TKC051021
|
P01375 |
Tumor necrosis factor |
None |
9 |
nM |
Kd |
TKC051029
|
P01375 |
Tumor necrosis factor |
None |
9 |
nM |
Kd |
TKC055869
|
P01375 |
Tumor necrosis factor |
None |
10880 |
nM |
IC50 |
TKC063751
|
P01375 |
Tumor necrosis factor |
None |
19 |
nM |
Kd |
TKC064986
|
P01375 |
Tumor necrosis factor |
None |
3 |
nM |
Kd |
TKC075769
|
P01375 |
Tumor necrosis factor |
None |
376 |
nM |
Potency |
TKC101833
|
P01375 |
Tumor necrosis factor |
None |
8 |
nM |
Kd |
TKC145547
|
P01375 |
Tumor necrosis factor |
None |
2 |
nM |
Kd |
TKC148618
|
P01375 |
Tumor necrosis factor |
None |
17 |
nM |
Kd |
TKC151763
|
P01375 |
Tumor necrosis factor |
None |
8 |
nM |
Kd |
TKC151876
|
P01375 |
Tumor necrosis factor |
None |
6 |
% |
Inhibition |
TKC008187
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
30200 |
nM |
IC50 |
TKC023515
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
53 |
% |
Inhibition |
TKC025574
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
52 |
% |
Inhibition |
TKC026893
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
21 |
% |
Inhibition |
TKC026895
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
61 |
% |
Inhibition |
TKC057019
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
22300 |
nM |
IC50 |
TKC100777
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
30 |
% |
Inhibition |
TKC101031
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
1500 |
nM |
IC50 |
TKC101538
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
39 |
% |
Inhibition |
TKC101847
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
1000 |
nM |
IC50 |
TKC103703
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
40 |
% |
Inhibition |
TKC137314
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
8400 |
nM |
IC50 |
TKC138471
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
21700 |
nM |
IC50 |
TKC017639
|
P04054 |
Phospholipase A2 |
None |
95 |
% |
Activity |
TKC017706
|
P04054 |
Phospholipase A2 |
None |
5 |
% |
Activity |
TKC045776
|
P04054 |
Phospholipase A2 |
None |
1600 |
nM |
IC50 |
TKC045777
|
P04054 |
Phospholipase A2 |
None |
3700 |
nM |
IC50 |
TKC045872
|
P04054 |
Phospholipase A2 |
None |
44 |
% |
Activity |
TKC046211
|
P04054 |
Phospholipase A2 |
None |
3900 |
nM |
IC50 |
TKC046211
|
P04054 |
Phospholipase A2 |
None |
13000 |
nM |
IC50 |
TKC055219
|
P04054 |
Phospholipase A2 |
None |
2040 |
nM |
IC50 |
TKC055219
|
P04054 |
Phospholipase A2 |
None |
2040 |
nM |
IC50 |
TKC077689
|
P04054 |
Phospholipase A2 |
None |
3000 |
nM |
IC50 |
TKC105149
|
P04054 |
Phospholipase A2 |
None |
8 |
% |
Activity |
TKC106090
|
P04054 |
Phospholipase A2 |
None |
95 |
% |
Activity |
TKC106091
|
P04054 |
Phospholipase A2 |
None |
90 |
% |
Activity |
TKC106240
|
P04054 |
Phospholipase A2 |
None |
5 |
% |
Activity |
TKC109622
|
P04054 |
Phospholipase A2 |
None |
10000 |
nM |
Kd |
TKC110322
|
P04054 |
Phospholipase A2 |
None |
67 |
% |
Inhibition |
TKC110427
|
P04054 |
Phospholipase A2 |
None |
13800 |
nM |
IC50 |
TKC112787
|
P04054 |
Phospholipase A2 |
None |
40 |
% |
Activity |
TKC115260
|
P04054 |
Phospholipase A2 |
None |
55 |
% |
Inhibition |
TKC146194
|
P04054 |
Phospholipase A2 |
None |
5 |
% |
Activity |
TKC151364
|
P04054 |
Phospholipase A2 |
None |
30 |
