TKC010047
|
P00441 |
Superoxide dismutase [Cu-Zn] |
None |
56600 |
nM |
IC50 |
TKC055903
|
P00734 |
Prothrombin |
None |
4 |
nM |
IC50 |
TKC055903
|
P00734 |
Prothrombin |
None |
50 |
nM |
IC50 |
TKC064786
|
P00734 |
Prothrombin |
None |
130 |
nM |
IC50 |
TKC064787
|
P00734 |
Prothrombin |
None |
70 |
nM |
IC50 |
TKC101989
|
P00734 |
Prothrombin |
None |
4000 |
nM |
IC50 |
TKC106074
|
P00734 |
Prothrombin |
None |
>50000 |
nM |
IC50 |
TKC106074
|
P00734 |
Prothrombin |
None |
>50000 |
nM |
IC50 |
TKC122980
|
P00734 |
Prothrombin |
None |
9200 |
nM |
IC50 |
TKC139119
|
P00734 |
Prothrombin |
None |
90 |
nM |
IC50 |
TKC141433
|
P00734 |
Prothrombin |
None |
18 |
nM |
IC50 |
TKC005744
|
P00742 |
Coagulation factor X |
None |
27900 |
nM |
IC50 |
TKC012492
|
P00742 |
Coagulation factor X |
None |
13385 |
nM |
Ki |
TKC013400
|
P00742 |
Coagulation factor X |
None |
2500 |
nM |
IC50 |
TKC013430
|
P00742 |
Coagulation factor X |
None |
11418 |
nM |
IC50 |
TKC055903
|
P00742 |
Coagulation factor X |
None |
>20000 |
nM |
IC50 |
TKC107140
|
P00742 |
Coagulation factor X |
None |
7991 |
nM |
Ki |
TKC124270
|
P00742 |
Coagulation factor X |
None |
27558 |
nM |
Ki |
TKC128698
|
P00742 |
Coagulation factor X |
None |
7200 |
nM |
IC50 |
TKC128699
|
P00742 |
Coagulation factor X |
None |
7165 |
nM |
IC50 |
TKC205733
|
P00742 |
Coagulation factor X |
None |
1023 |
nM |
IC50 |
TKC073833
|
P00749 |
Urokinase-type plasminogen activator |
None |
58479 |
nM |
Potency |
TKC076529
|
P00749 |
Urokinase-type plasminogen activator |
None |
23281 |
nM |
Potency |
TKC082279
|
P00749 |
Urokinase-type plasminogen activator |
None |
52119 |
nM |
Potency |
TKC008187
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
30200 |
nM |
IC50 |
TKC023515
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
53 |
% |
Inhibition |
TKC025574
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
52 |
% |
Inhibition |
TKC026893
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
21 |
% |
Inhibition |
TKC026895
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
61 |
% |
Inhibition |
TKC057019
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
22300 |
nM |
IC50 |
TKC100777
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
30 |
% |
Inhibition |
TKC101031
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
1500 |
nM |
IC50 |
TKC101538
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
39 |
% |
Inhibition |
TKC101847
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
1000 |
nM |
IC50 |
TKC103703
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
40 |
% |
Inhibition |
TKC137314
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
8400 |
nM |
IC50 |
TKC138471
|
P04035 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
None |
21700 |
nM |
IC50 |
TKC022234
|
P08246 |
Neutrophil elastase |
None |
>1 |
% |
Inhibition |
TKC022237
|
P08246 |
Neutrophil elastase |
None |
100000 |
nM |
IC50 |
TKC022245
|
P08246 |
Neutrophil elastase |
None |
18000 |
nM |
IC50 |
TKC055903
|
P08246 |
Neutrophil elastase |
None |
