TKC050429
|
O14920 |
Inhibitor of nuclear factor kappa-B kinase subunit beta |
None |
2620 |
nM |
IC50 |
TKC077819
|
O14920 |
Inhibitor of nuclear factor kappa-B kinase subunit beta |
None |
4240 |
nM |
IC50 |
TKC118419
|
O14920 |
Inhibitor of nuclear factor kappa-B kinase subunit beta |
None |
96 |
% |
Activity |
TKC013753
|
P03372 |
Estrogen receptor |
None |
8913 |
nM |
Potency |
TKC019072
|
P03372 |
Estrogen receptor |
None |
78 |
% |
Activity |
TKC022931
|
P03372 |
Estrogen receptor |
None |
1995 |
nM |
Potency |
TKC022961
|
P03372 |
Estrogen receptor |
None |
54 |
% |
Activity |
TKC028029
|
P03372 |
Estrogen receptor |
None |
0 |
% |
Activity |
TKC028034
|
P03372 |
Estrogen receptor |
None |
<0 |
% |
Activity |
TKC028037
|
P03372 |
Estrogen receptor |
None |
1 |
% |
Activity |
TKC028038
|
P03372 |
Estrogen receptor |
None |
<0 |
% |
Activity |
TKC028041
|
P03372 |
Estrogen receptor |
None |
<0 |
% |
Activity |
TKC034016
|
P03372 |
Estrogen receptor |
None |
51 |
% |
Activity |
TKC034337
|
P03372 |
Estrogen receptor |
None |
2800000 |
nM |
IC50 |
TKC034640
|
P03372 |
Estrogen receptor |
None |
>1000000 |
nM |
Ki |
TKC035208
|
P03372 |
Estrogen receptor |
None |
39 |
% |
Activity |
TKC035272
|
P03372 |
Estrogen receptor |
None |
2551 |
nM |
IC50 |
TKC035462
|
P03372 |
Estrogen receptor |
None |
42 |
% |
Activity |
TKC066169
|
P03372 |
Estrogen receptor |
None |
39811 |
nM |
Potency |
TKC075769
|
P03372 |
Estrogen receptor |
None |
251 |
nM |
Potency |
TKC079320
|
P03372 |
Estrogen receptor |
None |
<0 |
% |
Activity |
TKC079321
|
P03372 |
Estrogen receptor |
None |
<0 |
% |
Activity |
TKC087664
|
P03372 |
Estrogen receptor |
None |
3162 |
nM |
Potency |
TKC087988
|
P03372 |
Estrogen receptor |
None |
631 |
nM |
Potency |
TKC087991
|
P03372 |
Estrogen receptor |
None |
4467 |
nM |
Potency |
TKC092297
|
P03372 |
Estrogen receptor |
None |
15849 |
nM |
Potency |
TKC092348
|
P03372 |
Estrogen receptor |
None |
8913 |
nM |
Potency |
TKC096012
|
P03372 |
Estrogen receptor |
None |
126 |
nM |
Potency |
TKC100644
|
P03372 |
Estrogen receptor |
None |
31623 |
nM |
Potency |
TKC101365
|
P03372 |
Estrogen receptor |
None |
12570 |
nM |
EC50 |
TKC102448
|
P03372 |
Estrogen receptor |
None |
2550 |
nM |
EC50 |
TKC107086
|
P03372 |
Estrogen receptor |
None |
8913 |
nM |
Potency |
TKC107735
|
P03372 |
Estrogen receptor |
None |
50119 |
nM |
Potency |
TKC111727
|
P03372 |
Estrogen receptor |
None |
0 |
nM |
Ki |
TKC111738
|
P03372 |
Estrogen receptor |
None |
1 |
nM |
EC50 |
TKC111738
|
P03372 |
Estrogen receptor |
None |
166 |
nM |
IC50 |
TKC111738
|
P03372 |
Estrogen receptor |
None |
210 |
nM |
IC50 |
TKC111738
|
P03372 |
Estrogen receptor |
None |
96 |
nM |
IC50 |
TKC112923
|
P03372 |
Estrogen receptor |
None |
26 |
nM |
EC50 |
TKC115268
|
P03372 |
Estrogen receptor |
None |
15849 |
nM |
Potency |
TKC129821
|
P03372 |
Estrogen receptor |
None |
70 |
% |
Activity |
TKC151345
|
P03372 |
Estrogen receptor |
None |
35 |
% |
Activity |
TKC151713
|
P03372 |
Estrogen receptor |
None |
40 |
% |
Activity |
TKC151765
|
P03372 |
Estrogen receptor |
None |
81 |
% |
Activity |
TKC206549
|
P03372 |
Estrogen receptor |
None |
3548 |
nM |
Potency |
TKC206608
|
P03372 |
Estrogen receptor |
None |
8170 |
nM |
EC50 |
TKC206652
|
P03372 |
Estrogen receptor |
None |
112 |
nM |
Potency |
TKC206725
|
P03372 |
Estrogen receptor |
None |
8 |
nM |
Ki |
TKC206726
|
P03372 |
Estrogen receptor |
None |
72 |
nM |
EC50 |
TKC206759
|
P03372 |
Estrogen receptor |
None |
>10000 |
nM |
IC50 |
TKC206759
|
P03372 |
Estrogen receptor |
None |
>10000 |
nM |
IC50 |
TKC206760
|
P03372 |
Estrogen receptor |
