| Uniport ID | P08684 |
| Organism | Homo sapiens |
| Protein | Cytochrome P450 3A4 |
| Gene | CYP3A4 |
| Molecule Number | 197 |
| ID | Uniport | Pref Name | Value | Unit | Type |
|---|---|---|---|---|---|
| TKC000602 | P08684 | Cytochrome P450 3A4 | >100000 | nM | IC50 |
| TKC003636 | P08684 | Cytochrome P450 3A4 | >100000 | nM | IC50 |
| TKC003637 | P08684 | Cytochrome P450 3A4 | >100000 | nM | IC50 |
| TKC004452 | P08684 | Cytochrome P450 3A4 | >100000 | nM | IC50 |
| TKC004454 | P08684 | Cytochrome P450 3A4 | >100000 | nM | IC50 |
| TKC004758 | P08684 | Cytochrome P450 3A4 | >100000 | nM | IC50 |
| TKC025230 | P08684 | Cytochrome P450 3A4 | >10000 | nM | IC50 |
| TKC025231 | P08684 | Cytochrome P450 3A4 | >10000 | nM | IC50 |
| TKC030239 | P08684 | Cytochrome P450 3A4 | >19953 | nM | Potency |
| TKC030239 | P08684 | Cytochrome P450 3A4 | >50000 | nM | IC50 |
| TKC075769 | P08684 | Cytochrome P450 3A4 | >50000 | nM | IC50 |
| TKC112653 | P08684 | Cytochrome P450 3A4 | >100000 | nM | IC50 |
| TKC112655 | P08684 | Cytochrome P450 3A4 | >100000 | nM | IC50 |
| TKC122980 | P08684 | Cytochrome P450 3A4 | >100000 | nM | IC50 |
| TKC146761 | P08684 | Cytochrome P450 3A4 | 125000.0 | nM | IC50 |
| TKC032983 | P08684 | Cytochrome P450 3A4 | 98200.0 | nM | IC50 |
| TKC077034 | P08684 | Cytochrome P450 3A4 | 62500.0 | nM | IC50 |
| TKC097717 | P08684 | Cytochrome P450 3A4 | 48400.0 | nM | IC50 |
| TKC037686 | P08684 | Cytochrome P450 3A4 | 42600.0 | nM | IC50 |
| TKC008359 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC013304 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC096012 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC098345 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC101920 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC102204 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC102439 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC104404 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC104602 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC105168 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC106240 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC132834 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC135961 | P08684 | Cytochrome P450 3A4 | 39811.0 | nM | Potency |
| TKC134571 | P08684 | Cytochrome P450 3A4 | 35500.0 | nM | IC50 |
| TKC035272 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | AC50 |
| TKC045513 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC057133 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC078496 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC087991 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC090094 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC103257 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC104767 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC105530 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC105784 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC106198 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC106301 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC107201 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC115268 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC117710 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC151675 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC151875 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC206114 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC206386 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC206760 | P08684 | Cytochrome P450 3A4 | 31623.0 | nM | Potency |
| TKC012971 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | AC50 |
| TKC031954 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC032619 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC040026 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC079001 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC092348 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC101020 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC103736 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC105034 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC107818 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC108109 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC108732 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC111349 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC138780 | P08684 | Cytochrome P450 3A4 | 25119.0 | nM | Potency |
