Basic Information

Name [ICD-11: 5C80]
Protein Number 19
Molecule Number 737

Active subnetwork

Terpenoid-protein target Activity Association

ID Uniport Pref_name Gene name value unit type
TKC013753 P03372 Estrogen receptor None 8913 nM Potency
TKC019072 P03372 Estrogen receptor None 78 % Activity
TKC022931 P03372 Estrogen receptor None 1995 nM Potency
TKC022961 P03372 Estrogen receptor None 54 % Activity
TKC028029 P03372 Estrogen receptor None 0 % Activity
TKC028034 P03372 Estrogen receptor None <0 % Activity
TKC028037 P03372 Estrogen receptor None 1 % Activity
TKC028038 P03372 Estrogen receptor None <0 % Activity
TKC028041 P03372 Estrogen receptor None <0 % Activity
TKC034016 P03372 Estrogen receptor None 51 % Activity
TKC034337 P03372 Estrogen receptor None 2800000 nM IC50
TKC034640 P03372 Estrogen receptor None >1000000 nM Ki
TKC035208 P03372 Estrogen receptor None 39 % Activity
TKC035272 P03372 Estrogen receptor None 2551 nM IC50
TKC035462 P03372 Estrogen receptor None 42 % Activity
TKC066169 P03372 Estrogen receptor None 39811 nM Potency
TKC075769 P03372 Estrogen receptor None 251 nM Potency
TKC079320 P03372 Estrogen receptor None <0 % Activity
TKC079321 P03372 Estrogen receptor None <0 % Activity
TKC087664 P03372 Estrogen receptor None 3162 nM Potency
TKC087988 P03372 Estrogen receptor None 631 nM Potency
TKC087991 P03372 Estrogen receptor None 4467 nM Potency
TKC092297 P03372 Estrogen receptor None 15849 nM Potency
TKC092348 P03372 Estrogen receptor None 8913 nM Potency
TKC096012 P03372 Estrogen receptor None 126 nM Potency
TKC100644 P03372 Estrogen receptor None 31623 nM Potency
TKC101365 P03372 Estrogen receptor None 12570 nM EC50
TKC102448 P03372 Estrogen receptor None 2550 nM EC50
TKC107086 P03372 Estrogen receptor None 8913 nM Potency
TKC107735 P03372 Estrogen receptor None 50119 nM Potency
TKC111727 P03372 Estrogen receptor None 0 nM Ki
TKC111738 P03372 Estrogen receptor None 1 nM EC50
TKC111738 P03372 Estrogen receptor None 166 nM IC50
TKC111738 P03372 Estrogen receptor None 210 nM IC50
TKC111738 P03372 Estrogen receptor None 96 nM IC50
TKC112923 P03372 Estrogen receptor None 26 nM EC50
TKC115268 P03372 Estrogen receptor None 15849 nM Potency
TKC129821 P03372 Estrogen receptor None 70 % Activity
TKC151345 P03372 Estrogen receptor None 35 % Activity
TKC151713 P03372 Estrogen receptor None 40 % Activity
TKC151765 P03372 Estrogen receptor None 81 % Activity
TKC206549 P03372 Estrogen receptor None 3548 nM Potency
TKC206608 P03372 Estrogen receptor None 8170 nM EC50
TKC206652 P03372 Estrogen receptor None 112 nM Potency
TKC206725 P03372 Estrogen receptor None 8 nM Ki
TKC206726 P03372 Estrogen receptor None 72 nM EC50
TKC206759 P03372 Estrogen receptor None >10000 nM IC50
TKC206759 P03372 Estrogen receptor None >10000 nM IC50
TKC206760 P03372 Estrogen receptor None 25119 nM Potency
TKC206764 P03372 Estrogen receptor None 0 % RBA
TKC206770 P03372 Estrogen receptor None 5012 nM Potency
TKC206779 P03372 Estrogen receptor None 6310 nM Potency
TKC206812 P03372 Estrogen receptor None 62000 nM IC50
TKC206812 P03372 Estrogen receptor None 39811 nM Potency
TKC206816 P03372 Estrogen receptor None >1000 nM IC50
TKC206816 P03372 Estrogen receptor None >1000 nM IC50
TKC008187 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 30200 nM IC50
TKC023515 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 53 % Inhibition
TKC025574 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 52 % Inhibition
TKC026893 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 21 % Inhibition
TKC026895 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 61 % Inhibition
TKC057019 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 22300 nM IC50
TKC100777 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 30 % Inhibition
TKC101031 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 1500 nM IC50
TKC101538 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 39 % Inhibition
TKC101847 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 1000 nM IC50
TKC103703 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 40 % Inhibition
TKC137314 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 8400 nM IC50
TKC138471 P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase None 21700 nM IC50
TKC057132 P10613 Lanosterol 14-alpha demethylase None 7400 nM Km
TKC206812 P10827 Thyroid hormone receptor alpha None >100000 nM EC50
TKC005454 P10828 Thyroid hormone receptor beta None 50119 nM Potency
TKC017379 P10828 Thyroid hormone receptor beta None 35481 nM Potency
TKC019353 P10828 Thyroid hormone receptor beta None 4467 nM Potency
TKC020732 P10828 Thyroid hormone receptor beta None 794328 nM Potency
TKC026870 P10828 Thyroid hormone receptor beta None 2239 nM Potency
TKC034632 P10828 Thyroid hormone receptor beta None 63096 nM Potency
TKC035272 P10828 Thyroid hormone receptor beta None 22387 nM Potency
TKC042351 P10828 Thyroid hormone receptor beta None 2512 nM Potency
TKC075769 P10828 Thyroid hormone receptor beta None 126 nM Potency
TKC079004 P10828 Thyroid hormone receptor beta None 89125 nM Potency
TKC079006 P10828 Thyroid hormone receptor beta None 89125 nM Potency
TKC087988 P10828 Thyroid hormone receptor beta None 22387 nM Potency
TKC088230 P10828 Thyroid hormone receptor beta None 25119 nM Potency
TKC092297 P10828 Thyroid hormone receptor beta None 39811 nM Potency
TKC096012 P10828 Thyroid hormone receptor beta None 3 nM Potency
TKC102144 P10828 Thyroid hormone receptor beta None 4 nM Potency
TKC102407 P10828 Thyroid hormone receptor beta None 1 nM Potency
TKC107086 P10828 Thyroid hormone receptor beta None 8913 nM Potency
TKC107515 P10828 Thyroid hormone receptor beta None 25119 nM Potency
TKC108536 P10828 Thyroid hormone receptor beta None 44668 nM Potency
TKC109617 P10828 Thyroid hormone receptor beta None 36 nM Potency
TKC113161 P10828 Thyroid hormone receptor beta None 18 nM Potency
TKC113663 P10828 Thyroid hormone receptor beta None 3 nM Potency
TKC115268 P10828 Thyroid hormone receptor beta None 44668 nM Potency
TKC118419 P10828 Thyroid hormone receptor beta None 31623 nM Potency
