Basic Information

Name [ICD-11: 2A80-2A86]
Protein Number 27
Molecule Number 347

Active subnetwork

Terpenoid-protein target Activity Association

ID Uniport Pref_name Gene name value unit type
TKC118419 O00329 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform None 4 nM IC50
TKC118419 O00329 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform None 9 nM IC50
TKC118419 O00329 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform None 9 nM IC50
TKC118419 O00329 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform None 5.5 nM Kd
TKC118419 O14757 Serine/threonine-protein kinase Chk1 None 87 % Activity
TKC011761 O15530 3-phosphoinositide-dependent protein kinase 1 None 46 % Inhibition
TKC118419 O15530 3-phosphoinositide-dependent protein kinase 1 None 91 % Activity
TKC007127 P00533 Epidermal growth factor receptor None 19 % Inhibition
TKC025462 P00533 Epidermal growth factor receptor None >200 ug.mL-1 IC50
TKC025466 P00533 Epidermal growth factor receptor None >200 ug.mL-1 IC50
TKC025475 P00533 Epidermal growth factor receptor None 197 ug.mL-1 IC50
TKC071640 P00533 Epidermal growth factor receptor None >20000 nM IC50
TKC076041 P00533 Epidermal growth factor receptor None 75 % Inhibition
TKC077689 P00533 Epidermal growth factor receptor None >20000 nM IC50
TKC106319 P00533 Epidermal growth factor receptor None 56 nM IC50
TKC108557 P00533 Epidermal growth factor receptor None 0.82 nM Kd
TKC151761 P00533 Epidermal growth factor receptor None >10000 nM IC50
TKC200866 P00533 Epidermal growth factor receptor None >10000 nM IC50
TKC025462 P04626 Receptor tyrosine-protein kinase erbB-2 None >200 ug.mL-1 IC50
TKC025466 P04626 Receptor tyrosine-protein kinase erbB-2 None >200 ug.mL-1 IC50
TKC025475 P04626 Receptor tyrosine-protein kinase erbB-2 None 125 ug.mL-1 IC50
TKC026211 P04626 Receptor tyrosine-protein kinase erbB-2 None 6 ug.mL-1 IC50
TKC026214 P04626 Receptor tyrosine-protein kinase erbB-2 None 8 ug.mL-1 IC50
TKC026217 P04626 Receptor tyrosine-protein kinase erbB-2 None 4 ug.mL-1 IC50
TKC026229 P04626 Receptor tyrosine-protein kinase erbB-2 None 8 ug.mL-1 IC50
TKC012929 P05771 Protein kinase C beta type None 2 nM Ki
TKC055602 P05771 Protein kinase C beta type None >150000 nM IC50
TKC075924 P05771 Protein kinase C beta type None 90 % Inhibition
TKC090435 P05771 Protein kinase C beta type None 0.2 nM Kd
TKC103074 P05771 Protein kinase C beta type None >150000 nM IC50
TKC104128 P05771 Protein kinase C beta type None >150000 nM IC50
TKC104703 P05771 Protein kinase C beta type None >150000 nM IC50
TKC105956 P05771 Protein kinase C beta type None 2 nM Ki
TKC123088 P05771 Protein kinase C beta type None >150000 nM IC50
TKC151276 P05771 Protein kinase C beta type None >150000 nM IC50
TKC151326 P05771 Protein kinase C beta type None 1 nM Kd
TKC151326 P05771 Protein kinase C beta type None 1.3 nM Kd
TKC151326 P05771 Protein kinase C beta type None 1.3 nM Kd
TKC151326 P05771 Protein kinase C beta type None 1.8 nM Ki
TKC151326 P05771 Protein kinase C beta type None 1.3 nM Kd
TKC151326 P05771 Protein kinase C beta type None 1.3 nM Kd
TKC152742 P05771 Protein kinase C beta type None >150000 nM IC50
TKC000192 P08575 Receptor-type tyrosine-protein phosphatase C None >19000 nM IC50
TKC005454 P08575 Receptor-type tyrosine-protein phosphatase C None 41400 nM IC50
TKC031060 P08575 Receptor-type tyrosine-protein phosphatase C None 10000 nM IC50