% |
Activity |
TKC152148
|
P04054 |
Phospholipase A2 |
None |
47 |
% |
Inhibition |
TKC206812
|
P04054 |
Phospholipase A2 |
None |
35 |
% |
Activity |
TKC206849
|
P04054 |
Phospholipase A2 |
None |
80 |
% |
Activity |
TKC206884
|
P04054 |
Phospholipase A2 |
None |
150000 |
nM |
Kd |
TKC012971
|
P04637 |
Cellular tumor antigen p53 |
None |
15849 |
nM |
Potency |
TKC013753
|
P04637 |
Cellular tumor antigen p53 |
None |
13 |
nM |
Potency |
TKC014568
|
P04637 |
Cellular tumor antigen p53 |
None |
2512 |
nM |
Potency |
TKC016418
|
P04637 |
Cellular tumor antigen p53 |
None |
15849 |
nM |
Potency |
TKC018710
|
P04637 |
Cellular tumor antigen p53 |
None |
5 |
nM |
Potency |
TKC020116
|
P04637 |
Cellular tumor antigen p53 |
None |
1585 |
nM |
Potency |
TKC020117
|
P04637 |
Cellular tumor antigen p53 |
None |
12589 |
nM |
Potency |
TKC020732
|
P04637 |
Cellular tumor antigen p53 |
None |
3162 |
nM |
Potency |
TKC022945
|
P04637 |
Cellular tumor antigen p53 |
None |
10000 |
nM |
Potency |
TKC032619
|
P04637 |
Cellular tumor antigen p53 |
None |
15849 |
nM |
Potency |
TKC034083
|
P04637 |
Cellular tumor antigen p53 |
None |
31623 |
nM |
Potency |
TKC035272
|
P04637 |
Cellular tumor antigen p53 |
None |
12589 |
nM |
Potency |
TKC039869
|
P04637 |
Cellular tumor antigen p53 |
None |
25119 |
nM |
Potency |
TKC052854
|
P04637 |
Cellular tumor antigen p53 |
None |
25119 |
nM |
Potency |
TKC062321
|
P04637 |
Cellular tumor antigen p53 |
None |
10000 |
nM |
Potency |
TKC075769
|
P04637 |
Cellular tumor antigen p53 |
None |
159 |
nM |
Potency |
TKC084075
|
P04637 |
Cellular tumor antigen p53 |
None |
8 |
nM |
Potency |
TKC091895
|
P04637 |
Cellular tumor antigen p53 |
None |
50119 |
nM |
Potency |
TKC092297
|
P04637 |
Cellular tumor antigen p53 |
None |
15849 |
nM |
Potency |
TKC095493
|
P04637 |
Cellular tumor antigen p53 |
None |
3162 |
nM |
Potency |
TKC100636
|
P04637 |
Cellular tumor antigen p53 |
None |
1585 |
nM |
Potency |
TKC100701
|
P04637 |
Cellular tumor antigen p53 |
None |
10000 |
nM |
Potency |
TKC101020
|
P04637 |
Cellular tumor antigen p53 |
None |
12589 |
nM |
Potency |
TKC101618
|
P04637 |
Cellular tumor antigen p53 |
None |
12589 |
nM |
Potency |
TKC102204
|
P04637 |
Cellular tumor antigen p53 |
None |
31623 |
nM |
Potency |
TKC102540
|
P04637 |
Cellular tumor antigen p53 |
None |
31623 |
nM |
Potency |
TKC103149
|
P04637 |
Cellular tumor antigen p53 |
None |
12589 |
nM |
Potency |
TKC103210
|
P04637 |
Cellular tumor antigen p53 |
None |
40 |
nM |
Potency |
TKC103257
|
P04637 |
Cellular tumor antigen p53 |
None |
10000 |
nM |
Potency |
TKC103736
|
P04637 |
Cellular tumor antigen p53 |
None |
2512 |
nM |
Potency |
TKC104070
|
P04637 |
Cellular tumor antigen p53 |
None |
63 |
nM |
Potency |
TKC104071
|
P04637 |
Cellular tumor antigen p53 |
None |
50 |
nM |
Potency |
TKC104072
|
P04637 |
Cellular tumor antigen p53 |
None |
126 |
nM |
Potency |
TKC104073
|
P04637 |
Cellular tumor antigen p53 |
None |
63 |
nM |
Potency |
TKC104114
|
P04637 |
Cellular tumor antigen p53 |
None |
79 |
nM |
Potency |
TKC105153
|
P04637 |
Cellular tumor antigen p53 |
None |
5012 |
nM |
Potency |
TKC105168
|
P04637 |
Cellular tumor antigen p53 |
None |
12589 |
nM |
Potency |
TKC105360
|
P04637 |