None |
25119 |
nM |
Potency |
TKC206764
|
P03372 |
Estrogen receptor |
None |
0 |
% |
RBA |
TKC206770
|
P03372 |
Estrogen receptor |
None |
5012 |
nM |
Potency |
TKC206779
|
P03372 |
Estrogen receptor |
None |
6310 |
nM |
Potency |
TKC206812
|
P03372 |
Estrogen receptor |
None |
62000 |
nM |
IC50 |
TKC206812
|
P03372 |
Estrogen receptor |
None |
39811 |
nM |
Potency |
TKC206816
|
P03372 |
Estrogen receptor |
None |
>1000 |
nM |
IC50 |
TKC206816
|
P03372 |
Estrogen receptor |
None |
>1000 |
nM |
IC50 |
TKC009193
|
P08253 |
72 kDa type IV collagenase |
None |
33260 |
nM |
IC50 |
TKC020117
|
P08253 |
72 kDa type IV collagenase |
None |
90 |
% |
Inhibition |
TKC023429
|
P08253 |
72 kDa type IV collagenase |
None |
0 |
ug.mL-1 |
IC50 |
TKC020967
|
P0DPI0 |
Botulinum neurotoxin type A |
None |
0 |
/M/s |
Ratio |
TKC123088
|
P0DPI0 |
Botulinum neurotoxin type A |
None |
14300 |
nM |
Ki |
TKC141147
|
P0DPI0 |
Botulinum neurotoxin type A |
None |
<100000 |
nM |
IC50 |
TKC141164
|
P0DPI0 |
Botulinum neurotoxin type A |
None |
<100000 |
nM |
IC50 |
TKC151761
|
P0DPI0 |
Botulinum neurotoxin type A |
None |
5200 |
nM |
IC50 |
TKC200866
|
P0DPI0 |
Botulinum neurotoxin type A |
None |
5200 |
nM |
IC50 |
TKC001669
|
P10275 |
Androgen receptor |
None |
260 |
nM |
IC50 |
TKC006934
|
P10275 |
Androgen receptor |
None |
50119 |
nM |
Potency |
TKC013304
|
P10275 |
Androgen receptor |
None |
70795 |
nM |
Potency |
TKC019571
|
P10275 |
Androgen receptor |
None |
19953 |
nM |
Potency |
TKC021325
|
P10275 |
Androgen receptor |
None |
31623 |
nM |
Potency |
TKC021332
|
P10275 |
Androgen receptor |
None |
31623 |
nM |
Potency |
TKC023246
|
P10275 |
Androgen receptor |
None |
449 |
nM |
IC50 |
TKC030239
|
P10275 |
Androgen receptor |
None |
14 |
nM |
Potency |
TKC035272
|
P10275 |
Androgen receptor |
None |
15849 |
nM |
Potency |
TKC056140
|
P10275 |
Androgen receptor |
None |
50 |
% |
Activity |
TKC066169
|
P10275 |
Androgen receptor |
None |
3981 |
nM |
Potency |
TKC074867
|
P10275 |
Androgen receptor |
None |
28184 |
nM |
Potency |
TKC075769
|
P10275 |
Androgen receptor |
None |
355 |
nM |
Potency |
TKC079001
|
P10275 |
Androgen receptor |
None |
1 |
nM |
Potency |
TKC096012
|
P10275 |
Androgen receptor |
None |
178 |
nM |
Potency |
TKC100644
|
P10275 |
Androgen receptor |
None |
35481 |
nM |
Potency |
TKC102407
|
P10275 |
Androgen receptor |
None |
44668 |
nM |
Potency |
TKC106878
|
P10275 |
Androgen receptor |
None |
238 |
nM |
IC50 |
TKC107086
|
P10275 |
Androgen receptor |
None |
17783 |
nM |
Potency |
TKC107735
|
P10275 |
Androgen receptor |
None |
3981 |
nM |
Potency |
TKC111738
|
P10275 |
Androgen receptor |
None |
17783 |
nM |
Potency |
TKC112923
|
P10275 |
Androgen receptor |
None |
212 |
nM |
IC50 |
TKC114095
|
P10275 |
Androgen receptor |
None |
1790 |
nM |
IC50 |
TKC114511
|
P10275 |
Androgen receptor |
None |
315 |
nM |
Ki |
TKC115268
|
P10275 |
Androgen receptor |
None |
35481 |
nM |
Potency |
TKC115284
|
P10275 |
Androgen receptor |
None |
1 |
nM |
Ki |
TKC117154
|
P10275 |
Androgen receptor |
None |
580 |
nM |
IC50 |
TKC120161
|
P10275 |
Androgen receptor |
None |
44668 |
nM |
Potency |
TKC122884
|
P10275 |
Androgen receptor |
None |
39811 |
nM |
Potency |
TKC122892
|
P10275 |
Androgen receptor |
None |
10000 |
nM |
IC50 |
TKC134780
|
P10275 |
Androgen receptor |
None |
2 |
nM |
Potency |
TKC147240
|
P10275 |
Androgen receptor |
None |
50 |
% |
Activity |
TKC206652
|
P10275 |
Androgen receptor |
None |
50 |
nM |
Potency |
TKC206688
|
P10275 |
Androgen receptor |
None |
224 |
nM |
Potency |
TKC206690
|
P10275 |
Androgen receptor |
None |
36 |
nM |
Potency |