TKC045915 P08575 Receptor-type tyrosine-protein phosphatase C None >30000 nM IC50
TKC045916 P08575 Receptor-type tyrosine-protein phosphatase C None >27000 nM IC50
TKC077689 P08575 Receptor-type tyrosine-protein phosphatase C None 1000 nM IC50
TKC096804 P08575 Receptor-type tyrosine-protein phosphatase C None 1200 nM IC50
TKC105683 P08575 Receptor-type tyrosine-protein phosphatase C None 9000 nM IC50
TKC106945 P08575 Receptor-type tyrosine-protein phosphatase C None >16000 nM IC50
TKC156704 P08575 Receptor-type tyrosine-protein phosphatase C None >16000 nM IC50
TKC191566 P08575 Receptor-type tyrosine-protein phosphatase C None >19000 nM IC50
TKC035272 P10415 Apoptosis regulator Bcl-2 None 170 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 260 nM IC50
TKC035272 P10415 Apoptosis regulator Bcl-2 None 320 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 440 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 440 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 1191 nM IC50
TKC035272 P10415 Apoptosis regulator Bcl-2 None 450 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 320 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 600 nM IC50
TKC035272 P10415 Apoptosis regulator Bcl-2 None 420 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 10100 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 4800 nM Kd
TKC035272 P10415 Apoptosis regulator Bcl-2 None 2110 nM IC50
TKC035272 P10415 Apoptosis regulator Bcl-2 None 558 nM Ki
TKC035272 P10415 Apoptosis regulator Bcl-2 None 320 nM Ki
TKC134945 P10415 Apoptosis regulator Bcl-2 None 1460 nM Ki
TKC151761 P10415 Apoptosis regulator Bcl-2 None >10000 nM GI50
TKC200866 P10415 Apoptosis regulator Bcl-2 None >10000 nM GI50
TKC014892 P11387 DNA topoisomerase 1 None 3 ug.mL-1 MIC
TKC014893 P11387 DNA topoisomerase 1 None 13 ug.mL-1 MIC
TKC017201 P11387 DNA topoisomerase 1 None 13 ug.mL-1 MIC
TKC048122 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC048308 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC048324 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC048330 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC048341 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC049414 P11387 DNA topoisomerase 1 None 25000 nM IC50
TKC049417 P11387 DNA topoisomerase 1 None 55000 nM IC50
TKC056419 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC056423 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC056425 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC056427 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC056430 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC058891 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC058895 P11387 DNA topoisomerase 1 None 48600 nM IC50
TKC058897 P11387 DNA topoisomerase 1 None 45100 nM IC50
TKC058919 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC058921 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC058935 P11387 DNA topoisomerase 1 None 109300 nM IC50
TKC058949 P11387 DNA topoisomerase 1 None 250000 nM IC50
TKC058950 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC058953 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC058979 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC059000 P11387 DNA topoisomerase 1 None 53700 nM IC50
TKC059030 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC059045 P11387 DNA topoisomerase 1 None 131700 nM IC50
