TKC205544
|
P14416 |
D(2) dopamine receptor |
None |
687 |
nM |
Ki |
TKC205544
|
P14416 |
D(2) dopamine receptor |
None |
280 |
nM |
Ki |
TKC205544
|
P14416 |
D(2) dopamine receptor |
None |
398.1 |
nM |
Ki |
TKC206544
|
P14416 |
D(2) dopamine receptor |
None |
>10000 |
nM |
Ki |
TKC005313
|
P21728 |
D(1A) dopamine receptor |
None |
517 |
nM |
Potency |
TKC035272
|
P21728 |
D(1A) dopamine receptor |
None |
12589 |
nM |
Potency |
TKC035984
|
P21728 |
D(1A) dopamine receptor |
None |
20 |
nM |
Potency |
TKC084630
|
P21728 |
D(1A) dopamine receptor |
None |
14125 |
nM |
Potency |
TKC092297
|
P21728 |
D(1A) dopamine receptor |
None |
2909 |
nM |
Potency |
TKC205544
|
P21728 |
D(1A) dopamine receptor |
None |
2909 |
nM |
Potency |
TKC205544
|
P21728 |
D(1A) dopamine receptor |
None |
>10000 |
nM |
Ki |
TKC206544
|
P21728 |
D(1A) dopamine receptor |
None |
>10000 |
nM |
Ki |
TKC206622
|
P21728 |
D(1A) dopamine receptor |
None |
231 |
nM |
Potency |
TKC206690
|
P21728 |
D(1A) dopamine receptor |
None |
26 |
nM |
Potency |
TKC206777
|
P21728 |
D(1A) dopamine receptor |
None |
23109 |
nM |
Potency |
TKC206816
|
P21728 |
D(1A) dopamine receptor |
None |
14125 |
nM |
Potency |
TKC002194
|
P35372 |
Mu-type opioid receptor |
None |
760 |
nM |
Ke |
TKC005708
|
P35372 |
Mu-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC093001
|
P35372 |
Mu-type opioid receptor |
None |
10000 |
nM |
Ki |
TKC093006
|
P35372 |
Mu-type opioid receptor |
None |
>1000 |
nM |
Ki |
TKC093006
|
P35372 |
Mu-type opioid receptor |
None |
>1000 |
nM |
Ki |
TKC093010
|
P35372 |
Mu-type opioid receptor |
None |
41 |
nM |
Ki |
TKC093012
|
P35372 |
Mu-type opioid receptor |
None |
390 |
nM |
Ki |
TKC101289
|
P35372 |
Mu-type opioid receptor |
None |
>5800 |
nM |
Ki |
TKC101290
|
P35372 |
Mu-type opioid receptor |
None |
777 |
nM |
Ki |
TKC104953
|
P35372 |
Mu-type opioid receptor |
None |
3650 |
nM |
Ke |
TKC105684
|
P35372 |
Mu-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC105685
|
P35372 |
Mu-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC109881
|
P35372 |
Mu-type opioid receptor |
None |
>92466 |
nM |
EC50 |
TKC156630
|
P35372 |
Mu-type opioid receptor |
None |
>1900 |
nM |
Ki |
TKC206544
|
P35372 |
Mu-type opioid receptor |
None |
>0 |
% |
Emax |
TKC206544
|
P35372 |
Mu-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC206544
|
P35372 |
Mu-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC206544
|
P35372 |
Mu-type opioid receptor |
None |
4370 |
nM |
Ki |
TKC206544
|
P35372 |
Mu-type opioid receptor |
None |
>1000 |
nM |
Ki |
TKC206544
|
P35372 |
Mu-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC206544
|
P35372 |
Mu-type opioid receptor |
None |
2860 |
nM |
EC50 |
TKC206544
|
P35372 |
Mu-type opioid receptor |
None |
1370 |
nM |
Ki |
TKC206544
|
P35372 |
Mu-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC205544
|
P35462 |
D(3) dopamine receptor |
None |
2489 |
nM |
Ki |
TKC205544
|
P35462 |
D(3) dopamine receptor |
None |
3981.07 |
nM |
Ki |
TKC206544
|
P35462 |
D(3) dopamine receptor |
None |
>10000 |
nM |
Ki |
TKC002194
|
P41143 |
Delta-type opioid receptor |
None |
2830 |
nM |
Ke |
TKC005708
|
P41143 |
Delta-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC045774
|
P41143 |
Delta-type opioid receptor |
None |
>64582 |
nM |
EC50 |
TKC093001
|
P41143 |
Delta-type opioid receptor |
None |
10000 |
nM |
Ki |
TKC093006
|
P41143 |
Delta-type opioid receptor |
None |
6690 |
nM |
Ki |
TKC093006
|
P41143 |
Delta-type opioid receptor |
None |
6690 |
nM |
Ki |
TKC093010
|
P41143 |
Delta-type opioid receptor |
None |
1017 |
nM |
Ki |
TKC093012
|
P41143 |
Delta-type opioid receptor |
None |
2840 |
nM |
Ki |
TKC101289
|
P41143 |
Delta-type opioid receptor |
None |
>5000 |
nM |
Ki |
TKC101290
|
P41143 |
Delta-type opioid receptor |
None |
>5000 |
nM |
Ki |
TKC104953
|
P41143 |
Delta-type opioid receptor |
None |
964 |
nM |
Ke |
TKC105684
|
P41143 |
Delta-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC105685
|
P41143 |
Delta-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC109881
|
P41143 |
Delta-type opioid receptor |
None |
>92466 |
nM |
EC50 |
TKC109881
|
P41143 |
Delta-type opioid receptor |
None |
>92466 |
nM |
EC50 |
TKC156630
|
P41143 |
Delta-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC206544
|
P41143 |
Delta-type opioid receptor |
None |
3990 |
nM |
Ki |
TKC206544
|
P41143 |
Delta-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC206544
|
P41143 |
Delta-type opioid receptor |
None |
5790 |
nM |
Ki |
TKC206544
|
P41143 |
Delta-type opioid receptor |
None |
5790 |
nM |
Ki |
TKC206544
|
P41143 |
Delta-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC206544
|
P41143 |
Delta-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC206544