TKC206759
|
P10275 |
Androgen receptor |
None |
2 |
nM |
Potency |
TKC206759
|
P10275 |
Androgen receptor |
None |
3.9 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
4.7 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
4.2 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
29 |
nM |
Ki |
TKC206759
|
P10275 |
Androgen receptor |
None |
1.1 |
nM |
EC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
2.7 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
2.7 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
2.7 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
30 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
4.57 |
nM |
IC50 |
TKC206770
|
P10275 |
Androgen receptor |
None |
224 |
nM |
Potency |
TKC206779
|
P10275 |
Androgen receptor |
None |
2 |
nM |
Potency |
TKC206812
|
P10275 |
Androgen receptor |
None |
220 |
nM |
IC50 |
TKC206816
|
P10275 |
Androgen receptor |
None |
9 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
8.5 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
8.5 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
8.5 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
8.5 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
37 |
nM |
IC50 |
TKC206816
|
P10275 |
Androgen receptor |
None |
8.5 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
35 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
14 |
nM |
IC50 |
TKC000075
|
P11473 |
Vitamin D3 receptor |
None |
70795 |
nM |
Potency |
TKC002371
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC005454
|
P11473 |
Vitamin D3 receptor |
None |
7080 |
nM |
Potency |
TKC008359
|
P11473 |
Vitamin D3 receptor |
None |
28184 |
nM |
Potency |
TKC011412
|
P11473 |
Vitamin D3 receptor |
None |
19953 |
nM |
Potency |
TKC013736
|
P11473 |
Vitamin D3 receptor |
None |
11220 |
nM |
Potency |
TKC013755
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC013760
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC014568
|
P11473 |
Vitamin D3 receptor |
None |
63096 |
nM |
Potency |
TKC016371
|
P11473 |
Vitamin D3 receptor |
None |
56234 |
nM |
Potency |
TKC017379
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC020031
|
P11473 |
Vitamin D3 receptor |
None |
100000 |
nM |
Potency |
TKC020117
|
P11473 |
Vitamin D3 receptor |
None |
56234 |
nM |
Potency |
TKC027192
|
P11473 |
Vitamin D3 receptor |
None |
35481 |
nM |
Potency |
TKC030239
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC032619
|
P11473 |
Vitamin D3 receptor |
None |
31623 |
nM |
Potency |
TKC032913
|
P11473 |
Vitamin D3 receptor |
None |
70795 |
nM |
Potency |
TKC034083
|
P11473 |
Vitamin D3 receptor |
None |
39811 |
nM |
Potency |
TKC034760
|
P11473 |
Vitamin D3 receptor |
None |
35481 |
nM |
Potency |
TKC035208
|
P11473 |
Vitamin D3 receptor |
None |
39811 |
nM |
Potency |
TKC035272
|
P11473 |
Vitamin D3 receptor |
None |
6310 |
nM |
Potency |
TKC037521
|
P11473 |
Vitamin D3 receptor |
None |
79433 |
nM |
Potency |
TKC038268
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC038273
|
P11473 |
Vitamin D3 receptor |
None |
56234 |
nM |
Potency |
TKC038706
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC041160
|
P11473 |
Vitamin D3 receptor |
None |
79433 |
nM |
Potency |
TKC043519
|
P11473 |
Vitamin D3 receptor |
None |
79433 |
nM |
Potency |
TKC053095
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC053227
|
P11473 |
Vitamin D3 receptor |
None |
14125 |
nM |
Potency |
TKC053825
|
P11473 |
Vitamin D3 receptor |
None |
35481 |
nM |
Potency |
TKC055219
|
P11473 |
Vitamin D3 receptor |
None |
100000 |
nM |
Potency |
TKC057133
|
P11473 |
Vitamin D3 receptor |
None |
39811 |