TKC120161 P10828 Thyroid hormone receptor beta None 36 nM Potency
TKC136852 P10828 Thyroid hormone receptor beta None 501 nM Potency
TKC151274 P10828 Thyroid hormone receptor beta None 18 nM Potency
TKC205928 P10828 Thyroid hormone receptor beta None 1000000 nM Potency
TKC206348 P10828 Thyroid hormone receptor beta None 2818 nM Potency
TKC206652 P10828 Thyroid hormone receptor beta None 71 nM Potency
TKC206688 P10828 Thyroid hormone receptor beta None 35481 nM Potency
TKC206760 P10828 Thyroid hormone receptor beta None 22387 nM Potency
TKC206812 P10828 Thyroid hormone receptor beta None 44668 nM Potency
TKC206816 P10828 Thyroid hormone receptor beta None 44668 nM Potency
TKC206884 P10828 Thyroid hormone receptor beta None 1585 nM Potency
TKC002411 P11597 Cholesteryl ester transfer protein None 196000 nM IC50
TKC026245 P11597 Cholesteryl ester transfer protein None 25000 nM IC50
TKC026309 P11597 Cholesteryl ester transfer protein None 6000 nM IC50
TKC026600 P11597 Cholesteryl ester transfer protein None 100000 nM IC50
TKC027200 P11597 Cholesteryl ester transfer protein None 5000 nM IC50
TKC027200 P11597 Cholesteryl ester transfer protein None 5200 nM IC50
TKC027201 P11597 Cholesteryl ester transfer protein None 1000 nM IC50
TKC027201 P11597 Cholesteryl ester transfer protein None 5200 nM IC50
TKC056482 P11597 Cholesteryl ester transfer protein None 46600 nM IC50
TKC077689 P11597 Cholesteryl ester transfer protein None 10 % Inhibition
TKC094496 P11597 Cholesteryl ester transfer protein None 46000 nM IC50
TKC097288 P11597 Cholesteryl ester transfer protein None 600 nM IC50
TKC106450 P11597 Cholesteryl ester transfer protein None 5200 nM IC50
TKC123088 P11597 Cholesteryl ester transfer protein None 31 % Inhibition
TKC005454 P23141 Liver carboxylesterase 1 None 544 nM Ki
TKC012269 P23141 Liver carboxylesterase 1 None 2530 nM Ki
TKC014568 P23141 Liver carboxylesterase 1 None 26250 nM Ki
TKC088678 P23141 Liver carboxylesterase 1 None 20970 nM IC50
TKC088715 P23141 Liver carboxylesterase 1 None 49860 nM IC50
TKC101270 P23141 Liver carboxylesterase 1 None 23610 nM IC50
TKC103069 P23141 Liver carboxylesterase 1 None 49860 nM IC50
TKC107319 P23141 Liver carboxylesterase 1 None >100000 nM Ki
TKC141401 P23141 Liver carboxylesterase 1 None 10530 nM IC50
TKC141510 P23141 Liver carboxylesterase 1 None 22360 nM IC50
TKC151739 P23141 Liver carboxylesterase 1 None >100000 nM IC50
TKC000611 P23219 Prostaglandin G/H synthase 1 None 40000 nM IC50
TKC001618 P23219 Prostaglandin G/H synthase 1 None 34000 nM IC50
TKC009896 P23219 Prostaglandin G/H synthase 1 None 791100 nM IC50
TKC019819 P23219 Prostaglandin G/H synthase 1 None 48 % Inhibition
TKC019859 P23219 Prostaglandin G/H synthase 1 None 54 % Inhibition
TKC020491 P23219 Prostaglandin G/H synthase 1 None 4000 nM IC50
TKC020796 P23219 Prostaglandin G/H synthase 1 None 30 % Inhibition
TKC021940 P23219 Prostaglandin G/H synthase 1 None 40 % Inhibition
TKC022833 P23219 Prostaglandin G/H synthase 1 None 43 % Inhibition
TKC022834 P23219 Prostaglandin G/H synthase 1 None 43 % Inhibition
TKC022961 P23219 Prostaglandin G/H synthase 1 None 44 % Inhibition
TKC024587 P23219 Prostaglandin G/H synthase 1 None 3300 nM IC50
TKC024587 P23219 Prostaglandin G/H synthase 1 None 3300 nM IC50
TKC031258 P23219 Prostaglandin G/H synthase 1 None 3600 nM IC50
TKC034201 P23219 Prostaglandin G/H synthase 1 None >200000 nM IC50
TKC034358 P23219 Prostaglandin G/H synthase 1 None 39000 nM IC50
TKC034359 P23219 Prostaglandin G/H synthase 1 None 39000 nM IC50
TKC036372 P23219 Prostaglandin G/H synthase 1 None 14000 nM IC50
TKC037595 P23219 Prostaglandin G/H synthase 1 None 36000 nM IC50
TKC043613 P23219 Prostaglandin G/H synthase 1 None 43000 nM IC50
TKC049750 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC049818 P23219 Prostaglandin G/H synthase 1 None 44 ug IC50
TKC054011 P23219 Prostaglandin G/H synthase 1 None 8800 nM IC50
TKC054031 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC054081 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC054090 P23219 Prostaglandin G/H synthase 1 None 7500 nM IC50
TKC054099 P23219 Prostaglandin G/H synthase 1 None 8800 nM IC50
TKC054100 P23219 Prostaglandin G/H synthase 1 None 8900 nM IC50
TKC054101 P23219 Prostaglandin G/H synthase 1 None 7600 nM IC50
TKC054240 P23219 Prostaglandin G/H synthase 1 None 7800 nM IC50
TKC054241 P23219 Prostaglandin G/H synthase 1 None 6300 nM IC50
TKC056482 P23219 Prostaglandin G/H synthase 1 None 210000 nM IC50
TKC060184 P23219 Prostaglandin G/H synthase 1 None 8300 nM IC50
TKC060216 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC060284 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC060302 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC060303 P23219 Prostaglandin G/H synthase 1 None 7800 nM IC50
TKC060304 P23219 Prostaglandin G/H synthase 1 None 8000 nM IC50
TKC060399 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC060602 P23219 Prostaglandin G/H synthase 1 None 5900 nM IC50
TKC066954 P23219 Prostaglandin G/H synthase 1 None 38 % Inhibition
TKC068533 P23219 Prostaglandin G/H synthase 1 None 28000 nM IC50
TKC071010 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC077689 P23219 Prostaglandin G/H synthase 1 None 380000 nM IC50
TKC077689 P23219 Prostaglandin G/H synthase 1 None 380000 nM IC50
TKC095276 P23219 Prostaglandin G/H synthase 1 None 48 % Inhibition
TKC113936 P23219 Prostaglandin G/H synthase 1 None 65 % Inhibition
TKC122543 P23219 Prostaglandin G/H synthase 1 None 35 % Inhibition
TKC130084 P23219 Prostaglandin G/H synthase 1 None 39 % Inhibition
TKC130119 P23219 Prostaglandin G/H synthase 1 None 33 % Inhibition
TKC130577 P23219 Prostaglandin G/H synthase 1 None <43 % Inhibition
TKC130901 P23219 Prostaglandin G/H synthase 1 None 36 % Inhibition
TKC133309 P23219 Prostaglandin G/H synthase 1 None >200000 nM IC50
TKC133517 P23219 Prostaglandin G/H synthase 1 None 1300 nM IC50
TKC133656 P23219 Prostaglandin G/H synthase 1 None >200000 nM IC50
TKC134278 P23219 Prostaglandin G/H synthase 1 None >200000 nM IC50