TKC059148 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC059149 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC059160 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC059165 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC059317 P11387 DNA topoisomerase 1 None 250000 nM IC50
TKC059337 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC059344 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC059345 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC059425 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC072969 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC072970 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC096715 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC100727 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC103324 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC105545 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC137826 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC137841 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC138033 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC138054 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC143022 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC143033 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC143055 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC143114 P11387 DNA topoisomerase 1 None 250000 nM IC50
TKC143115 P11387 DNA topoisomerase 1 None 23800 nM IC50
TKC145932 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC146257 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC147779 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC147805 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC148618 P11387 DNA topoisomerase 1 None 106000 nM IC50
TKC205544 P11387 DNA topoisomerase 1 None 30000 nM IC50
TKC205878 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC207002 P11387 DNA topoisomerase 1 None >250000 nM IC50
TKC205544 P14416 D(2) dopamine receptor None 687 nM Ki
TKC205544 P14416 D(2) dopamine receptor None 280 nM Ki
TKC205544 P14416 D(2) dopamine receptor None 398.1 nM Ki
TKC206544 P14416 D(2) dopamine receptor None >10000 nM Ki
TKC006896 P14902 Indoleamine 2,3-dioxygenase 1 None 7700 nM IC50
TKC014575 P14902 Indoleamine 2,3-dioxygenase 1 None 4680 nM IC50
TKC024473 P14902 Indoleamine 2,3-dioxygenase 1 None 10000 nM IC50
TKC024474 P14902 Indoleamine 2,3-dioxygenase 1 None 11000 nM IC50
TKC104241 P14902 Indoleamine 2,3-dioxygenase 1 None 0 nM EC50
TKC118419 P24941 Cyclin-dependent kinase 2 None 95 % Activity
TKC206292 P24941 Cyclin-dependent kinase 2 None 4800 nM Kd
TKC011761 P31749 RAC-alpha serine/threonine-protein kinase None 54 % Inhibition
TKC016414 P31749 RAC-alpha serine/threonine-protein kinase None 36 % Activity
TKC024886 P31749 RAC-alpha serine/threonine-protein kinase None 48400 nM IC50
TKC025690 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC044763 P31749 RAC-alpha serine/threonine-protein kinase None 100 % Inhibition
TKC115259 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC115261 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC115272 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC115273 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC118419 P31749 RAC-alpha serine/threonine-protein kinase None 96 % Inhibition
TKC152148 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC152157 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC174547 P31749 RAC-alpha serine/threonine-protein kinase None >100000 nM IC50