Cellular tumor antigen p53 |
None |
15849 |
nM |
Potency |
TKC105424
|
P04637 |
Cellular tumor antigen p53 |
None |
25119 |
nM |
Potency |
TKC105784
|
P04637 |
Cellular tumor antigen p53 |
None |
25119 |
nM |
Potency |
TKC105891
|
P04637 |
Cellular tumor antigen p53 |
None |
10000 |
nM |
Potency |
TKC106232
|
P04637 |
Cellular tumor antigen p53 |
None |
15849 |
nM |
Potency |
TKC107086
|
P04637 |
Cellular tumor antigen p53 |
None |
12589 |
nM |
Potency |
TKC107104
|
P04637 |
Cellular tumor antigen p53 |
None |
12589 |
nM |
Potency |
TKC107201
|
P04637 |
Cellular tumor antigen p53 |
None |
19953 |
nM |
Potency |
TKC107332
|
P04637 |
Cellular tumor antigen p53 |
None |
10000 |
nM |
Potency |
TKC107525
|
P04637 |
Cellular tumor antigen p53 |
None |
31623 |
nM |
Potency |
TKC107627
|
P04637 |
Cellular tumor antigen p53 |
None |
25119 |
nM |
Potency |
TKC107818
|
P04637 |
Cellular tumor antigen p53 |
None |
12589 |
nM |
Potency |
TKC108536
|
P04637 |
Cellular tumor antigen p53 |
None |
5 |
nM |
Potency |
TKC108732
|
P04637 |
Cellular tumor antigen p53 |
None |
19953 |
nM |
Potency |
TKC109484
|
P04637 |
Cellular tumor antigen p53 |
None |
20 |
nM |
Potency |
TKC109519
|
P04637 |
Cellular tumor antigen p53 |
None |
10000 |
nM |
Potency |
TKC109561
|
P04637 |
Cellular tumor antigen p53 |
None |
159 |
nM |
Potency |
TKC109569
|
P04637 |
Cellular tumor antigen p53 |
None |
32 |
nM |
Potency |
TKC110010
|
P04637 |
Cellular tumor antigen p53 |
None |
56234 |
nM |
Potency |
TKC112576
|
P04637 |
Cellular tumor antigen p53 |
None |
50 |
nM |
Potency |
TKC112784
|
P04637 |
Cellular tumor antigen p53 |
None |
31623 |
nM |
Potency |
TKC112792
|
P04637 |
Cellular tumor antigen p53 |
None |
25119 |
nM |
Potency |
TKC115268
|
P04637 |
Cellular tumor antigen p53 |
None |
70795 |
nM |
Potency |
TKC117625
|
P04637 |
Cellular tumor antigen p53 |
None |
3162 |
nM |
Potency |
TKC117993
|
P04637 |
Cellular tumor antigen p53 |
None |
501 |
nM |
Potency |
TKC117994
|
P04637 |
Cellular tumor antigen p53 |
None |
40 |
nM |
Potency |
TKC118006
|
P04637 |
Cellular tumor antigen p53 |
None |
100 |
nM |
Potency |
TKC118895
|
P04637 |
Cellular tumor antigen p53 |
None |
31623 |
nM |
Potency |
TKC132609
|
P04637 |
Cellular tumor antigen p53 |
None |
11220 |
nM |
Potency |
TKC134635
|
P04637 |
Cellular tumor antigen p53 |
None |
56234 |
nM |
Potency |
TKC138777
|
P04637 |
Cellular tumor antigen p53 |
None |
15849 |
nM |
Potency |
TKC140757
|
P04637 |
Cellular tumor antigen p53 |
None |
31623 |
nM |
Potency |
TKC147290
|
P04637 |
Cellular tumor antigen p53 |
None |
12589 |
nM |
Potency |
TKC148482
|
P04637 |
Cellular tumor antigen p53 |
None |
19953 |
nM |
Potency |
TKC149827
|
P04637 |
Cellular tumor antigen p53 |
None |
1000 |
nM |
Potency |
TKC150706
|
P04637 |
Cellular tumor antigen p53 |
None |
31623 |
nM |
Potency |
TKC151237
|
P04637 |
Cellular tumor antigen p53 |
None |
35481 |
nM |
Potency |
TKC151303
|
P04637 |
Cellular tumor antigen p53 |
None |
31623 |
nM |
Potency |
TKC151571
|
P04637 |
Cellular tumor antigen p53 |
None |
6310 |
nM |
Potency |
TKC151758
|
P04637 |
Cellular tumor antigen p53 |
None |
19953 |
nM |
Potency |
TKC173955
|
P04637 |
Cellular tumor antigen p53 |
None |
31623 |
nM |
Potency |
