Basic Information

Name [ICD-11: EA90]
Protein Number 34
Molecule Number 526

Active subnetwork

Terpenoid-protein target Activity Association

ID Uniport Pref_name Gene name value unit type
TKC118419 O75116 Rho-associated protein kinase 2 None 99 % Activity
TKC007127 P00533 Epidermal growth factor receptor None 19 % Inhibition
TKC025462 P00533 Epidermal growth factor receptor None >200 ug.mL-1 IC50
TKC025466 P00533 Epidermal growth factor receptor None >200 ug.mL-1 IC50
TKC025475 P00533 Epidermal growth factor receptor None 197 ug.mL-1 IC50
TKC071640 P00533 Epidermal growth factor receptor None >20000 nM IC50
TKC076041 P00533 Epidermal growth factor receptor None 75 % Inhibition
TKC077689 P00533 Epidermal growth factor receptor None >20000 nM IC50
TKC106319 P00533 Epidermal growth factor receptor None 56 nM IC50
TKC108557 P00533 Epidermal growth factor receptor None 0.82 nM Kd
TKC151761 P00533 Epidermal growth factor receptor None >10000 nM IC50
TKC200866 P00533 Epidermal growth factor receptor None >10000 nM IC50
TKC005744 P00742 Coagulation factor X None 27900 nM IC50
TKC012492 P00742 Coagulation factor X None 13385 nM Ki
TKC013400 P00742 Coagulation factor X None 2500 nM IC50
TKC013430 P00742 Coagulation factor X None 11418 nM IC50
TKC055903 P00742 Coagulation factor X None >20000 nM IC50
TKC107140 P00742 Coagulation factor X None 7991 nM Ki
TKC124270 P00742 Coagulation factor X None 27558 nM Ki
TKC128698 P00742 Coagulation factor X None 7200 nM IC50
TKC128699 P00742 Coagulation factor X None 7165 nM IC50
TKC205733 P00742 Coagulation factor X None 1023 nM IC50
TKC051021 P01375 Tumor necrosis factor None 9 nM Kd
TKC051029 P01375 Tumor necrosis factor None 9 nM Kd
TKC055869 P01375 Tumor necrosis factor None 10880 nM IC50
TKC063751 P01375 Tumor necrosis factor None 19 nM Kd
TKC064986 P01375 Tumor necrosis factor None 3 nM Kd
TKC075769 P01375 Tumor necrosis factor None 376 nM Potency
TKC101833 P01375 Tumor necrosis factor None 8 nM Kd
TKC145547 P01375 Tumor necrosis factor None 2 nM Kd
TKC148618 P01375 Tumor necrosis factor None 17 nM Kd
TKC151763 P01375 Tumor necrosis factor None 8 nM Kd
TKC151876 P01375 Tumor necrosis factor None 6 % Inhibition
TKC206051 P07858 Cathepsin B None 103500 nM IC50
TKC024886 P08069 Insulin-like growth factor 1 receptor None 11800 nM IC50
TKC025690 P08069 Insulin-like growth factor 1 receptor None 3310 nM IC50
TKC115259 P08069 Insulin-like growth factor 1 receptor None 3160 nM IC50
TKC115261 P08069 Insulin-like growth factor 1 receptor None 2420 nM IC50
TKC115272 P08069 Insulin-like growth factor 1 receptor None >100000 nM IC50
TKC115273 P08069 Insulin-like growth factor 1 receptor None 2300 nM IC50
TKC152148 P08069 Insulin-like growth factor 1 receptor None 2770 nM IC50
TKC152157 P08069 Insulin-like growth factor 1 receptor None 2460 nM IC50
TKC174547 P08069 Insulin-like growth factor 1 receptor None >100000 nM IC50
TKC151523 P08908 5-hydroxytryptamine receptor 1A None >100000 nM Ki
TKC205544 P08908 5-hydroxytryptamine receptor 1A None 4500 nM Ki
TKC205544 P08908 5-hydroxytryptamine receptor 1A None 1500 nM Ki
TKC205544 P08908 5-hydroxytryptamine receptor 1A None 642 nM Ki
TKC205544 P08908 5-hydroxytryptamine receptor 1A None 1258.92 nM Ki
TKC206544 P08908 5-hydroxytryptamine receptor 1A None >10000 nM Ki
TKC206549 P08908 5-hydroxytryptamine receptor 1A None 30 pM well-1 cAMP
TKC020117 P09917 Polyunsaturated fatty acid 5-lipoxygenase None -67 % Inhibition
TKC024485 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >50000 nM IC50
TKC024587 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 600 nM IC50
TKC024956 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 18000 nM IC50
TKC024992 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 450 nM IC50
TKC024993 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 14000 nM IC50
TKC025965 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >150000 nM IC50
TKC026303 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 4600 nM IC50
TKC026309 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 680 nM IC50
TKC027255 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >67 % Activity
TKC034201 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >200000 nM IC50
TKC040026 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 72 % Inhibition