TKC206776 P31749 RAC-alpha serine/threonine-protein kinase None 3 uM Activity
TKC205544 P35462 D(3) dopamine receptor None 2489 nM Ki
TKC205544 P35462 D(3) dopamine receptor None 3981.07 nM Ki
TKC206544 P35462 D(3) dopamine receptor None >10000 nM Ki
TKC022945 P42345 Serine/threonine-protein kinase mTOR None 4645 nM Potency
TKC032619 P42345 Serine/threonine-protein kinase mTOR None 2931 nM Potency
TKC035272 P42345 Serine/threonine-protein kinase mTOR None 2612 nM Potency
TKC035984 P42345 Serine/threonine-protein kinase mTOR None 4 nM Potency
TKC084630 P42345 Serine/threonine-protein kinase mTOR None 3690 nM Potency
TKC087988 P42345 Serine/threonine-protein kinase mTOR None 4645 nM Potency
TKC092297 P42345 Serine/threonine-protein kinase mTOR None 13092 nM Potency
TKC118419 P42345 Serine/threonine-protein kinase mTOR None 40 nM IC50
TKC118419 P42345 Serine/threonine-protein kinase mTOR None 9200 nM Kd
TKC205544 P42345 Serine/threonine-protein kinase mTOR None 14689 nM Potency
TKC206622 P42345 Serine/threonine-protein kinase mTOR None 23281 nM Potency
TKC206688 P42345 Serine/threonine-protein kinase mTOR None 16482 nM Potency
TKC108557 P43405 Tyrosine-protein kinase SYK None 0.2 nM IC50
TKC112367 P46531 Neurogenic locus notch homolog protein 1 None 300 nM IC50
TKC112399 P46531 Neurogenic locus notch homolog protein 1 None 2400 nM IC50
TKC117085 P46531 Neurogenic locus notch homolog protein 1 None 17300 nM IC50
TKC118351 P46531 Neurogenic locus notch homolog protein 1 None 400 nM IC50
TKC118354 P46531 Neurogenic locus notch homolog protein 1 None 2000 nM IC50
TKC118356 P46531 Neurogenic locus notch homolog protein 1 None 300 nM IC50
TKC118360 P46531 Neurogenic locus notch homolog protein 1 None 700 nM IC50
TKC206738 P46531 Neurogenic locus notch homolog protein 1 None 800 nM IC50
TKC025058 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 1000 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 5 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 19 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 55 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 55000 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 89 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 5 nM IC50
TKC118419 P48736 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform None 15 nM Kd
TKC027726 P52732 Kinesin-like protein KIF11 None 3500 nM IC50
TKC035272 P52732 Kinesin-like protein KIF11 None 10800 nM IC50
TKC035272 P52732 Kinesin-like protein KIF11 None 25000 nM IC50
TKC108557 P52732 Kinesin-like protein KIF11 None 0.3 nM IC50
TKC001786 P53350 Serine/threonine-protein kinase PLK1 None 23778 nM Potency
TKC005454 P53350 Serine/threonine-protein kinase PLK1 None 26680 nM Potency
TKC011384 P53350 Serine/threonine-protein kinase PLK1 None 18888 nM Potency
TKC014568 P53350 Serine/threonine-protein kinase PLK1 None 26680 nM Potency
TKC016277 P53350 Serine/threonine-protein kinase PLK1 None 29935 nM Potency
TKC018288 P53350 Serine/threonine-protein kinase PLK1 None 13371 nM Potency
TKC020967 P53350 Serine/threonine-protein kinase PLK1 None 2180 nM IC50
TKC020987 P53350 Serine/threonine-protein kinase PLK1 None 23778 nM Potency
TKC024886 P53350 Serine/threonine-protein kinase PLK1 None 21700 nM IC50
TKC025690 P53350 Serine/threonine-protein kinase PLK1 None >100000 nM IC50