>10000 |
nM |
IC50 |
TKC056482
|
P08246 |
Neutrophil elastase |
None |
416 |
nM |
IC50 |
TKC093449
|
P08246 |
Neutrophil elastase |
None |
100000 |
nM |
IC50 |
TKC093451
|
P08246 |
Neutrophil elastase |
None |
>40 |
% |
Inhibition |
TKC104777
|
P08246 |
Neutrophil elastase |
None |
1560 |
nM |
IC50 |
TKC020117
|
P08254 |
Stromelysin-1 |
None |
98 |
% |
Inhibition |
TKC042585
|
P08254 |
Stromelysin-1 |
None |
300 |
nM |
MIC50 |
TKC042586
|
P08254 |
Stromelysin-1 |
None |
300 |
nM |
MIC50 |
TKC042587
|
P08254 |
Stromelysin-1 |
None |
300 |
nM |
MIC50 |
TKC002411
|
P11597 |
Cholesteryl ester transfer protein |
None |
196000 |
nM |
IC50 |
TKC026245
|
P11597 |
Cholesteryl ester transfer protein |
None |
25000 |
nM |
IC50 |
TKC026309
|
P11597 |
Cholesteryl ester transfer protein |
None |
6000 |
nM |
IC50 |
TKC026600
|
P11597 |
Cholesteryl ester transfer protein |
None |
100000 |
nM |
IC50 |
TKC027200
|
P11597 |
Cholesteryl ester transfer protein |
None |
5000 |
nM |
IC50 |
TKC027200
|
P11597 |
Cholesteryl ester transfer protein |
None |
5200 |
nM |
IC50 |
TKC027201
|
P11597 |
Cholesteryl ester transfer protein |
None |
1000 |
nM |
IC50 |
TKC027201
|
P11597 |
Cholesteryl ester transfer protein |
None |
5200 |
nM |
IC50 |
TKC056482
|
P11597 |
Cholesteryl ester transfer protein |
None |
46600 |
nM |
IC50 |
TKC077689
|
P11597 |
Cholesteryl ester transfer protein |
None |
10 |
% |
Inhibition |
TKC094496
|
P11597 |
Cholesteryl ester transfer protein |
None |
46000 |
nM |
IC50 |
TKC097288
|
P11597 |
Cholesteryl ester transfer protein |
None |
600 |
nM |
IC50 |
TKC106450
|
P11597 |
Cholesteryl ester transfer protein |
None |
5200 |
nM |
IC50 |
TKC123088
|
P11597 |
Cholesteryl ester transfer protein |
None |
31 |
% |
Inhibition |
TKC032440
|
P25101 |
Endothelin-1 receptor |
None |
135000 |
nM |
IC50 |
TKC032443
|
P25101 |
Endothelin-1 receptor |
None |
62000 |
nM |
IC50 |
TKC082111
|
P25116 |
Proteinase-activated receptor 1 |
None |
20000 |
nM |
IC50 |
TKC113091
|
P27487 |
Dipeptidyl peptidase 4 |
None |
35600 |
nM |
IC50 |
TKC122980
|
P27487 |
Dipeptidyl peptidase 4 |
None |
28840 |
nM |
IC50 |
TKC123088
|
P27487 |
Dipeptidyl peptidase 4 |
None |
55820 |
nM |
IC50 |
TKC038273
|
P30556 |
Type-1 angiotensin II receptor |
None |
21974 |
nM |
IC50 |
TKC038273
|
P30556 |
Type-1 angiotensin II receptor |
None |
21974 |
nM |
IC50 |
TKC134702
|
P30556 |
Type-1 angiotensin II receptor |
None |
18639 |
nM |
IC50 |
TKC134702
|
P30556 |
Type-1 angiotensin II receptor |
None |
18639 |
nM |
IC50 |
TKC012971
|
P40225 |
Thrombopoietin |
None |
12589 |
nM |
Potency |
TKC092297
|
P40225 |
Thrombopoietin |
None |
10000 |
nM |
Potency |
TKC101618
|
P40225 |
Thrombopoietin |
None |
3162 |
nM |
Potency |
TKC103149
|
P40225 |
Thrombopoietin |
None |
50 |
nM |
Potency |
TKC106232
|
P40225 |
Thrombopoietin |
None |
12589 |
nM |
Potency |
TKC114511
|
P40225 |
Thrombopoietin |
None |
7943 |
nM |
Potency |
TKC151571
|
P40225 |
Thrombopoietin |
None |
10000 |
nM |
Potency |
TKC206453
|
P40225 |
Thrombopoietin |
None |