TKC139036 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC140627 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC141365 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC143641 P23219 Prostaglandin G/H synthase 1 None >50000 nM IC50
TKC151113 P23219 Prostaglandin G/H synthase 1 None 116400 nM IC50
TKC151284 P23219 Prostaglandin G/H synthase 1 None 51 % Inhibition
TKC151765 P23219 Prostaglandin G/H synthase 1 None 48 % Inhibition
TKC151792 P23219 Prostaglandin G/H synthase 1 None 14000 nM IC50
TKC172853 P23219 Prostaglandin G/H synthase 1 None 43700 nM IC50
TKC012378 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 56 % Inhibition
TKC036177 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 13 nM IC50
TKC036177 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 13 nM IC50
TKC047464 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None <50 % Inhibition
TKC049301 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 22 % Inhibition
TKC049302 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 6 % Inhibition
TKC049559 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 11400 nM IC50
TKC049666 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 3800 nM IC50
TKC049832 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 395 nM IC50
TKC049833 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 34 nM IC50
TKC050879 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None >10000 nM IC50
TKC051029 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 46 % Inhibition
TKC051154 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 63 % Inhibition
TKC052452 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None >10000 nM IC50
TKC053100 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 3200 nM IC50
TKC053930 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 6 nM IC50
TKC055403 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 1400 nM IC50
TKC055404 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 4100 nM IC50
TKC055890 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 105 nM IC50
TKC056332 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None >10000 nM IC50
TKC056482 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 1900 nM IC50
TKC057835 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 2300 nM IC50
TKC063150 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None <50 % Inhibition
TKC063649 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 72 nM IC50
TKC064069 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 76 nM IC50
TKC064070 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 195 nM IC50
TKC064071 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 15 nM IC50
TKC064939 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 45 % Inhibition
TKC064940 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 3740 nM IC50
TKC075891 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 6 nM IC50
TKC076051 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None >35 % Inhibition
TKC077375 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 97 % Inhibition
TKC079733 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 82 % Inhibition
TKC080267 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 40 % Inhibition
TKC088620 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 62 nM Ki
TKC088678 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 9 nM IC50
TKC088678 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 29 nM IC50
TKC088678 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 13 nM IC50
TKC088678 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 778 nM IC50
TKC088678 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 778 nM IC50
TKC088678 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 11.78 nM IC50
TKC088678 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 11 nM IC50
TKC088678 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 29 nM IC50
TKC088678 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 8.8 nM IC50
TKC088715 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 800 nM IC50
TKC088715 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 7138 nM IC50
TKC088715 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 7100 nM IC50
TKC088961 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 929 nM IC50
TKC088962 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 825 nM IC50
TKC088963 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 626 nM IC50
TKC088981 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 504 nM IC50
TKC102290 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None >10000 nM IC50
TKC103069 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 800 nM IC50
TKC104256 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 2060 nM IC50
TKC104829 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 20 % Inhibition
TKC105165 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 4 % Activity
TKC106140 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 17 % Inhibition
TKC107137 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 910 nM IC50
TKC138609 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None <50 % Inhibition
TKC139322 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 810 nM IC50
TKC139355 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 5200 nM IC50
TKC139366 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 52 % Inhibition
TKC141002 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None <50 % Inhibition
TKC145231 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None <50 % Inhibition
TKC145651 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 9400 nM IC50
TKC145901 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 1350 nM IC50
TKC151633 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 1236 nM IC50
TKC151739 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 619 nM IC50
TKC151798 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 1417 nM IC50
TKC205472 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None >9900 nM IC50
