TKC039202
|
P13612 |
Integrin alpha-4 |
None |
3150 |
nM |
EC50 |
TKC009214
|
P14867 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
None |
-21 |
% |
Activity |
TKC009484
|
P14867 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
None |
29 |
% |
Activity |
TKC009488
|
P14867 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
None |
9 |
% |
Activity |
TKC009489
|
P14867 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
None |
24 |
% |
Activity |
TKC021304
|
P14867 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
None |
91 |
% |
Activity |
TKC086929
|
P14867 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
None |
226 |
% |
Activity |
TKC095084
|
P14867 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
None |
91 |
% |
Activity |
TKC130495
|
P14867 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
None |
280 |
% |
Activity |
TKC136411
|
P14867 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
None |
19000 |
nM |
EC50 |
TKC206157
|
P14867 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
None |
-30 |
% |
Activity |
TKC206777
|
P14867 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
None |
22 |
nM |
IC50 |
TKC206777
|
P14867 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
None |
160 |
nM |
EC50 |
TKC034640
|
P21397 |
Amine oxidase [flavin-containing] A |
None |
>1000000 |
nM |
Ki |
TKC146423
|
P21397 |
Amine oxidase [flavin-containing] A |
None |
170000 |
nM |
IC50 |
TKC205544
|
P28221 |
5-hydroxytryptamine receptor 1D |
None |
40 |
nM |
Ki |
TKC205544
|
P28221 |
5-hydroxytryptamine receptor 1D |
None |
59 |
nM |
Ki |
TKC205544
|
P28221 |
5-hydroxytryptamine receptor 1D |
None |
15.84 |
nM |
Ki |
TKC205544
|
P28221 |
5-hydroxytryptamine receptor 1D |
None |
19.95 |
nM |
Ki |
TKC206544
|
P28221 |
5-hydroxytryptamine receptor 1D |
None |
>10000 |
nM |
Ki |
TKC020967
|
P29466 |
Caspase-1 |
None |
1080 |
nM |
IC50 |
TKC035272
|
P29466 |
Caspase-1 |
None |
12589 |
nM |
Potency |
TKC035272
|
P29466 |
Caspase-1 |
None |
1230 |
nM |
IC50 |
TKC036497
|
P29466 |
Caspase-1 |
None |
100000 |
nM |
IC50 |
TKC042585
|
P29466 |
Caspase-1 |
None |
30000 |
nM |
MIC50 |
TKC042586
|
P29466 |
Caspase-1 |
None |
30000 |
nM |
MIC50 |
TKC042587
|
P29466 |
Caspase-1 |
None |
30000 |
nM |
MIC50 |
TKC096499
|
P29466 |
Caspase-1 |
None |
90000 |
nM |
IC50 |
TKC149924
|
P29466 |
Caspase-1 |
None |
4 |
/s |
Kinact |
TKC019353
|
P46098 |
5-hydroxytryptamine receptor 3A |
None |
141254 |
nM |
IC50 |
TKC019571
|
P46098 |
5-hydroxytryptamine receptor 3A |
None |
257040 |
nM |
IC50 |
TKC206544
|
P46098 |
5-hydroxytryptamine receptor 3A |
None |
>10000 |
nM |
Ki |
TKC046324
|
P49840 |
Glycogen synthase kinase-3 alpha |
None |
1600 |
nM |
IC50 |
TKC118938
|
Q05586 |
Glutamate receptor ionotropic, NMDA 1 |
None |
150 |
nM |
EC50 |
TKC206917
|
Q05586 |
Glutamate receptor ionotropic, NMDA 1 |
None |
55 |
nM |
EC50 |
TKC206783
|
Q12879 |
Glutamate receptor ionotropic, NMDA 2A |
None |
21000 |
nM |
EC50 |
TKC206783
|
Q13224 |
Glutamate receptor ionotropic, NMDA 2B |
None |
33000 |
nM |
EC50 |
TKC206544
|
Q14416 |
Metabotropic glutamate receptor 2 |
None |
>10000 |
nM |
Ki |
TKC112754
|
Q9Y6A2 |
Cholesterol 24-hydroxylase |
None |
56 |
% |
Activity |
TKC112826
|
Q9Y6A2 |
Cholesterol 24-hydroxylase |
None |
53 |
% |
Activity |
TKC112827
|
Q9Y6A2 |
Cholesterol 24-hydroxylase |
None |
30 |
% |
Activity |
TKC113159
|
Q9Y6A2 |
Cholesterol 24-hydroxylase |
None |
32 |
% |
Activity |
TKC119202
|
Q9Y6A2 |
Cholesterol 24-hydroxylase |
None |
50 |
nM |
Kd |
TKC122884
|
Q9Y6A2 |
Cholesterol 24-hydroxylase |
None |
670 |
nM |
Kd |
TKC206783
|
Q9Y6A2 |
Cholesterol 24-hydroxylase |
None |
2500 |
nM |
Ki |