|
TKC151761
|
P00519 |
Tyrosine-protein kinase ABL1 |
None |
>10000 |
nM |
IC50 |
|
TKC200866
|
P00519 |
Tyrosine-protein kinase ABL1 |
None |
>10000 |
nM |
IC50 |
|
TKC055903
|
P00734 |
Prothrombin |
None |
4 |
nM |
IC50 |
|
TKC055903
|
P00734 |
Prothrombin |
None |
50 |
nM |
IC50 |
|
TKC064786
|
P00734 |
Prothrombin |
None |
130 |
nM |
IC50 |
|
TKC064787
|
P00734 |
Prothrombin |
None |
70 |
nM |
IC50 |
|
TKC101989
|
P00734 |
Prothrombin |
None |
4000 |
nM |
IC50 |
|
TKC106074
|
P00734 |
Prothrombin |
None |
>50000 |
nM |
IC50 |
|
TKC106074
|
P00734 |
Prothrombin |
None |
>50000 |
nM |
IC50 |
|
TKC122980
|
P00734 |
Prothrombin |
None |
9200 |
nM |
IC50 |
|
TKC139119
|
P00734 |
Prothrombin |
None |
90 |
nM |
IC50 |
|
TKC141433
|
P00734 |
Prothrombin |
None |
18 |
nM |
IC50 |
|
TKC000611
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
40000 |
nM |
IC50 |
|
TKC001618
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
34000 |
nM |
IC50 |
|
TKC009896
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
791100 |
nM |
IC50 |
|
TKC019819
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
48 |
% |
Inhibition |
|
TKC019859
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
54 |
% |
Inhibition |
|
TKC020491
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
4000 |
nM |
IC50 |
|
TKC020796
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
30 |
% |
Inhibition |
|
TKC021940
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
40 |
% |
Inhibition |
|
TKC022833
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
43 |
% |
Inhibition |
|
TKC022834
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
43 |
% |
Inhibition |
|
TKC022961
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
44 |
% |
Inhibition |
|
TKC024587
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
3300 |
nM |
IC50 |
|
TKC024587
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
3300 |
nM |
IC50 |
|
TKC031258
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
3600 |
nM |
IC50 |
|
TKC034201
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>200000 |
nM |
IC50 |
|
TKC034358
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
39000 |
nM |
IC50 |
|
TKC034359
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
39000 |
nM |
IC50 |
|
TKC036372
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
14000 |
nM |
IC50 |
|
TKC037595
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
36000 |
nM |
IC50 |
|
TKC043613
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
43000 |
nM |
IC50 |
|
TKC049750
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>50000 |
nM |
IC50 |
|
TKC049818
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
44 |
ug |
IC50 |
|
TKC054011
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
8800 |
nM |
IC50 |
|
TKC054031
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>50000 |
nM |
IC50 |
|
TKC054081
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>50000 |
nM |
IC50 |
|
TKC054090
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
7500 |
nM |
IC50 |
|
TKC054099
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
8800 |
nM |
IC50 |
|
TKC054100
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
8900 |
nM |
IC50 |
|
TKC054101
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
7600 |
nM |
IC50 |
|
TKC054240
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
7800 |
nM |
IC50 |
|
TKC054241
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
6300 |
nM |
IC50 |
|
TKC056482
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
210000 |
nM |
IC50 |
|
TKC060184
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
8300 |
nM |
IC50 |
|
TKC060216
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>50000 |
nM |
IC50 |
|
TKC060284
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>50000 |
nM |
IC50 |
|
TKC060302
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>50000 |
nM |
IC50 |
|
TKC060303
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
7800 |
nM |
IC50 |
|
TKC060304
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
8000 |
nM |
IC50 |
|
TKC060399
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>50000 |
nM |
IC50 |
|
TKC060602
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
5900 |
nM |
IC50 |
|
TKC066954
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
38 |
% |
Inhibition |
|
TKC068533
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
28000 |
nM |
IC50 |
|
TKC071010
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>50000 |
nM |
IC50 |
|
TKC077689
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
380000 |
nM |
IC50 |
|
TKC077689
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
380000 |
nM |
IC50 |
|
TKC095276
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
48 |
% |
Inhibition |
|
TKC113936
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
65 |
% |
Inhibition |
|
TKC122543
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
35 |
% |
Inhibition |
|
TKC130084
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
39 |
% |
Inhibition |
|
TKC130119
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
33 |
% |
Inhibition |
|
TKC130577
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
<43 |
% |
Inhibition |
|
TKC130901
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
36 |
% |
Inhibition |
|
TKC133309
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>200000 |
nM |
IC50 |
|
TKC133517
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
1300 |
nM |
IC50 |
|
TKC133656
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>200000 |
nM |
IC50 |
|
TKC134278
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>200000 |
nM |
IC50 |
|
TKC139036
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>50000 |
nM |
IC50 |
|
TKC140627
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>50000 |
nM |
IC50 |
|
TKC141365
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>50000 |
nM |
IC50 |
|
TKC143641
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
>50000 |
nM |
IC50 |
|
TKC151113
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
116400 |
nM |
IC50 |
|
TKC151284
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
51 |
% |
Inhibition |
|
TKC151765
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
48 |
% |
Inhibition |
|
TKC151792
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
14000 |
nM |
IC50 |
|
TKC172853
|
P23219 |
Prostaglandin G/H synthase 1 |
None |
43700 |
nM |
IC50 |
|
TKC072774
|
Q08828 |
Adenylate cyclase type 1 |
None |
150 |
nM |
IC50 |
|
TKC100973
|
Q08828 |
Adenylate cyclase type 1 |
None |
150 |
nM |
IC50 |
|
TKC103970
|
Q08828 |
Adenylate cyclase type 1 |
None |
150 |
nM |
IC50 |
|
TKC105066
|
Q08828 |
Adenylate cyclase type 1 |
None |
150 |
nM |
IC50 |
|
TKC105796
|
Q08828 |
Adenylate cyclase type 1 |
None |
150 |
nM |
IC50 |
|
TKC105904
|
Q08828 |
Adenylate cyclase type 1 |
None |
150 |
nM |
IC50 |
|
TKC108085
|
Q08828 |
Adenylate cyclase type 1 |
None |
150 |
nM |
IC50 |
|
TKC206549
|
Q08828 |
Adenylate cyclase type 1 |
None |
41 |
nM |
IC50 |
|
TKC206783
|
Q12879 |
Glutamate receptor ionotropic, NMDA 2A |
None |
21000 |
nM |
EC50 |