TKC205869 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None >1900 nM IC50
TKC206764 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 81 % Inhibition
TKC207256 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None >353700 nM Ki
TKC207257 P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 None 13500 nM Ki
TKC008359 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC010020 P35354 Prostaglandin G/H synthase 2 None 61 % Inhibition
TKC010022 P35354 Prostaglandin G/H synthase 2 None 55 % Inhibition
TKC010023 P35354 Prostaglandin G/H synthase 2 None 57 % Inhibition
TKC010024 P35354 Prostaglandin G/H synthase 2 None 42 % Inhibition
TKC010025 P35354 Prostaglandin G/H synthase 2 None 78 % Inhibition
TKC010026 P35354 Prostaglandin G/H synthase 2 None 17 % Inhibition
TKC011599 P35354 Prostaglandin G/H synthase 2 None 64 % Inhibition
TKC012919 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC012941 P35354 Prostaglandin G/H synthase 2 None 8500 nM IC50
TKC012956 P35354 Prostaglandin G/H synthase 2 None 2200 nM IC50
TKC012962 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC015443 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC015459 P35354 Prostaglandin G/H synthase 2 None 2200 nM IC50
TKC015537 P35354 Prostaglandin G/H synthase 2 None 0 % Inhibition
TKC016794 P35354 Prostaglandin G/H synthase 2 None 40 nM IC50
TKC019436 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC019466 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC019819 P35354 Prostaglandin G/H synthase 2 None 35 % Inhibition
TKC019859 P35354 Prostaglandin G/H synthase 2 None <33 % Inhibition
TKC020479 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC020796 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC021940 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC022833 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC022834 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC022961 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC026245 P35354 Prostaglandin G/H synthase 2 None 2300 nM IC50
TKC027200 P35354 Prostaglandin G/H synthase 2 None 700 nM IC50
TKC028143 P35354 Prostaglandin G/H synthase 2 None 100 % Inhibition
TKC031202 P35354 Prostaglandin G/H synthase 2 None 3800 nM IC50
TKC031223 P35354 Prostaglandin G/H synthase 2 None 45 % Inhibition
TKC032234 P35354 Prostaglandin G/H synthase 2 None 400 nM IC50
TKC035208 P35354 Prostaglandin G/H synthase 2 None 7 uM IC60
TKC037534 P35354 Prostaglandin G/H synthase 2 None 97 % Inhibition
TKC038330 P35354 Prostaglandin G/H synthase 2 None 2900 nM IC50
TKC041884 P35354 Prostaglandin G/H synthase 2 None 18000 nM IC50
TKC043993 P35354 Prostaglandin G/H synthase 2 None 98 % Inhibition
TKC045188 P35354 Prostaglandin G/H synthase 2 None 98 % Inhibition
TKC048282 P35354 Prostaglandin G/H synthase 2 None 370 nM IC50
TKC049750 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC049818 P35354 Prostaglandin G/H synthase 2 None 5 ug IC50
TKC051154 P35354 Prostaglandin G/H synthase 2 None >61 % Activity
TKC054011 P35354 Prostaglandin G/H synthase 2 None 9000 nM IC50
TKC054031 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC054081 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC054090 P35354 Prostaglandin G/H synthase 2 None 8900 nM IC50
TKC054099 P35354 Prostaglandin G/H synthase 2 None 7800 nM IC50
TKC054100 P35354 Prostaglandin G/H synthase 2 None 7900 nM IC50
TKC054101 P35354 Prostaglandin G/H synthase 2 None 8800 nM IC50
TKC054240 P35354 Prostaglandin G/H synthase 2 None 6700 nM IC50
TKC054241 P35354 Prostaglandin G/H synthase 2 None 6100 nM IC50
TKC056482 P35354 Prostaglandin G/H synthase 2 None 40000 nM IC50
TKC056482 P35354 Prostaglandin G/H synthase 2 None 86000 nM IC50
TKC056482 P35354 Prostaglandin G/H synthase 2 None 130000 nM IC50
TKC057308 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC058811 P35354 Prostaglandin G/H synthase 2 None >85 % Activity
TKC058812 P35354 Prostaglandin G/H synthase 2 None >78 % Activity
TKC060184 P35354 Prostaglandin G/H synthase 2 None 8500 nM IC50
TKC060216 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC060284 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC060302 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC060303 P35354 Prostaglandin G/H synthase 2 None 7200 nM IC50
TKC060304 P35354 Prostaglandin G/H synthase 2 None 7600 nM IC50
TKC060399 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC060602 P35354 Prostaglandin G/H synthase 2 None 6700 nM IC50
TKC061939 P35354 Prostaglandin G/H synthase 2 None >10000 nM IC50
TKC061968 P35354 Prostaglandin G/H synthase 2 None >10000 nM IC50
TKC061969 P35354 Prostaglandin G/H synthase 2 None >10000 nM IC50
TKC064374 P35354 Prostaglandin G/H synthase 2 None >73 % Activity
TKC064407 P35354 Prostaglandin G/H synthase 2 None >78 % Activity
TKC065375 P35354 Prostaglandin G/H synthase 2 None >70 % Activity
TKC066954 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC070952 P35354 Prostaglandin G/H synthase 2 None >100000 nM IC50
TKC071010 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC071640 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC076350 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC077689 P35354 Prostaglandin G/H synthase 2 None 40000 nM IC50
TKC077689 P35354 Prostaglandin G/H synthase 2 None 295000 nM IC50
TKC077689 P35354 Prostaglandin G/H synthase 2 None 295000 nM IC50
TKC077689 P35354 Prostaglandin G/H synthase 2 None 87000 nM IC50
TKC077703 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC078194 P35354 Prostaglandin G/H synthase 2 None >74 % Activity
TKC085168 P35354 Prostaglandin G/H synthase 2 None <60 % Inhibition
TKC088678 P35354 Prostaglandin G/H synthase 2 None >72 % Activity
TKC095276 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC095567 P35354 Prostaglandin G/H synthase 2 None >10000 nM IC50
TKC110247 P35354 Prostaglandin G/H synthase 2 None >10 ug.mL-1 IC50
TKC113936 P35354 Prostaglandin G/H synthase 2 None 60 % Inhibition
TKC122543 P35354 Prostaglandin G/H synthase 2 None 30 % Inhibition
TKC123028 P35354 Prostaglandin G/H synthase 2 None >72 % Activity
