappa-type opioid receptor	None	29	nM	Ki
TKC093022	P41145	Kappa-type opioid receptor	None	31	nM	Ki
TKC093023	P41145	Kappa-type opioid receptor	None	3	nM	Ki
TKC093024	P41145	Kappa-type opioid receptor	None	4	nM	Ki
TKC093025	P41145	Kappa-type opioid receptor	None	>81	%	Emax
TKC101289	P41145	Kappa-type opioid receptor	None	10	nM	EC50
TKC101289	P41145	Kappa-type opioid receptor	None	1233	nM	Ki
TKC101290	P41145	Kappa-type opioid receptor	None	7	nM	Ki
TKC103606	P41145	Kappa-type opioid receptor	None	0	nM	Ki
TKC104953	P41145	Kappa-type opioid receptor	None	7	nM	EC50
TKC104953	P41145	Kappa-type opioid receptor	None	424	nM	Ki
TKC104956	P41145	Kappa-type opioid receptor	None	41	nM	Ki
TKC105684	P41145	Kappa-type opioid receptor	None	6	nM	Ki
TKC105684	P41145	Kappa-type opioid receptor	None	3	nM	EC50
TKC105685	P41145	Kappa-type opioid receptor	None	300	nM	Ki
TKC106987	P41145	Kappa-type opioid receptor	None	641	nM	Ki
TKC106989	P41145	Kappa-type opioid receptor	None	>1000	nM	Ki
TKC156630	P41145	Kappa-type opioid receptor	None	1900	nM	Ki
TKC206540	P41145	Kappa-type opioid receptor	None	>0	%	Emax
TKC206544	P41145	Kappa-type opioid receptor	None	0	nM	EC50
TKC206544	P41145	Kappa-type opioid receptor	None	16	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	10	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	38	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	1.3	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	0.75	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	40	nM	EC50
TKC206544	P41145	Kappa-type opioid receptor	None	7.4	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	0.36	nM	EC50
TKC206544	P41145	Kappa-type opioid receptor	None	40	nM	EC50
TKC206544	P41145	Kappa-type opioid receptor	None	0.03	nM	EC50
TKC206544	P41145	Kappa-type opioid receptor	None	1.7	nM	EC50
TKC206544	P41145	Kappa-type opioid receptor	None	45	nM	EC50
TKC206544	P41145	Kappa-type opioid receptor	None	1.9	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	1.3	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	2.82	nM	EC50
TKC206544	P41145	Kappa-type opioid receptor	None	1.24	nM	EC50
TKC206544	P41145	Kappa-type opioid receptor	None	1.3	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	2.5	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	7.5	nM	EC50
TKC206544	P41145	Kappa-type opioid receptor	None	7.4	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	3	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	45	nM	EC50
TKC206544	P41145	Kappa-type opioid receptor	None	2.4	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	0.21	nM	EC50
TKC206544	P41145	Kappa-type opioid receptor	None	0.8	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	1.9	nM	Ki
TKC206544	P41145	Kappa-type opioid receptor	None	10	nM	EC50
TKC118419	P42338	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	None	8	nM	Kd
TKC118419	P42338	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	None	7.6	nM	Kd
TKC118419	P42338	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	None	10	nM	IC50
TKC118419	P42338	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	None	15	nM	IC50
TKC118419	P42338	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	None	14	nM	IC50
TKC022945	P42345	Serine/threonine-protein kinase mTOR	None	4645	nM	Potency
TKC032619	P42345	Serine/threonine-protein kinase mTOR	None	2931	nM	Potency
TKC035272	P42345	Serine/threonine-protein kinase mTOR	None	2612	nM	Potency
TKC035984	P42345	Serine/threonine-protein kinase mTOR	None	4	nM	Potency
TKC084630	P42345	Serine/threonine-protein kinase mTOR	None	3690	nM	Potency
TKC087988	P42345	Serine/threonine-protein kinase mTOR	None	4645	nM	Potency
TKC092297	P42345	Serine/threonine-protein kinase mTOR	None	13092	nM	Potency
TKC118419	P42345	Serine/threonine-protein kinase mTOR	None	40	nM	IC50