15849 |
nM |
Potency |
TKC206688
|
P40225 |
Thrombopoietin |
None |
1259 |
nM |
Potency |
TKC206777
|
P40225 |
Thrombopoietin |
None |
7943 |
nM |
Potency |
TKC206816
|
P40225 |
Thrombopoietin |
None |
10000 |
nM |
Potency |
TKC206901
|
P40225 |
Thrombopoietin |
None |
3162 |
nM |
Potency |
TKC025058
|
P48736 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
None |
1000 |
nM |
IC50 |
TKC118419
|
P48736 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
None |
5 |
nM |
IC50 |
TKC118419
|
P48736 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
None |
19 |
nM |
IC50 |
TKC118419
|
P48736 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
None |
55 |
nM |
IC50 |
TKC118419
|
P48736 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
None |
55000 |
nM |
IC50 |
TKC118419
|
P48736 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
None |
89 |
nM |
IC50 |
TKC118419
|
P48736 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
None |
5 |
nM |
IC50 |
TKC118419
|
P48736 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
None |
15 |
nM |
Kd |
TKC009521
|
Q05655 |
Protein kinase C delta type |
None |
4 |
nM |
EC50 |
TKC009534
|
Q05655 |
Protein kinase C delta type |
None |
5 |
nM |
EC50 |
TKC009557
|
Q05655 |
Protein kinase C delta type |
None |
5 |
nM |
EC50 |
TKC011761
|
Q05655 |
Protein kinase C delta type |
None |
1 |
% |
Inhibition |
TKC012929
|
Q05655 |
Protein kinase C delta type |
None |
1 |
nM |
Ki |
TKC012929
|
Q05655 |
Protein kinase C delta type |
None |
5170 |
nM |
EC50 |
TKC012929
|
Q05655 |
Protein kinase C delta type |
None |
290 |
nM |
EC50 |
TKC015409
|
Q05655 |
Protein kinase C delta type |
None |
24.6 |
nM |
Ki |
TKC070351
|
Q05655 |
Protein kinase C delta type |
None |
1.31 |
nM |
Ki |
TKC070919
|
Q05655 |
Protein kinase C delta type |
None |
0.56 |
nM |
Ki |
TKC090435
|
Q05655 |
Protein kinase C delta type |
None |
0.33 |
nM |
Kd |
TKC090508
|
Q05655 |
Protein kinase C delta type |
None |
0.177 |
nM |
Kd |
TKC103074
|
Q05655 |
Protein kinase C delta type |
None |
49000 |
nM |
IC50 |
TKC105956
|
Q05655 |
Protein kinase C delta type |
None |
1 |
nM |
Ki |
TKC107460
|
Q05655 |
Protein kinase C delta type |
None |
6 |
nM |
EC50 |
TKC149470
|
Q05655 |
Protein kinase C delta type |
None |
0.55 |
nM |
Ki |
TKC151326
|
Q05655 |
Protein kinase C delta type |
None |
0 |
nM |
Kd |
TKC151326
|
Q05655 |
Protein kinase C delta type |
None |
273 |
nM |
Kd |
TKC151326
|
Q05655 |
Protein kinase C delta type |
None |
52 |
nM |
Kd |
TKC151326
|
Q05655 |
Protein kinase C delta type |
None |
0.53 |
nM |
Kd |
TKC151326
|
Q05655 |
Protein kinase C delta type |
None |
12 |
nM |
Ki |
TKC151326
|
Q05655 |
Protein kinase C delta type |
None |
107 |
nM |
Ki |
TKC151326
|
Q05655 |
Protein kinase C delta type |
None |
0.53 |
nM |
Kd |
TKC151326
|
Q05655 |
Protein kinase C delta type |
None |
0.53 |
nM |
Kd |
TKC087988
|
Q16539 |
Mitogen-activated protein kinase 14 |
None |
2529 |
nM |
IC50 |
TKC118419
|
Q16539 |
Mitogen-activated protein kinase 14 |
None |
86 |
% |
Inhibition |