TKC206652
|
P04637 |
Cellular tumor antigen p53 |
None |
32 |
nM |
Potency |
TKC206657
|
P04637 |
Cellular tumor antigen p53 |
None |
8 |
nM |
Potency |
TKC206760
|
P04637 |
Cellular tumor antigen p53 |
None |
31623 |
nM |
Potency |
TKC206760
|
P04637 |
Cellular tumor antigen p53 |
None |
15000 |
nM |
Kd |
TKC206812
|
P04637 |
Cellular tumor antigen p53 |
None |
31623 |
nM |
Potency |
TKC206872
|
P04637 |
Cellular tumor antigen p53 |
None |
631 |
nM |
Potency |
TKC206889
|
P04637 |
Cellular tumor antigen p53 |
None |
501 |
nM |
Potency |
TKC206901
|
P04637 |
Cellular tumor antigen p53 |
None |
2512 |
nM |
Potency |
TKC020117
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
-67 |
% |
Inhibition |
TKC024485
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>50000 |
nM |
IC50 |
TKC024587
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
600 |
nM |
IC50 |
TKC024956
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
18000 |
nM |
IC50 |
TKC024992
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
450 |
nM |
IC50 |
TKC024993
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
14000 |
nM |
IC50 |
TKC025965
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>150000 |
nM |
IC50 |
TKC026303
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
4600 |
nM |
IC50 |
TKC026309
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
680 |
nM |
IC50 |
TKC027255
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>67 |
% |
Activity |
TKC034201
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>200000 |
nM |
IC50 |
TKC040026
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
72 |
% |
Inhibition |
TKC051154
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
2700 |
nM |
IC50 |
TKC056482
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>64 |
% |
Activity |
TKC058811
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
42000 |
nM |
IC50 |
TKC058812
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>93 |
% |
Activity |
TKC064374
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
42000 |
nM |
IC50 |
TKC064407
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>72 |
% |
Activity |
TKC065375
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>70 |
% |
Activity |
TKC071640
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>60 |
% |
Activity |
TKC076350
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
100 |
% |
Activity |
TKC077689
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
100 |
% |
Activity |
TKC077703
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>86 |
% |
Activity |
TKC078194
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
31800 |
nM |
IC50 |
TKC082039
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
48 |
% |
Inhibition |
TKC088678
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
24800 |
nM |
IC50 |
TKC089448
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
35 |
% |
Inhibition |
TKC094647
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
97 |
% |
Activity |
TKC107943
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
2000 |
nM |
IC50 |
TKC123028
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
30400 |
nM |
IC50 |
TKC124303
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
750 |
nM |
IC50 |
TKC133309