TKC118419	P42345	Serine/threonine-protein kinase mTOR	None	9200	nM	Kd
TKC205544	P42345	Serine/threonine-protein kinase mTOR	None	14689	nM	Potency
TKC206622	P42345	Serine/threonine-protein kinase mTOR	None	23281	nM	Potency
TKC206688	P42345	Serine/threonine-protein kinase mTOR	None	16482	nM	Potency
TKC025058	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	1000	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	5	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	19	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	55	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	55000	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	89	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	5	nM	IC50
TKC118419	P48736	Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	None	15	nM	Kd
TKC118419	P53778	Mitogen-activated protein kinase 12	None	75	%	Inhibition
TKC016794	P55085	Proteinase-activated receptor 2	None	14	nM	IC50
TKC206816	P56373	P2X purinoceptor 3	None	1600	nM	IC50
TKC000046	Q12809	Potassium voltage-gated channel subfamily H member 2	None	14	%	Inhibition
TKC000047	Q12809	Potassium voltage-gated channel subfamily H member 2	None	14	%	Inhibition
TKC005704	Q12809	Potassium voltage-gated channel subfamily H member 2	None	0	%	Inhibition
TKC005753	Q12809	Potassium voltage-gated channel subfamily H member 2	None	19	%	Inhibition
TKC006670	Q12809	Potassium voltage-gated channel subfamily H member 2	None	12	%	Inhibition
TKC006671	Q12809	Potassium voltage-gated channel subfamily H member 2	None	0	%	Inhibition
TKC012725	Q12809	Potassium voltage-gated channel subfamily H member 2	None	51	%	Inhibition
TKC013753	Q12809	Potassium voltage-gated channel subfamily H member 2	None	15849	nM	Potency
TKC020459	Q12809	Potassium voltage-gated channel subfamily H member 2	None	1585	nM	Potency
TKC038011	Q12809	Potassium voltage-gated channel subfamily H member 2	None	109648	nM	IC50
TKC070824	Q12809	Potassium voltage-gated channel subfamily H member 2	None	2	%	Inhibition
TKC073696	Q12809	Potassium voltage-gated channel subfamily H member 2	None	3	%	Inhibition
TKC078496	Q12809	Potassium voltage-gated channel subfamily H member 2	None	39811	nM	Potency
TKC084630	Q12809	Potassium voltage-gated channel subfamily H member 2	None	1413	nM	Potency
TKC087664	Q12809	Potassium voltage-gated channel subfamily H member 2	None	14125	nM	Potency
TKC087988	Q12809	Potassium voltage-gated channel subfamily H member 2	None	5623	nM	Potency
TKC087991	Q12809	Potassium voltage-gated channel subfamily H member 2	None	39811	nM	Potency
TKC092297	Q12809	Potassium voltage-gated channel subfamily H member 2	None	35481	nM	Potency
TKC101269	Q12809	Potassium voltage-gated channel subfamily H member 2	None	43	%	Inhibition
TKC101481	Q12809	Potassium voltage-gated channel subfamily H member 2	None	55	%	Inhibition
TKC103025	Q12809	Potassium voltage-gated channel subfamily H member 2	None	4	%	Inhibition
TKC103150	Q12809	Potassium voltage-gated channel subfamily H member 2	None	22387	nM	Potency
TKC105356	Q12809	Potassium voltage-gated channel subfamily H member 2	None	112	nM	Potency
TKC106909	Q12809	Potassium voltage-gated channel subfamily H member 2	None	>40	%	Inhibition
TKC107086	Q12809	Potassium voltage-gated channel subfamily H member 2	None	25119	nM	Potency
TKC112576	Q12809	Potassium voltage-gated channel subfamily H member 2	None	5800	nM	IC50
TKC112576	Q12809	Potassium voltage-gated channel subfamily H member 2	None	5800	nM	IC50
TKC112745	Q12809	Potassium voltage-gated channel subfamily H member 2	None	25119	nM	Potency
TKC118419	Q12809	Potassium voltage-gated channel subfamily H member 2	None	17783	nM	Potency
TKC205892	Q12809	Potassium voltage-gated channel subfamily H member 2	None	11	%	Inhibition