|
P41143 |
Delta-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC206544
|
P41143 |
Delta-type opioid receptor |
None |
>10000 |
nM |
Ki |
TKC004780
|
P41145 |
Kappa-type opioid receptor |
None |
1 |
nM |
Ki |
TKC004780
|
P41145 |
Kappa-type opioid receptor |
None |
140 |
nM |
Ki |
TKC004780
|
P41145 |
Kappa-type opioid receptor |
None |
4.6 |
nM |
Ki |
TKC004780
|
P41145 |
Kappa-type opioid receptor |
None |
31.6 |
nM |
Ki |
TKC005708
|
P41145 |
Kappa-type opioid receptor |
None |
390 |
nM |
Ki |
TKC080736
|
P41145 |
Kappa-type opioid receptor |
None |
>2000 |
nM |
EC50 |
TKC093001
|
P41145 |
Kappa-type opioid receptor |
None |
17 |
nM |
Ki |
TKC093006
|
P41145 |
Kappa-type opioid receptor |
None |
2 |
nM |
Ki |
TKC093006
|
P41145 |
Kappa-type opioid receptor |
None |
7.2 |
nM |
Ki |
TKC093006
|
P41145 |
Kappa-type opioid receptor |
None |
1.8 |
nM |
Ki |
TKC093008
|
P41145 |
Kappa-type opioid receptor |
None |
5 |
nM |
Ki |
TKC093010
|
P41145 |
Kappa-type opioid receptor |
None |
0 |
nM |
EC50 |
TKC093011
|
P41145 |
Kappa-type opioid receptor |
None |
2 |
nM |
Ki |
TKC093012
|
P41145 |
Kappa-type opioid receptor |
None |
0 |
nM |
EC50 |
TKC093013
|
P41145 |
Kappa-type opioid receptor |
None |
2 |
nM |
Ki |
TKC093014
|
P41145 |
Kappa-type opioid receptor |
None |
147 |
nM |
Ki |
TKC093016
|
P41145 |
Kappa-type opioid receptor |
None |
35 |
nM |
Ki |
TKC093018
|
P41145 |
Kappa-type opioid receptor |
None |
2 |
nM |
Ki |
TKC093019
|
P41145 |
Kappa-type opioid receptor |
None |
141 |
nM |
Ki |
TKC093021
|
P41145 |
Kappa-type opioid receptor |
None |
29 |
nM |
Ki |
TKC093022
|
P41145 |
Kappa-type opioid receptor |
None |
31 |
nM |
Ki |
TKC093023
|
P41145 |
Kappa-type opioid receptor |
None |
3 |
nM |
Ki |
TKC093024
|
P41145 |
Kappa-type opioid receptor |
None |
4 |
nM |
Ki |
TKC093025
|
P41145 |
Kappa-type opioid receptor |
None |
>81 |
% |
Emax |
TKC101289
|
P41145 |
Kappa-type opioid receptor |
None |
10 |
nM |
EC50 |
TKC101289
|
P41145 |
Kappa-type opioid receptor |
None |
1233 |
nM |
Ki |
TKC101290
|
P41145 |
Kappa-type opioid receptor |
None |
7 |
nM |
Ki |
TKC103606
|
P41145 |
Kappa-type opioid receptor |
None |
0 |
nM |
Ki |
TKC104953
|
P41145 |
Kappa-type opioid receptor |
None |
7 |
nM |
EC50 |
TKC104953
|
P41145 |
Kappa-type opioid receptor |
None |
424 |
nM |
Ki |
TKC104956
|
P41145 |
Kappa-type opioid receptor |
None |
41 |
nM |
Ki |
TKC105684
|
P41145 |
Kappa-type opioid receptor |
None |
6 |
nM |
Ki |
TKC105684
|
P41145 |
Kappa-type opioid receptor |
None |
3 |
nM |
EC50 |
TKC105685
|
P41145 |
Kappa-type opioid receptor |
None |
300 |
nM |
Ki |
TKC106987
|
P41145 |
Kappa-type opioid receptor |
None |
641 |
nM |
Ki |
TKC106989
|
P41145 |
Kappa-type opioid receptor |
None |
>1000 |
nM |
Ki |
TKC156630
|
P41145 |
Kappa-type opioid receptor |
None |
1900 |
nM |
Ki |
TKC206540
|
P41145 |
Kappa-type opioid receptor |
None |
>0 |
% |
Emax |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
0 |
nM |
EC50 |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
16 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
10 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
38 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
1.3 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
0.75 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
40 |
nM |
EC50 |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
7.4 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
0.36 |
nM |
EC50 |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
40 |
nM |
EC50 |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
0.03 |
nM |
EC50 |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
1.7 |
nM |
EC50 |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
45 |
nM |
EC50 |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
1.9 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
1.3 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
2.82 |
nM |
EC50 |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
1.24 |
nM |
EC50 |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
1.3 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
2.5 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
7.5 |
nM |
EC50 |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
7.4 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
3 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
45 |
nM |
EC50 |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
2.4 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
0.21 |
nM |
EC50 |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
0.8 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
1.9 |
nM |
Ki |
TKC206544
|
P41145 |
Kappa-type opioid receptor |
None |
10 |
nM |
EC50 |