nM |
Potency |
TKC062321
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC062327
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC062332
|
P11473 |
Vitamin D3 receptor |
None |
70795 |
nM |
Potency |
TKC062333
|
P11473 |
Vitamin D3 receptor |
None |
39811 |
nM |
Potency |
TKC062669
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC066096
|
P11473 |
Vitamin D3 receptor |
None |
28184 |
nM |
Potency |
TKC066169
|
P11473 |
Vitamin D3 receptor |
None |
7943 |
nM |
Potency |
TKC073833
|
P11473 |
Vitamin D3 receptor |
None |
56234 |
nM |
Potency |
TKC073873
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC074866
|
P11473 |
Vitamin D3 receptor |
None |
1 |
nM |
Potency |
TKC075769
|
P11473 |
Vitamin D3 receptor |
None |
562 |
nM |
Potency |
TKC082279
|
P11473 |
Vitamin D3 receptor |
None |
70795 |
nM |
Potency |
TKC082378
|
P11473 |
Vitamin D3 receptor |
None |
25119 |
nM |
Potency |
TKC083025
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC086929
|
P11473 |
Vitamin D3 receptor |
None |
39811 |
nM |
Potency |
TKC087533
|
P11473 |
Vitamin D3 receptor |
None |
56234 |
nM |
Potency |
TKC087664
|
P11473 |
Vitamin D3 receptor |
None |
100000 |
nM |
Potency |
TKC087988
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC091895
|
P11473 |
Vitamin D3 receptor |
None |
79433 |
nM |
Potency |
TKC092297
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC092348
|
P11473 |
Vitamin D3 receptor |
None |
39811 |
nM |
Potency |
TKC093161
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC095442
|
P11473 |
Vitamin D3 receptor |
None |
39811 |
nM |
Potency |
TKC095452
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC096012
|
P11473 |
Vitamin D3 receptor |
None |
31623 |
nM |
Potency |
TKC097937
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC098345
|
P11473 |
Vitamin D3 receptor |
None |
28184 |
nM |
Potency |
TKC098704
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC099703
|
P11473 |
Vitamin D3 receptor |
None |
39811 |
nM |
Potency |
TKC100636
|
P11473 |
Vitamin D3 receptor |
None |
3981 |
nM |
Potency |
TKC100644
|
P11473 |
Vitamin D3 receptor |
None |
35481 |
nM |
Potency |
TKC100701
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC101052
|
P11473 |
Vitamin D3 receptor |
None |
56234 |
nM |
Potency |
TKC101598
|
P11473 |
Vitamin D3 receptor |
None |
56234 |
nM |
Potency |
TKC102204
|
P11473 |
Vitamin D3 receptor |
None |
28184 |
nM |
Potency |
TKC102407
|
P11473 |
Vitamin D3 receptor |
None |
15849 |
nM |
Potency |
TKC102540
|
P11473 |
Vitamin D3 receptor |
None |
35481 |
nM |
Potency |
TKC102593
|
P11473 |
Vitamin D3 receptor |
None |
7080 |
nM |
Potency |
TKC102939
|
P11473 |
Vitamin D3 receptor |
None |
63096 |
nM |
Potency |
TKC103023
|
P11473 |
Vitamin D3 receptor |
None |
28184 |
nM |
Potency |
TKC103159
|
P11473 |
Vitamin D3 receptor |
None |
100000 |
nM |
Potency |
TKC103257
|
P11473 |
Vitamin D3 receptor |
None |
3162 |
nM |
Potency |
TKC103542
|
P11473 |
Vitamin D3 receptor |
None |
28184 |
nM |
Potency |
TKC103736
|
P11473 |
Vitamin D3 receptor |
None |
3548 |
nM |
Potency |
TKC104404
|
P11473 |
Vitamin D3 receptor |
None |
28184 |
nM |
Potency |
TKC104960
|
P11473 |
Vitamin D3 receptor |
None |
79433 |
nM |
Potency |
TKC104961
|
P11473 |
Vitamin D3 receptor |
None |
35481 |
nM |
Potency |
TKC105153
|
P11473 |
Vitamin D3 receptor |
None |
7943 |
nM |
Potency |
TKC105295
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC105424
|
P11473 |
Vitamin D3 receptor |
None |
19953 |
nM |
Potency |
TKC105932
|
P11473 |
Vitamin D3 receptor |
None |
63096 |
nM |
Potency |
TKC106240
|
P11473 |
Vitamin D3 receptor |