TKC206041	Q12809	Potassium voltage-gated channel subfamily H member 2	None	13	%	Inhibition
TKC206760	Q12809	Potassium voltage-gated channel subfamily H member 2	None	50119	nM	Potency
TKC206770	Q12809	Potassium voltage-gated channel subfamily H member 2	None	31623	nM	Potency
TKC206812	Q12809	Potassium voltage-gated channel subfamily H member 2	None	17783	nM	Potency
TKC206816	Q12809	Potassium voltage-gated channel subfamily H member 2	None	50119	nM	Potency
TKC206544	Q13255	Metabotropic glutamate receptor 1	None	>10000	nM	Ki
TKC109622	Q13822	Ectonucleotide pyrophosphatase/phosphodiesterase family member 2	None	10300	nM	IC50
TKC087988	Q16539	Mitogen-activated protein kinase 14	None	2529	nM	IC50
TKC118419	Q16539	Mitogen-activated protein kinase 14	None	86	%	Inhibition
TKC019571	Q7Z2W7	Transient receptor potential cation channel subfamily M member 8	None	100	uM	Activity
TKC074866	Q7Z2W7	Transient receptor potential cation channel subfamily M member 8	None	5900000	nM	EC50
TKC085168	Q7Z2W7	Transient receptor potential cation channel subfamily M member 8	None	10100	nM	EC50
TKC086929	Q7Z2W7	Transient receptor potential cation channel subfamily M member 8	None	3000	nM	EC50
TKC013738	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	24	nM	Ki
TKC013738	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	23	nM	Ki
TKC013738	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	14	nM	Ki
TKC013739	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	129	nM	Ki
TKC023433	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	5000	nM	IC50
TKC027364	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	1300	nM	EC50
TKC027373	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	6200	nM	EC50
TKC027397	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	6600	nM	EC50
TKC033765	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	176	%	Activity
TKC034016	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	94	%	Activity
TKC036488	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	22	%	Activity
TKC074866	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	>102	uM	Activity
TKC090445	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	0	nM	Ki
TKC092268	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	0	nM	EC50
TKC092268	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	0.48	nM	Ki
TKC092268	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	1.2	nM	Ki
TKC092268	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	19	nM	EC50
TKC092268	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	0.92	nM	EC50
TKC098861	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	115	%	Activity
TKC116435	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	1400	nM	IC50
TKC122664	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	31	%	Activity
TKC146124	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	45	%	Activity
TKC151092	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	115	%	Activity
TKC205687	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	1	nM	Kd
TKC206945	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	6	nM	Ki
TKC206945	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	4000	nM	IC50
TKC206945	Q8NER1	Transient receptor potential cation channel subfamily V member 1	None	5.9	nM	Ki
TKC022931	Q8NET8	Transient receptor potential cation channel subfamily V member 3	None	100	uM	Activity
TKC206688	Q99720	Sigma non-opioid intracellular receptor 1	None	35600	nM	Ki
TKC206759	Q99720	Sigma non-opioid intracellular receptor 1	None	1200	nM	Ki
TKC206816	Q99720	Sigma non-opioid intracellular receptor 1	None	260	nM	Ki
TKC119168	Q9Y5Y9	Sodium channel protein type 10 subunit alpha	None	88	%	Inhibition
TKC119169	Q9Y5Y9	Sodium channel protein type 10 subunit alpha	None	9000	nM	IC50