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>200000 |
nM |
IC50 |
TKC133656
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
25100 |
nM |
IC50 |
TKC134278
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>200000 |
nM |
IC50 |
TKC139322
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>67 |
% |
Activity |
TKC139366
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
3000 |
nM |
IC50 |
TKC141401
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
42000 |
nM |
IC50 |
TKC141499
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
25700 |
nM |
IC50 |
TKC141805
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>53 |
% |
Activity |
TKC142849
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>70 |
% |
Activity |
TKC142897
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
30600 |
nM |
IC50 |
TKC142922
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>61 |
% |
Activity |
TKC143539
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
100 |
% |
Activity |
TKC145848
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
42000 |
nM |
IC50 |
TKC145932
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>56 |
% |
Activity |
TKC145968
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
100 |
% |
Activity |
TKC146774
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>63 |
% |
Activity |
TKC149759
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>73 |
% |
Activity |
TKC150706
|
P09917 |
Polyunsaturated fatty acid 5-lipoxygenase |
None |
>62 |
% |
Activity |
TKC002411
|
P11597 |
Cholesteryl ester transfer protein |
None |
196000 |
nM |
IC50 |
TKC026245
|
P11597 |
Cholesteryl ester transfer protein |
None |
25000 |
nM |
IC50 |
TKC026309
|
P11597 |
Cholesteryl ester transfer protein |
None |
6000 |
nM |
IC50 |
TKC026600
|
P11597 |
Cholesteryl ester transfer protein |
None |
100000 |
nM |
IC50 |
TKC027200
|
P11597 |
Cholesteryl ester transfer protein |
None |
5000 |
nM |
IC50 |
TKC027200
|
P11597 |
Cholesteryl ester transfer protein |
None |
5200 |
nM |
IC50 |
TKC027201
|
P11597 |
Cholesteryl ester transfer protein |
None |
1000 |
nM |
IC50 |
TKC027201
|
P11597 |
Cholesteryl ester transfer protein |
None |
5200 |
nM |
IC50 |
TKC056482
|
P11597 |
Cholesteryl ester transfer protein |
None |
46600 |
nM |
IC50 |
TKC077689
|
P11597 |
Cholesteryl ester transfer protein |
None |
10 |
% |
Inhibition |
TKC094496
|
P11597 |
Cholesteryl ester transfer protein |
None |
46000 |
nM |
IC50 |
TKC097288
|
P11597 |
Cholesteryl ester transfer protein |
None |
600 |
nM |
IC50 |
TKC106450
|
P11597 |
Cholesteryl ester transfer protein |
None |
5200 |
nM |
IC50 |
TKC123088
|
P11597 |
Cholesteryl ester transfer protein |
None |
31 |
% |
Inhibition |
TKC075756
|
P17948 |
Vascular endothelial growth factor receptor 1 |
None |
1001 |
nM |
Ki |
TKC005454
|
P23141 |
Liver carboxylesterase 1 |
None |
544 |
nM |
Ki |
TKC012269
|
P23141 |
Liver carboxylesterase 1 |
None |
2530 |
nM |
Ki |
TKC014568
|
P23141 |
Liver carboxylesterase 1 |
None |
26250 |
nM |
Ki |
TKC088678
|
P23141 |
Liver carboxylesterase 1 |
None |
20970 |
nM |
IC50 |
TKC088715
|
P23141 |
Liver carboxylesterase 1 |
None |
49860 |
nM |
IC50 |
TKC101270
|
P23141 |
Liver carboxylesterase 1 |
None |
23610 |
nM |
IC50 |