TKC129152 P35354 Prostaglandin G/H synthase 2 None >100000 nM IC50
TKC130084 P35354 Prostaglandin G/H synthase 2 None 37 % Inhibition
TKC130119 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC130223 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC130577 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC130901 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC135264 P35354 Prostaglandin G/H synthase 2 None 400 nM IC50
TKC135559 P35354 Prostaglandin G/H synthase 2 None 4600 nM IC50
TKC139036 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC139322 P35354 Prostaglandin G/H synthase 2 None >82 % Activity
TKC139366 P35354 Prostaglandin G/H synthase 2 None 40000 nM IC50
TKC140627 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC141365 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC141401 P35354 Prostaglandin G/H synthase 2 None >75 % Activity
TKC141499 P35354 Prostaglandin G/H synthase 2 None >87 % Activity
TKC141601 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC141602 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC141622 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC141805 P35354 Prostaglandin G/H synthase 2 None 40000 nM IC50
TKC142150 P35354 Prostaglandin G/H synthase 2 None 450000 nM IC50
TKC142203 P35354 Prostaglandin G/H synthase 2 None >10000 nM IC50
TKC142208 P35354 Prostaglandin G/H synthase 2 None >10000 nM IC50
TKC142849 P35354 Prostaglandin G/H synthase 2 None >69 % Activity
TKC142897 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC142922 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC143527 P35354 Prostaglandin G/H synthase 2 None 97 % Inhibition
TKC143539 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC143641 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC145295 P35354 Prostaglandin G/H synthase 2 None 22 % Inhibition
TKC145848 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC145932 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC145968 P35354 Prostaglandin G/H synthase 2 None >94 % Activity
TKC146116 P35354 Prostaglandin G/H synthase 2 None >5.0e+4 nM IC50
TKC146774 P35354 Prostaglandin G/H synthase 2 None >78 % Activity
TKC146857 P35354 Prostaglandin G/H synthase 2 None 600 nM IC50
TKC149251 P35354 Prostaglandin G/H synthase 2 None 1100 nM IC50
TKC149759 P35354 Prostaglandin G/H synthase 2 None 100 % Activity
TKC149924 P35354 Prostaglandin G/H synthase 2 None 800 nM IC50
TKC149926 P35354 Prostaglandin G/H synthase 2 None 800 nM IC50
TKC150635 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC150706 P35354 Prostaglandin G/H synthase 2 None >76 % Activity
TKC150907 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC151280 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC151284 P35354 Prostaglandin G/H synthase 2 None 33 % Inhibition
TKC151765 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC152742 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC152813 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC156345 P35354 Prostaglandin G/H synthase 2 None 25 % Inhibition
TKC156572 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC156716 P35354 Prostaglandin G/H synthase 2 None 2200 nM IC50
TKC170277 P35354 Prostaglandin G/H synthase 2 None >50000 nM IC50
TKC172853 P35354 Prostaglandin G/H synthase 2 None 4700 nM IC50
TKC174442 P35354 Prostaglandin G/H synthase 2 None 10000 nM IC50
TKC205509 P35354 Prostaglandin G/H synthase 2 None 540000 nM IC50
TKC205699 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC205700 P35354 Prostaglandin G/H synthase 2 None <30 % Inhibition
TKC206319 P35354 Prostaglandin G/H synthase 2 None 99 % Inhibition
TKC005728 P37231 Peroxisome proliferator-activated receptor gamma None >100000 nM EC50
TKC005729 P37231 Peroxisome proliferator-activated receptor gamma None 16700 nM EC50
TKC013753 P37231 Peroxisome proliferator-activated receptor gamma None 2818 nM Potency
TKC021262 P37231 Peroxisome proliferator-activated receptor gamma None 21700 nM EC50
TKC035272 P37231 Peroxisome proliferator-activated receptor gamma None 7943 nM Potency
TKC066169 P37231 Peroxisome proliferator-activated receptor gamma None 28184 nM Potency
TKC075769 P37231 Peroxisome proliferator-activated receptor gamma None 316 nM Potency
TKC079000 P37231 Peroxisome proliferator-activated receptor gamma None 50119 nM Potency
TKC087664 P37231 Peroxisome proliferator-activated receptor gamma None 44668 nM Potency
TKC087991 P37231 Peroxisome proliferator-activated receptor gamma None 3162 nM Potency
TKC088230 P37231 Peroxisome proliferator-activated receptor gamma None 44668 nM Potency
TKC092297 P37231 Peroxisome proliferator-activated receptor gamma None 15849 nM Potency
TKC096012 P37231 Peroxisome proliferator-activated receptor gamma None 316 nM Potency
TKC100644 P37231 Peroxisome proliferator-activated receptor gamma None 44668 nM Potency
TKC102407 P37231 Peroxisome proliferator-activated receptor gamma None 50119 nM Potency
TKC107086 P37231 Peroxisome proliferator-activated receptor gamma None 28184 nM Potency
TKC107735 P37231 Peroxisome proliferator-activated receptor gamma None 39811 nM Potency
TKC108536 P37231 Peroxisome proliferator-activated receptor gamma None 44668 nM Potency
TKC110634 P37231 Peroxisome proliferator-activated receptor gamma None 6400 nM EC50
TKC110635 P37231 Peroxisome proliferator-activated receptor gamma None 8200 nM EC50
TKC111200 P37231 Peroxisome proliferator-activated receptor gamma None 22300 nM EC50
TKC111271 P37231 Peroxisome proliferator-activated receptor gamma None >50000 nM EC50
TKC111272 P37231 Peroxisome proliferator-activated receptor gamma None 18700 nM EC50
TKC111273 P37231 Peroxisome proliferator-activated receptor gamma None >50000 nM EC50
TKC111274 P37231 Peroxisome proliferator-activated receptor gamma None 20600 nM EC50
TKC111276 P37231 Peroxisome proliferator-activated receptor gamma None >50000 nM EC50
TKC111284 P37231 Peroxisome proliferator-activated receptor gamma None >50000 nM EC50
TKC111466 P37231 Peroxisome proliferator-activated receptor gamma None >50000 nM EC50