TKC051154 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 2700 nM IC50
TKC056482 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >64 % Activity
TKC058811 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 42000 nM IC50
TKC058812 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >93 % Activity
TKC064374 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 42000 nM IC50
TKC064407 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >72 % Activity
TKC065375 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >70 % Activity
TKC071640 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >60 % Activity
TKC076350 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 100 % Activity
TKC077689 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 100 % Activity
TKC077703 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >86 % Activity
TKC078194 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 31800 nM IC50
TKC082039 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 48 % Inhibition
TKC088678 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 24800 nM IC50
TKC089448 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 35 % Inhibition
TKC094647 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 97 % Activity
TKC107943 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 2000 nM IC50
TKC123028 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 30400 nM IC50
TKC124303 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 750 nM IC50
TKC133309 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >200000 nM IC50
TKC133656 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 25100 nM IC50
TKC134278 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >200000 nM IC50
TKC139322 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >67 % Activity
TKC139366 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 3000 nM IC50
TKC141401 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 42000 nM IC50
TKC141499 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 25700 nM IC50
TKC141805 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >53 % Activity
TKC142849 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >70 % Activity
TKC142897 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 30600 nM IC50
TKC142922 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >61 % Activity
TKC143539 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 100 % Activity
TKC145848 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 42000 nM IC50
TKC145932 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >56 % Activity
TKC145968 P09917 Polyunsaturated fatty acid 5-lipoxygenase None 100 % Activity
TKC146774 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >63 % Activity
TKC149759 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >73 % Activity
TKC150706 P09917 Polyunsaturated fatty acid 5-lipoxygenase None >62 % Activity
TKC087988 P0DMS8 Adenosine receptor A3 None 2357 nM Ki
TKC096012 P0DMS8 Adenosine receptor A3 None 2982 nM Ki
TKC205544 P0DMS8 Adenosine receptor A3 None 95 nM IC50
TKC206779 P0DMS8 Adenosine receptor A3 None 2674 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 170 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 260 nM IC50
TKC035272 P10415 Apoptosis regulator Bcl-2 None 320 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 440 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 440 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 1191 nM IC50
TKC035272 P10415 Apoptosis regulator Bcl-2 None 450 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 320 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 600 nM IC50
TKC035272 P10415 Apoptosis regulator Bcl-2 None 420 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 10100 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 4800 nM Kd
TKC035272 P10415 Apoptosis regulator Bcl-2 None 2110 nM IC50
TKC035272 P10415 Apoptosis regulator Bcl-2 None 558 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 320 nM Ki
TKC134945 P10415 Apoptosis regulator Bcl-2 None 1460 nM Ki
TKC151761 P10415 Apoptosis regulator Bcl-2 None >10000 nM GI50
TKC200866 P10415 Apoptosis regulator Bcl-2 None >10000 nM GI50
TKC000075 P11473 Vitamin D3 receptor None 70795 nM Potency
TKC002371 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC005454 P11473 Vitamin D3 receptor None 7080 nM Potency