TKC037521 P53350 Serine/threonine-protein kinase PLK1 None 18888 nM Potency
TKC040032 P53350 Serine/threonine-protein kinase PLK1 None 29935 nM Potency
TKC055219 P53350 Serine/threonine-protein kinase PLK1 None 13371 nM Potency
TKC055869 P53350 Serine/threonine-protein kinase PLK1 None 33588 nM Potency
TKC066096 P53350 Serine/threonine-protein kinase PLK1 None 2119 nM Potency
TKC066411 P53350 Serine/threonine-protein kinase PLK1 None 2994 nM Potency
TKC077689 P53350 Serine/threonine-protein kinase PLK1 None 26680 nM Potency
TKC082378 P53350 Serine/threonine-protein kinase PLK1 None 15003 nM Potency
TKC087988 P53350 Serine/threonine-protein kinase PLK1 None 26680 nM Potency
TKC088678 P53350 Serine/threonine-protein kinase PLK1 None 37686 nM Potency
TKC091895 P53350 Serine/threonine-protein kinase PLK1 None 26680 nM Potency
TKC098704 P53350 Serine/threonine-protein kinase PLK1 None 26680 nM Potency
TKC101726 P53350 Serine/threonine-protein kinase PLK1 None 26680 nM Potency
TKC104088 P53350 Serine/threonine-protein kinase PLK1 None 33588 nM Potency
TKC107557 P53350 Serine/threonine-protein kinase PLK1 None 26680 nM Potency
TKC112826 P53350 Serine/threonine-protein kinase PLK1 None 33588 nM Potency
TKC115259 P53350 Serine/threonine-protein kinase PLK1 None >100000 nM IC50
TKC115261 P53350 Serine/threonine-protein kinase PLK1 None >100000 nM IC50
TKC115272 P53350 Serine/threonine-protein kinase PLK1 None >100000 nM IC50
TKC115273 P53350 Serine/threonine-protein kinase PLK1 None 100000 nM IC50
TKC118419 P53350 Serine/threonine-protein kinase PLK1 None 6 nM IC50
TKC118419 P53350 Serine/threonine-protein kinase PLK1 None 1500 nM Ki
TKC118419 P53350 Serine/threonine-protein kinase PLK1 None 24 nM IC50
TKC141147 P53350 Serine/threonine-protein kinase PLK1 None 13371 nM Potency
TKC150277 P53350 Serine/threonine-protein kinase PLK1 None 23778 nM Potency
TKC151609 P53350 Serine/threonine-protein kinase PLK1 None 23778 nM Potency
TKC151885 P53350 Serine/threonine-protein kinase PLK1 None 6702 nM Potency
TKC151902 P53350 Serine/threonine-protein kinase PLK1 None 26680 nM Potency
TKC151910 P53350 Serine/threonine-protein kinase PLK1 None 18888 nM Potency
TKC152148 P53350 Serine/threonine-protein kinase PLK1 None >100000 nM IC50
TKC152157 P53350 Serine/threonine-protein kinase PLK1 None >100000 nM IC50
TKC159332 P53350 Serine/threonine-protein kinase PLK1 None 21192 nM Potency
TKC171689 P53350 Serine/threonine-protein kinase PLK1 None 23778 nM Potency
TKC174547 P53350 Serine/threonine-protein kinase PLK1 None >100000 nM IC50
TKC206362 P53350 Serine/threonine-protein kinase PLK1 None 13371 nM Potency
TKC206589 P53350 Serine/threonine-protein kinase PLK1 None 29935 nM Potency
TKC206760 P53350 Serine/threonine-protein kinase PLK1 None 21192 nM Potency
TKC021620 P60568 Interleukin-2 None 3 nM Kd
TKC116180 P60568 Interleukin-2 None 0 nM Kd
TKC005454 Q16665 Hypoxia-inducible factor 1-alpha None 1360 nM IC50
TKC005475 Q16665 Hypoxia-inducible factor 1-alpha None 7340 nM IC50
TKC010010 Q16665 Hypoxia-inducible factor 1-alpha None >20000 nM IC50
TKC011921 Q16665 Hypoxia-inducible factor 1-alpha None 1995 nM Potency
TKC012261 Q16665 Hypoxia-inducible factor 1-alpha None 280 nM IC50
TKC012262 Q16665 Hypoxia-inducible factor 1-alpha None 3180 nM IC50
TKC012971 Q16665 Hypoxia-inducible factor 1-alpha None 25119 nM Potency
TKC014568 Q16665 Hypoxia-inducible factor 1-alpha None 8510 nM IC50