None |
>50000 |
nM |
IC50 |
TKC106250
|
P11473 |
Vitamin D3 receptor |
None |
>50000 |
nM |
IC50 |
TKC106301
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC106364
|
P11473 |
Vitamin D3 receptor |
None |
7080 |
nM |
Potency |
TKC106367
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC106426
|
P11473 |
Vitamin D3 receptor |
None |
14125 |
nM |
Potency |
TKC107086
|
P11473 |
Vitamin D3 receptor |
None |
31623 |
nM |
Potency |
TKC107332
|
P11473 |
Vitamin D3 receptor |
None |
19953 |
nM |
Potency |
TKC107625
|
P11473 |
Vitamin D3 receptor |
None |
56234 |
nM |
Potency |
TKC107627
|
P11473 |
Vitamin D3 receptor |
None |
35481 |
nM |
Potency |
TKC107735
|
P11473 |
Vitamin D3 receptor |
None |
17783 |
nM |
Potency |
TKC107775
|
P11473 |
Vitamin D3 receptor |
None |
100000 |
nM |
Potency |
TKC107830
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC109619
|
P11473 |
Vitamin D3 receptor |
None |
>50000 |
nM |
IC50 |
TKC109849
|
P11473 |
Vitamin D3 receptor |
None |
>100000 |
nM |
IC50 |
TKC109996
|
P11473 |
Vitamin D3 receptor |
None |
100000 |
nM |
Potency |
TKC111464
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC112754
|
P11473 |
Vitamin D3 receptor |
None |
79433 |
nM |
Potency |
TKC112759
|
P11473 |
Vitamin D3 receptor |
None |
70795 |
nM |
Potency |
TKC112784
|
P11473 |
Vitamin D3 receptor |
None |
19953 |
nM |
Potency |
TKC112785
|
P11473 |
Vitamin D3 receptor |
None |
>40100 |
nM |
IC50 |
TKC112787
|
P11473 |
Vitamin D3 receptor |
None |
>14500 |
nM |
IC50 |
TKC112792
|
P11473 |
Vitamin D3 receptor |
None |
28184 |
nM |
Potency |
TKC112906
|
P11473 |
Vitamin D3 receptor |
None |
25119 |
nM |
Potency |
TKC113063
|
P11473 |
Vitamin D3 receptor |
None |
5805 |
nM |
Potency |
TKC113146
|
P11473 |
Vitamin D3 receptor |
None |
39811 |
nM |
Potency |
TKC113150
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC113161
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC113663
|
P11473 |
Vitamin D3 receptor |
None |
35481 |
nM |
Potency |
TKC114511
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC114568
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC114819
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC115268
|
P11473 |
Vitamin D3 receptor |
None |
0 |
nM |
EC50 |
TKC115284
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC115284
|
P11473 |
Vitamin D3 receptor |
None |
>2408 |
uM |
Activity |
TKC118419
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC122884
|
P11473 |
Vitamin D3 receptor |
None |
35481 |
nM |
Potency |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
2 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
1 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.08 |
nM |
IC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
7.7 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.7 |
nM |
IC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.8 |
nM |
IC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
322 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.06 |
nM |
IC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.35 |
nM |
IC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
3.9 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
10 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.3 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.16 |
nM |
IC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.065 |
nM |
Kd |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
9 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.5 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.555 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
1 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