TKC115268 P37231 Peroxisome proliferator-activated receptor gamma None 44668 nM Potency
TKC170559 P37231 Peroxisome proliferator-activated receptor gamma None 1000 nM EC50
TKC206549 P37231 Peroxisome proliferator-activated receptor gamma None 126 nM Potency
TKC206652 P37231 Peroxisome proliferator-activated receptor gamma None 316 nM Potency
TKC206672 P37231 Peroxisome proliferator-activated receptor gamma None 31623 nM Potency
TKC206759 P37231 Peroxisome proliferator-activated receptor gamma None 12589 nM Potency
TKC206760 P37231 Peroxisome proliferator-activated receptor gamma None 17783 nM Potency
TKC206812 P37231 Peroxisome proliferator-activated receptor gamma None 27000 nM IC50
TKC206812 P37231 Peroxisome proliferator-activated receptor gamma None 50119 nM Potency
TKC206816 P37231 Peroxisome proliferator-activated receptor gamma None 39811 nM Potency
TKC073907 P37268 Squalene synthase None 2300 nM Km
TKC122582 P37268 Squalene synthase None 2300 nM Km
TKC147153 P37268 Squalene synthase None 2300 nM Km
TKC038192 Q02127 Dihydroorotate dehydrogenase None 3 % Inhibition
TKC039868 Q02127 Dihydroorotate dehydrogenase None 0 % Inhibition
TKC043742 Q02127 Dihydroorotate dehydrogenase None 0 % Inhibition
TKC079733 Q02127 Dihydroorotate dehydrogenase None 28 % Inhibition
TKC136181 Q02127 Dihydroorotate dehydrogenase None 12 % Inhibition
TKC020732 Q03181 Peroxisome proliferator-activated receptor delta None 1258925 nM Potency
TKC021262 Q03181 Peroxisome proliferator-activated receptor delta None 48500 nM EC50
TKC021321 Q03181 Peroxisome proliferator-activated receptor delta None 50119 nM Potency
TKC034760 Q03181 Peroxisome proliferator-activated receptor delta None 50119 nM Potency
TKC035272 Q03181 Peroxisome proliferator-activated receptor delta None 10000 nM Potency
TKC038473 Q03181 Peroxisome proliferator-activated receptor delta None 14125 nM Potency
TKC066169 Q03181 Peroxisome proliferator-activated receptor delta None 15849 nM Potency
TKC074866 Q03181 Peroxisome proliferator-activated receptor delta None 1 nM Potency
TKC075769 Q03181 Peroxisome proliferator-activated receptor delta None 141 nM Potency
TKC079001 Q03181 Peroxisome proliferator-activated receptor delta None 50119 nM Potency
TKC087664 Q03181 Peroxisome proliferator-activated receptor delta None 50119 nM Potency
TKC092297 Q03181 Peroxisome proliferator-activated receptor delta None 44668 nM Potency
TKC096012 Q03181 Peroxisome proliferator-activated receptor delta None 44668 nM Potency
TKC100644 Q03181 Peroxisome proliferator-activated receptor delta None 15849 nM Potency
TKC102407 Q03181 Peroxisome proliferator-activated receptor delta None 22387 nM Potency
TKC107086 Q03181 Peroxisome proliferator-activated receptor delta None 39811 nM Potency
TKC107735 Q03181 Peroxisome proliferator-activated receptor delta None 12589 nM Potency
TKC108536 Q03181 Peroxisome proliferator-activated receptor delta None 2 nM Potency
TKC110634 Q03181 Peroxisome proliferator-activated receptor delta None 100 % Activity
TKC110635 Q03181 Peroxisome proliferator-activated receptor delta None 100 % Activity
TKC115268 Q03181 Peroxisome proliferator-activated receptor delta None 39811 nM Potency
TKC122884 Q03181 Peroxisome proliferator-activated receptor delta None 79433 nM Potency
TKC136411 Q03181 Peroxisome proliferator-activated receptor delta None 31623 nM Potency
TKC206652 Q03181 Peroxisome proliferator-activated receptor delta None 251 nM Potency
TKC206672 Q03181 Peroxisome proliferator-activated receptor delta None 17783 nM Potency
TKC206759 Q03181 Peroxisome proliferator-activated receptor delta None 50119 nM Potency
TKC206760 Q03181 Peroxisome proliferator-activated receptor delta None 35481 nM Potency
TKC206770 Q03181 Peroxisome proliferator-activated receptor delta None 31623 nM Potency
TKC206812 Q03181 Peroxisome proliferator-activated receptor delta None 22387 nM Potency
TKC206816 Q03181 Peroxisome proliferator-activated receptor delta None 25119 nM Potency
TKC021262 Q07869 Peroxisome proliferator-activated receptor alpha None 19500 nM EC50
TKC021666 Q07869 Peroxisome proliferator-activated receptor alpha None 28 % Activity
TKC021674 Q07869 Peroxisome proliferator-activated receptor alpha None 25 % Activity
TKC035272 Q07869 Peroxisome proliferator-activated receptor alpha None 15849 nM Potency
TKC056482 Q07869 Peroxisome proliferator-activated receptor alpha None 259 % Activity
TKC057132 Q07869 Peroxisome proliferator-activated receptor alpha None 12589 nM Potency
TKC088526 Q07869 Peroxisome proliferator-activated receptor alpha None 12 % Activity
TKC100644 Q07869 Peroxisome proliferator-activated receptor alpha None 8913 nM Potency
TKC108536 Q07869 Peroxisome proliferator-activated receptor alpha None 50119 nM Potency
TKC110634 Q07869 Peroxisome proliferator-activated receptor alpha None 309 % Activity
TKC110635 Q07869 Peroxisome proliferator-activated receptor alpha None 289 % Activity
TKC170559 Q07869 Peroxisome proliferator-activated receptor alpha None 1000 nM EC50
TKC171329 Q07869 Peroxisome proliferator-activated receptor alpha None 184 nM EC50
TKC206812 Q07869 Peroxisome proliferator-activated receptor alpha None >20000 nM IC50
TKC106240 Q12908 Ileal sodium/bile acid cotransporter None 3300 nM Ki
TKC106250 Q12908 Ileal sodium/bile acid cotransporter None 75000 nM Ki
TKC109619 Q12908 Ileal sodium/bile acid cotransporter None 75000 nM Ki
TKC109621 Q12908 Ileal sodium/bile acid cotransporter None 4100 nM Km
TKC109622 Q12908 Ileal sodium/bile acid cotransporter None 28000 nM Ki
TKC109625 Q12908 Ileal sodium/bile acid cotransporter None 2000 nM Km
TKC206670 Q12908 Ileal sodium/bile acid cotransporter None 5700 nM Km
TKC206671 Q12908 Ileal sodium/bile acid cotransporter None 6100 nM Ki
TKC206672 Q12908 Ileal sodium/bile acid cotransporter None 6300 nM Ki
TKC206849 Q12908 Ileal sodium/bile acid cotransporter None 41500 nM Ki
TKC023246 Q92731 Estrogen receptor beta None >10000 nM IC50
TKC028029 Q92731 Estrogen receptor beta None <1 % Activity
TKC028037 Q92731 Estrogen receptor beta None 10 % Activity