TKC008359 P11473 Vitamin D3 receptor None 28184 nM Potency
TKC011412 P11473 Vitamin D3 receptor None 19953 nM Potency
TKC013736 P11473 Vitamin D3 receptor None 11220 nM Potency
TKC013755 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC013760 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC014568 P11473 Vitamin D3 receptor None 63096 nM Potency
TKC016371 P11473 Vitamin D3 receptor None 56234 nM Potency
TKC017379 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC020031 P11473 Vitamin D3 receptor None 100000 nM Potency
TKC020117 P11473 Vitamin D3 receptor None 56234 nM Potency
TKC027192 P11473 Vitamin D3 receptor None 35481 nM Potency
TKC030239 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC032619 P11473 Vitamin D3 receptor None 31623 nM Potency
TKC032913 P11473 Vitamin D3 receptor None 70795 nM Potency
TKC034083 P11473 Vitamin D3 receptor None 39811 nM Potency
TKC034760 P11473 Vitamin D3 receptor None 35481 nM Potency
TKC035208 P11473 Vitamin D3 receptor None 39811 nM Potency
TKC035272 P11473 Vitamin D3 receptor None 6310 nM Potency
TKC037521 P11473 Vitamin D3 receptor None 79433 nM Potency
TKC038268 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC038273 P11473 Vitamin D3 receptor None 56234 nM Potency
TKC038706 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC041160 P11473 Vitamin D3 receptor None 79433 nM Potency
TKC043519 P11473 Vitamin D3 receptor None 79433 nM Potency
TKC053095 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC053227 P11473 Vitamin D3 receptor None 14125 nM Potency
TKC053825 P11473 Vitamin D3 receptor None 35481 nM Potency
TKC055219 P11473 Vitamin D3 receptor None 100000 nM Potency
TKC057133 P11473 Vitamin D3 receptor None 39811 nM Potency
TKC062321 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC062327 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC062332 P11473 Vitamin D3 receptor None 70795 nM Potency
TKC062333 P11473 Vitamin D3 receptor None 39811 nM Potency
TKC062669 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC066096 P11473 Vitamin D3 receptor None 28184 nM Potency
TKC066169 P11473 Vitamin D3 receptor None 7943 nM Potency
TKC073833 P11473 Vitamin D3 receptor None 56234 nM Potency
TKC073873 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC074866 P11473 Vitamin D3 receptor None 1 nM Potency
TKC075769 P11473 Vitamin D3 receptor None 562 nM Potency
TKC082279 P11473 Vitamin D3 receptor None 70795 nM Potency
TKC082378 P11473 Vitamin D3 receptor None 25119 nM Potency
TKC083025 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC086929 P11473 Vitamin D3 receptor None 39811 nM Potency
TKC087533 P11473 Vitamin D3 receptor None 56234 nM Potency
TKC087664 P11473 Vitamin D3 receptor None 100000 nM Potency
TKC087988 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC091895 P11473 Vitamin D3 receptor None 79433 nM Potency
TKC092297 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC092348 P11473 Vitamin D3 receptor None 39811 nM Potency
TKC093161 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC095442 P11473 Vitamin D3 receptor None 39811 nM Potency
TKC095452 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC096012 P11473 Vitamin D3 receptor None 31623 nM Potency
TKC097937 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC098345 P11473 Vitamin D3 receptor None 28184 nM Potency
TKC098704 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC099703 P11473 Vitamin D3 receptor None 39811 nM Potency
TKC100636 P11473 Vitamin D3 receptor None 3981 nM Potency
TKC100644 P11473 Vitamin D3 receptor None 35481 nM Potency
TKC100701 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC101052 P11473 Vitamin D3 receptor None 56234 nM Potency
TKC101598 P11473 Vitamin D3 receptor None 56234 nM Potency
TKC102204 P11473 Vitamin D3 receptor None 28184 nM Potency
TKC102407 P11473 Vitamin D3 receptor None 15849 nM Potency
TKC102540 P11473 Vitamin D3 receptor None 35481 nM Potency
TKC102593 P11473 Vitamin D3 receptor None 7080 nM Potency
TKC102939 P11473 Vitamin D3 receptor None 63096 nM Potency
TKC103023 P11473 Vitamin D3 receptor None 28184 nM Potency
TKC103159 P11473 Vitamin D3 receptor None 100000 nM Potency
TKC103257 P11473 Vitamin D3 receptor None 3162 nM Potency
TKC103542 P11473 Vitamin D3 receptor None 28184 nM Potency