13 |
nM |
IC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
1.24 |
nM |
IC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.04 |
nM |
IC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
>0.900000 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
3 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.026 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
7.7 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
15 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
1.6 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.0953 |
nM |
IC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
0.011 |
nM |
EC50 |
TKC122892
|
P11473 |
Vitamin D3 receptor |
None |
24 |
nM |
Kd |
TKC134702
|
P11473 |
Vitamin D3 receptor |
None |
31623 |
nM |
Potency |
TKC136931
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC143885
|
P11473 |
Vitamin D3 receptor |
None |
79433 |
nM |
Potency |
TKC147290
|
P11473 |
Vitamin D3 receptor |
None |
25119 |
nM |
Potency |
TKC147303
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC148601
|
P11473 |
Vitamin D3 receptor |
None |
35481 |
nM |
Potency |
TKC149827
|
P11473 |
Vitamin D3 receptor |
None |
14125 |
nM |
Potency |
TKC151237
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC151571
|
P11473 |
Vitamin D3 receptor |
None |
22387 |
nM |
Potency |
TKC151609
|
P11473 |
Vitamin D3 receptor |
None |
79433 |
nM |
Potency |
TKC151675
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC151758
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC151784
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC151885
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC174441
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC205788
|
P11473 |
Vitamin D3 receptor |
None |
0 |
nM |
ED50 |
TKC205791
|
P11473 |
Vitamin D3 receptor |
None |
1 |
nM |
IC50 |
TKC205796
|
P11473 |
Vitamin D3 receptor |
None |
631 |
nM |
Potency |
TKC205798
|
P11473 |
Vitamin D3 receptor |
None |
11 |
% |
Activity |
TKC206385
|
P11473 |
Vitamin D3 receptor |
None |
>44 |
uM |
Activity |
TKC206544
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC206652
|
P11473 |
Vitamin D3 receptor |
None |
562 |
nM |
Potency |
TKC206669
|
P11473 |
Vitamin D3 receptor |
None |
>50000 |
nM |
IC50 |
TKC206672
|
P11473 |
Vitamin D3 receptor |
None |
>50000 |
nM |
IC50 |
TKC206758
|
P11473 |
Vitamin D3 receptor |
None |
56234 |
nM |
Potency |
TKC206760
|
P11473 |
Vitamin D3 receptor |
None |
8913 |
nM |
Potency |
TKC206760
|
P11473 |
Vitamin D3 receptor |
None |
6 |
% |
Activity |
TKC206760
|
P11473 |
Vitamin D3 receptor |
None |
330 |
nM |
Kd |
TKC206761
|
P11473 |
Vitamin D3 receptor |
None |
>15100 |
nM |
IC50 |
TKC206780
|
P11473 |
Vitamin D3 receptor |
None |
89125 |
nM |
Potency |
TKC206812
|
P11473 |
Vitamin D3 receptor |
None |
44668 |
nM |
Potency |
TKC206812
|
P11473 |
Vitamin D3 receptor |
None |
2000 |
nM |
IC50 |
TKC206816
|
P11473 |
Vitamin D3 receptor |
None |
15849 |
nM |
Potency |
TKC206876
|
P11473 |
Vitamin D3 receptor |
None |
79433 |
nM |
Potency |
TKC206884
|
P11473 |
Vitamin D3 receptor |
None |
50119 |
nM |
Potency |
TKC206884
|
P11473 |
Vitamin D3 receptor |
None |
>150000 |
nM |
EC50 |
TKC206901
|
P11473 |
Vitamin D3 receptor |
None |
31623 |
nM |
Potency |
TKC206902
|
P11473 |
Vitamin D3 receptor |
None |
35481 |
nM |
Potency |
TKC206960
|
P11473 |
Vitamin D3 receptor |
None |
17783 |
nM |
Potency |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
1 |
nM |
Kd |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
148 |
nM |
Kd |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
45 |
nM |
