TKC151523
|
P08908 |
5-hydroxytryptamine receptor 1A |
None |
>100000 |
nM |
Ki |
TKC205544
|
P08908 |
5-hydroxytryptamine receptor 1A |
None |
4500 |
nM |
Ki |
TKC205544
|
P08908 |
5-hydroxytryptamine receptor 1A |
None |
1500 |
nM |
Ki |
TKC205544
|
P08908 |
5-hydroxytryptamine receptor 1A |
None |
642 |
nM |
Ki |
TKC205544
|
P08908 |
5-hydroxytryptamine receptor 1A |
None |
1258.92 |
nM |
Ki |
TKC206544
|
P08908 |
5-hydroxytryptamine receptor 1A |
None |
>10000 |
nM |
Ki |
TKC206549
|
P08908 |
5-hydroxytryptamine receptor 1A |
None |
30 |
pM well-1 |
cAMP |
TKC001669
|
P10275 |
Androgen receptor |
None |
260 |
nM |
IC50 |
TKC006934
|
P10275 |
Androgen receptor |
None |
50119 |
nM |
Potency |
TKC013304
|
P10275 |
Androgen receptor |
None |
70795 |
nM |
Potency |
TKC019571
|
P10275 |
Androgen receptor |
None |
19953 |
nM |
Potency |
TKC021325
|
P10275 |
Androgen receptor |
None |
31623 |
nM |
Potency |
TKC021332
|
P10275 |
Androgen receptor |
None |
31623 |
nM |
Potency |
TKC023246
|
P10275 |
Androgen receptor |
None |
449 |
nM |
IC50 |
TKC030239
|
P10275 |
Androgen receptor |
None |
14 |
nM |
Potency |
TKC035272
|
P10275 |
Androgen receptor |
None |
15849 |
nM |
Potency |
TKC056140
|
P10275 |
Androgen receptor |
None |
50 |
% |
Activity |
TKC066169
|
P10275 |
Androgen receptor |
None |
3981 |
nM |
Potency |
TKC074867
|
P10275 |
Androgen receptor |
None |
28184 |
nM |
Potency |
TKC075769
|
P10275 |
Androgen receptor |
None |
355 |
nM |
Potency |
TKC079001
|
P10275 |
Androgen receptor |
None |
1 |
nM |
Potency |
TKC096012
|
P10275 |
Androgen receptor |
None |
178 |
nM |
Potency |
TKC100644
|
P10275 |
Androgen receptor |
None |
35481 |
nM |
Potency |
TKC102407
|
P10275 |
Androgen receptor |
None |
44668 |
nM |
Potency |
TKC106878
|
P10275 |
Androgen receptor |
None |
238 |
nM |
IC50 |
TKC107086
|
P10275 |
Androgen receptor |
None |
17783 |
nM |
Potency |
TKC107735
|
P10275 |
Androgen receptor |
None |
3981 |
nM |
Potency |
TKC111738
|
P10275 |
Androgen receptor |
None |
17783 |
nM |
Potency |
TKC112923
|
P10275 |
Androgen receptor |
None |
212 |
nM |
IC50 |
TKC114095
|
P10275 |
Androgen receptor |
None |
1790 |
nM |
IC50 |
TKC114511
|
P10275 |
Androgen receptor |
None |
315 |
nM |
Ki |
TKC115268
|
P10275 |
Androgen receptor |
None |
35481 |
nM |
Potency |
TKC115284
|
P10275 |
Androgen receptor |
None |
1 |
nM |
Ki |
TKC117154
|
P10275 |
Androgen receptor |
None |
580 |
nM |
IC50 |
TKC120161
|
P10275 |
Androgen receptor |
None |
44668 |
nM |
Potency |
TKC122884
|
P10275 |
Androgen receptor |
None |
39811 |
nM |
Potency |
TKC122892
|
P10275 |
Androgen receptor |
None |
10000 |
nM |
IC50 |
TKC134780
|
P10275 |
Androgen receptor |
None |
2 |
nM |
Potency |
TKC147240
|
P10275 |
Androgen receptor |
None |
50 |
% |
Activity |
TKC206652
|
P10275 |
Androgen receptor |
None |
50 |
nM |
Potency |
TKC206688
|
P10275 |
Androgen receptor |
None |
224 |
nM |
Potency |
TKC206690
|
P10275 |
Androgen receptor |
None |
36 |
nM |
Potency |
TKC206759
|
P10275 |
Androgen receptor |
None |
2 |
nM |
Potency |
TKC206759
|
P10275 |
Androgen receptor |
None |
3.9 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
4.7 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
4.2 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
29 |
nM |
Ki |
TKC206759
|
P10275 |
Androgen receptor |
None |
1.1 |
nM |
EC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
2.7 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
2.7 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
2.7 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
30 |
nM |
IC50 |
TKC206759
|
P10275 |
Androgen receptor |
None |
4.57 |
nM |
IC50 |
TKC206770
|
P10275 |
Androgen receptor |
None |
224 |
nM |
Potency |
TKC206779
|
P10275 |
Androgen receptor |
None |
2 |
nM |
Potency |
TKC206812
|
P10275 |
Androgen receptor |
None |
220 |
nM |
IC50 |
TKC206816
|
P10275 |
Androgen receptor |
None |
9 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
8.5 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