TKC103736 P11473 Vitamin D3 receptor None 3548 nM Potency
TKC104404 P11473 Vitamin D3 receptor None 28184 nM Potency
TKC104960 P11473 Vitamin D3 receptor None 79433 nM Potency
TKC104961 P11473 Vitamin D3 receptor None 35481 nM Potency
TKC105153 P11473 Vitamin D3 receptor None 7943 nM Potency
TKC105295 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC105424 P11473 Vitamin D3 receptor None 19953 nM Potency
TKC105932 P11473 Vitamin D3 receptor None 63096 nM Potency
TKC106240 P11473 Vitamin D3 receptor None >50000 nM IC50
TKC106250 P11473 Vitamin D3 receptor None >50000 nM IC50
TKC106301 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC106364 P11473 Vitamin D3 receptor None 7080 nM Potency
TKC106367 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC106426 P11473 Vitamin D3 receptor None 14125 nM Potency
TKC107086 P11473 Vitamin D3 receptor None 31623 nM Potency
TKC107332 P11473 Vitamin D3 receptor None 19953 nM Potency
TKC107625 P11473 Vitamin D3 receptor None 56234 nM Potency
TKC107627 P11473 Vitamin D3 receptor None 35481 nM Potency
TKC107735 P11473 Vitamin D3 receptor None 17783 nM Potency
TKC107775 P11473 Vitamin D3 receptor None 100000 nM Potency
TKC107830 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC109619 P11473 Vitamin D3 receptor None >50000 nM IC50
TKC109849 P11473 Vitamin D3 receptor None >100000 nM IC50
TKC109996 P11473 Vitamin D3 receptor None 100000 nM Potency
TKC111464 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC112754 P11473 Vitamin D3 receptor None 79433 nM Potency
TKC112759 P11473 Vitamin D3 receptor None 70795 nM Potency
TKC112784 P11473 Vitamin D3 receptor None 19953 nM Potency
TKC112785 P11473 Vitamin D3 receptor None >40100 nM IC50
TKC112787 P11473 Vitamin D3 receptor None >14500 nM IC50
TKC112792 P11473 Vitamin D3 receptor None 28184 nM Potency
TKC112906 P11473 Vitamin D3 receptor None 25119 nM Potency
TKC113063 P11473 Vitamin D3 receptor None 5805 nM Potency
TKC113146 P11473 Vitamin D3 receptor None 39811 nM Potency
TKC113150 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC113161 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC113663 P11473 Vitamin D3 receptor None 35481 nM Potency
TKC114511 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC114568 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC114819 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC115268 P11473 Vitamin D3 receptor None 0 nM EC50
TKC115284 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC115284 P11473 Vitamin D3 receptor None >2408 uM Activity
TKC118419 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC122884 P11473 Vitamin D3 receptor None 35481 nM Potency
TKC122892 P11473 Vitamin D3 receptor None 0 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 2 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 1 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 0.08 nM IC50
TKC122892 P11473 Vitamin D3 receptor None 7.7 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 0.7 nM IC50
TKC122892 P11473 Vitamin D3 receptor None 0.8 nM IC50
TKC122892 P11473 Vitamin D3 receptor None 322 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 0.06 nM IC50
TKC122892 P11473 Vitamin D3 receptor None 0.35 nM IC50
TKC122892 P11473 Vitamin D3 receptor None 3.9 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 10 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 0.3 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 0.16 nM IC50
TKC122892 P11473 Vitamin D3 receptor None 0.065 nM Kd
TKC122892 P11473 Vitamin D3 receptor None 9 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 0.5 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 0.555 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 1 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 13 nM IC50
TKC122892 P11473 Vitamin D3 receptor None 1.24 nM IC50
TKC122892 P11473 Vitamin D3 receptor None 0.04 nM IC50
TKC122892 P11473 Vitamin D3 receptor None >0.900000 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 3 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 0.026 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 7.7 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 15 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 1.6 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 0.0953 nM IC50