EC50 |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
74 |
nM |
EC50 |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
6 |
nM |
EC50 |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
12 |
nM |
EC50 |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
45 |
nM |
EC50 |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
1 |
nM |
Ki |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
148 |
nM |
Kd |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
6 |
nM |
EC50 |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
4 |
nM |
EC50 |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
6 |
nM |
EC50 |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
45 |
nM |
EC50 |
TKC013755
|
P13631 |
Retinoic acid receptor gamma |
None |
22 |
nM |
Kd |
TKC092297
|
P13631 |
Retinoic acid receptor gamma |
None |
>400 |
nM |
Ki |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
0 |
nM |
Ki |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
18 |
nM |
Kd |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
18 |
nM |
Kd |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
6 |
nM |
EC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
16 |
nM |
Kd |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
19 |
nM |
EC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
18 |
nM |
IC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
19 |
nM |
Kd |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
33 |
nM |
EC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
20 |
nM |
EC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
0.5 |
nM |
EC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
8 |
nM |
EC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
0.3 |
nM |
Kd |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
18 |
nM |
Kd |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
10 |
nM |
EC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
18 |
nM |
Kd |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
18 |
nM |
Kd |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
3 |
nM |
Kd |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
0.5 |
nM |
IC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
0.62 |
nM |
IC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
0.7 |
nM |
Ki |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
0.2 |
nM |
Kd |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
0.2 |
nM |
EC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
0.5 |
nM |
EC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
0.5 |
nM |
Ki |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
10 |
nM |
EC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
0.5 |
nM |
EC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
0.6 |
nM |
Ki |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
15 |
nM |
EC50 |
TKC096012
|
P13631 |
Retinoic acid receptor gamma |
None |
18 |
nM |
Kd |
TKC206482
|
P13631 |
Retinoic acid receptor gamma |
None |
6 |
nM |
EC50 |
TKC206812
|
P13631 |
Retinoic acid receptor gamma |
None |
>100000 |
nM |
EC50 |
TKC112925
|
P18405 |
3-oxo-5-alpha-steroid 4-dehydrogenase 1 |
None |
2700 |
nM |
IC50 |
TKC206770
|
P18405 |
3-oxo-5-alpha-steroid 4-dehydrogenase 1 |
None |
2700 |
nM |
IC50 |
TKC039202
|
P21453 |
Sphingosine 1-phosphate receptor 1 |
None |
4962 |
nM |
IC50 |
TKC096012
|
P21453 |
Sphingosine 1-phosphate receptor 1 |
None |
34120 |
nM |
EC50 |
TKC096012
|
P21453 |
Sphingosine 1-phosphate receptor 1 |
None |
>95100 |
nM |
EC50 |
TKC096012
|
P21453 |
Sphingosine 1-phosphate receptor 1 |
None |
25400 |
nM |
EC50 |
TKC075756
|
P33032 |
Melanocortin receptor 5 |
None |
3639 |
nM |
Ki |