TKC103069
|
P23141 |
Liver carboxylesterase 1 |
None |
49860 |
nM |
IC50 |
TKC107319
|
P23141 |
Liver carboxylesterase 1 |
None |
>100000 |
nM |
Ki |
TKC141401
|
P23141 |
Liver carboxylesterase 1 |
None |
10530 |
nM |
IC50 |
TKC141510
|
P23141 |
Liver carboxylesterase 1 |
None |
22360 |
nM |
IC50 |
TKC151739
|
P23141 |
Liver carboxylesterase 1 |
None |
>100000 |
nM |
IC50 |
TKC082111
|
P25116 |
Proteinase-activated receptor 1 |
None |
20000 |
nM |
IC50 |
TKC011761
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
54 |
% |
Inhibition |
TKC016414
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
36 |
% |
Activity |
TKC024886
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
48400 |
nM |
IC50 |
TKC025690
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
>100000 |
nM |
IC50 |
TKC044763
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
100 |
% |
Inhibition |
TKC115259
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
>100000 |
nM |
IC50 |
TKC115261
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
>100000 |
nM |
IC50 |
TKC115272
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
>100000 |
nM |
IC50 |
TKC115273
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
>100000 |
nM |
IC50 |
TKC118419
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
96 |
% |
Inhibition |
TKC152148
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
>100000 |
nM |
IC50 |
TKC152157
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
>100000 |
nM |
IC50 |
TKC174547
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
>100000 |
nM |
IC50 |
TKC206776
|
P31749 |
RAC-alpha serine/threonine-protein kinase |
None |
3 |
uM |
Activity |
TKC073907
|
P37268 |
Squalene synthase |
None |
2300 |
nM |
Km |
TKC122582
|
P37268 |
Squalene synthase |
None |
2300 |
nM |
Km |
TKC147153
|
P37268 |
Squalene synthase |
None |
2300 |
nM |
Km |
TKC205544
|
P43119 |
Prostacyclin receptor |
None |
8 |
% |
Inhibition |
TKC013304
|
P51449 |
Nuclear receptor ROR-gamma |
None |
66824 |
nM |
Potency |
TKC013753
|
P51449 |
Nuclear receptor ROR-gamma |
None |
29849 |
nM |
Potency |
TKC013755
|
P51449 |
Nuclear receptor ROR-gamma |
None |
14000 |
nM |
EC50 |
TKC021977
|
P51449 |
Nuclear receptor ROR-gamma |
None |
42163 |
nM |
Potency |
TKC022931
|
P51449 |
Nuclear receptor ROR-gamma |
None |
84 |
nM |
Potency |
TKC056482
|
P51449 |
Nuclear receptor ROR-gamma |
None |
130 |
nM |
IC50 |
TKC066169
|
P51449 |
Nuclear receptor ROR-gamma |
None |
33492 |
nM |
Potency |
TKC075769
|
P51449 |
Nuclear receptor ROR-gamma |
None |
1980 |
nM |
IC50 |
TKC075769
|
P51449 |
Nuclear receptor ROR-gamma |
None |
109 |
nM |
Kd |
TKC075769
|
P51449 |
Nuclear receptor ROR-gamma |
None |
2000 |
nM |
IC50 |
TKC083807
|
P51449 |
Nuclear receptor ROR-gamma |
None |
10591 |
nM |
Potency |
TKC087664
|
P51449 |
Nuclear receptor ROR-gamma |
None |
47308 |
nM |
Potency |
TKC087991
|
P51449 |
Nuclear receptor ROR-gamma |
None |
21132 |
nM |
Potency |
TKC088230
|
P51449 |
Nuclear receptor ROR-gamma |
None |
1333 |
nM |
Potency |
TKC088231
|
P51449 |
Nuclear receptor ROR-gamma |
None |
23710 |
nM |
Potency |
TKC092297
|
P51449 |
Nuclear receptor ROR-gamma |
None |
26603 |
nM |
Potency |
TKC096012
|
P51449 |
Nuclear receptor ROR-gamma |