TKC035272 Q92731 Estrogen receptor beta None >50000 nM IC50
TKC100932 Q92731 Estrogen receptor beta None 25300 nM EC50
TKC101365 Q92731 Estrogen receptor beta None 17690 nM EC50
TKC102448 Q92731 Estrogen receptor beta None 4680 nM EC50
TKC106878 Q92731 Estrogen receptor beta None >10000 nM IC50
TKC110673 Q92731 Estrogen receptor beta None 2.78E+11 M-1 Ka
TKC111721 Q92731 Estrogen receptor beta None 1520000000 M-1 Ka
TKC111727 Q92731 Estrogen receptor beta None 614000000 M-1 Ka
TKC111727 Q92731 Estrogen receptor beta None 0 nM EC50
TKC111738 Q92731 Estrogen receptor beta None 2 nM EC50
TKC111738 Q92731 Estrogen receptor beta None 4 % RSA
TKC111738 Q92731 Estrogen receptor beta None 26 nM IC50
TKC111738 Q92731 Estrogen receptor beta None 540 nM IC50
TKC111738 Q92731 Estrogen receptor beta None 8 nM EC50
TKC112923 Q92731 Estrogen receptor beta None 6 nM EC50
TKC206608 Q92731 Estrogen receptor beta None 4280 nM EC50
TKC206725 Q92731 Estrogen receptor beta None 24 nM Ki
TKC206726 Q92731 Estrogen receptor beta None 11 nM EC50
TKC206759 Q92731 Estrogen receptor beta None >10000 nM IC50
TKC206759 Q92731 Estrogen receptor beta None >10000 nM IC50
TKC206764 Q92731 Estrogen receptor beta None 1 % RBA
TKC206765 Q92731 Estrogen receptor beta None 18000000 M-1 Ka
TKC206769 Q92731 Estrogen receptor beta None 27000000 M-1 Ka
TKC206812 Q92731 Estrogen receptor beta None >5000 nM IC50
TKC206816 Q92731 Estrogen receptor beta None 1000000 nM IC50
TKC013753 Q96RI1 Bile acid receptor None 16 nM Potency
TKC016414 Q96RI1 Bile acid receptor None 9700 nM IC50
TKC016817 Q96RI1 Bile acid receptor None 3900 nM IC50
TKC017639 Q96RI1 Bile acid receptor None 1 % Activity
TKC019374 Q96RI1 Bile acid receptor None 4 nM Potency
TKC021321 Q96RI1 Bile acid receptor None 39811 nM Potency
TKC021365 Q96RI1 Bile acid receptor None 28184 nM Potency
TKC021425 Q96RI1 Bile acid receptor None 28184 nM Potency
TKC022931 Q96RI1 Bile acid receptor None 50119 nM Potency
TKC026455 Q96RI1 Bile acid receptor None 17000 nM IC50
TKC027095 Q96RI1 Bile acid receptor None 1500 nM IC50
TKC027096 Q96RI1 Bile acid receptor None 1500 nM IC50
TKC027225 Q96RI1 Bile acid receptor None 5900 nM IC50
TKC035272 Q96RI1 Bile acid receptor None 22387 nM Potency
TKC045729 Q96RI1 Bile acid receptor None >100000 nM IC50
TKC045739 Q96RI1 Bile acid receptor None 60400 nM IC50
TKC045844 Q96RI1 Bile acid receptor None 24800 nM IC50
TKC045846 Q96RI1 Bile acid receptor None 81100 nM IC50
TKC046058 Q96RI1 Bile acid receptor None 31600 nM IC50
TKC046480 Q96RI1 Bile acid receptor None 24000 nM EC50
TKC048922 Q96RI1 Bile acid receptor None 8800 nM EC50
TKC048923 Q96RI1 Bile acid receptor None 3570 nM EC50
TKC048938 Q96RI1 Bile acid receptor None 15100 nM EC50
TKC048939 Q96RI1 Bile acid receptor None 25290 nM EC50
TKC048940 Q96RI1 Bile acid receptor None 4740 nM EC50
TKC048951 Q96RI1 Bile acid receptor None 3260 nM EC50
TKC050873 Q96RI1 Bile acid receptor None 3030 nM EC50
TKC050874 Q96RI1 Bile acid receptor None 140 nM EC50
TKC050875 Q96RI1 Bile acid receptor None 2400 nM EC50
TKC052230 Q96RI1 Bile acid receptor None 13300 nM EC50
TKC052231 Q96RI1 Bile acid receptor None 5660 nM EC50
TKC052444 Q96RI1 Bile acid receptor None 10400 nM EC50
TKC053303 Q96RI1 Bile acid receptor None 40740 nM EC50
TKC054499 Q96RI1 Bile acid receptor None 20240 nM EC50
TKC055291 Q96RI1 Bile acid receptor None 0 nM EC50
TKC055602 Q96RI1 Bile acid receptor None 0 nM EC50
TKC056482 Q96RI1 Bile acid receptor None 0 nM EC50
TKC061474 Q96RI1 Bile acid receptor None 4 nM Potency
TKC062736 Q96RI1 Bile acid receptor None 5640 nM EC50
TKC063162 Q96RI1 Bile acid receptor None 29680 nM EC50
TKC063163 Q96RI1 Bile acid receptor None 10160 nM EC50
TKC063164 Q96RI1 Bile acid receptor None 15310 nM EC50
TKC063165 Q96RI1 Bile acid receptor None 64890 nM EC50
TKC063168 Q96RI1 Bile acid receptor None 940 nM EC50
TKC063169 Q96RI1 Bile acid receptor None 8900 nM EC50
TKC064374 Q96RI1 Bile acid receptor None 0 nM EC50
TKC064856 Q96RI1 Bile acid receptor None 6000 nM EC50
TKC064857 Q96RI1 Bile acid receptor None 12140 nM EC50
TKC064858 Q96RI1 Bile acid receptor None 15470 nM EC50
TKC064860 Q96RI1 Bile acid receptor None 24090 nM EC50
TKC066169 Q96RI1 Bile acid receptor None 35481 nM Potency
TKC074296 Q96RI1 Bile acid receptor None 20150 nM EC50
TKC074867 Q96RI1 Bile acid receptor None 1 nM Potency
TKC075769 Q96RI1 Bile acid receptor None 18 nM Potency
TKC077533 Q96RI1 Bile acid receptor None 0 nM EC50
TKC077595 Q96RI1 Bile acid receptor None 0 nM EC50
TKC077599 Q96RI1 Bile acid receptor None 0 nM EC50
TKC077601 Q96RI1 Bile acid receptor None 0 nM EC50
TKC077608 Q96RI1 Bile acid receptor None 0 nM EC50
TKC077609 Q96RI1 Bile acid receptor None 0 nM EC50
TKC077612 Q96RI1 Bile acid receptor None 0 nM EC50
TKC077626 Q96RI1 Bile acid receptor None 0 nM EC50
TKC077689 Q96RI1 Bile acid receptor None 0 nM EC50
TKC082589 Q96RI1 Bile acid receptor None 0 nM EC50
TKC082597 Q96RI1 Bile acid receptor None 0 nM EC50
TKC082600 Q96RI1 Bile acid receptor None 0 nM EC50
TKC082608 Q96RI1 Bile acid receptor None 0 nM EC50
TKC082609 Q96RI1 Bile acid receptor None 0 nM EC50
TKC082639 Q96RI1 Bile acid receptor None 0 nM EC50
TKC082652 Q96RI1 Bile acid receptor None 0 nM EC50
TKC082703 Q96RI1 Bile acid receptor None 0 nM EC50
TKC082710 Q96RI1 Bile acid receptor None 0 nM EC50
TKC082711 Q96RI1 Bile acid receptor None 0 nM EC50
TKC082712 Q96RI1 Bile acid receptor None 0 nM EC50
TKC086929 Q96RI1 Bile acid receptor None 2 nM Potency
TKC087988 Q96RI1 Bile acid receptor None 7080 nM Potency
TKC087991 Q96RI1 Bile acid receptor None 70795 nM Potency
TKC092297 Q96RI1 Bile acid receptor None 39811 nM Potency
TKC092348 Q96RI1 Bile acid receptor None 25119 nM Potency
TKC093375 Q96RI1 Bile acid receptor None 9000 nM IC50
TKC096012 Q96RI1 Bile acid receptor None 17783 nM Potency
TKC100644 Q96RI1 Bile acid receptor None 39811 nM Potency
TKC102407 Q96RI1 Bile acid receptor None 22387 nM Potency
TKC103074 Q96RI1 Bile acid receptor None 0 nM EC50
TKC104925 Q96RI1 Bile acid receptor None 0 nM EC50