TKC122892 P11473 Vitamin D3 receptor None 0.011 nM EC50
TKC122892 P11473 Vitamin D3 receptor None 24 nM Kd
TKC134702 P11473 Vitamin D3 receptor None 31623 nM Potency
TKC136931 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC143885 P11473 Vitamin D3 receptor None 79433 nM Potency
TKC147290 P11473 Vitamin D3 receptor None 25119 nM Potency
TKC147303 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC148601 P11473 Vitamin D3 receptor None 35481 nM Potency
TKC149827 P11473 Vitamin D3 receptor None 14125 nM Potency
TKC151237 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC151571 P11473 Vitamin D3 receptor None 22387 nM Potency
TKC151609 P11473 Vitamin D3 receptor None 79433 nM Potency
TKC151675 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC151758 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC151784 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC151885 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC174441 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC205788 P11473 Vitamin D3 receptor None 0 nM ED50
TKC205791 P11473 Vitamin D3 receptor None 1 nM IC50
TKC205796 P11473 Vitamin D3 receptor None 631 nM Potency
TKC205798 P11473 Vitamin D3 receptor None 11 % Activity
TKC206385 P11473 Vitamin D3 receptor None >44 uM Activity
TKC206544 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC206652 P11473 Vitamin D3 receptor None 562 nM Potency
TKC206669 P11473 Vitamin D3 receptor None >50000 nM IC50
TKC206672 P11473 Vitamin D3 receptor None >50000 nM IC50
TKC206758 P11473 Vitamin D3 receptor None 56234 nM Potency
TKC206760 P11473 Vitamin D3 receptor None 8913 nM Potency
TKC206760 P11473 Vitamin D3 receptor None 6 % Activity
TKC206760 P11473 Vitamin D3 receptor None 330 nM Kd
TKC206761 P11473 Vitamin D3 receptor None >15100 nM IC50
TKC206780 P11473 Vitamin D3 receptor None 89125 nM Potency
TKC206812 P11473 Vitamin D3 receptor None 44668 nM Potency
TKC206812 P11473 Vitamin D3 receptor None 2000 nM IC50
TKC206816 P11473 Vitamin D3 receptor None 15849 nM Potency
TKC206876 P11473 Vitamin D3 receptor None 79433 nM Potency
TKC206884 P11473 Vitamin D3 receptor None 50119 nM Potency
TKC206884 P11473 Vitamin D3 receptor None >150000 nM EC50
TKC206901 P11473 Vitamin D3 receptor None 31623 nM Potency
TKC206902 P11473 Vitamin D3 receptor None 35481 nM Potency
TKC206960 P11473 Vitamin D3 receptor None 17783 nM Potency
TKC021325 P11509 Cytochrome P450 2A6 None 840 nM Ki
TKC021325 P11509 Cytochrome P450 2A6 None 2000 nM Ki
TKC021332 P11509 Cytochrome P450 2A6 None 840 nM Ki
TKC039868 P11509 Cytochrome P450 2A6 None 15 % Drug metabolism
TKC110956 P11509 Cytochrome P450 2A6 None <0 pmol/min Drug metabolism
TKC026583 P11802 Cyclin-dependent kinase 4 None 9 ug.mL-1 IC50
TKC113582 P11802 Cyclin-dependent kinase 4 None 10 ug.mL-1 IC50
TKC013755 P13631 Retinoic acid receptor gamma None 1 nM Kd
TKC013755 P13631 Retinoic acid receptor gamma None 148 nM Kd
TKC013755 P13631 Retinoic acid receptor gamma None 45 nM EC50
TKC013755 P13631 Retinoic acid receptor gamma None 74 nM EC50
TKC013755 P13631 Retinoic acid receptor gamma None 6 nM EC50
TKC013755 P13631 Retinoic acid receptor gamma None 12 nM EC50
TKC013755 P13631 Retinoic acid receptor gamma None 45 nM EC50
TKC013755 P13631 Retinoic acid receptor gamma None 1 nM Ki
TKC013755 P13631 Retinoic acid receptor gamma None 148 nM Kd
TKC013755 P13631 Retinoic acid receptor gamma None 6 nM EC50
TKC013755 P13631 Retinoic acid receptor gamma None 4 nM EC50
TKC013755 P13631 Retinoic acid receptor gamma None 6 nM EC50
TKC013755 P13631 Retinoic acid receptor gamma None 45 nM EC50
TKC013755 P13631 Retinoic acid receptor gamma None 22 nM Kd
TKC092297 P13631 Retinoic acid receptor gamma None >400 nM Ki
TKC096012 P13631 Retinoic acid receptor gamma None 0 nM Ki
TKC096012 P13631 Retinoic acid receptor gamma None 18 nM Kd
TKC096012 P13631 Retinoic acid receptor gamma None 18 nM Kd
TKC096012 P13631 Retinoic acid receptor gamma None 6 nM EC50
TKC096012 P13631 Retinoic acid receptor gamma None 16 nM Kd
TKC096012 P13631 Retinoic acid receptor gamma None 19 nM EC50
TKC096012 P13631 Retinoic acid receptor gamma None 18 nM IC50
TKC096012 P13631 Retinoic acid receptor gamma None 19 nM Kd
TKC096012 P13631 Retinoic acid receptor gamma None 33 nM EC50
TKC096012 P13631 Retinoic acid receptor gamma None 20 nM EC50