8.5 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
8.5 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
8.5 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
37 |
nM |
IC50 |
TKC206816
|
P10275 |
Androgen receptor |
None |
8.5 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
35 |
nM |
Ki |
TKC206816
|
P10275 |
Androgen receptor |
None |
14 |
nM |
IC50 |
TKC205544
|
P25100 |
Alpha-1D adrenergic receptor |
None |
2 |
nM |
Ki |
TKC205544
|
P25100 |
Alpha-1D adrenergic receptor |
None |
158.48 |
nM |
Ki |
TKC205544
|
P25100 |
Alpha-1D adrenergic receptor |
None |
954.99 |
nM |
Ki |
TKC205544
|
P25100 |
Alpha-1D adrenergic receptor |
None |
289 |
nM |
Ki |
TKC205544
|
P28223 |
5-hydroxytryptamine receptor 2A |
None |
>10000 |
nM |
Ki |
TKC205544
|
P28223 |
5-hydroxytryptamine receptor 2A |
None |
252 |
nM |
Ki |
TKC205544
|
P28223 |
5-hydroxytryptamine receptor 2A |
None |
288.4 |
nM |
Ki |
TKC205544
|
P28223 |
5-hydroxytryptamine receptor 2A |
None |
1000 |
nM |
Ki |
TKC206781
|
P28223 |
5-hydroxytryptamine receptor 2A |
None |
1.4 |
nM |
Ki |
TKC112925
|
P31213 |
3-oxo-5-alpha-steroid 4-dehydrogenase 2 |
None |
84 |
nM |
IC50 |
TKC206770
|
P31213 |
3-oxo-5-alpha-steroid 4-dehydrogenase 2 |
None |
84 |
nM |
IC50 |
TKC013725
|
P35348 |
Alpha-1A adrenergic receptor |
None |
13 |
nM |
IC50 |
TKC100416
|
P35348 |
Alpha-1A adrenergic receptor |
None |
32 |
nM |
Kd |
TKC205544
|
P35348 |
Alpha-1A adrenergic receptor |
None |
398 |
nM |
Kd |
TKC205544
|
P35348 |
Alpha-1A adrenergic receptor |
None |
148 |
nM |
Kd |
TKC205544
|
P35348 |
Alpha-1A adrenergic receptor |
None |
770 |
nM |
Ki |
TKC205544
|
P35348 |
Alpha-1A adrenergic receptor |
None |
199.52 |
nM |
Ki |
TKC205544
|
P35348 |
Alpha-1A adrenergic receptor |
None |
3162.28 |
nM |
Ki |
TKC205544
|
P35348 |
Alpha-1A adrenergic receptor |
None |
1057 |
nM |
Ki |
TKC206544
|
P35348 |
Alpha-1A adrenergic receptor |
None |
>10000 |
nM |
Ki |
TKC023246
|
Q92731 |
Estrogen receptor beta |
None |
>10000 |
nM |
IC50 |
TKC028029
|
Q92731 |
Estrogen receptor beta |
None |
<1 |
% |
Activity |
TKC028037
|
Q92731 |
Estrogen receptor beta |
None |
10 |
% |
Activity |
TKC035272
|
Q92731 |
Estrogen receptor beta |
None |
>50000 |
nM |
IC50 |
TKC100932
|
Q92731 |
Estrogen receptor beta |
None |
25300 |
nM |
EC50 |
TKC101365
|
Q92731 |
Estrogen receptor beta |
None |
17690 |
nM |
EC50 |
TKC102448
|
Q92731 |
Estrogen receptor beta |
None |
4680 |
nM |
EC50 |
TKC106878
|
Q92731 |
Estrogen receptor beta |
None |
>10000 |
nM |
IC50 |
TKC110673
|
Q92731 |
Estrogen receptor beta |
None |
2.78E+11 |
M-1 |
Ka |
TKC111721
|
Q92731 |
Estrogen receptor beta |
None |
1520000000 |
M-1 |
Ka |
TKC111727
|
Q92731 |
Estrogen receptor beta |
None |
614000000 |
M-1 |
Ka |
TKC111727
|
Q92731 |
Estrogen receptor beta |
None |
0 |
nM |
EC50 |
TKC111738
|
Q92731 |
Estrogen receptor beta |
None |
2 |
nM |
EC50 |
TKC111738
|
Q92731 |
Estrogen receptor beta |
None |
4 |
% |
RSA |
TKC111738
|
Q92731 |
Estrogen receptor beta |
None |
26 |
nM |
IC50 |
TKC111738
|
Q92731 |
Estrogen receptor beta |
None |
540 |
nM |
IC50 |
TKC111738
|
Q92731 |
Estrogen receptor beta |
None |
8 |
nM |
EC50 |
TKC112923
|
Q92731 |
Estrogen receptor beta |
None |
6 |
nM |
EC50 |
TKC206608
|
Q92731 |
Estrogen receptor beta |
None |
4280 |
nM |
EC50 |
TKC206725
|
Q92731 |
Estrogen receptor beta |
None |
24 |
nM |
Ki |
TKC206726
|
Q92731 |
Estrogen receptor beta |
None |
11 |
nM |
EC50 |
TKC206759
|
Q92731 |
Estrogen receptor beta |
None |
>10000 |
nM |
IC50 |
TKC206759
|
Q92731 |
Estrogen receptor beta |
None |
>10000 |
nM |
IC50 |
TKC206764
|
Q92731 |
Estrogen receptor beta |
None |
1 |
% |
RBA |
TKC206765
|
Q92731 |
Estrogen receptor beta |
None |
18000000 |
M-1 |
Ka |
TKC206769
|
Q92731 |
Estrogen receptor beta |
None |
27000000 |
M-1 |
Ka |
TKC206812
|
Q92731 |
Estrogen receptor beta |
None |
>5000 |
nM |
IC50 |
TKC206816
|
Q92731 |
Estrogen receptor beta |
None |
1000000 |
nM |
IC50 |