TKC105149 Q96RI1 Bile acid receptor None 1 % Activity
TKC106240 Q96RI1 Bile acid receptor None 3400 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 13000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 27000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 8300 nM EC50
TKC106240 Q96RI1 Bile acid receptor None >01000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None >10000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None >10000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None >10000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 18000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 18000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 18000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 13000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 21000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 10000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 8660 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 9000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 8660 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 8660 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 3500 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 11700 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 8660 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 13000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 6310 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 13000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 27000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 13000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 15000 nM EC50
TKC106240 Q96RI1 Bile acid receptor None 8660 nM EC50
TKC106240 Q96RI1 Bile acid receptor None >10000 nM EC50
TKC106250 Q96RI1 Bile acid receptor None 50000 nM EC50
TKC107086 Q96RI1 Bile acid receptor None 28184 nM Potency
TKC107735 Q96RI1 Bile acid receptor None 15849 nM Potency
TKC108191 Q96RI1 Bile acid receptor None 0 nM EC50
TKC108536 Q96RI1 Bile acid receptor None 4 nM Potency
TKC109619 Q96RI1 Bile acid receptor None 50000 nM EC50
TKC109622 Q96RI1 Bile acid receptor None 2 % Activity
TKC111390 Q96RI1 Bile acid receptor None 80 % Inhibition
TKC112787 Q96RI1 Bile acid receptor None 5 % Activity
TKC113499 Q96RI1 Bile acid receptor None 30 % Activity
TKC114511 Q96RI1 Bile acid receptor None 12000 nM EC50
TKC114511 Q96RI1 Bile acid receptor None 100000 nM IC50
TKC114511 Q96RI1 Bile acid receptor None 10000 nM IC50
TKC114511 Q96RI1 Bile acid receptor None 12000 nM IC50
TKC114511 Q96RI1 Bile acid receptor None 89360 nM IC50
TKC114511 Q96RI1 Bile acid receptor None 4100 nM IC50
TKC114511 Q96RI1 Bile acid receptor None 41000 nM IC50
TKC114511 Q96RI1 Bile acid receptor None 44000 nM IC50
TKC115268 Q96RI1 Bile acid receptor None 44668 nM Potency
TKC117705 Q96RI1 Bile acid receptor None >9 % Efficacy
TKC117716 Q96RI1 Bile acid receptor None 33180 nM EC50
TKC117717 Q96RI1 Bile acid receptor None 10230 nM EC50
TKC123088 Q96RI1 Bile acid receptor None 0 nM EC50
TKC131507 Q96RI1 Bile acid receptor None 2500 nM IC50
TKC134780 Q96RI1 Bile acid receptor None 35481 nM Potency
TKC137135 Q96RI1 Bile acid receptor None 2400 nM IC50
TKC137137 Q96RI1 Bile acid receptor None 75000 nM IC50
TKC137142 Q96RI1 Bile acid receptor None 24000 nM IC50
TKC137199 Q96RI1 Bile acid receptor None 64500 nM IC50
TKC137200 Q96RI1 Bile acid receptor None 25300 nM IC50
TKC141147 Q96RI1 Bile acid receptor None 0 nM EC50
TKC141164 Q96RI1 Bile acid receptor None 0 nM EC50
TKC141622 Q96RI1 Bile acid receptor None 0 nM EC50
TKC144889 Q96RI1 Bile acid receptor None 189050 nM EC50
TKC145498 Q96RI1 Bile acid receptor None 3360 nM EC50
TKC145848 Q96RI1 Bile acid receptor None 0 nM EC50
TKC145932 Q96RI1 Bile acid receptor None 0 nM EC50
TKC147336 Q96RI1 Bile acid receptor None 34190 nM EC50
TKC150706 Q96RI1 Bile acid receptor None 0 nM EC50
TKC151412 Q96RI1 Bile acid receptor None 110 nM EC50
TKC151556 Q96RI1 Bile acid receptor None 2100 nM EC50
TKC152742 Q96RI1 Bile acid receptor None 0 nM EC50
TKC152765 Q96RI1 Bile acid receptor None 0 nM EC50
TKC152829 Q96RI1 Bile acid receptor None 0 nM EC50
TKC166596 Q96RI1 Bile acid receptor None 0 nM EC50
TKC167188 Q96RI1 Bile acid receptor None 8100 nM IC50
TKC170602 Q96RI1 Bile acid receptor None 0 nM EC50
TKC170603 Q96RI1 Bile acid receptor None 0 nM EC50
TKC203882 Q96RI1 Bile acid receptor None 7320 nM EC50
TKC206249 Q96RI1 Bile acid receptor None 12430 nM EC50
TKC206344 Q96RI1 Bile acid receptor None 90 nM EC50
TKC206652 Q96RI1 Bile acid receptor None 447 nM Potency
TKC206670 Q96RI1 Bile acid receptor None 3000 nM EC50
TKC206671 Q96RI1 Bile acid receptor None 3000 nM EC50
TKC206672 Q96RI1 Bile acid receptor None 45000 nM EC50
TKC206688 Q96RI1 Bile acid receptor None 28184 nM Potency
TKC206759 Q96RI1 Bile acid receptor None 22387 nM Potency
TKC206760 Q96RI1 Bile acid receptor None 100000 nM EC50
TKC206760 Q96RI1 Bile acid receptor None 18 nM IC50
TKC206760 Q96RI1 Bile acid receptor None 20000 nM EC50
TKC206760 Q96RI1 Bile acid receptor None 6700 nM EC50
TKC206812 Q96RI1 Bile acid receptor None 130 nM EC50
TKC206812 Q96RI1 Bile acid receptor None 5000 nM Ki
TKC206816 Q96RI1 Bile acid receptor None 12589 nM Potency
TKC206884 Q96RI1 Bile acid receptor None 25119 nM Potency
TKC206884 Q96RI1 Bile acid receptor None 2 % Efficacy
TKC206884 Q96RI1 Bile acid receptor None >100000 nM EC50
TKC206884 Q96RI1 Bile acid receptor None >100000 nM EC50
TKC206885 Q96RI1 Bile acid receptor None 100000 nM EC50
TKC206927 Q96RI1 Bile acid receptor None 520 nM EC50
TKC112754 Q9UHC9 NPC1-like intracellular cholesterol transporter 1 None >10000 nM EC50
TKC112813 Q9UHC9 NPC1-like intracellular cholesterol transporter 1 None 3400 nM EC50
TKC112826 Q9UHC9 NPC1-like intracellular cholesterol transporter 1 None 8700 nM EC50
TKC118895 Q9UHC9 NPC1-like intracellular cholesterol transporter 1 None 1700 nM EC50
TKC206458 Q9UHC9 NPC1-like intracellular cholesterol transporter 1 None 2900 nM EC50
TKC206915 Q9UHC9 NPC1-like intracellular cholesterol transporter 1 None 3400 nM EC50