TKC096012 P13631 Retinoic acid receptor gamma None 0.5 nM EC50
TKC096012 P13631 Retinoic acid receptor gamma None 8 nM EC50
TKC096012 P13631 Retinoic acid receptor gamma None 0.3 nM Kd
TKC096012 P13631 Retinoic acid receptor gamma None 18 nM Kd
TKC096012 P13631 Retinoic acid receptor gamma None 10 nM EC50
TKC096012 P13631 Retinoic acid receptor gamma None 18 nM Kd
TKC096012 P13631 Retinoic acid receptor gamma None 18 nM Kd
TKC096012 P13631 Retinoic acid receptor gamma None 3 nM Kd
TKC096012 P13631 Retinoic acid receptor gamma None 0.5 nM IC50
TKC096012 P13631 Retinoic acid receptor gamma None 0.62 nM IC50
TKC096012 P13631 Retinoic acid receptor gamma None 0.7 nM Ki
TKC096012 P13631 Retinoic acid receptor gamma None 0.2 nM Kd
TKC096012 P13631 Retinoic acid receptor gamma None 0.2 nM EC50
TKC096012 P13631 Retinoic acid receptor gamma None 0.5 nM EC50
TKC096012 P13631 Retinoic acid receptor gamma None 0.5 nM Ki
TKC096012 P13631 Retinoic acid receptor gamma None 10 nM EC50
TKC096012 P13631 Retinoic acid receptor gamma None 0.5 nM EC50
TKC096012 P13631 Retinoic acid receptor gamma None 0.6 nM Ki
TKC096012 P13631 Retinoic acid receptor gamma None 15 nM EC50
TKC096012 P13631 Retinoic acid receptor gamma None 18 nM Kd
TKC206482 P13631 Retinoic acid receptor gamma None 6 nM EC50
TKC206812 P13631 Retinoic acid receptor gamma None >100000 nM EC50
TKC205544 P14416 D(2) dopamine receptor None 687 nM Ki
TKC205544 P14416 D(2) dopamine receptor None 280 nM Ki
TKC205544 P14416 D(2) dopamine receptor None 398.1 nM Ki
TKC206544 P14416 D(2) dopamine receptor None >10000 nM Ki
TKC003173 P20701 Integrin alpha-L None 50000 nM IC50
TKC062636 P20701 Integrin alpha-L None 1360 nM IC50
TKC062646 P20701 Integrin alpha-L None >50000 nM IC50
TKC062669 P20701 Integrin alpha-L None 950 nM IC50
TKC062671 P20701 Integrin alpha-L None 180 nM IC50
TKC089595 P20701 Integrin alpha-L None 25 ug.mL-1 IC50
TKC093960 P20701 Integrin alpha-L None 25 ug.mL-1 IC50
TKC103159 P20701 Integrin alpha-L None 300 nM IC50
TKC105374 P20701 Integrin alpha-L None >50000 nM IC50
TKC156472 P20701 Integrin alpha-L None 25 ug.mL-1 IC50
TKC039202 P21453 Sphingosine 1-phosphate receptor 1 None 4962 nM IC50
TKC096012 P21453 Sphingosine 1-phosphate receptor 1 None 34120 nM EC50
TKC096012 P21453 Sphingosine 1-phosphate receptor 1 None >95100 nM EC50
TKC096012 P21453 Sphingosine 1-phosphate receptor 1 None 25400 nM EC50
TKC066433 P22001 Potassium voltage-gated channel subfamily A member 3 None 100 nM Kd
TKC107279 P22001 Potassium voltage-gated channel subfamily A member 3 None 100 nM IC50
TKC007073 P25105 Platelet-activating factor receptor None 5 uM Binding affinity
TKC105026 P25105 Platelet-activating factor receptor None 575 nM IC50
TKC105028 P25105 Platelet-activating factor receptor None 575 nM IC50
TKC106540 P25105 Platelet-activating factor receptor None 964 nM Ki
TKC147486 P25105 Platelet-activating factor receptor None 4 uM Binding affinity
TKC147612 P25105 Platelet-activating factor receptor None 5 uM Binding affinity
TKC151784 P25105 Platelet-activating factor receptor None 128 nM IC50
TKC205457 P25105 Platelet-activating factor receptor None 1259 nM IC50
TKC113091 P27487 Dipeptidyl peptidase 4 None 35600 nM IC50
TKC122980 P27487 Dipeptidyl peptidase 4 None 28840 nM IC50
TKC123088 P27487 Dipeptidyl peptidase 4 None 55820 nM IC50
TKC206549 P35869 Aryl hydrocarbon receptor None 17783 nM Potency
TKC003060 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC005454 P40763 Signal transducer and activator of transcription 3 None 4600 nM IC50
TKC016414 P40763 Signal transducer and activator of transcription 3 None >10000 nM EC50
TKC020636 P40763 Signal transducer and activator of transcription 3 None 6900 nM IC50
TKC020796 P40763 Signal transducer and activator of transcription 3 None 22900 nM IC50
TKC020867 P40763 Signal transducer and activator of transcription 3 None 26 % Inhibition
TKC020868 P40763 Signal transducer and activator of transcription 3 None 31 % Inhibition
TKC020869 P40763 Signal transducer and activator of transcription 3 None 49 % Inhibition
TKC022393 P40763 Signal transducer and activator of transcription 3 None 89500 nM IC50
TKC022771 P40763 Signal transducer and activator of transcription 3 None >100000 nM IC50
TKC028367 P40763 Signal transducer and activator of transcription 3 None 4100 nM IC50