TKC017189 Q16665 Hypoxia-inducible factor 1-alpha None 10600 nM IC50
TKC017192 Q16665 Hypoxia-inducible factor 1-alpha None 1700 nM IC50
TKC017193 Q16665 Hypoxia-inducible factor 1-alpha None 2300 nM IC50
TKC020116 Q16665 Hypoxia-inducible factor 1-alpha None 501 nM Potency
TKC022945 Q16665 Hypoxia-inducible factor 1-alpha None 2512 nM Potency
TKC023570 Q16665 Hypoxia-inducible factor 1-alpha None 15800 nM IC50
TKC030239 Q16665 Hypoxia-inducible factor 1-alpha None 200 nM Potency
TKC035272 Q16665 Hypoxia-inducible factor 1-alpha None 10000 nM Potency
TKC037547 Q16665 Hypoxia-inducible factor 1-alpha None 10 % Activity
TKC038977 Q16665 Hypoxia-inducible factor 1-alpha None 820 nM IC50
TKC045710 Q16665 Hypoxia-inducible factor 1-alpha None 500 nM IC50
TKC045931 Q16665 Hypoxia-inducible factor 1-alpha None 2900 nM IC50
TKC045946 Q16665 Hypoxia-inducible factor 1-alpha None 2900 nM IC50
TKC047694 Q16665 Hypoxia-inducible factor 1-alpha None 63 nM IC50
TKC047695 Q16665 Hypoxia-inducible factor 1-alpha None 68 nM IC50
TKC056482 Q16665 Hypoxia-inducible factor 1-alpha None >100000 nM IC50
TKC056482 Q16665 Hypoxia-inducible factor 1-alpha None >100000 nM IC50
TKC062172 Q16665 Hypoxia-inducible factor 1-alpha None 15000 nM IC50
TKC062175 Q16665 Hypoxia-inducible factor 1-alpha None 20000 nM IC50
TKC062182 Q16665 Hypoxia-inducible factor 1-alpha None 20000 nM IC50
TKC062192 Q16665 Hypoxia-inducible factor 1-alpha None 20000 nM IC50
TKC062193 Q16665 Hypoxia-inducible factor 1-alpha None >30000 nM IC50
TKC065782 Q16665 Hypoxia-inducible factor 1-alpha None >30000 nM IC50
TKC081893 Q16665 Hypoxia-inducible factor 1-alpha None 400 nM IC50
TKC092297 Q16665 Hypoxia-inducible factor 1-alpha None 39811 nM Potency
TKC094057 Q16665 Hypoxia-inducible factor 1-alpha None >30000 nM IC50
TKC094058 Q16665 Hypoxia-inducible factor 1-alpha None >20000 nM IC50
TKC095493 Q16665 Hypoxia-inducible factor 1-alpha None 3162 nM Potency
TKC096011 Q16665 Hypoxia-inducible factor 1-alpha None 1 nM Potency
TKC096012 Q16665 Hypoxia-inducible factor 1-alpha None 251 nM Potency
TKC100416 Q16665 Hypoxia-inducible factor 1-alpha None 25119 nM Potency
TKC100643 Q16665 Hypoxia-inducible factor 1-alpha None 12589 nM Potency
TKC100990 Q16665 Hypoxia-inducible factor 1-alpha None 159 nM Potency
TKC101618 Q16665 Hypoxia-inducible factor 1-alpha None 15849 nM Potency
TKC102145 Q16665 Hypoxia-inducible factor 1-alpha None 1259 nM Potency
TKC102589 Q16665 Hypoxia-inducible factor 1-alpha None 8000 nM EC50
TKC103149 Q16665 Hypoxia-inducible factor 1-alpha None 31623 nM Potency
TKC103159 Q16665 Hypoxia-inducible factor 1-alpha None 270 nM IC50
TKC103433 Q16665 Hypoxia-inducible factor 1-alpha None >30000 nM IC50
TKC103494 Q16665 Hypoxia-inducible factor 1-alpha None 79 nM Potency
TKC103496 Q16665 Hypoxia-inducible factor 1-alpha None 20 nM Potency
TKC104070 Q16665 Hypoxia-inducible factor 1-alpha None 40 nM Potency
TKC104071 Q16665 Hypoxia-inducible factor 1-alpha None 100 nM Potency
TKC104114 Q16665 Hypoxia-inducible factor 1-alpha None 126 nM Potency
TKC104664 Q16665 Hypoxia-inducible factor 1-alpha None 794 nM Potency
TKC105037 Q16665 Hypoxia-inducible factor 1-alpha None 794 nM Potency
TKC105510 Q16665 Hypoxia-inducible factor 1-alpha None 6000 nM EC50
TKC105710 Q16665 Hypoxia-inducible factor 1-alpha None 12589 nM Potency
TKC106426 Q16665 Hypoxia-inducible factor 1-alpha None 1000 nM Potency