None |
200 |
nM |
IC50 |
TKC096012
|
P51449 |
Nuclear receptor ROR-gamma |
None |
18000 |
nM |
EC50 |
TKC097944
|
P51449 |
Nuclear receptor ROR-gamma |
None |
4216 |
nM |
Potency |
TKC102407
|
P51449 |
Nuclear receptor ROR-gamma |
None |
21132 |
nM |
Potency |
TKC107086
|
P51449 |
Nuclear receptor ROR-gamma |
None |
3758 |
nM |
Potency |
TKC115268
|
P51449 |
Nuclear receptor ROR-gamma |
None |
37578 |
nM |
Potency |
TKC118648
|
P51449 |
Nuclear receptor ROR-gamma |
None |
80 |
nM |
EC50 |
TKC118652
|
P51449 |
Nuclear receptor ROR-gamma |
None |
110 |
nM |
EC50 |
TKC118929
|
P51449 |
Nuclear receptor ROR-gamma |
None |
10 |
nM |
Ki |
TKC118938
|
P51449 |
Nuclear receptor ROR-gamma |
None |
10 |
nM |
Ki |
TKC122884
|
P51449 |
Nuclear receptor ROR-gamma |
None |
20 |
nM |
EC50 |
TKC136411
|
P51449 |
Nuclear receptor ROR-gamma |
None |
37578 |
nM |
Potency |
TKC151274
|
P51449 |
Nuclear receptor ROR-gamma |
None |
60 |
nM |
Potency |
TKC206457
|
P51449 |
Nuclear receptor ROR-gamma |
None |
20 |
nM |
EC50 |
TKC206457
|
P51449 |
Nuclear receptor ROR-gamma |
None |
20 |
nM |
EC50 |
TKC206457
|
P51449 |
Nuclear receptor ROR-gamma |
None |
20 |
nM |
EC50 |
TKC206458
|
P51449 |
Nuclear receptor ROR-gamma |
None |
20 |
nM |
EC50 |
TKC206459
|
P51449 |
Nuclear receptor ROR-gamma |
None |
7 |
degrees C |
T |
TKC206672
|
P51449 |
Nuclear receptor ROR-gamma |
None |
42163 |
nM |
Potency |
TKC206688
|
P51449 |
Nuclear receptor ROR-gamma |
None |
23710 |
nM |
Potency |
TKC206759
|
P51449 |
Nuclear receptor ROR-gamma |
None |
26603 |
nM |
Potency |
TKC206760
|
P51449 |
Nuclear receptor ROR-gamma |
None |
74978 |
nM |
Potency |
TKC206770
|
P51449 |
Nuclear receptor ROR-gamma |
None |
33492 |
nM |
Potency |
TKC206812
|
P51449 |
Nuclear receptor ROR-gamma |
None |
47308 |
nM |
Potency |
TKC206816
|
P51449 |
Nuclear receptor ROR-gamma |
None |
8413 |
nM |
Potency |
TKC206915
|
P51449 |
Nuclear receptor ROR-gamma |
None |
10 |
nM |
Ki |
TKC016794
|
P55085 |
Proteinase-activated receptor 2 |
None |
14 |
nM |
IC50 |
TKC021262
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
19500 |
nM |
EC50 |
TKC021666
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
28 |
% |
Activity |
TKC021674
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
25 |
% |
Activity |
TKC035272
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
15849 |
nM |
Potency |
TKC056482
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
259 |
% |
Activity |
TKC057132
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
12589 |
nM |
Potency |
TKC088526
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
12 |
% |
Activity |
TKC100644
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
8913 |
nM |
Potency |
TKC108536
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
50119 |
nM |
Potency |
TKC110634
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
309 |
% |
Activity |
TKC110635
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
289 |
% |
Activity |
TKC170559
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
1000 |
nM |
EC50 |
TKC171329
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
184 |
nM |
EC50 |
TKC206812
|
Q07869 |
Peroxisome proliferator-activated receptor alpha |
None |
>20000 |
nM |
IC50 |