TKC030728 P40763 Signal transducer and activator of transcription 3 None 2 % Inhibition
TKC033506 P40763 Signal transducer and activator of transcription 3 None 2400 nM IC50
TKC033507 P40763 Signal transducer and activator of transcription 3 None 2300 nM IC50
TKC036334 P40763 Signal transducer and activator of transcription 3 None 4 % Inhibition
TKC038766 P40763 Signal transducer and activator of transcription 3 None 1 % Inhibition
TKC039282 P40763 Signal transducer and activator of transcription 3 None 2 % Inhibition
TKC042554 P40763 Signal transducer and activator of transcription 3 None 6300 nM IC50
TKC042556 P40763 Signal transducer and activator of transcription 3 None 110000 nM IC50
TKC044507 P40763 Signal transducer and activator of transcription 3 None 4 % Inhibition
TKC044595 P40763 Signal transducer and activator of transcription 3 None 4 % Inhibition
TKC044621 P40763 Signal transducer and activator of transcription 3 None 3 % Inhibition
TKC044669 P40763 Signal transducer and activator of transcription 3 None 4 % Inhibition
TKC047957 P40763 Signal transducer and activator of transcription 3 None 17100 nM IC50
TKC047959 P40763 Signal transducer and activator of transcription 3 None >30000 nM IC50
TKC047961 P40763 Signal transducer and activator of transcription 3 None >30000 nM IC50
TKC048029 P40763 Signal transducer and activator of transcription 3 None 270 nM IC50
TKC048030 P40763 Signal transducer and activator of transcription 3 None 19200 nM IC50
TKC048031 P40763 Signal transducer and activator of transcription 3 None 590 nM IC50
TKC051029 P40763 Signal transducer and activator of transcription 3 None 60000 nM MIC
TKC060882 P40763 Signal transducer and activator of transcription 3 None >25000 nM IC50
TKC075769 P40763 Signal transducer and activator of transcription 3 None 1862 nM IC50
TKC077689 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC078334 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC087623 P40763 Signal transducer and activator of transcription 3 None >100000 nM IC50
TKC087625 P40763 Signal transducer and activator of transcription 3 None 7000 nM IC50
TKC093311 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC100739 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC101161 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC103159 P40763 Signal transducer and activator of transcription 3 None 3000 nM IC50
TKC103189 P40763 Signal transducer and activator of transcription 3 None 32500 nM IC50
TKC103191 P40763 Signal transducer and activator of transcription 3 None 24800 nM IC50
TKC105152 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC107659 P40763 Signal transducer and activator of transcription 3 None 4 % Inhibition
TKC108773 P40763 Signal transducer and activator of transcription 3 None >50000 nM IC50
TKC112576 P40763 Signal transducer and activator of transcription 3 None 1154 nM IC50
TKC134761 P40763 Signal transducer and activator of transcription 3 None 48 % Inhibition
TKC135961 P40763 Signal transducer and activator of transcription 3 None 73000 nM IC50
TKC135978 P40763 Signal transducer and activator of transcription 3 None 14210 nM IC50
TKC136653 P40763 Signal transducer and activator of transcription 3 None 2 % Inhibition
TKC148207 P40763 Signal transducer and activator of transcription 3 None 15840 nM IC50
TKC149924 P40763 Signal transducer and activator of transcription 3 None 74 % Inhibition
TKC151284 P40763 Signal transducer and activator of transcription 3 None 14000 nM IC50
TKC156528 P40763 Signal transducer and activator of transcription 3 None >30000 nM IC50
TKC206318 P40763 Signal transducer and activator of transcription 3 None 12200 nM IC50
TKC206468 P40763 Signal transducer and activator of transcription 3 None 46 % Inhibition
TKC206627 P40763 Signal transducer and activator of transcription 3 None >100000 nM IC50
TKC206646 P40763 Signal transducer and activator of transcription 3 None 67000 nM IC50
TKC206652 P40763 Signal transducer and activator of transcription 3 None 700 nM IC50
TKC013304 P51449 Nuclear receptor ROR-gamma None 66824 nM Potency
TKC013753 P51449 Nuclear receptor ROR-gamma None 29849 nM Potency
TKC013755 P51449 Nuclear receptor ROR-gamma None 14000 nM EC50
TKC021977 P51449 Nuclear receptor ROR-gamma None 42163 nM Potency