| TKC151523 | P08684 | Cytochrome P450 3A4 | 23200.0 | nM | Ki |
| TKC077038 | P08684 | Cytochrome P450 3A4 | 21800.0 | nM | IC50 |
| TKC034979 | P08684 | Cytochrome P450 3A4 | 20000.0 | nM | Ki |
| TKC103023 | P08684 | Cytochrome P450 3A4 | 19953.0 | nM | Potency |
| TKC103041 | P08684 | Cytochrome P450 3A4 | 19953.0 | nM | Potency |
| TKC207209 | P08684 | Cytochrome P450 3A4 | 19953.0 | nM | Potency |
| TKC005454 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC016418 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC068076 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC074866 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC087664 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC088678 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC092297 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC101907 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC107332 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC107830 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC108295 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC112745 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC112754 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC118004 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC148601 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC150706 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC206453 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC206754 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC206777 | P08684 | Cytochrome P450 3A4 | 15849.0 | nM | Potency |
| TKC013753 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC034640 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC034641 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC039869 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC040829 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC102032 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC102120 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC103799 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC104293 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC104656 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC105033 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | AC50 |
| TKC105037 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | AC50 |
| TKC105346 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC106426 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | AC50 |
| TKC106840 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC112909 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC147290 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC151571 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | AC50 |
| TKC206452 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | AC50 |
| TKC206783 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | AC50 |
| TKC206884 | P08684 | Cytochrome P450 3A4 | 12589.0 | nM | Potency |
| TKC011526 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC034078 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC062321 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC101092 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC104091 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC105378 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC107593 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC112906 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC112914 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC113146 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC135244 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC205806 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC206690 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | Potency |
| TKC206759 | P08684 | Cytochrome P450 3A4 | 10000.0 | nM | IC50 |
| TKC040094 | P08684 | Cytochrome P450 3A4 | 8800.0 | nM | IC50 |
| TKC013736 | P08684 | Cytochrome P450 3A4 | 8700.0 | nM | Km |
| TKC034083 | P08684 | Cytochrome P450 3A4 | 7943.0 | nM | Potency |
| TKC066013 | P08684 | Cytochrome P450 3A4 | 7943.0 | nM | Potency |
| TKC101617 | P08684 | Cytochrome P450 3A4 | 7943.0 | nM | AC50 |
| TKC104977 | P08684 | Cytochrome P450 3A4 | 7943.0 | nM | Potency |
| TKC206688 | P08684 | Cytochrome P450 3A4 | 7943.0 | nM | Potency |