TKC106576 Q16665 Hypoxia-inducible factor 1-alpha None 13000 nM EC50
TKC107086 Q16665 Hypoxia-inducible factor 1-alpha None 19953 nM Potency
TKC109561 Q16665 Hypoxia-inducible factor 1-alpha None 251 nM Potency
TKC110002 Q16665 Hypoxia-inducible factor 1-alpha None 63 nM Potency
TKC110007 Q16665 Hypoxia-inducible factor 1-alpha None 7943 nM Potency
TKC111738 Q16665 Hypoxia-inducible factor 1-alpha None 16 nM Potency
TKC112789 Q16665 Hypoxia-inducible factor 1-alpha None 1000 nM Potency
TKC112906 Q16665 Hypoxia-inducible factor 1-alpha None 5012 nM Potency
TKC114819 Q16665 Hypoxia-inducible factor 1-alpha None 12589 nM Potency
TKC117993 Q16665 Hypoxia-inducible factor 1-alpha None 2000 nM EC50
TKC117997 Q16665 Hypoxia-inducible factor 1-alpha None 40 nM EC50
TKC118004 Q16665 Hypoxia-inducible factor 1-alpha None 2512 nM Potency
TKC118012 Q16665 Hypoxia-inducible factor 1-alpha None 600 nM EC50
TKC118131 Q16665 Hypoxia-inducible factor 1-alpha None 126 nM Potency
TKC134897 Q16665 Hypoxia-inducible factor 1-alpha None 3400 nM IC50
TKC137120 Q16665 Hypoxia-inducible factor 1-alpha None 200 nM IC50
TKC137126 Q16665 Hypoxia-inducible factor 1-alpha None 2400 nM IC50
TKC137243 Q16665 Hypoxia-inducible factor 1-alpha None 200 nM IC50
TKC144475 Q16665 Hypoxia-inducible factor 1-alpha None 25000 nM IC50
TKC151571 Q16665 Hypoxia-inducible factor 1-alpha None 7943 nM Potency
TKC205806 Q16665 Hypoxia-inducible factor 1-alpha None 5012 nM Potency
TKC206042 Q16665 Hypoxia-inducible factor 1-alpha None 6310 nM Potency
TKC206395 Q16665 Hypoxia-inducible factor 1-alpha None 12589 nM Potency
TKC206453 Q16665 Hypoxia-inducible factor 1-alpha None 25119 nM Potency
TKC206617 Q16665 Hypoxia-inducible factor 1-alpha None 12700 nM IC50
TKC206688 Q16665 Hypoxia-inducible factor 1-alpha None 63 nM Potency
TKC206726 Q16665 Hypoxia-inducible factor 1-alpha None 79 nM Potency
TKC206760 Q16665 Hypoxia-inducible factor 1-alpha None 50119 nM Potency
TKC206780 Q16665 Hypoxia-inducible factor 1-alpha None 3981 nM Potency
TKC206812 Q16665 Hypoxia-inducible factor 1-alpha None 79433 nM Potency
TKC206816 Q16665 Hypoxia-inducible factor 1-alpha None 12589 nM Potency
TKC206872 Q16665 Hypoxia-inducible factor 1-alpha None 1000 nM Potency
TKC206889 Q16665 Hypoxia-inducible factor 1-alpha None 501 nM Potency
TKC206890 Q16665 Hypoxia-inducible factor 1-alpha None 20 nM EC50
TKC206901 Q16665 Hypoxia-inducible factor 1-alpha None 159 nM Potency
TKC076129 Q16790 Carbonic anhydrase 9 None 980 nM Ki
TKC020117 Q92769 Histone deacetylase 2 None 15 nM Ki
TKC118419 Q9BUB5 MAP kinase-interacting serine/threonine-protein kinase 1 None 81 % Activity
TKC118419 Q9HBH9 MAP kinase-interacting serine/threonine-protein kinase 2 None 97 % Activity
TKC011761 Q9UM73 ALK tyrosine kinase receptor None 18 % Inhibition
TKC024886 Q9UM73 ALK tyrosine kinase receptor None 2190 nM IC50
TKC025690 Q9UM73 ALK tyrosine kinase receptor None 3380 nM IC50
TKC115259 Q9UM73 ALK tyrosine kinase receptor None 9330 nM IC50
TKC115261 Q9UM73 ALK tyrosine kinase receptor None 4160 nM IC50
TKC115272 Q9UM73 ALK tyrosine kinase receptor None >100000 nM IC50
TKC115273 Q9UM73 ALK tyrosine kinase receptor None 4360 nM IC50
TKC152148 Q9UM73 ALK tyrosine kinase receptor None 7550 nM IC50
TKC152157 Q9UM73 ALK tyrosine kinase receptor None 4730 nM IC50
TKC174547 Q9UM73 ALK tyrosine kinase receptor None >100000 nM IC50