TKC022931 P51449 Nuclear receptor ROR-gamma None 84 nM Potency
TKC056482 P51449 Nuclear receptor ROR-gamma None 130 nM IC50
TKC066169 P51449 Nuclear receptor ROR-gamma None 33492 nM Potency
TKC075769 P51449 Nuclear receptor ROR-gamma None 1980 nM IC50
TKC075769 P51449 Nuclear receptor ROR-gamma None 109 nM Kd
TKC075769 P51449 Nuclear receptor ROR-gamma None 2000 nM IC50
TKC083807 P51449 Nuclear receptor ROR-gamma None 10591 nM Potency
TKC087664 P51449 Nuclear receptor ROR-gamma None 47308 nM Potency
TKC087991 P51449 Nuclear receptor ROR-gamma None 21132 nM Potency
TKC088230 P51449 Nuclear receptor ROR-gamma None 1333 nM Potency
TKC088231 P51449 Nuclear receptor ROR-gamma None 23710 nM Potency
TKC092297 P51449 Nuclear receptor ROR-gamma None 26603 nM Potency
TKC096012 P51449 Nuclear receptor ROR-gamma None 200 nM IC50
TKC096012 P51449 Nuclear receptor ROR-gamma None 18000 nM EC50
TKC097944 P51449 Nuclear receptor ROR-gamma None 4216 nM Potency
TKC102407 P51449 Nuclear receptor ROR-gamma None 21132 nM Potency
TKC107086 P51449 Nuclear receptor ROR-gamma None 3758 nM Potency
TKC115268 P51449 Nuclear receptor ROR-gamma None 37578 nM Potency
TKC118648 P51449 Nuclear receptor ROR-gamma None 80 nM EC50
TKC118652 P51449 Nuclear receptor ROR-gamma None 110 nM EC50
TKC118929 P51449 Nuclear receptor ROR-gamma None 10 nM Ki
TKC118938 P51449 Nuclear receptor ROR-gamma None 10 nM Ki
TKC122884 P51449 Nuclear receptor ROR-gamma None 20 nM EC50
TKC136411 P51449 Nuclear receptor ROR-gamma None 37578 nM Potency
TKC151274 P51449 Nuclear receptor ROR-gamma None 60 nM Potency
TKC206457 P51449 Nuclear receptor ROR-gamma None 20 nM EC50
TKC206457 P51449 Nuclear receptor ROR-gamma None 20 nM EC50
TKC206457 P51449 Nuclear receptor ROR-gamma None 20 nM EC50
TKC206458 P51449 Nuclear receptor ROR-gamma None 20 nM EC50
TKC206459 P51449 Nuclear receptor ROR-gamma None 7 degrees C T
TKC206672 P51449 Nuclear receptor ROR-gamma None 42163 nM Potency
TKC206688 P51449 Nuclear receptor ROR-gamma None 23710 nM Potency
TKC206759 P51449 Nuclear receptor ROR-gamma None 26603 nM Potency
TKC206760 P51449 Nuclear receptor ROR-gamma None 74978 nM Potency
TKC206770 P51449 Nuclear receptor ROR-gamma None 33492 nM Potency
TKC206812 P51449 Nuclear receptor ROR-gamma None 47308 nM Potency
TKC206816 P51449 Nuclear receptor ROR-gamma None 8413 nM Potency
TKC206915 P51449 Nuclear receptor ROR-gamma None 10 nM Ki
TKC205544 P51685 C-C chemokine receptor type 8 None 5 % Inhibition
TKC009486 P52333 Tyrosine-protein kinase JAK3 None >100 nM IC50
TKC009499 P52333 Tyrosine-protein kinase JAK3 None >100 nM IC50
TKC011761 P52333 Tyrosine-protein kinase JAK3 None 100 nM IC50
TKC031094 P52333 Tyrosine-protein kinase JAK3 None >25 % Inhibition
TKC107626 P52333 Tyrosine-protein kinase JAK3 None 25 % Inhibition
TKC120591 P52333 Tyrosine-protein kinase JAK3 None >100 nM IC50
TKC120592 P52333 Tyrosine-protein kinase JAK3 None >100 nM IC50
TKC120593 P52333 Tyrosine-protein kinase JAK3 None >100 nM IC50
TKC134702 P52333 Tyrosine-protein kinase JAK3 None 25 % Inhibition
TKC151713 P52333 Tyrosine-protein kinase JAK3 None 25 % Inhibition
TKC118419 P53778 Mitogen-activated protein kinase 12 None 75 % Inhibition
TKC016794 P55085 Proteinase-activated receptor 2 None 14 nM IC50
TKC205544 P61073 C-X-C chemokine receptor type 4 None 21 % Inhibition
TKC051063 Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D None >20000 nM IC50
TKC104905 Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D None 245 nM IC50
TKC104906 Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D None 542 nM IC50
TKC146367 Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D None >20000 nM IC50
TKC023254 Q15722 Leukotriene B4 receptor 1 None 44500 nM IC50
TKC118419 Q15759 Mitogen-activated protein kinase 11 None 74 % Inhibition
TKC087988 Q16539 Mitogen-activated protein kinase 14 None 2529 nM IC50
TKC118419 Q16539 Mitogen-activated protein kinase 14 None 86 % Inhibition
TKC105649 Q16881 Thioredoxin reductase 1, cytoplasmic None 280 nM Ki
TKC066096 Q9NR96 Toll-like receptor 9 None 3015 nM IC50
TKC076529 Q9NR96 Toll-like receptor 9 None >49739 nM IC50
TKC076529 Q9NR96 Toll-like receptor 9 None >49739 nM IC50
TKC082378 Q9NR96 Toll-like receptor 9 None 7929 nM IC50
TKC082378 Q9NR96 Toll-like receptor 9 None 7929 nM IC50