| TKC206901 | P08684 | Cytochrome P450 3A4 | 7943.0 | nM | AC50 |
| TKC207071 | P08684 | Cytochrome P450 3A4 | 7500.0 | nM | Km |
| TKC062333 | P08684 | Cytochrome P450 3A4 | 6310.0 | nM | Potency |
| TKC023263 | P08684 | Cytochrome P450 3A4 | 5070.0 | nM | IC50 |
| TKC102407 | P08684 | Cytochrome P450 3A4 | 5012.0 | nM | Potency |
| TKC106184 | P08684 | Cytochrome P450 3A4 | 5012.0 | nM | Potency |
| TKC107067 | P08684 | Cytochrome P450 3A4 | 5012.0 | nM | Potency |
| TKC141032 | P08684 | Cytochrome P450 3A4 | 5012.0 | nM | Potency |
| TKC207099 | P08684 | Cytochrome P450 3A4 | 5012.0 | nM | Potency |
| TKC011412 | P08684 | Cytochrome P450 3A4 | 4300.0 | nM | Ki |
| TKC053825 | P08684 | Cytochrome P450 3A4 | 3981.0 | nM | Potency |
| TKC100649 | P08684 | Cytochrome P450 3A4 | 3981.0 | nM | Potency |
| TKC102540 | P08684 | Cytochrome P450 3A4 | 3981.0 | nM | Potency |
| TKC103149 | P08684 | Cytochrome P450 3A4 | 3981.0 | nM | AC50 |
| TKC106358 | P08684 | Cytochrome P450 3A4 | 3981.0 | nM | Potency |
| TKC114819 | P08684 | Cytochrome P450 3A4 | 3981.0 | nM | Potency |
| TKC151522 | P08684 | Cytochrome P450 3A4 | 3981.0 | nM | Potency |
| TKC206816 | P08684 | Cytochrome P450 3A4 | 3981.0 | nM | Potency |
| TKC107021 | P08684 | Cytochrome P450 3A4 | 3162.0 | nM | Potency |
| TKC109561 | P08684 | Cytochrome P450 3A4 | 3162.0 | nM | AC50 |
| TKC113150 | P08684 | Cytochrome P450 3A4 | 3162.0 | nM | Potency |
| TKC114511 | P08684 | Cytochrome P450 3A4 | 3162.0 | nM | Potency |
| TKC207282 | P08684 | Cytochrome P450 3A4 | 3162.0 | nM | AC50 |
| TKC011075 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | Potency |
| TKC055066 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | Potency |
| TKC055209 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | Potency |
| TKC101111 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | Potency |
| TKC104435 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | Potency |
| TKC105295 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | Potency |
| TKC105424 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | Potency |
| TKC106212 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | AC50 |
| TKC107104 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | Potency |
| TKC107525 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | Potency |
| TKC107944 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | Potency |
| TKC113125 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | Potency |
| TKC138777 | P08684 | Cytochrome P450 3A4 | 2512.0 | nM | Potency |
| TKC038725 | P08684 | Cytochrome P450 3A4 | 1995.0 | nM | Potency |
| TKC100701 | P08684 | Cytochrome P450 3A4 | 1995.0 | nM | Potency |
| TKC106232 | P08684 | Cytochrome P450 3A4 | 1995.0 | nM | AC50 |
| TKC111738 | P08684 | Cytochrome P450 3A4 | 1995.0 | nM | Potency |
| TKC062327 | P08684 | Cytochrome P450 3A4 | 1585.0 | nM | Potency |
| TKC062332 | P08684 | Cytochrome P450 3A4 | 1585.0 | nM | Potency |
| TKC095493 | P08684 | Cytochrome P450 3A4 | 1585.0 | nM | AC50 |
| TKC113149 | P08684 | Cytochrome P450 3A4 | 1585.0 | nM | Potency |
| TKC148482 | P08684 | Cytochrome P450 3A4 | 1585.0 | nM | Potency |
| TKC066332 | P08684 | Cytochrome P450 3A4 | 1259.0 | nM | Potency |
| TKC104979 | P08684 | Cytochrome P450 3A4 | 1259.0 | nM | Potency |
| TKC102743 | P08684 | Cytochrome P450 3A4 | 1000.0 | nM | Potency |
| TKC206365 | P08684 | Cytochrome P450 3A4 | 1000.0 | nM | Potency |
| TKC206687 | P08684 | Cytochrome P450 3A4 | 1000.0 | nM | Potency |
| TKC206812 | P08684 | Cytochrome P450 3A4 | 1000.0 | nM | Potency |
| TKC020117 | P08684 | Cytochrome P450 3A4 | 631.0 | nM | Potency |
| TKC105153 | P08684 | Cytochrome P450 3A4 | 501.0 | nM | Potency |
| TKC100636 | P08684 | Cytochrome P450 3A4 | 398.0 | nM | Potency |
| TKC104664 | P08684 | Cytochrome P450 3A4 | 398.0 | nM | Potency |
| TKC151758 | P08684 | Cytochrome P450 3A4 | 316.0 | nM | Potency |
| TKC205809 | P08684 | Cytochrome P450 3A4 | 66.0 | % | Activity |
| TKC110956 | P08684 | Cytochrome P450 3A4 | 26.0 | pmol/min | Drug metabolism |
| TKC206689 | P08684 | Cytochrome P450 3A4 | 25.0 | nM | Potency |
| TKC039868 | P08684 | Cytochrome P450 3A4 | 10.0 | % | Drug metabolism |
| TKC122904 | P08684 | Cytochrome P450 3A4 | 9.0 | pmol/min | Vmax |
| TKC101618 | P08684 | Cytochrome P450 3A4 | 6.0 | nM | Potency |
| TKC110481 | P08684 | Cytochrome P450 3A4 | 1.0 | uL/mg/min | Vmax/Km |